Page last updated: 2024-08-21

thiazolidines and Prostatic Neoplasms

thiazolidines has been researched along with Prostatic Neoplasms in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19902 (16.67)18.7374
1990's0 (0.00)18.2507
2000's2 (16.67)29.6817
2010's6 (50.00)24.3611
2020's2 (16.67)2.80

Authors

AuthorsStudies
Ahmad, A; Alam, MA; Alam, O; Haider, MR; Husain, A; Iqbal, MA; Khan, SA1
Ben-Salha, I; Costa, H; Echeverria, LMC; Freeman, A; Gately, KA; Haider, A; Heavey, S; Jameson, C; Kelly, JD; Kumar, C; Luszczak, S; Pye, H; Ratynska, M; Sathyadevan, VK; Shaw, G; Simpson, BS; Sridhar, A; Stopka-Farooqui, U; Whitaker, HC1
Devi, R; Divakar, S; Elancheran, R; Kabilan, S; Kotoky, J; Kumari, S; Maruthanila, VL; Ramanathan, M; Saravanan, K1
Peng, F; Xie, F1
Abdulkadir, SA; Ahdesmaki, M; Anderson, PD; Everett, JH; Franco-Coronel, OE; Grosskurth, SE; Hameed, O; Huszar, D; Keeton, EK; Kirschner, AN; Kushner, MH; van der Meer, R; Wang, J1
Kraft, AS; Sainz, AG; Song, JH; Warfel, NA1
Awad, HM; El-Sayed, WA; El-Sofany, WI; Flefel, EM; Mohamed, AM1
Kopeček, J; Yang, J; Zhou, Y1
Davis, JJ; Dong, F; Fang, B; Guo, W; Inoue, S; Teraishi, F; Wu, S; Zhang, L1
Awate, B; Khanfar, MA; Liu, Y; Muralidharan, A; Nagle, DG; Sayed, KA; Shah, G; Shallal, HM; Youssef, DT; Zhou, YD1
Black, J; Ip, MM; Shea, WK1
Ip, MM; Schenkel, L; Sylvester, PW1

Other Studies

12 other study(ies) available for thiazolidines and Prostatic Neoplasms

ArticleYear
Design, synthesis, and biological evaluation of imidazopyridine-linked thiazolidinone as potential anticancer agents.
    Archiv der Pharmazie, 2020, Volume: 353, Issue:10

    Topics: A549 Cells; Animals; Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Drug Design; Female; Humans; Imidazoles; Lung Neoplasms; Male; MCF-7 Cells; Molecular Docking Simulation; Prostatic Neoplasms; Pyridines; Rats; Rats, Wistar; Thiazolidines; Toxicity Tests

2020
Co-targeting PIM and PI3K/mTOR using multikinase inhibitor AUM302 and a combination of AZD-1208 and BEZ235 in prostate cancer.
    Scientific reports, 2020, 09-01, Volume: 10, Issue:1

    Topics: Antineoplastic Agents; Biphenyl Compounds; Cell Line, Tumor; Cell Proliferation; Cohort Studies; Drug Therapy, Combination; Gene Expression Regulation, Neoplastic; Humans; Imidazoles; Male; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Prostatic Neoplasms; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-pim-1; Pyridines; Pyrimidines; Quinolines; RNA, Messenger; Signal Transduction; Thiazolidines; Thiophenes; TOR Serine-Threonine Kinases

2020
Design, Synthesis and Biological Evaluation of Novel 1, 3- thiazolidine-2, 4-diones as Anti-prostate Cancer Agents.
    Anti-cancer agents in medicinal chemistry, 2017, Volume: 17, Issue:13

    Topics: Antineoplastic Agents; Cell Line, Tumor; Crystallography, X-Ray; Drug Design; Drug Screening Assays, Antitumor; Humans; Male; Molecular Docking Simulation; Prostatic Neoplasms; Thiazolidines

2017
Anticancer Activity of Copper Complex of (4R)-(-)-2-Thioxo-4-thiazolidinecarboxylic Acid and 3-Rhodaninepropionic Acid on Prostate and Breast Cancer Cells by Fluorescent Microscopic Imaging.
    Journal of fluorescence, 2018, Volume: 28, Issue:1

    Topics: Antineoplastic Agents; Apoptosis; Breast Neoplasms; Cell Proliferation; Coordination Complexes; Copper; Female; Humans; Male; Microscopy, Fluorescence; Propionates; Prostatic Neoplasms; Thiazolidines; Tumor Cells, Cultured

2018
PIM kinase inhibitor AZD1208 for treatment of MYC-driven prostate cancer.
    Journal of the National Cancer Institute, 2015, Volume: 107, Issue:2

    Topics: Administration, Oral; Allografts; Animals; Antineoplastic Agents; Apoptosis; Biphenyl Compounds; Cell Hypoxia; Cell Proliferation; Down-Regulation; Gene Expression Regulation, Enzymologic; Gene Expression Regulation, Neoplastic; Genes, myc; Humans; Male; Mice; Prostatic Neoplasms; Prostatic Neoplasms, Castration-Resistant; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-pim-1; Thiazolidines; Tumor Suppressor Protein p53; Xenograft Model Antitumor Assays

2015
PIM Kinase Inhibitors Kill Hypoxic Tumor Cells by Reducing Nrf2 Signaling and Increasing Reactive Oxygen Species.
    Molecular cancer therapeutics, 2016, Volume: 15, Issue:7

    Topics: Animals; Biphenyl Compounds; Cell Line, Tumor; Cell Proliferation; Cell Survival; Disease Models, Animal; Humans; Hypoxia; Hypoxia-Inducible Factor 1, alpha Subunit; Male; Mice; Models, Biological; Neoplasms; NF-E2-Related Factor 2; Prostatic Neoplasms; Protein Binding; Protein Kinase Inhibitors; Protein Transport; Proto-Oncogene Proteins c-pim-1; Reactive Oxygen Species; Signal Transduction; Thiazolidines; Xenograft Model Antitumor Assays

2016
Synthesis and Anticancer Activity of New 1-Thia-4-azaspiro[4.5]decane, Their Derived Thiazolopyrimidine and 1,3,4-Thiadiazole Thioglycosides.
    Molecules (Basel, Switzerland), 2017, Jan-20, Volume: 22, Issue:1

    Topics: Antineoplastic Agents; Carcinoma, Hepatocellular; Cell Line, Tumor; Colorectal Neoplasms; Glycosylation; HCT116 Cells; Hep G2 Cells; Humans; Liver Neoplasms; Male; Prostatic Neoplasms; Spiro Compounds; Structure-Activity Relationship; Thiadiazoles; Thiazolidines; Thioglycosides

2017
Selective inhibitory effect of HPMA copolymer-cyclopamine conjugate on prostate cancer stem cells.
    Biomaterials, 2012, Volume: 33, Issue:6

    Topics: Antineoplastic Agents; Biomarkers, Tumor; Cell Line, Tumor; Cell Separation; Cell Survival; Hedgehog Proteins; Humans; Male; Methacrylates; Neoplastic Stem Cells; Polymers; Prostatic Neoplasms; Signal Transduction; Thiazolidines; Veratrum Alkaloids

2012
Antitumor activity and downregulation of pro-angiogenic molecules in human prostate cancer cells by a novel thiazolidione compound.
    The Prostate, 2006, Mar-01, Volume: 66, Issue:4

    Topics: Apoptosis; Blotting, Western; Cell Cycle; Cell Proliferation; Down-Regulation; Enzyme-Linked Immunosorbent Assay; Flow Cytometry; Humans; Male; Neovascularization, Pathologic; Phosphorylation; Prostatic Neoplasms; Thiazoles; Thiazolidines; Tumor Cells, Cultured

2006
Latrunculin A and its C-17-O-carbamates inhibit prostate tumor cell invasion and HIF-1 activation in breast tumor cells.
    Journal of natural products, 2008, Volume: 71, Issue:3

    Topics: Animals; Breast Neoplasms; Bridged Bicyclo Compounds, Heterocyclic; Carbamates; Drug Screening Assays, Antitumor; Humans; Hypoxia-Inducible Factor 1; Male; Molecular Structure; Porifera; Prostatic Neoplasms; Thiazolidines

2008
Short-term primary culture of rat prostate tumor epithelial cells on reconstituted basement membrane as a useful in vitro model to assess drug action on prostatic cancer: efficacy of the thiazolidinedione derivative CGP 19984.
    The Prostate, 1989, Volume: 15, Issue:2

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Basement Membrane; Disease Models, Animal; Epithelium; Male; Prostatic Neoplasms; Rats; Thiazoles; Thiazolidines; Tumor Cells, Cultured

1989
Antitumor efficacy in rats of CGP 19984, a thiazolidinedione derivative that inhibits luteinizing hormone secretion.
    Cancer research, 1986, Volume: 46, Issue:4 Pt 1

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Castration; Corticosterone; Female; Luteinizing Hormone; Male; Mammary Neoplasms, Experimental; Neoplasms, Hormone-Dependent; Prolactin; Prostatic Neoplasms; Rats; Rats, Inbred F344; Testosterone; Thiazoles; Thiazolidines

1986