Page last updated: 2024-08-26

u 69593 and Muscle Contraction

u 69593 has been researched along with Muscle Contraction in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19902 (16.67)18.7374
1990's6 (50.00)18.2507
2000's4 (33.33)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Ananthan, S; Bartlett, JL; Bilsky, EJ; Davis, P; Dersch, CM; Khare, NK; Porreca, F; Rothman, RB; Saini, SK; Seitz, LE1
Arvidsson, S; Bayati, A; Ekman, C; Larsson, M1
Levendusky, MC; Levin, RM; Longhurst, PA; Matsumoto, S; Millington, WR1
Beattie, DT; Cheruvu, M; Johnson-Rabidoux, S; Kaufman, E; Mai, N; O'Keefe, M; Peterson, C; Vickery, R1
Davis, P; DeLeon, IA; Hruby, VJ; Li, G; Lou, BS; Lung, FD; Meyer, JP; Porreca, F; Xiang, L; Yamamura, HI1
Demedts, MG; Dupont, LJ; Pype, JL; Verleden, GM1
Corbett, AD; Davies, MR; Glen, T; Menzies, JR; Paterson, SJ1
Gu, ZF; Jensen, RT; Maton, PN; Pradhan, T; Zhang, L1
Birch, PJ; Hayes, AG; Hayward, NJ; Judd, DB; Naylor, A; Rogers, H; Scopes, DI; Sheehan, MJ; Tyers, MB1
Dissanayake, VU; Hill, RG; Hughes, J; Hunter, JC1
Bruce, DS; Nuchols, PA; Oeltgen, PR; Spurrier, WA; Su, TP; Welborn, JR1
Birch, PP; Cavicchini, E; Hayes, AG1

Other Studies

12 other study(ies) available for u 69593 and Muscle Contraction

ArticleYear
Identification of opioid ligands possessing mixed micro agonist/delta antagonist activity among pyridomorphinans derived from naloxone, oxymorphone, and hydromorphone [correction of hydropmorphone].
    Journal of medicinal chemistry, 2004, Mar-11, Volume: 47, Issue:6

    Topics: Analgesics; Animals; Binding Sites; Brain; Drug Tolerance; Electric Stimulation; Guinea Pigs; Hydromorphone; Ileum; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred ICR; Morphinans; Muscle Contraction; Muscle, Smooth; Naloxone; Oxymorphone; Pyridines; Radioligand Assay; Rats; Receptors, Opioid, delta; Receptors, Opioid, mu; Vas Deferens

2004
A model for chronic quantitative studies of colorectal sensitivity using balloon distension in conscious mice -- effects of opioid receptor agonists.
    Neurogastroenterology and motility, 2003, Volume: 15, Issue:4

    Topics: Abdominal Muscles; Analgesics, Opioid; Animals; Benzeneacetamides; Colon; Consciousness; Electromyography; Female; Fentanyl; Male; Mice; Models, Animal; Muscle Contraction; Nociceptors; Pain Measurement; Physical Stimulation; Pyrrolidines; Receptors, Opioid; Rectum; Sex Characteristics

2003
Activation of mu opioid receptors in the ventrolateral periaqueductal gray inhibits reflex micturition in anesthetized rats.
    Neuroscience letters, 2004, Jun-10, Volume: 363, Issue:2

    Topics: Administration, Intravesical; Anesthetics; Animals; Benzeneacetamides; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Female; Microinjections; Morphine; Muscle Contraction; Narcotics; Periaqueductal Gray; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, kappa; Receptors, Opioid, mu; Reflex; Sodium Chloride; Urinary Bladder; Urination

2004
The in vitro pharmacology of the peripherally restricted opioid receptor antagonists, alvimopan, ADL 08-0011 and methylnaltrexone.
    Naunyn-Schmiedeberg's archives of pharmacology, 2007, Volume: 375, Issue:3

    Topics: Analgesics, Opioid; Animals; Benzeneacetamides; CHO Cells; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Guanosine 5'-O-(3-Thiotriphosphate); Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Morphine; Muscle Contraction; Naltrexone; Narcotic Antagonists; Oligopeptides; Piperidines; Pyrrolidines; Quaternary Ammonium Compounds; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Recombinant Proteins; Transfection

2007
Effects of modifications of residues in position 3 of dynorphin A(1-11)-NH2 on kappa receptor selectivity and potency.
    Journal of medicinal chemistry, 1996, Jun-21, Volume: 39, Issue:13

    Topics: Amino Acid Sequence; Analgesics; Animals; Benzeneacetamides; Brain; Dynorphins; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalins; Guinea Pigs; Ileum; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Peptide Fragments; Protein Binding; Protein Conformation; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Structure-Activity Relationship

1996
Opioids modulate the cholinergic contraction but not the nonadrenergic relaxation in guinea-pig airways in vitro.
    The European respiratory journal, 1996, Volume: 9, Issue:11

    Topics: Animals; Benzeneacetamides; Cholinergic Fibers; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Pyrrolidines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Trachea

1996
In vitro agonist effects of nociceptin and [Phe(1)psi(CH(2)-NH)Gly(2)]nociceptin(1-13)NH(2) in the mouse and rat colon and the mouse vas deferens.
    European journal of pharmacology, 1999, Dec-03, Volume: 385, Issue:2-3

    Topics: Animals; Benzeneacetamides; Benzofurans; Colon; Dose-Response Relationship, Drug; Electric Stimulation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; In Vitro Techniques; Ligands; Male; Mice; Mice, Inbred DBA; Muscle Contraction; Narcotic Antagonists; Nociceptin; Nociceptin Receptor; Opioid Peptides; Peptide Fragments; Pyrrolidines; Rats; Rats, Wistar; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tetrodotoxin; Vas Deferens

1999
Characterization of opioid receptors on smooth muscle cells from guinea pig stomach.
    The American journal of physiology, 1992, Volume: 262, Issue:3 Pt 1

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Animals; Benzeneacetamides; Binding, Competitive; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalins; Gastric Mucosa; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Naloxone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid; Stomach

1992
A series of novel, highly potent and selective agonists for the kappa-opioid receptor.
    British journal of pharmacology, 1990, Volume: 101, Issue:4

    Topics: Abdomen; Analgesics; Animals; Benzeneacetamides; Cricetinae; Electric Stimulation; In Vitro Techniques; Male; Mesocricetus; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Naloxone; Narcotic Antagonists; Pyrrolidines; Rabbits; Rats; Receptors, Opioid; Receptors, Opioid, kappa; Urination; Vas Deferens

1990
Characterization of kappa-opioid receptors in the guinea-pig ileum.
    European journal of pharmacology, 1990, Jun-21, Volume: 182, Issue:1

    Topics: Animals; Benzeneacetamides; Benzomorphans; Binding, Competitive; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, D-Penicillamine (2,5)-; Enkephalin, Leucine; Enkephalin, Leucine-2-Alanine; Enkephalins; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Naloxone; Pyrroles; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Thiophenes

1990
Opioids and hibernation. II. Effects of kappa opioid U69593 on induction of hibernation in summer-active ground squirrels by "hibernation induction trigger" (HIT).
    Life sciences, 1987, Nov-02, Volume: 41, Issue:18

    Topics: Animals; Benzeneacetamides; Electric Stimulation; Female; Guinea Pigs; Hibernation; Ileum; Infusion Pumps; Male; Marmota; Muscle Contraction; Naloxone; Peptides; Proteins; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa; Sciuridae; Seasons

1987
Evidence that the kappa agonist U50488H has non-opioid actions.
    The Journal of pharmacy and pharmacology, 1988, Volume: 40, Issue:10

    Topics: 3,4-Dichloro-N-methyl-N-(2-(1-pyrrolidinyl)-cyclohexyl)-benzeneacetamide, (trans)-Isomer; Analgesics; Animals; Benzeneacetamides; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; Postural Balance; Pyrrolidines; Receptors, Opioid; Receptors, Opioid, kappa

1988