Page last updated: 2024-08-21

thiazoles and Staphylococcal Infections

thiazoles has been researched along with Staphylococcal Infections in 57 studies

Research

Studies (57)

Timeframe	Studies, this research(%)	All Research%
pre-1990	12 (21.05)	18.7374
1990's	9 (15.79)	18.2507
2000's	4 (7.02)	29.6817
2010's	28 (49.12)	24.3611
2020's	4 (7.02)	2.80

Authors

Authors	Studies
Akhir, A; Chopra, S; Goel, A; Kaul, G; Rawat, KS; Rode, HB; Sangu, KG; Sharma, CP; Shukla, M	1
Akbar, S; Ganapathi, T; Ganesh Kumar, C; Kamal, A; Khan, I; Nagendra Babu, B; Sayeed, IB; Shareef, MA; Sirisha, K	1
Abutaleb, NS; Elsebaei, MM; Hagras, M; Li, D; Mahgoub, AA; Mayhoub, AS; Mohammad, H; Seleem, MN	1
Kirmusaoglu, S	1
Abutaleb, NS; Alhashimi, M; Kassab, AE; Mayhoub, AS; Mohamed, KO; Seleem, MN; Shahin, IG; Taher, AT	1
Ahmed, N; Ali, S; Farooq, S; Hussain, M; Khan, MA; Khan, S; Shamim, S	1
Lan, D; Qi, G; Zhao, G	1
Abouf, M; Abutaleb, NS; Chen, L; Elsebaei, MM; Ghiaty, A; Hegazy, YA; Malwal, SR; Mayhoub, AS; Mohammad, H; Oldfield, E; Seleem, MN; Zhang, J	1
Abutaleb, NS; Bayoumi, A; Ghiaty, A; Hagras, M; Kotb, A; Mayhoub, AS; Mohammad, H; Seleem, MA; Seleem, MN	1
Barraja, P; Carbone, A; Cascioferro, S; Cirrincione, G; Cusimano, MG; Diana, P; Montalbano, A; Parrino, B; Schillaci, D; Spanò, V	1
Abdel-Aleem, JA; Abutaleb, NS; Ali, AO; Elsebaei, MM; Hagras, M; Mayhoub, AS; Seleem, MN	1
Hagiya, H; Kokado, R; Okuno, H; Tomono, K	1
Beaufrère, H; Field, CL; MacLean, R; Rademacher, N; Wakamatsu, N	1
Kaul, M; Lavoie, EJ; Mark, L; Parhi, AK; Pilch, DS; Zhang, Y	1
Alm, R; Basarab, GS; Bist, S; Dangel, PB; Eakin, AE; Garner, CE; Green, O; Hauck, S; Hill, PJ; Hull, K; Illingworth, R; Manchester, JI; Rooney, M; Sherer, BA; Uria-Nickelsen, M; Zhou, F	1
Jaudzems, K; Leonchiks, A; Rudevica, Z; Turks, M; Zhulenkovs, D	1
Cushman, M; Mayhoub, AS; Mohammad, H; Seleem, MN	1
Kaul, M; LaVoie, EJ; Lyu, YL; Mark, L; Parhi, AK; Pawlak, J; Pilch, DS; Saravolatz, LD; Saravolatz, S; Weinstein, MP; Zhang, Y	1
Gong, T; Han, H; Han, S; Liu, H; Peschel, A; Qu, D; Wu, Y; Xu, T; Zhao, D; Zhao, Y	1
Cushman, M; Hammac, GK; Mayhoub, AS; Mohammad, H; Monteleone, D; Reddy, PV; Seleem, MN	1
Ang, W; Chang, Y; Chen, G; Li, G; Liu, Y; Long, H; Luo, Y; Sang, Z; Tang, J; Wang, Z; Wei, Y; Yang, S; Yang, T; Yang, X; Zhang, J	1
Cascioferro, S; Daidone, G; Maggio, B; Raffa, D; Raimondi, MV; Schillaci, D	1
Fischer, D; Hartmann, A; Kershaw, O; Lierz, M; Maier, K; Pendl, H; Prenger-Berninghoff, E; Schmidt, MJ	1
Cushman, M; Mohammad, H; Seleem, MN	1
Chittoor Neelakantan, S; Kuppuswamy, AA; Lowrence, RC; Makala, HV; Mani, A; Nagarajan, S; Raman, T; Subramaniapillai, SG; Ulaganathan, V	1
Aiwale, ST; Baker, PJ; Barynin, VV; Bennett, JM; Brown, DR; Chauhan, PK; Collins, I; Czaplewski, LG; Errington, J; Galbraith, G; Haydon, DJ; Heal, JR; Rice, DW; Sedelnikova, SE; Sheridan, JM; Srivastava, A; Stokes, NR; Taneja, A; Ure, R	1
LENZI, G; TRIA, E	1
Aman, AT; Busscher, HJ; Iravati, S; Krom, BP; Nuryastuti, T; van der Mei, HC	1
Beanland, J; Bennett, JM; Brown, D; Chauhan, PK; Collins, I; Czaplewski, L; Galbraith, G; Hall, R; Haydon, DJ; Henstock, V; Lancett, P; Macdonald, R; Nayal, N; Noula, C; Rockley, C; Srivastava, A; Stokes, NR; Sutariya, JK	1
Brewer, JT; Bushell, SM; Deng, G; Dewhurst, JM; Dzink-Fox, J; Gangl, E; Jain, A; LaMarche, MJ; Lee, L; Leeds, JA; Lilly, M; Manni, K; Mullin, S; Neckermann, G; Osborne, C; Palestrant, D; Patane, MA; Raimondi, A; Ranjitkar, S; Rann, EM; Sachdeva, M; Shao, J; Tiamfook, S; Whitehead, L; Yu, D	1
Han, SQ; Hu, J; Huang, RZ; Jiang, DB; Liu, HY; Pan, B; Qu, D; Wang, W; Wu, Y; Wu, YC; Zheng, LK; Zhu, T	1
Baryshnikova, A; Benton-Perdomo, L; Caron, A; Claveau, D; Daigneault, E; Deschamps, K; Elsen, NL; Gill, CJ; Kramer, S; Landry, F; Langlois, E; Lebeau-Jacob, C; Lee, SH; Liang, L; Lu, J; Lumb, KJ; Maxwell, E; Meredith, TC; Monteiro, JM; Parthasarathy, G; Pereira, PM; Petcu, M; Pinho, MG; Ramtohul, Y; Reid, JC; Roemer, T; Sharma, S; Sillaots, S; Skorey, K; Soisson, SM; Tam, J; Tan, CM; Therien, AG; Vaillancourt, J; Wang, H; Wang-Jarantow, L; Wong, S; Wu, J	1
Elsen, NL; Lu, J; Lumb, KJ; Parthasarathy, G; Reid, JC; Sharma, S; Soisson, SM	1
Fenical, W; Haste, NM; Hensler, ME; Jensen, PR; Loesgen, S; Nam, SJ; Nizet, V; Sakoulas, G; Sun, P; Thienphrapa, W; Tran, DN	1
Dorrestein, PC; Walsh, CT; Young, TS	1
ROMANO, C	1
GIUBERTONI, C	1
RANGONI, AG	1
CONTERNO, G; MATONE, S; PUPITA, F	1
MANZOLI, U; RUBERTI, A; VALLINI, A	1
PIROLI, G	1
Hawser, SP	1
Barrett, JF; Dorso, K; Gill, C; Herath, K; Hickey, E; Jayasuriya, H; Masurekar, P; Motyl, M; Occi, J; Overbye, KM; Singh, SB	1
Ciciliato, I; Colombo, L; Ferrari, P; Goldstein, BP; Landini, P; Le Monnier, F; Marinelli, F; Montanini, N; Selva, E; Stella, S	1
Connolly, RJ; Dinarello, CA; Dirkes, K; Gelfand, JA; Harris, BH; Schwaitzberg, SD	1
Inoue, Y; Jinbo, Y; Kondo, H; Sakamoto, F; Taguchi, M; Tsukamoto, G	2
DeJoy, SQ; Jeyaseelan, R; Kerwar, SS; Oronsky, AL; Pickett, WC; Torley, LW; Wick, MM; Wissner, A	1
Broom, NJ; Elder, JS; Hannan, PC; O'Hanlon, PJ; Pons, JE; Walker, G; Wilson, J; Woodall, P	1
Abson, A; Broom, NJ; Coates, PA; Elder, JS; Forrest, AK; Hannan, PC; Hicks, AJ; Masson, ND; O'Hanlon, PJ; Pearson, ND; Pons, JE; Wilson, JM	1
Blizzard, TA; DiNinno, FP; Dorso, K; Epstein-Toney, JH; Gill, CJ; Hajdu, R; Hammond, GG; Hammond, ML; Heck, JV; Huber, J; Jackson, JJ; Kohler, J; Kozarich, JW; Kropp, H; Lankas, G; Pelak, BA; Ratcliffe, RW; Rosen, H; Silver, L; Sundelof, JG; Thompson, R; Wildonger, KJ; Wilkening, RR	1
Beretta, G; Ferrari, P; Gastaldo, L; Goldstein, BP; Landini, P; Lorenzetti, R; Montanini, N; Ripamonti, F; Saddler, GS; Selva, E	1
Reyes-Javier, PD	1
Bormioli, P; D'Alessandro, A; Dominici, A; Ravagnan, L	1
Micetich, RG; Raap, R	2
Closier, MD; Islip, PJ	1

Other Studies

57 other study(ies) available for thiazoles and Staphylococcal Infections

Article	Year
Nitazoxanide potentiates linezolid against linezolid-resistant Staphylococcus aureus in vitro and in vivo. The Journal of antimicrobial chemotherapy, 2022, 08-25, Volume: 77, Issue:9 Topics: Anti-Bacterial Agents; Humans; Linezolid; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Nitro Compounds; Staphylococcal Infections; Staphylococcus aureus; Thiazoles	2022
Synthesis of new triazole fused imidazo[2,1-b]thiazole hybrids with emphasis on Staphylococcus aureus virulence factors. Bioorganic & medicinal chemistry letters, 2019, 10-01, Volume: 29, Issue:19 Topics: Anti-Bacterial Agents; Biofilms; Molecular Docking Simulation; Molecular Structure; Staphylococcal Infections; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles; Triazoles; Virulence Factors	2019
Phenylthiazoles with nitrogenous side chain: An approach to overcome molecular obesity. European journal of medicinal chemistry, 2019, Nov-15, Volume: 182 Topics: Amines; Animals; Anti-Bacterial Agents; Cell Line; Dose-Response Relationship, Drug; Drug Resistance, Multiple, Bacterial; Humans; Macrophages; Male; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Molecular Structure; Obesity; Rats; Rats, Sprague-Dawley; Staphylococcal Infections; Structure-Activity Relationship; Thiazoles	2019
Improved β-Lactam Susceptibility Against ica-Dependent Biofilm-Embedded Staphylococcus aureus by 2-Aminothiazole. Clinical laboratory, 2020, Jan-01, Volume: 66, Issue:1 Topics: Anti-Bacterial Agents; beta-Lactams; Biofilms; Drug Resistance, Bacterial; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Staphylococcal Infections; Thiazoles	2020
Evaluation of N-phenyl-2-aminothiazoles for treatment of multi-drug resistant and intracellular Staphylococcus aureus infections. European journal of medicinal chemistry, 2020, Sep-15, Volume: 202 Topics: Animals; Anti-Bacterial Agents; Cell Line; Cell Survival; Dose-Response Relationship, Drug; Humans; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Microsomes, Liver; Molecular Structure; Staphylococcal Infections; Structure-Activity Relationship; Thiazoles	2020
Antimicrobial and synergistic activity of thiazoline derivatives in combination with conventional antibiotics against multidrug resistant Staphylococcus aureus isolated from abscess drainage samples. Pakistan journal of pharmaceutical sciences, 2020, Volume: 33, Issue:5(Suppleme Topics: Abscess; Anti-Bacterial Agents; Disk Diffusion Antimicrobial Tests; Drainage; Drug Resistance, Multiple, Bacterial; Drug Synergism; Drug Therapy, Combination; Humans; Ribotyping; Staphylococcal Infections; Staphylococcus aureus; Thiazoles; Thiazolidines	2020
Design and development of some thiazole-based flavanoids as novel antibacterial against pathogens causing surgical site infection for possible benefit in bone trauma via inhibition of DNA gyrase. Chemical biology & drug design, 2017, Volume: 90, Issue:5 Topics: Animals; Anti-Bacterial Agents; DNA Gyrase; Drug Design; Flavonoids; Humans; Male; Molecular Docking Simulation; Rats, Sprague-Dawley; Staphylococcal Infections; Staphylococcus aureus; Surgical Wound Infection; Thiazoles; Topoisomerase II Inhibitors	2017
Alkynyl-containing phenylthiazoles: Systemically active antibacterial agents effective against methicillin-resistant Staphylococcus aureus (MRSA). European journal of medicinal chemistry, 2018, Mar-25, Volume: 148 Topics: Alkynes; Animals; Anti-Bacterial Agents; Half-Life; Methicillin-Resistant Staphylococcus aureus; Mice; Microsomes, Liver; Staphylococcal Infections; Thiazoles	2018
Phenylthiazoles with tert-Butyl side chain: Metabolically stable with anti-biofilm activity. European journal of medicinal chemistry, 2018, May-10, Volume: 151 Topics: Animals; Anti-Bacterial Agents; Biofilms; Caco-2 Cells; Humans; Male; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Rats, Sprague-Dawley; Staphylococcal Infections; Thiazoles	2018
New Thiazole Nortopsentin Analogues Inhibit Bacterial Biofilm Formation. Marine drugs, 2018, Aug-04, Volume: 16, Issue:8 Topics: Anti-Bacterial Agents; Aquatic Organisms; Biofilms; Drug Resistance, Bacterial; Humans; Imidazoles; Indoles; Inhibitory Concentration 50; Staphylococcal Infections; Staphylococcus aureus; Thiazoles	2018
Naphthylthiazoles: Targeting Multidrug-Resistant and Intracellular Staphylococcus aureus with Biofilm Disruption Activity. ACS infectious diseases, 2018, 12-14, Volume: 4, Issue:12 Topics: Animals; Anti-Bacterial Agents; Biofilms; Cell Line; Drug Design; Drug Resistance, Multiple, Bacterial; Enterococcus; Humans; Microbial Sensitivity Tests; Staphylococcal Infections; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles	2018
Daptomycin-associated myopathy induced by concomitant administration of mirabegron. Infection, 2019, Volume: 47, Issue:2 Topics: Acetanilides; Anti-Bacterial Agents; Daptomycin; Female; Humans; Methicillin-Resistant Staphylococcus aureus; Middle Aged; Muscular Diseases; Staphylococcal Infections; Thiazoles; Urological Agents	2019
Discospondylitis caused by Staphylococcus aureus in an African black-footed penguin (Spheniscus demersus). Journal of avian medicine and surgery, 2012, Volume: 26, Issue:4 Topics: Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Antifungal Agents; Bird Diseases; Doxycycline; Female; Itraconazole; Meloxicam; Spheniscidae; Spondylitis; Staphylococcal Infections; Thiazines; Thiazoles	2012
An FtsZ-targeting prodrug with oral antistaphylococcal efficacy in vivo. Antimicrobial agents and chemotherapy, 2013, Volume: 57, Issue:12 Topics: Animals; Anti-Bacterial Agents; Bacterial Proteins; Benzamides; Biological Availability; Biotransformation; Chlorocebus aethiops; Cytoskeletal Proteins; Female; Half-Life; Male; Methicillin-Resistant Staphylococcus aureus; Mice; Mice, Inbred BALB C; Microbial Sensitivity Tests; Prodrugs; Pyridines; Staphylococcal Infections; Thiazoles; Vero Cells	2013
Optimization of pyrrolamide topoisomerase II inhibitors toward identification of an antibacterial clinical candidate (AZD5099). Journal of medicinal chemistry, 2014, Jul-24, Volume: 57, Issue:14 Topics: Adenosine Triphosphatases; Amides; Animals; Anti-Bacterial Agents; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Humans; Mice; Mice, Knockout; Microbial Sensitivity Tests; Models, Molecular; Molecular Structure; Pyrroles; Rats; Rats, Wistar; Staphylococcal Infections; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles; Topoisomerase II Inhibitors	2014
Discovery and structure-activity relationship studies of irreversible benzisothiazolinone-based inhibitors against Staphylococcus aureus sortase A transpeptidase. Bioorganic & medicinal chemistry, 2014, Nov-01, Volume: 22, Issue:21 Topics: Aminoacyltransferases; Bacterial Proteins; Cysteine Endopeptidases; Enzyme Inhibitors; Fluorescence Resonance Energy Transfer; High-Throughput Screening Assays; Humans; Molecular Docking Simulation; Staphylococcal Infections; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles	2014
Anti-biofilm activity and synergism of novel thiazole compounds with glycopeptide antibiotics against multidrug-resistant staphylococci. The Journal of antibiotics, 2015, Volume: 68, Issue:4 Topics: Anti-Bacterial Agents; Biofilms; Drug Resistance, Multiple, Bacterial; Drug Synergism; Glycopeptides; Humans; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Staphylococcal Infections; Staphylococcus aureus; Staphylococcus epidermidis; Thiazoles; Vancomycin; Vancomycin Resistance	2015
TXA709, an FtsZ-Targeting Benzamide Prodrug with Improved Pharmacokinetics and Enhanced In Vivo Efficacy against Methicillin-Resistant Staphylococcus aureus. Antimicrobial agents and chemotherapy, 2015, Volume: 59, Issue:8 Topics: Animals; Anti-Bacterial Agents; Bacterial Proteins; Benzamides; Cells, Cultured; Cytoskeletal Proteins; Daptomycin; Dogs; Half-Life; Humans; Linezolid; Methicillin; Methicillin Resistance; Methicillin-Resistant Staphylococcus aureus; Mice; Mice, Inbred BALB C; Microbial Sensitivity Tests; Prodrugs; Pyridines; Rats; Staphylococcal Infections; Thiazoles; Vancomycin	2015
Antibacterial and anti-biofilm activities of thiazolidione derivatives against clinical staphylococcus strains. Emerging microbes & infections, 2015, Volume: 4, Issue:1 Topics: Anti-Bacterial Agents; Biofilms; China; Hospitals, Teaching; Humans; Methicillin Resistance; Methicillin-Resistant Staphylococcus aureus; Microbial Sensitivity Tests; Microscopy, Confocal; Retrospective Studies; Staphylococcal Infections; Staphylococcus aureus; Staphylococcus epidermidis; Tertiary Care Centers; Thiazoles	2015
Antibacterial Characterization of Novel Synthetic Thiazole Compounds against Methicillin-Resistant Staphylococcus pseudintermedius. PloS one, 2015, Volume: 10, Issue:6 Topics: Animals; Anti-Bacterial Agents; Cell Line; Cell Survival; Dog Diseases; Dogs; Lysostaphin; Methicillin; Methicillin Resistance; Mice; Microbial Sensitivity Tests; Oxacillin; Rifampin; Staphylococcal Infections; Staphylococcus; Thiazoles; Vancomycin	2015
Discovery of a Teraryl Oxazolidinone Compound (S)-N-((3-(3-Fluoro-4-(4-(pyridin-2-yl)-1H-pyrazol-1-yl)phenyl)-2-oxooxazolidin-5-yl)methyl)acetamide Phosphate as a Novel Antimicrobial Agent with Enhanced Safety Profile and Efficacies. Journal of medicinal chemistry, 2015, Aug-27, Volume: 58, Issue:16 Topics: Acetamides; Animals; Anti-Infective Agents; Bacteria; Biological Availability; Drug Design; Ether-A-Go-Go Potassium Channels; Linezolid; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Models, Molecular; Oxazoles; Oxazolidinones; Potassium Channel Blockers; Staphylococcal Infections; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles	2015
Sortase A Inhibitors: Recent Advances and Future Perspectives. Journal of medicinal chemistry, 2015, Dec-10, Volume: 58, Issue:23 Topics: Adamantane; Aminoacyltransferases; Animals; Anti-Bacterial Agents; Bacterial Adhesion; Bacterial Proteins; Benzoates; Carbolines; Cysteine Endopeptidases; Enzyme Inhibitors; Humans; Models, Molecular; Nitriles; Protein Conformation; Rhodanine; Small Molecule Libraries; Staphylococcal Infections; Staphylococcus aureus; Thiazoles; Thiones	2015
Vertebral Osteomyelitis and Septic Arthritis Associated With Staphylococcus hyicus in a Juvenile Peregrine Falcon ( Falco peregrinus ). Journal of avian medicine and surgery, 2015, Volume: 29, Issue:3 Topics: Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Infectious; Bird Diseases; Falconiformes; Fluoroquinolones; Male; Meloxicam; Osteomyelitis; Spine; Staphylococcal Infections; Staphylococcus hyicus; Thiazines; Thiazoles	2015
Antibacterial Evaluation of Synthetic Thiazole Compounds In Vitro and In Vivo in a Methicillin-Resistant Staphylococcus aureus (MRSA) Skin Infection Mouse Model. PloS one, 2015, Volume: 10, Issue:11 Topics: Administration, Topical; Animals; Drug Therapy, Combination; Humans; Keratinocytes; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Mupirocin; Staphylococcal Infections; Staphylococcal Skin Infections; Thiazoles	2015
Dithiazole thione derivative as competitive NorA efflux pump inhibitor to curtail multi drug resistant clinical isolate of MRSA in a zebrafish infection model. Applied microbiology and biotechnology, 2016, Volume: 100, Issue:21 Topics: Animals; Anti-Bacterial Agents; Bacterial Load; Bacterial Proteins; Ciprofloxacin; Disease Models, Animal; Drug Resistance, Multiple, Bacterial; Enzyme Inhibitors; Gene Expression Profiling; Methicillin-Resistant Staphylococcus aureus; Multidrug Resistance-Associated Proteins; Muscles; Real-Time Polymerase Chain Reaction; Skin; Staphylococcal Infections; Thiazoles; Thiones; Treatment Outcome; Zebrafish	2016
An inhibitor of FtsZ with potent and selective anti-staphylococcal activity. Science (New York, N.Y.), 2008, Sep-19, Volume: 321, Issue:5896 Topics: Amino Acid Sequence; Animals; Anti-Bacterial Agents; Bacillus subtilis; Bacterial Proteins; Binding Sites; Cell Division; Crystallography, X-Ray; Cytoskeletal Proteins; Drug Resistance, Bacterial; Drug Resistance, Multiple, Bacterial; Ligands; Methicillin Resistance; Mice; Microbial Sensitivity Tests; Models, Molecular; Molecular Sequence Data; Mutation; Protein Conformation; Pyridines; Staphylococcal Infections; Staphylococcus aureus; Thiazoles; Tubulin	2008
Research on the action of penicillin and vitamin BI on the development of staphylococcus in vitro. Rivista critica di clinica medica, 1947, Volume: 47, Issue:1-3 Topics: Penicillins; Staphylococcal Infections; Staphylococcus; Thiamine; Thiazoles	1947
Effect of cinnamon oil on icaA expression and biofilm formation by Staphylococcus epidermidis. Applied and environmental microbiology, 2009, Volume: 75, Issue:21 Topics: Anti-Bacterial Agents; Bacterial Proteins; Biofilms; Drug Synergism; Gene Expression Profiling; Gene Expression Regulation, Bacterial; Humans; Microbial Sensitivity Tests; Microbial Viability; Oils, Volatile; Staphylococcal Infections; Staphylococcus epidermidis; Tetrazolium Salts; Thiazoles	2009
Creating an antibacterial with in vivo efficacy: synthesis and characterization of potent inhibitors of the bacterial cell division protein FtsZ with improved pharmaceutical properties. Journal of medicinal chemistry, 2010, May-27, Volume: 53, Issue:10 Topics: Animals; Anti-Bacterial Agents; Bacterial Proteins; Biological Availability; Blood Proteins; Caco-2 Cells; Cell Division; Cell Membrane Permeability; Cytoskeletal Proteins; Hepatocytes; Humans; Mice; Microbial Sensitivity Tests; Models, Molecular; Protein Binding; Pyridines; Staphylococcal Infections; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles	2010
In vitro and in vivo activities of novel, semisynthetic thiopeptide inhibitors of bacterial elongation factor Tu. Antimicrobial agents and chemotherapy, 2011, Volume: 55, Issue:11 Topics: Animals; Anti-Bacterial Agents; Cell Line; Cell Survival; Female; Hep G2 Cells; Humans; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Molecular Structure; Peptide Elongation Factor Tu; Peptides, Cyclic; Staphylococcal Infections; Thiazoles	2011
Thiazolidione derivatives targeting the histidine kinase YycG are effective against both planktonic and biofilm-associated Staphylococcus epidermidis. Acta pharmacologica Sinica, 2012, Volume: 33, Issue:3 Topics: Anti-Bacterial Agents; Biofilms; Histidine Kinase; Plankton; Protein Kinase Inhibitors; Protein Kinases; Staphylococcal Infections; Staphylococcus epidermidis; Thiazoles	2012
Restoring methicillin-resistant Staphylococcus aureus susceptibility to β-lactam antibiotics. Science translational medicine, 2012, Mar-21, Volume: 4, Issue:126 Topics: Animals; Anti-Bacterial Agents; Bacterial Proteins; beta-Lactams; Cell Division; Crystallography, X-Ray; Cytoskeletal Proteins; Disease Models, Animal; Drug Resistance, Bacterial; Drug Synergism; Gene Regulatory Networks; Guanosine Diphosphate; Imipenem; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Mutation; Protein Structure, Secondary; Protein Transport; Pyridines; Staphylococcal Infections; Thiazoles; Virulence	2012
Mechanism of action of the cell-division inhibitor PC190723: modulation of FtsZ assembly cooperativity. Journal of the American Chemical Society, 2012, Aug-01, Volume: 134, Issue:30 Topics: Anti-Bacterial Agents; Bacterial Proteins; Cytoskeletal Proteins; Humans; Molecular Docking Simulation; Protein Conformation; Protein Structure, Tertiary; Pyridines; Staphylococcal Infections; Staphylococcus aureus; Thiazoles	2012
Activity of the thiopeptide antibiotic nosiheptide against contemporary strains of methicillin-resistant Staphylococcus aureus. The Journal of antibiotics, 2012, Volume: 65, Issue:12 Topics: Animals; Anti-Bacterial Agents; Disease Models, Animal; Dose-Response Relationship, Drug; Female; HeLa Cells; Humans; Methicillin-Resistant Staphylococcus aureus; Mice; Microbial Sensitivity Tests; Staphylococcal Infections; Streptomyces; Thiazoles; Time Factors; Vancomycin	2012
Codon randomization for rapid exploration of chemical space in thiopeptide antibiotic variants. Chemistry & biology, 2012, Dec-21, Volume: 19, Issue:12 Topics: Amino Acid Sequence; Anti-Bacterial Agents; Base Sequence; Codon; Gene Expression; Genetic Engineering; Humans; Methicillin-Resistant Staphylococcus aureus; Molecular Sequence Data; Mutagenesis; Peptides, Cyclic; Staphylococcal Infections; Streptomyces; Thiazoles	2012
[FIRST CLINICAL RESULTS OF THE USE IN UROLOGY OF A NEW NITROFURAN DERIVATIVE]. Minerva medica, 1963, Aug-29, Volume: 54 Topics: Escherichia coli Infections; Humans; Nitrofurans; Proteus Infections; Pseudomonas Infections; Staphylococcal Infections; Streptococcal Infections; Thiazoles; Urinary Tract Infections; Urology	1963
[CLINICAL EXPERIENCES WITH THE INTESTINAL ANTIBACTERIAL ACTIVITY OF 2ACETAMIDO-4-(5-NITRO-2-FURYL)-THIAZOLE]. Minerva medica, 1963, Aug-29, Volume: 54 Topics: Anti-Bacterial Agents; Bronchitis; Child; Dyspepsia; Enteritis; Escherichia coli Infections; Humans; Infant; Influenza, Human; Nitrofurans; Staphylococcal Infections; Thiazoles	1963
[A FURTHER CONTRIBUTION TO THE THERAPY OF URINARY INFECTIONS: FURIUM]. Minerva medica, 1963, Aug-29, Volume: 54 Topics: Enterobacter aerogenes; Escherichia coli Infections; Humans; Male; Nitrofurans; Prostatitis; Proteus Infections; Pseudomonas Infections; Staphylococcal Infections; Thiazoles; Urinary Calculi; Urinary Tract Infections	1963
[CLINICAL AND BACTERIOLOGICAL STUDY OF THE CHEMOTHERAPEUTIC ACTIVITY OF 2-ACETAMIDO-4-(5-NITRO-2-FURYL)-THIAZOLE]. La Clinica terapeutica, 1964, Jul-15, Volume: 30 Topics: Bacillus; Cholangitis; Cholecystitis; Cystitis; Dysentery; Dysentery, Bacillary; Enterocolitis; Escherichia coli Infections; Humans; Male; Nitrofurans; Prostatitis; Proteus Infections; Staphylococcal Infections; Thiazoles; Urethritis	1964
[2-ACETAMIDO-4-(5-NITRO-2-FURYL)-THIAZOLE IN VARIOUS PICTURES OF INFECTIVE PATHOLOGY. CLINICO-LABORATORY STUDY]. Minerva medica, 1964, Nov-03, Volume: 55 Topics: Biomedical Research; Brucellosis; Drug Therapy; Escherichia coli Infections; Humans; Meningitis; Meningitis, Meningococcal; Nitrofurans; Pharmacology; Salmonella Infections; Staphylococcal Infections; Streptococcal Infections; Thiazoles	1964
[On the behavior of the complementary power in toto in complications of staphylococcal pneumopathy in infancy]. Rassegna internazionale di clinica e terapia, 1960, May-15, Volume: 40 Topics: Child; Complement System Proteins; Humans; Infant; Pneumonia; Quinolinium Compounds; Staphylococcal Infections; Staphylococcus; Thiazoles	1960
Antibacterial drug discovery and development--SRI's 11th Annual Summit. IDrugs : the investigational drugs journal, 2006, Volume: 9, Issue:6 Topics: Aminoglycosides; Animals; Anti-Bacterial Agents; Cephalosporins; Clinical Trials as Topic; Drug Design; Humans; Incidence; Lipoglycopeptides; Methicillin Resistance; Minocycline; Molecular Structure; Oxazolidinones; Staphylococcal Infections; Staphylococcus aureus; Thiazoles; Tigecycline	2006
Antibacterial evaluations of thiazomycin- a potent thiazolyl peptide antibiotic from Amycolatopsis fastidiosa. The Journal of antibiotics, 2007, Volume: 60, Issue:9 Topics: Actinomycetales; Animals; Anti-Bacterial Agents; Drug Resistance, Bacterial; Mice; Microbial Sensitivity Tests; Mutation; Peptides; Peptides, Cyclic; Protein Synthesis Inhibitors; RNA, Ribosomal; Staphylococcal Infections; Staphylococcus aureus; Thiazoles	2007
Antibiotic GE37468 A: a new inhibitor of bacterial protein synthesis. I. Isolation and characterization. The Journal of antibiotics, 1995, Volume: 48, Issue:8 Topics: Animals; Anti-Bacterial Agents; Bacillus subtilis; Bacterial Proteins; Bacteroides fragilis; Chromatography, High Pressure Liquid; Female; Gram-Positive Bacteria; Male; Mice; Microbial Sensitivity Tests; Molecular Structure; Peptides, Cyclic; Rats; Staphylococcal Infections; Streptomyces; Thiazoles	1995
Platelet activating factor-antagonist improves survival in experimental staphylococcal septicemia. Journal of pediatric surgery, 1994, Volume: 29, Issue:8 Topics: Animals; Hemodynamics; Leukocyte Count; Organophosphorus Compounds; Platelet Activating Factor; Platelet Count; Rabbits; Sepsis; Staphylococcal Infections; Staphylococcus epidermidis; Thiazoles	1994
Synthesis and antibacterial activity of thiazolopyrazine-incorporated tetracyclic quinolone antibacterial agents. 2. Journal of medicinal chemistry, 1994, Aug-19, Volume: 37, Issue:17 Topics: 4-Quinolones; Animals; Anti-Infective Agents; Gram-Negative Bacteria; Gram-Positive Bacteria; Indicators and Reagents; Magnetic Resonance Spectroscopy; Mice; Microbial Sensitivity Tests; Molecular Structure; Optical Rotation; Pyrazines; Staphylococcal Infections; Staphylococcus aureus; Structure-Activity Relationship; Thiazoles	1994
Synthesis and antibacterial activity of thiazolopyrazine-incorporated tetracyclic quinolone antibacterials. Journal of medicinal chemistry, 1994, Mar-04, Volume: 37, Issue:5 Topics: Animals; Drug Resistance, Microbial; Gram-Negative Bacteria; Gram-Positive Bacteria; Male; Methicillin; Mice; Microbial Sensitivity Tests; Ofloxacin; Quinolones; Staphylococcal Infections; Thiazoles; Topoisomerase II Inhibitors	1994
Effect of CL 184,005, a platelet-activating factor antagonist in a murine model of Staphylococcus aureus-induced gram-positive sepsis. The Journal of infectious diseases, 1994, Volume: 169, Issue:1 Topics: Animals; Blood Pressure; Disease Models, Animal; Dose-Response Relationship, Drug; Enterotoxins; Interleukin-6; Male; Mice; Mice, Inbred BALB C; Mice, Nude; Organophosphorus Compounds; Platelet Activating Factor; Staphylococcal Infections; Thiazoles; Time Factors; Tumor Necrosis Factor-alpha	1994
The chemistry of pseudomonic acid. Part 14. Synthesis and in vivo biological activity of heterocyclyl substituted oxazole derivatives. The Journal of antibiotics, 1995, Volume: 48, Issue:11 Topics: Animals; Anti-Bacterial Agents; Furans; Humans; Isoxazoles; Mice; Mupirocin; Oxazoles; Pyrazoles; Pyridines; Sepsis; Staphylococcal Infections; Thiazoles; Thiophenes	1995
Chemistry of pseudomonic acid. Part 16. Aryl and heteroaryl ketone derivatives of monic acid. The Journal of antibiotics, 1996, Volume: 49, Issue:4 Topics: Animals; Anti-Bacterial Agents; Humans; Ketones; Male; Mice; Mice, Inbred Strains; Microbial Sensitivity Tests; Mupirocin; Sepsis; Staphylococcal Infections; Structure-Activity Relationship; Thiazoles	1996
Reduced immunotoxicity and preservation of antibacterial activity in a releasable side-chain carbapenem antibiotic. Science (New York, N.Y.), 1999, Jan-29, Volume: 283, Issue:5402 Topics: Animals; Antibodies; Bacterial Proteins; Carbapenems; Carrier Proteins; Dipeptidases; Drug Design; Drug Resistance, Microbial; Drug Resistance, Multiple; Enterococcus; Erythrocytes; Haptens; Hexosyltransferases; Humans; Immunodominant Epitopes; Immunoglobulin G; Lactams; Lymphocyte Activation; Macaca mulatta; Mice; Mice, Inbred DBA; Microbial Sensitivity Tests; Muramoylpentapeptide Carboxypeptidase; Penicillin-Binding Proteins; Peptidyl Transferases; Staphylococcal Infections; Staphylococcus; Thiazoles	1999
Antibiotic GE2270 a: a novel inhibitor of bacterial protein synthesis. I. Isolation and characterization. The Journal of antibiotics, 1991, Volume: 44, Issue:7 Topics: Actinomycetales; Animals; Anti-Bacterial Agents; Bacteria, Anaerobic; Bacterial Proteins; Bacteroides fragilis; Gram-Positive Bacteria; Mice; Microbial Sensitivity Tests; Molecular Structure; Moraxella catarrhalis; Mycobacterium tuberculosis; Peptides; Peptides, Cyclic; Propionibacterium acnes; Protein Synthesis Inhibitors; Staphylococcal Infections; Thiazoles	1991
Epicillin in the treatment of acute superficial and soft tissue infections. Current therapeutic research, clinical and experimental, 1971, Volume: 13, Issue:9 Topics: Acetamides; Adult; Child; Cyclohexanes; Escherichia coli Infections; Humans; Penicillanic Acid; Penicillins; Skin Diseases, Infectious; Staphylococcal Infections; Thiazoles	1971
[Hetacillin: protective action and serum and tissue levels]. Antibiotica, 1969, Volume: 7, Issue:4 Topics: Administration, Oral; Ampicillin; Animals; Escherichia coli Infections; Imidazoles; Injections, Intraperitoneal; Lethal Dose 50; Male; Mice; Penicillanic Acid; Penicillins; Rabbits; Staphylococcal Infections; Thiazoles; Time Factors	1969
Penicillins from 3- and 5-phenylisothiazole-4-carboxylic acids and alkoxy derivatives. Journal of medicinal chemistry, 1968, Volume: 11, Issue:1 Topics: Acids; Animals; Methods; Mice; Oxacillin; Penicillin G; Penicillin Resistance; Penicillins; Staphylococcal Infections; Staphylococcus; Streptococcus pneumoniae; Streptococcus pyogenes; Thiazoles	1968
Penicillins and cephalosporins from isothiazolylacetic acids. Journal of medicinal chemistry, 1968, Volume: 11, Issue:1 Topics: Acetates; Amides; Ampicillin; Animals; Anti-Bacterial Agents; Cephalosporins; Cephalothin; Escherichia coli; Klebsiella; Klebsiella Infections; Methods; Mice; Penicillin G; Penicillins; Salmonella; Salmonella typhi; Staphylococcal Infections; Staphylococcus; Streptococcus pneumoniae; Streptococcus pyogenes; Thiazoles	1968
Nitrofuryl heterocyclics. 2. Journal of medicinal chemistry, 1971, Volume: 14, Issue:5 Topics: Amides; Animals; Enterococcus faecalis; Mice; Nitrofurans; Shigella sonnei; Staphylococcal Infections; Staphylococcus; Streptococcal Infections; Thiazoles; Urea	1971