Page last updated: 2024-09-03

ym 12617 and Muscle Contraction

ym 12617 has been researched along with Muscle Contraction in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19905 (55.56)18.7374
1990's4 (44.44)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Blaylock, NA; Wilson, VG2
Guarneri, L; Leonardi, A; Poggesi, E; Simonazzi, I; Taddei, C; Testa, R1
Andersson, KE; Hedlund, H; Holmquist, F1
Honda, K; Miyata-Osawa, A; Shiono, K; Takenaka, T; Terai, M1
Furukawa, A; Kameda, H; Konno, F; Kubo, H; Takayanagi, I; Toyoda, T1
Honda, K; Nakagawa, C; Terai, M1
Itoh, T; Kuriyama, H; Nishiye, E; Seki, N; Suzuki, H1
Daly, CJ; Dunn, WR; McGrath, JC; Wilson, VG1

Other Studies

9 other study(ies) available for ym 12617 and Muscle Contraction

ArticleYear
Pharmacological characterization of noradrenaline-induced contractions of the porcine isolated palmar lateral vein and palmar common digital artery.
    British journal of pharmacology, 1995, Volume: 114, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Arteries; Berberine; Drug Interactions; Drug Synergism; Forelimb; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Prazosin; Receptors, Adrenergic, alpha; Reproducibility of Results; Sulfonamides; Swine; Veins; Yohimbine

1995
Mediation of noradrenaline-induced contractions of rat aorta by the alpha 1B-adrenoceptor subtype.
    British journal of pharmacology, 1995, Volume: 114, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Clonidine; Computer Simulation; Hippocampus; In Vitro Techniques; Liver; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phentolamine; Piperazines; Prazosin; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Regression Analysis; Spiperone; Stereoisomerism; Sulfonamides

1995
Preliminary evidence for noradrenaline and ATP as neurotransmitters in the porcine isolated palmar common digital artery.
    Journal of neural transmission. Supplementum, 1991, Volume: 34

    Topics: Adenosine Triphosphate; Adrenergic alpha-Antagonists; Animals; Arteries; Electric Stimulation; Forelimb; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Neurotransmitter Agents; Norepinephrine; Phentolamine; Receptors, Adrenergic, alpha; Receptors, Purinergic; Sulfonamides; Swine

1991
Effects of the alpha 1-adrenoceptor antagonist R-(-)-YM12617 on isolated human penile erectile tissue and vas deferens.
    European journal of pharmacology, 1990, Sep-04, Volume: 186, Issue:1

    Topics: Adrenergic alpha-Antagonists; Aged; Electric Stimulation; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Norepinephrine; Penile Erection; Penis; Prazosin; Sulfonamides; Vas Deferens

1990
Studies on YM-12617: a selective and potent antagonist of postsynaptic alpha 1-adrenoceptors.
    Naunyn-Schmiedeberg's archives of pharmacology, 1985, Volume: 328, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Blood Pressure; Brain; Brimonidine Tartrate; Clonidine; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Phenylephrine; Pulmonary Artery; Quinoxalines; Rabbits; Rats; Receptors, Adrenergic, alpha; Sulfonamides; Tritium; Vas Deferens

1985
A difference in mode of antagonism between optical isomers of a potent selective alpha 1-adrenoceptor blocker (YM-12617) and norepinephrine in isolated rabbit iris dilator and aorta.
    Japanese journal of pharmacology, 1986, Volume: 42, Issue:4

    Topics: Adrenergic alpha-Antagonists; Animals; Aorta; Dose-Response Relationship, Drug; In Vitro Techniques; Iris; Male; Muscle Contraction; Norepinephrine; Rabbits; Stereoisomerism; Sulfonamides

1986
Further studies on (+/-)-YM-12617, a potent and selective alpha 1-adrenoceptor antagonist and its individual optical enantiomers.
    Naunyn-Schmiedeberg's archives of pharmacology, 1987, Volume: 336, Issue:3

    Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Decerebrate State; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Rabbits; Rats; Receptors, Adrenergic, alpha; Stereoisomerism; Sulfonamides

1987
Electrical and mechanical properties of the capsular smooth muscles of the rabbit prostate in relation to the actions of the alpha 1-adrenoceptor blocker, YM-12617.
    British journal of pharmacology, 1988, Volume: 93, Issue:3

    Topics: Acetylcholine; Adrenergic alpha-Antagonists; Animals; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Prazosin; Prostate; Rabbits; Receptors, Adrenergic, alpha; Sulfonamides

1988
An attempt at selective protection from phenoxybenzamine of postjunctional alpha-adrenoceptor subtypes mediating contractions to noradrenaline in the rabbit isolated saphenous vein.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Adrenergic alpha-Antagonists; Animals; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenoxybenzamine; Prazosin; Rabbits; Receptors, Adrenergic, alpha; Saphenous Vein; Sulfonamides; Yohimbine

1988