Page last updated: 2024-08-18

thiophenes and Malaria, Falciparum

thiophenes has been researched along with Malaria, Falciparum in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (80.00)24.3611
2020's1 (20.00)2.80

Authors

AuthorsStudies
Banerjee, T; Ghosh, A1
Aponte, RA; Bonnert, R; Chaiyen, P; Charman, SA; Chitnumsub, P; Diederich, F; Freiberg, GM; Ittarat, W; Jaruwat, A; Kundu, A; Leartsakulpanich, U; Lloyd, M; Rottmann, M; Sadhukhan, S; Schäfer, A; Schwertz, G; Siggel, M; Srikumaran, M; White, KL; Witschel, MC; Zwyssig, A1
Bhunia, SS; Roy, KK; Saxena, AK1
Banerjee, T; Dwivedi, V; Kapoor, N; Sharma, SK; Surolia, A; Surolia, N1
Banerjee, T; Kapoor, N; Surolia, A; Surolia, N1

Other Studies

5 other study(ies) available for thiophenes and Malaria, Falciparum

ArticleYear
Nanotized curcumin-benzothiophene conjugate: A potential combination for treatment of cerebral malaria.
    IUBMB life, 2020, Volume: 72, Issue:12

    Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Antimalarials; Biological Availability; Curcumin; Malaria, Cerebral; Malaria, Falciparum; Mice; Mice, Inbred C57BL; Nanoparticles; Plasmodium berghei; Thiophenes

2020
Antimalarial Inhibitors Targeting Serine Hydroxymethyltransferase (SHMT) with in Vivo Efficacy and Analysis of their Binding Mode Based on X-ray Cocrystal Structures.
    Journal of medicinal chemistry, 2017, 06-22, Volume: 60, Issue:12

    Topics: Animals; Antimalarials; Arabidopsis Proteins; Chemistry Techniques, Synthetic; Crystallography, X-Ray; Cysteine; Drug Stability; Enzyme Inhibitors; Glycine Hydroxymethyltransferase; Half-Life; Ligands; Malaria, Falciparum; Mice, SCID; Plasmodium falciparum; Plasmodium vivax; Protein Conformation; Rats; Structure-Activity Relationship; Thiophenes

2017
CoMFA, CoMSIA, and docking studies on thiolactone-class of potent anti-malarials: identification of essential structural features modulating anti-malarial activity.
    Chemical biology & drug design, 2011, Volume: 78, Issue:3

    Topics: Antimalarials; Drug Design; Humans; Malaria, Falciparum; Models, Molecular; Plasmodium falciparum; Quantitative Structure-Activity Relationship; Thiophenes

2011
Benzothiophene carboxamide derivatives as inhibitors of Plasmodium falciparum enoyl-ACP reductase.
    IUBMB life, 2011, Volume: 63, Issue:12

    Topics: Antimalarials; Enoyl-(Acyl-Carrier-Protein) Reductase (NADH); Enzyme Inhibitors; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Molecular Structure; Plasmodium falciparum; Thiophenes

2011
Benzothiophene carboxamide derivatives as novel antimalarials.
    IUBMB life, 2011, Volume: 63, Issue:12

    Topics: Animals; Antimalarials; Disease Models, Animal; Malaria, Falciparum; Mice; Plasmodium berghei; Plasmodium falciparum; Thiophenes; Trophozoites

2011