Page last updated: 2024-08-24

triazoles and Muscle Relaxation

triazoles has been researched along with Muscle Relaxation in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19904 (15.38)18.7374
1990's13 (50.00)18.2507
2000's7 (26.92)29.6817
2010's2 (7.69)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cellai, I; Comeglio, P; Filippi, S; Gacci, M; Maggi, M; Mancina, R; Maneschi, E; Morelli, A; Sarchielli, E; Vannelli, GB; Vignozzi, L1
Amin, K; Antonsson, M; Broddefalk, J; Jensen, J; Jin, S; Lehmann, A; Nilsson, K; Plowright, AT; St-Onge, S; Tomaszewski, MJ; Tremblay, M; Ulander, J; Walpole, C; Wei, Z; Yang, H1
Baur, F; Fozard, JR; Wolber, C1
Abebe, W; Mozaffari, MS1
Biagi, G; Calderone, V; Giorgi, I; Livi, O; Martelli, A; Martinotti, E; Nardi, A1
Elmedal Laursen, B; Mulvany, MJ; Simonsen, U1
Carneiro, FS; Giachini, FR; Inscho, EW; Leite, R; Tostes, RC; Webb, RC1
Clarke, GD; Harling, EJ; Hassall, PA; Ross, JW; Smith, H; Spicer, BA; Taylor, JF1
Hourani, SM; Prentice, DJ2
Cross, AJ; Green, AR; Misra, A; Murray, TK; Snape, MF1
Andersson, RG; Grenegård, M; Johansson Rydberg, IG1
Van de Voorde, J; Vanheel, B1
Hayakawa, T; Kamei, C; Kishida, H; Mihara, T; Nakayama, Y; Sugimoto, Y1
Fujiwara, R; Hayakawa, T; Kamei, C; Kishida, H; Nakayama, Y; Sugimoto, Y1
Elmedal, B; Hernández, M; Mulvany, MJ; Simonsen, U1
Bertaccini, G; Coppelli, G; Coruzzi, G; Poli, E; Pozzoli, C1
Cseppentö, A; Kovács, P; Nagy, E; Szabó, JZ; Szentmiklósi, AJ; Ujfalusi, A1
Abebe, W; Arif Hasan, AZ; Mustafa, SJ1
Baragatti, B; Biagi, G; Calderone, V; Giorgi, I; Livi, O; Martinotti, E; Scartoni, V1
Chidester, C; Duchamp, DJ; Gall, M; Lahti, RA; Rudzik, AD; Scahill, T1
Anderson, WH; Fitzpatrick, DF; Hwang, DP; Krzanowski, JJ; Polson, JB; Szentivanyi, A1
Junnarkar, AY; Patnaik, GK; Shrotri, DS; Singh, PP1
Brown, GL; Douglas, FL; Kotake, AN; Mustafa, SJ; Sabouni, MH1
Conroy, DM; Piper, PJ; Samhoun, MN1
Benveniste, J; Brink, C; Brunelleschi, S; Fantozzi, R; Giotti, A; Ledda, F; Renzi, D1

Other Studies

26 other study(ies) available for triazoles and Muscle Relaxation

ArticleYear
Testosterone/estradiol ratio regulates NO-induced bladder relaxation and responsiveness to PDE5 inhibitors.
    The journal of sexual medicine, 2012, Volume: 9, Issue:12

    Topics: Androgens; Animals; Aromatase Inhibitors; Cyclic Nucleotide Phosphodiesterases, Type 5; Estradiol; Estrogens; Female; Gene Expression; Imidazoles; Letrozole; Male; Muscle Relaxation; Muscle, Smooth; Nitric Oxide Donors; Nitriles; Nitroprusside; Ovariectomy; Phosphodiesterase 5 Inhibitors; Piperazines; Progesterone; Progestins; Rats; Rats, Sprague-Dawley; RNA, Messenger; Sex Factors; Sulfones; Testosterone; Triazines; Triazoles; Urinary Bladder; Vardenafil Dihydrochloride

2012
Discovery of agonists of cannabinoid receptor 1 with restricted central nervous system penetration aimed for treatment of gastroesophageal reflux disease.
    Journal of medicinal chemistry, 2013, Jan-10, Volume: 56, Issue:1

    Topics: Administration, Oral; Animals; Aryl Hydrocarbon Hydroxylases; Benzamides; Biological Availability; Brain; Cell Line; Cricetinae; Cricetulus; Cytochrome P-450 CYP2C9; Cytochrome P-450 CYP3A; Cytochrome P-450 CYP3A Inhibitors; Dogs; ERG1 Potassium Channel; Esophageal Sphincter, Lower; Ether-A-Go-Go Potassium Channels; Gastroesophageal Reflux; High-Throughput Screening Assays; Humans; Muscle Relaxation; Pyrazines; Pyridines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Cannabinoid, CB1; Solubility; Structure-Activity Relationship; Sulfoxides; Triazoles

2013
Antagonist pharmacology of adenosine A2B receptors from rat, guinea pig and dog.
    European journal of pharmacology, 2003, Aug-15, Volume: 475, Issue:1-3

    Topics: Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Dogs; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Quinazolines; Rats; Receptor, Adenosine A2B; Species Specificity; Triazoles

2003
Effect of taurine deficiency on adenosine receptor-mediated relaxation of the rat aorta.
    Vascular pharmacology, 2003, Volume: 40, Issue:4

    Topics: 2-Chloroadenosine; Acetylcholine; Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Aorta, Thoracic; beta-Alanine; Endothelium, Vascular; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Phenylephrine; Rats; Rats, Inbred WKY; Receptors, Purinergic P1; Taurine; Triazines; Triazoles; Vasoconstrictor Agents; Vasodilator Agents

2003
1,5-Diarylsubstituted 1,2,3-triazoles as potassium channel activators. VI.
    Farmaco (Societa chimica italiana : 1989), 2004, Volume: 59, Issue:5

    Topics: Animals; Benzimidazoles; Inhibitory Concentration 50; Models, Chemical; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium Channels, Calcium-Activated; Rats; Triazoles; Vasodilator Agents

2004
Involvement of guanylyl cyclase, protein kinase A and Na+ K+ ATPase in relaxations of bovine isolated bronchioles induced by GEA 3175, an NO donor.
    Pulmonary pharmacology & therapeutics, 2006, Volume: 19, Issue:3

    Topics: Animals; Bronchi; Calcium; Cattle; Colforsin; Cyclic AMP; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Guanylate Cyclase; In Vitro Techniques; Molsidomine; Muscle Relaxation; Nitric Oxide; Nitric Oxide Donors; Ouabain; Oxadiazoles; Peptides; Potassium; Quinoxalines; S-Nitrosoglutathione; Serotonin; Sodium-Potassium-Exchanging ATPase; Thionucleotides; Triazoles

2006
Determination of adenosine effects and adenosine receptors in murine corpus cavernosum.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 322, Issue:2

    Topics: 2-Chloroadenosine; Adenosine; Adenosine A2 Receptor Agonists; Adenosine A2 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Atropine; Bretylium Tosylate; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; In Vitro Techniques; Male; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Penile Erection; Phenylephrine; Prazosin; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Pyrimidines; Receptor, Adenosine A2A; Receptor, Adenosine A2B; Receptors, Purinergic P1; Triazoles

2007
BRL 22321, a compound that has mast cell stabilizing activity similar to that of disodium cromoglycate and in addition has smooth muscle relaxing activity.
    Agents and actions, 1983, Volume: 13, Issue:4

    Topics: Animals; Cromolyn Sodium; Guinea Pigs; Histamine Release; Immunoglobulin E; Lung; Male; Mast Cells; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Passive Cutaneous Anaphylaxis; Rats; Rats, Inbred Strains; Triazoles

1983
Activation of multiple sites by adenosine analogues in the rat isolated aorta.
    British journal of pharmacology, 1996, Volume: 118, Issue:6

    Topics: Adenosine; Animals; Aorta, Thoracic; Endothelium, Vascular; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Purines; Rats; Rats, Wistar; Receptors, Purinergic P1; Sulfonamides; Theophylline; Triazines; Triazoles; Xanthines

1996
A behavioural and neurochemical study in rats of the pharmacology of loreclezole, a novel allosteric modulator of the GABAA receptor.
    Neuropharmacology, 1996, Volume: 35, Issue:9-10

    Topics: Allosteric Regulation; Animals; Behavior, Animal; Brain Chemistry; Bridged Bicyclo Compounds, Heterocyclic; Cerebral Cortex; Chlormethiazole; Dose-Response Relationship, Drug; GABA Modulators; Hypnotics and Sedatives; Male; Muscle Relaxation; Pentobarbital; Picrotoxin; Rats; Receptors, GABA-A; Seizures; Sesterterpenes; Triazoles

1996
Adenosine analogues relax guinea-pig taenia caeci via an adenosine A2B receptor and a xanthine-resistant site.
    European journal of pharmacology, 1997, Mar-26, Volume: 323, Issue:1

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Cecum; Dose-Response Relationship, Drug; Guinea Pigs; Male; Muscle Relaxation; Muscle, Smooth; Phenethylamines; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Theophylline; Triazines; Triazoles; Vasodilator Agents; Xanthines

1997
Effects of the nitric oxide-donor, GEA 3175, on guinea-pig airways.
    European journal of pharmacology, 1997, Jun-25, Volume: 329, Issue:2-3

    Topics: Acetylcholine; Animals; Cyclic GMP; Electric Stimulation; Enzyme Inhibitors; Guinea Pigs; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide; Okadaic Acid; Peptides; Phosphoprotein Phosphatases; Potassium Channel Blockers; Trachea; Triazoles

1997
Influence of cytochrome P-450 inhibitors on endothelium-dependent nitro-L-arginine-resistant relaxation and cromakalim-induced relaxation in rat mesenteric arteries.
    Journal of cardiovascular pharmacology, 1997, Volume: 29, Issue:6

    Topics: Acetylcholine; Animals; Benzopyrans; Biological Factors; Cromakalim; Cytochrome P-450 Enzyme Inhibitors; Fatty Acids, Unsaturated; Female; In Vitro Techniques; Mesenteric Arteries; Miconazole; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroarginine; Norepinephrine; Proadifen; Pyrroles; Rats; Rats, Wistar; Triazoles; Vasodilator Agents

1997
Effect of Apafant on bronchial hyperresponsiveness and down-regulation of beta-adrenoceptors induced by endotoxin in guinea pigs.
    Arzneimittel-Forschung, 1997, Volume: 47, Issue:7

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Azepines; Binding Sites; Bronchial Hyperreactivity; Bronchodilator Agents; Cardiography, Impedance; Down-Regulation; Endotoxins; Guinea Pigs; Histamine; In Vitro Techniques; Isoproterenol; Lipopolysaccharides; Lung; Male; Membranes; Muscle Contraction; Muscle Relaxation; Triazoles

1997
Effects of apafant on PAF-induced downregulation of beta-adrenoceptors in guinea pigs.
    Methods and findings in experimental and clinical pharmacology, 1997, Volume: 19, Issue:8

    Topics: Adrenergic beta-Agonists; Animals; Azepines; Binding, Competitive; Bronchi; Down-Regulation; Guinea Pigs; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Platelet Activating Factor; Platelet Aggregation Inhibitors; Receptors, Adrenergic, beta; Triazoles

1997
Mechanisms of relaxations of bovine isolated bronchioles by the nitric oxide donor, GEA 3175.
    British journal of pharmacology, 1998, Volume: 123, Issue:5

    Topics: Albuterol; Aminoquinolines; Animals; Apamin; Bronchi; Bronchodilator Agents; Cattle; Charybdotoxin; Female; Glyburide; Male; Molsidomine; Muscle Relaxation; Nitric Oxide; Oxyhemoglobins; Penicillamine; Peptides; Receptors, Adrenergic, beta-2; Superoxide Dismutase; Triazoles

1998
Effects of histamine H2 receptor agonists and antagonists on the isolated guinea pig gallbladder.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:1

    Topics: Animals; Benzothiazoles; Dopamine Agents; Famotidine; Gallbladder; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Phenoxypropanolamines; Piperidines; Pyridines; Receptors, Histamine H2; Sincalide; Thiazoles; Triazoles

1999
Sensitization by chronic diazepam treatment of A2A adenosine receptor-mediated relaxation in rat pulmonary artery.
    Life sciences, 1999, Volume: 64, Issue:2

    Topics: Adenosine; Animals; Carrier Proteins; Diazepam; Dinucleoside Phosphates; Dipyridamole; Dose-Response Relationship, Drug; Female; Heart; Heart Atria; Muscle Relaxation; Phenethylamines; Pulmonary Artery; Purinergic P1 Receptor Agonists; Purinergic P1 Receptor Antagonists; Rats; Rats, Wistar; Receptor, Adenosine A2A; Receptors, Purinergic P1; Thioinosine; Triazines; Triazoles; Verapamil

1999
Antagonism of coronary artery relaxation by adenosine A2A-receptor antagonist ZM241385.
    Journal of cardiovascular pharmacology, 2000, Volume: 35, Issue:2

    Topics: Adenosine; Adenosine-5'-(N-ethylcarboxamide); Animals; Antihypertensive Agents; Coronary Vessels; Dinoprost; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Phenethylamines; Purinergic P1 Receptor Antagonists; Pyrimidines; Receptors, Purinergic P1; Swine; Triazines; Triazoles; Vasodilator Agents

2000
Triazolyl-benzimidazolones and triazolyl-benzotriazoles: new potential potassium channel activators. II.
    European journal of medicinal chemistry, 2000, Volume: 35, Issue:10

    Topics: Animals; Aorta, Thoracic; Benzimidazoles; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Molecular Structure; Muscle Relaxation; Potassium Channels; Rats; Rats, Wistar; Triazoles

2000
Novel anxiolytic agents derived from alpha-amino-alpha-phenyl-o-tolyl-4H-triazoles and -imidazoles.
    Journal of medicinal chemistry, 1978, Volume: 21, Issue:6

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Brain; Crystallography; Hypnotics and Sedatives; Imidazoles; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Mice; Models, Molecular; Molecular Conformation; Muscle Relaxation; Nicotine; Pentylenetetrazole; Rats; Seizures; Semicarbazides; Triazoles

1978
Analysis of the relationship between pharmacological inhibition of cyclic nucleotide phosphodiesterase and relaxation of canine tracheal smooth muscle.
    Biochemical pharmacology, 1979, Apr-15, Volume: 28, Issue:8

    Topics: 1-Methyl-3-isobutylxanthine; 3',5'-Cyclic-AMP Phosphodiesterases; 3',5'-Cyclic-GMP Phosphodiesterases; Airway Resistance; Animals; Caffeine; Dogs; Etazolate; Female; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phosphodiesterase Inhibitors; Pyrazines; Theophylline; Trachea; Triazoles

1979
Neuropsychopharmacological study of 2,4-dihydro[1,2,4]triazolo[3,4-c][1,4]benzothiazine-1-one (IDPH-791).
    Pharmacological research, 1992, Volume: 26, Issue:2

    Topics: Administration, Oral; Animals; Brain; Hypnosis; Injections, Intraperitoneal; Lethal Dose 50; Mephenesin; Mice; Motor Activity; Muscle Relaxants, Central; Muscle Relaxation; Paralysis; Rabbits; Rats; Rats, Wistar; Seizures; Thiazines; Triazoles

1992
Effects of CGS-15943A on the relaxations produced by adenosine analogs in human blood vessels.
    European journal of pharmacology, 1990, Oct-23, Volume: 187, Issue:3

    Topics: Adenosine; Adult; Coronary Vessels; Humans; In Vitro Techniques; Mammary Arteries; Middle Aged; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium Chloride; Quinazolines; Saphenous Vein; Theophylline; Triazoles

1990
Relaxations of guinea-pig isolated trachea induced by platelet-activating factor are epithelial-dependent and are antagonised by WEB 2086.
    European journal of pharmacology, 1990, Sep-21, Volume: 186, Issue:2-3

    Topics: Albuterol; Animals; Azepines; Epithelium; Guinea Pigs; In Vitro Techniques; Indomethacin; Male; Muscle Relaxation; Muscle, Smooth; Platelet Activating Factor; Trachea; Triazoles

1990
Interference of WEB 2086 and BN 52021 with Paf-induced effects on guinea-pig trachea.
    British journal of pharmacology, 1989, Volume: 97, Issue:2

    Topics: Animals; Azepines; Dinoprostone; Diterpenes; Ginkgolides; Guinea Pigs; Histamine Antagonists; In Vitro Techniques; Lactones; Male; Muscle Relaxation; Muscle, Smooth; Platelet Activating Factor; Trachea; Triazines; Triazoles

1989