Page last updated: 2024-09-05

vx-745 and Adjuvant Arthritis

vx-745 has been researched along with Adjuvant Arthritis in 3 studies

Research

Studies (3)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (33.33)29.6817
2010's2 (66.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Balagué, C; Caturla, F; Domínguez, M; Esteve, C; Godessart, N; Huerta, JM; Lumeras, W; Orellana, A; Roca, R; Vidal, B; Vidal, L1
Balagué, C; Caturla, F; Domínguez, M; Lumeras, W; Maldonado, M; Orellana, A; Segarra, V; Vidal, B; Vidal, L1
Allémann, E; Doelker, E; Gabay, C; Jordan, O; Maudens, P; Pradal, J; Seemayer, CA; Waldburger, JM; Zuluaga, MF1

Other Studies

3 other study(ies) available for vx-745 and Adjuvant Arthritis

ArticleYear
Design, synthesis, and structure-activity relationships of aminopyridine N-oxides, a novel scaffold for the potent and selective inhibition of p38 mitogen activated protein kinase.
    Journal of medicinal chemistry, 2009, Sep-10, Volume: 52, Issue:17

    Topics: Aminopyridines; Animals; Arthritis, Experimental; Catalytic Domain; Cell Line; Drug Design; Humans; Inhibitory Concentration 50; Male; Models, Molecular; Oxides; p38 Mitogen-Activated Protein Kinases; Protein Kinase Inhibitors; Rats; Rats, Wistar; Structure-Activity Relationship; Substrate Specificity; Tumor Necrosis Factor-alpha

2009
1,7-Naphthyridine 1-oxides as novel potent and selective inhibitors of p38 mitogen activated protein kinase.
    Journal of medicinal chemistry, 2011, Nov-24, Volume: 54, Issue:22

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Binding Sites; Cell Line; Crystallography, X-Ray; Humans; Inflammation; Lipopolysaccharides; Male; Mice; Microsomes, Liver; Monocytes; Naphthyridines; p38 Mitogen-Activated Protein Kinases; Protein Binding; Protein Conformation; Rats; Rats, Wistar; Structure-Activity Relationship; Tumor Necrosis Factor-alpha

2011
Intra-articular bioactivity of a p38 MAPK inhibitor and development of an extended-release system.
    European journal of pharmaceutics and biopharmaceutics : official journal of Arbeitsgemeinschaft fur Pharmazeutische Verfahrenstechnik e.V, 2015, Volume: 93

    Topics: Animals; Anti-Inflammatory Agents; Arthritis, Experimental; Cells, Cultured; Chemistry, Pharmaceutical; Delayed-Action Preparations; Diffusion; Drug Carriers; Humans; Injections, Intra-Articular; Joints; Kinetics; Male; Mice, Inbred C57BL; p38 Mitogen-Activated Protein Kinases; Particle Size; Polymers; Protein Kinase Inhibitors; Pyridazines; Pyrimidines; Solubility; Synovial Membrane; Technology, Pharmaceutical

2015