thiazoles has been researched along with Muscle Contraction in 127 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 29 (22.83) | 18.7374 |
1990's | 38 (29.92) | 18.2507 |
2000's | 30 (23.62) | 29.6817 |
2010's | 22 (17.32) | 24.3611 |
2020's | 8 (6.30) | 2.80 |
Authors | Studies |
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Hennenberg, M; Huang, R; Stief, CG; Strittmatter, F; Tamalunas, A; Waidelich, R | 1 |
Chess-Williams, R; Lim, I | 1 |
Clodfelder-Miller, B; McNaught, J; Ness, TJ; Su, X | 1 |
Chermansky, C; Ikeda, Y; Kanai, A; Mizoguchi, S; Singh, N; Suzuki, T; Tyagi, P; Yoshimura, N; Zabbarova, I | 1 |
Budriesi, R; Caputo, L; Cavalluzzi, MM; Corazza, I; De Salvia, MA; Franchini, C; Gualdani, R; Lentini, G; Micucci, M; Milani, G; Piarulli, M; Quintieri, L; Rosato, A; Viale, M | 1 |
Chimoto, J; Morikawa, K; Okura, T; Shiho, M; Shinozuka, K; Wakuda, H; Yamada, S | 1 |
Jung, DW; Kim, HJ; Kim, JH; Kim, SW; Lee, JH; Um, J; Williams, DR | 1 |
Deshpande, DA; Javed, E; Kambayashi, T; Lim, JM; Nayak, AP; Pan, S; Panettieri, RA; Penn, RB; Shah, SD; Sharma, P; Yadav, SK | 1 |
Kida, J; Mashimo, H; Matsuya, H; Okada, H; Sekido, N; Wakamatsu, D | 1 |
Ciotkowska, A; Gratzke, C; Hennenberg, M; Herlemann, A; Rutz, B; Sterr, CM; Stief, CG; Strittmatter, F; Wang, X; Wang, Y; Yu, Q | 1 |
Antunes, E; Bertollotto, GM; Candido, TZ; De Nucci, G; de Oliveira, MG; Kiguti, LRA; Mónica, FZ; Pupo, AS; Rojas-Moscoso, JA | 1 |
Hatanaka, T; Masuda, N; Ohtake, A; Sato, S; Someya, A; Suzuki, M; Ueshima, K; Ukai, M; Watanabe, M | 1 |
Drake, MJ; Paton, JF; Pickering, AE; Sadananda, P | 1 |
Aizawa, N; Homma, Y; Igawa, Y | 2 |
Adeoye, OO; Bouthors, V; Hubbell, MC; Pearce, WJ; Williams, JM | 1 |
Atala, A | 1 |
de Groat, WC; Reese, JN; Rogers, MJ; Roppolo, JR; Schwen, Z; Shen, B; Tai, C; Wang, J; Xiao, Z | 1 |
Calvi, P; D' Agostino, G; Maria Condino, A | 1 |
Alexandre, EC; Antunes, E; Claudino, MA; Costa, FF; da Silva, FH; de Nucci, G; Fertrin, KY; Franco-Penteado, CF; Leiria, LO; Mónica, FZ; Renno, A | 1 |
Hirayama, M; Hori, Y; Ito, K; Kawabata, Y; Kawachi, M; Matsunaga, Y; Nagahama, K; Ozaki, T; Shiraishi, Y; Takei, M; Tanaka, T | 1 |
De Wachter, S; Eastham, J; Gillespie, J; Persyn, S; Wyndaele, JJ | 1 |
Bastide, B; Cieniewski-Bernard, C; Deracinois, B; Duban-Deweer, S; Dupont, E; Krzewinski, F; Lambert, M; Richard, E | 1 |
Alexandre, EC; Antunes, E; Calmasini, FB; Candido, TZ; da Silva, CPV; da Silva, FH; de Oliveira, MG; Mónica, FZ | 1 |
Baker, DJ; Constantin, D; Constantin-Teodosiu, D; Greenhaff, PL | 1 |
Hirayama, M; Hori, Y; Inoue, N; Ito, K; Kawabata, Y; Kawachi, M; Matsunaga, Y; Nagahama, K; Ozaki, T; Takei, M; Tanaka, T; Toda, R; Yoshii, K | 1 |
Andersson, KE; Beckmann, C; Göttinger, J; Gratzke, C; Hedlund, P; Hennenberg, M; Roosen, A; Schlenker, B; Stief, CG; Strittmatter, F; Walther, S | 1 |
Gao, W; Li, J; Lu, J; Morales, A; Xing, J | 1 |
Shafik, AN | 1 |
Joseph, L; Mei, L; Song, T; Wang, YX; Yadav, VR; Zheng, YM | 1 |
Andersson, KE; Bouchelouche, K; Bouchelouche, P; Korstanje, C; Nordling, J; Svalø, J | 1 |
Gros, G; Kleinke, T; Papadopoulos, S; Wetzel, P | 1 |
Ballabeni, V; Barocelli, E; Calcina, F; Impicciatore, M; Tognolini, M; Vicini, P | 1 |
Iida, KT; Iwama, Y; Kamata, K; Kawakami, Y; Mokuno, H; Shimada, K; Shimano, H; Sone, H; Suzuki, M; Toyoshima, H; Watanabe, Y; Yamada, N | 1 |
Akuzawa, S; Imanishi, N; Ito, H; Iwaoka, K; Kazuta, K; Kiso, T; Koshio, H; Mase, T; Nagashima, SY; Ohta, M; Sakamoto, S; Tsukamoto, S | 1 |
Albinsson, S; Hellstrand, P; Malmqvist, U; Nordström, I; Swärd, K; Zeidan, A | 1 |
Gosens, R; Meurs, H; Nelemans, SA; Schaafsma, D; Zaagsma, J | 1 |
Dhawan, J; Helfman, DM | 1 |
Dowell, ML; Fredberg, JJ; Gerthoffer, WT; Halayko, AJ; Lakser, OJ; Mitchell, RW; Solway, J; Stelmack, GL | 1 |
Chen, A; Chin, TY; Chueh, SH; Jin, JS; Ka, SM; Lee, HS; Lee, WH; Lin, YF; Sheu, LF; Yao, CW | 1 |
Mahesh, R; Pandi, PV; Perumal, RV | 1 |
An, SS; Butler, JP; Fabry, B; Fredberg, JJ; Laudadio, RE; Millet, EJ | 1 |
Comini, M; Menozzi, A; Morini, G; Poli, E; Pozzoli, C | 2 |
Orlando, KA; Pittman, RN; Stone, NL | 1 |
Han, DH; Holloszy, JO; Terada, S; Wicke, S | 1 |
Maruyama, T; Matsui, T; Miyata, K; Nagase, I; Sasamata, M; Sato, S; Takasu, T; Uchida, H; Ukai, M; Yamaguchi, O | 1 |
Dowell, ML; Lakser, OJ; Mitchell, RW; Solway, J | 1 |
Certa, K; Chism, LM; Mago, R; Pinninti, NR | 1 |
Angelico, P; Clarke, DE; Farina, P; Guarneri, L; Leonardi, A; Poggesi, E; Testa, R | 1 |
Vohra, MM | 1 |
Barker, LA | 1 |
Schunack, W; Spengler, JP | 1 |
Ito, K; Kanazawa, T; Morita, T; Nose, T | 1 |
Hachisu, M; Koeda, T; Sekizawa, Y; Shitoh, K | 1 |
Impicciatore, M; Plazzi, PV; Vitali, T | 1 |
Ito, K; Ito, KM; Murakami, K; Shindo, K | 1 |
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH | 1 |
Ogilvie, RW; Robinson, DM; Terjung, RL; Tullson, PC | 1 |
Kadowaki, S; Nakao, E; Takahashi, K; Umezu, K; Yamada, K; Yamada, N | 1 |
Baziard-Mouysset, G; Bonnafous, R; Payard, M; Stigliani, JL; Tchani, G; Tisne-Versailles, J | 1 |
Momose, K; Nobe, K; Ohata, H | 2 |
Elhilali, MM; Gagnon, C; Hassan, AA; Hassouna, MM; Taketo, T | 1 |
Davison, JS; Jennings, LJ; Lea, RW; Pozo, MJ; Salido, GM; Sharkey, KA; Singh, J | 1 |
Barazi, M; Dominguez, LJ; Igwe, R; Ram, JL; Song, J; Sowers, JR; Walsh, MF | 1 |
Maehr, H; Yang, R | 1 |
Capasso, A; Sorrentino, L | 1 |
Bourghli, M; Miller, JA; Peuler, JD; Soltis, EE; Sowers, JR; Zammam, HY | 1 |
Bocheva, A; Golovinsky, E; Stanchev, M; Todorov, S | 1 |
De Freitas, GA; Santos, AR; Vedana, EM | 1 |
Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C; Timmerman, H | 1 |
Arakida, Y; Honda, K; Miyata, K; Ohga, K; Suwa, K; Yamada, T; Yokota, M | 1 |
De Leyn, P; Demedts, MG; Deneffe, G; Dupont, LJ; Pype, JL; Verleden, GM | 1 |
Bertaccini, G; Coppelli, G; Coruzzi, G; Poli, E; Pozzoli, C | 1 |
Gunst, SJ; Mehta, D | 1 |
Glinka, R; Timmerman, H; Walczyński, K; Zhang, MQ; Zuiderveld, OP | 1 |
Fukamachi, H; Higa, T; Miura, T; Sakakibara, M; Sindo, K; Suzuki, H; Takei, M; Ueno, A | 1 |
Guryn, R; Timmerman, H; Walczyński, K; Zuiderveld, OP | 1 |
Kaibara, M; Kurimoto, T; Ogishima, M; Taniyama, K; Ueki, S | 1 |
Ito, Y; Nakajima, T; Nawata, H | 1 |
Adachi, Y; Karaki, H; Satake, N; Sato, K; Shibata, S | 1 |
Amoretti, L; Ballabeni, V; Barocelli, E; Tognolini, M; Vicini, P | 1 |
Andreani, A; Garaliene, V; Leoni, A; Locatelli, A; Morigi, R; Rambaldi, M; Recanatini, M | 1 |
Akuzawa, S; Ito, H; Iwaoka, K; Kamato, T; Kiso, T; Miyata, K; Nagakura, Y; Naitoh, Y; Sakai, H; Suzuki, M; Yamaguchi, T; Yamano, M; Yuki, H | 1 |
Boissard, C; Chung, NN; Keller, M; Lemieux, C; Mutter, M; Patiny, L; Schiller, PW | 1 |
Gros, G; Papadopoulos, S; Wetzel, P | 1 |
Hagen, JL; Hepple, RT; Krause, DJ | 1 |
Ito, H; Iwaoka, K; Kiso, T; Miyata, K; Nagakura, Y; Yamaguchi, T | 1 |
Clark, SJ; Poyser, RH | 1 |
Waldeck, B | 1 |
Berti, F; Folco, GC; Malandrino, S; Omini, C; Sautebin, L; Viganò, T | 1 |
Aono, S; Hara, Y; Miyagishi, A; Nakatani, H; Sato, E | 1 |
Iso, T; Iwao, J; Nishimura, K; Oya, M | 1 |
Colombo, M; Márquez, M; Roberts, DJ | 1 |
Morimoto, K; Nakayama, K; Nozawa, Y; Tanaka, Y | 1 |
Horiba, M; Nabe, T; Ohata, K; Watanabe-Kohno, S; Yamamura, H; Yasui, K | 1 |
Goto, S; Inagaki, N; Koda, A; Miura, T; Nagai, H; Yoshida, K | 1 |
Alonso, S; Artalejo, CR; Cillero, J; Fau de Casa-Juana, M; García, AG; González-Morales, MA; López, MG; Santos, L; Sunkel, CE; Villarroya, M | 1 |
Horiba, M; Nabe, T; Ohata, K; Watanabe-Kohno, S; Yamamura, H | 1 |
Eriks, JC; Sterk, GJ; Timmerman, H; van der Goot, H | 1 |
Crowley, HJ; O'Donnell, M; O'Neill, N; Welton, AF; Yaremko, B | 1 |
Eriks, JC; Sterk, GJ; Timmerman, H; van Acker, SA; van der Aar, EM; van der Goot, H | 1 |
Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P | 1 |
Calignano, A; Diurno, MV; Mazzoni, O; Piscopo, E | 1 |
Karibe, H; Oishi, K; Uchida, MK | 1 |
Bertrand, C; Landry, Y; Tschirhart, E | 1 |
Iso, T; Miyawaki, N; Nishimura, K; Yamauchi, H | 1 |
Bast, A; Leurs, R; Timmerman, H | 1 |
Egginton, S; Hargreaves, D; Hudlická, O | 1 |
Butler, RD; Evans, RL; McCrohan, CR | 1 |
Holzer, P; Lippe, IT | 1 |
Koch, P; Peters, T; Wilffert, B; Wilhelm, D | 1 |
Benveniste, J; Coëffier, E; Desquand, S; Floch, A; Lefort, J; Maridonneau-Parini, I; Randon, J; Sedivy, P; Vargaftig, BB | 1 |
Postius, S; Sattler, HJ; Schunack, W; Szelenyi, I; Trumm, KA | 1 |
Aono, M; Mizuta, K; Moriga, M; Narusawa, H | 1 |
Hashimoto, Y; Iwatsuki, N; Koga, Y | 1 |
Adami, M; Bertaccini, G; Coruzzi, G; Poli, E | 1 |
Hidaka, H; Ishikawa, T; Ito, M; Itoh, H; Kawamatsu, Y; Saitoh, M; Shin, T; Sugihara, H; Tanaka, T; Umekawa, H | 1 |
Chang, SW; Henson, PM; McMurtry, IF; Pfeffer, KD; Voelkel, NF; Worthen, SG | 1 |
Bian, K; Inatomi, A; Lu, W; Okamura, T; Toda, N | 1 |
Koch, P; Nebel, U; Peters, T; Wermelskirchen, D; Wilffert, B; Wilhelm, D | 1 |
Fujita, M; Iso, T; Iwao, J; Kato, E; Kawashima, Y; Oya, M; Tabashi, K; Yamamoto, K | 1 |
Dahlbom, R; Lindeke, B; Ringdahl, B | 1 |
Berkoz, B; Edwards, JA; Fried, JH; Halpern, O; Lewis, GS; Miller, LM; Roszkowski, AP; Strosberg, AM | 1 |
Ambrus, CM; Ambrus, JL | 1 |
Aceves, J; Erlij, D; Martínez-Marañón, R | 1 |
1 review(s) available for thiazoles and Muscle Contraction
Article | Year |
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Force fluctuation-induced relengthening of acetylcholine-contracted airway smooth muscle.
Topics: Acetylcholine; Actin Cytoskeleton; Animals; Asthma; Bridged Bicyclo Compounds, Heterocyclic; Depsipeptides; Humans; Mitogen-Activated Protein Kinases; Muscle Contraction; Muscle, Smooth; Myosins; Stress, Mechanical; Thiazoles; Thiazolidines | 2008 |
126 other study(ies) available for thiazoles and Muscle Contraction
Article | Year |
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Inhibition of Full Smooth Muscle Contraction in Isolated Human Detrusor Tissues by Mirabegron Is Limited to Off-Target Inhibition of Neurogenic Contractions.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetanilides; Carbachol; Endothelin-1; Female; Humans; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Receptors, Adrenergic; Thiazoles; Urinary Bladder, Overactive | 2022 |
Mirabegron attenuates porcine ureteral contractility via α1-adrenoceptor antagonism.
Topics: Acetanilides; Adrenergic beta-Antagonists; Animals; Muscle Contraction; Phenylephrine; Receptors, Adrenergic, alpha-1; Serotonin; Swine; Thiazoles | 2022 |
Medications used to treat bladder disorders may alter effects of neuromodulation.
Topics: Acetanilides; Animals; Cystitis; Electric Stimulation Therapy; Female; Mandelic Acids; Muscle Contraction; Pudendal Nerve; Rats; Rats, Sprague-Dawley; Thiazoles; Urological Agents | 2020 |
Excitatory effect of acotiamide on rat and human bladder: Implications for underactive bladder treatment.
Topics: Animals; Benzamides; Carbachol; Electric Stimulation; Humans; Male; Muscle Contraction; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder; Urinary Bladder, Underactive | 2020 |
Lubeluzole: from anti-ischemic drug to preclinical antidiarrheal studies.
Topics: Animals; Anti-Bacterial Agents; Antidiarrheals; Bacteria; Colon; Diarrhea; Dose-Response Relationship, Drug; Gram-Negative Bacterial Infections; Gram-Positive Bacterial Infections; Guinea Pigs; Ileum; Loperamide; Male; Microbial Sensitivity Tests; Muscle Contraction; Neuroprotective Agents; Piperidines; Quaternary Ammonium Compounds; Rats; Rats, Sprague-Dawley; Thiazoles | 2021 |
Possible Involvement of Muscarinic Receptor Blockade in Mirabegron Therapy for Patients with Overactive Bladder.
Topics: Acetanilides; Administration, Oral; Adrenergic beta-3 Receptor Agonists; Animals; Brain; Male; Muscarinic Antagonists; Muscle Contraction; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Thiazoles; Urinary Bladder; Urinary Bladder, Overactive; Urological Agents | 2021 |
Lithium Chloride Protects against Sepsis-Induced Skeletal Muscle Atrophy and Cancer Cachexia.
Topics: Animals; Body Weight; Cachexia; Cell Differentiation; Cell Proliferation; Culture Media, Conditioned; Glycogen Synthase Kinase 3 beta; Inflammation; Lipopolysaccharides; Lithium Chloride; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Muscle Contraction; Muscle Fibers, Skeletal; Muscle Proteins; Muscle, Skeletal; Muscular Atrophy; Neoplasms; RAW 264.7 Cells; RNA, Small Interfering; Sepsis; SKP Cullin F-Box Protein Ligases; Tetrazolium Salts; Thiazoles | 2021 |
Diacylglycerol Kinase Inhibition Reduces Airway Contraction by Negative Feedback Regulation of Gq-Signaling.
Topics: Bronchoconstriction; Cells, Cultured; Diacylglycerol Kinase; Gene Knockdown Techniques; GTP-Binding Protein alpha Subunits, Gq-G11; Humans; Muscle Contraction; Muscle, Smooth; Pyrimidinones; Signal Transduction; Thiazoles | 2021 |
Effects of an EP2 and EP3 Receptor Dual Agonist, ONO-8055, on a Radical Hysterectomy-Induced Underactive Bladder Model in Monkeys.
Topics: Animals; Cholinesterase Inhibitors; Disease Models, Animal; Female; Hysterectomy; Macaca fascicularis; Muscle Contraction; Pyridinium Compounds; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP3 Subtype; Rheology; Thiazoles; Urinary Bladder, Neurogenic; Urination | 2018 |
Inhibition of human prostate smooth muscle contraction by the LIM kinase inhibitors, SR7826 and LIMKi3.
Topics: Actin Depolymerizing Factors; Cell Survival; Cells, Cultured; Electric Stimulation; Humans; Lim Kinases; Male; Muscle Contraction; Muscle, Smooth; Prostatic Neoplasms; Protein Kinase Inhibitors; Pyrazoles; Thiazoles | 2018 |
Mirabegron elicits rat corpus cavernosum relaxation and increases in vivo erectile response.
Topics: Acetanilides; Animals; Arterial Pressure; Cyclic AMP; Cyclic GMP; Gene Expression Regulation; Intracellular Space; Male; Muscle Contraction; Muscle Relaxation; Penile Erection; Penis; Rats; Rats, Wistar; Receptors, Adrenergic, beta; RNA, Messenger; Thiazoles | 2019 |
Pharmacological profile of the selective β3-adrenoceptor agonist mirabegron in cynomolgus monkeys.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; CHO Cells; Cricetulus; Cyclic AMP; Female; In Vitro Techniques; Macaca fascicularis; Muscle Contraction; Muscle, Smooth; Receptors, Adrenergic, beta-3; RNA, Messenger; Thiazoles; Urinary Bladder | 2013 |
A functional analysis of the influence of β3-adrenoceptors on the rat micturition cycle.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Female; Muscle Contraction; Perfusion; Rats; Rats, Wistar; Receptors, Adrenergic, beta-3; Thiazoles; Urinary Bladder; Urination | 2013 |
Effects of L-arginine, mirabegron, and oxybutynin on the primary bladder afferent nerve activities synchronized with reflexic, rhythmic bladder contractions in the rat.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Arginine; Electric Stimulation; Female; Mandelic Acids; Mechanotransduction, Cellular; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Neurons, Afferent; Nitric Oxide; Periodicity; Pressure; Rats, Sprague-Dawley; Reflex; Thiazoles; Time Factors; Urinary Bladder | 2015 |
VEGF receptors mediate hypoxic remodeling of adult ovine carotid arteries.
Topics: Animals; Carotid Arteries; Contractile Proteins; Dasatinib; Hypoxia; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Phosphorylation; Phthalazines; Pyridines; Pyrimidines; Receptors, Vascular Endothelial Growth Factor; Sheep; Thiazoles; Vascular Endothelial Growth Factor A; Vascular Remodeling | 2014 |
Re: a functional analysis of the influence of β3-adrenoceptors on the rat micturition cycle.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Female; Muscle Contraction; Receptors, Adrenergic, beta-3; Thiazoles; Urinary Bladder; Urination | 2014 |
Role of spinal metabotropic glutamate receptor 5 in pudendal inhibition of the nociceptive bladder reflex in cats.
Topics: Acetic Acid; Action Potentials; Animals; Cats; Disease Models, Animal; Excitatory Amino Acid Antagonists; Female; Male; Muscle Contraction; Muscle, Smooth; Nerve Fibers, Unmyelinated; Neural Inhibition; Nociception; Nociceptors; Pudendal Nerve; Pyridines; Receptor, Metabotropic Glutamate 5; Reflex; Signal Transduction; Spinal Cord Injuries; Spinal Nerves; Thiazoles; Thoracic Vertebrae; Time Factors; Urinary Bladder; Urinary Bladder, Overactive; Urodynamics | 2015 |
Involvement of β3-adrenoceptors in the inhibitory control of cholinergic activity in human bladder: Direct evidence by [(3)H]-acetylcholine release experiments in the isolated detrusor.
Topics: Acetanilides; Acetylcholine; Adrenergic beta-3 Receptor Agonists; Aminophenols; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Humans; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta-3; Sulfonamides; Thiazoles; Urinary Bladder | 2015 |
Urinary Bladder Dysfunction in Transgenic Sickle Cell Disease Mice.
Topics: Acetanilides; Adenosine Triphosphate; Anemia, Sickle Cell; Animals; Atropine; Calcium Chloride; Carbachol; Disease Models, Animal; Diuresis; Electric Stimulation; Hemoglobin, Sickle; Humans; Isoproterenol; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle Contraction; Muscle, Smooth; Phenylephrine; Potassium Chloride; Thiazoles; Urethra; Urinary Bladder | 2015 |
Acotiamide Hydrochloride, a Therapeutic Agent for Functional Dyspepsia, Enhances Acetylcholine-induced Contraction via Inhibition of Acetylcholinesterase Activity in Circular Muscle Strips of Guinea Pig Stomach.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Benzamides; Benzyl Compounds; Carbachol; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Dyspepsia; Guinea Pigs; In Vitro Techniques; Male; Morpholines; Muscle Contraction; Muscle, Smooth; Neostigmine; Stomach; Thiazoles | 2016 |
The actions of isoprenaline and mirabegron in the isolated whole rat and guinea pig bladder.
Topics: Acetanilides; Animals; Arecoline; Carbachol; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Muscarinic Agonists; Muscle Contraction; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder | 2016 |
O-GlcNAcylation is a key modulator of skeletal muscle sarcomeric morphometry associated to modulation of protein-protein interactions.
Topics: Actinin; Acylation; Animals; Cell Line; Crystallins; Desmin; Mice; Microfilament Proteins; Muscle Contraction; Muscle Fibers, Skeletal; Muscle, Skeletal; Myofibrils; Protein Interaction Maps; Protein Processing, Post-Translational; Proteome; Pyrans; Sarcomeres; Thiazoles | 2016 |
Long-term treatment with the beta-3 adrenoceptor agonist, mirabegron ameliorates detrusor overactivity and restores cyclic adenosine monophosphate (cAMP) levels in obese mice.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Body Weight; Carbachol; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Muscle Contraction; Muscle, Smooth; Obesity; Thiazoles; Urinary Bladder; Urinary Bladder, Overactive; Urination | 2017 |
PPARdelta agonism inhibits skeletal muscle PDC activity, mitochondrial ATP production and force generation during prolonged contraction.
Topics: Adenosine Triphosphate; Animals; Carbohydrate Metabolism; Electric Stimulation; Glucose; Lactic Acid; Male; Mitochondria, Muscle; Muscle Contraction; Muscle, Skeletal; Oxidation-Reduction; PPAR delta; Pyruvate Dehydrogenase Complex; Rats; Rats, Wistar; Thiazoles | 2009 |
Acotiamide hydrochloride (Z-338) enhances gastric motility and emptying by inhibiting acetylcholinesterase activity in rats.
Topics: Acetylcholinesterase; Animals; Benzamides; Cholinesterase Inhibitors; Clonidine; Electric Stimulation; Gastric Emptying; Male; Muscle Contraction; Rats; Rats, Sprague-Dawley; Stomach; Thiazoles | 2011 |
Inhibition of adrenergic human prostate smooth muscle contraction by the inhibitors of c-Jun N-terminal kinase, SP600125 and BI-78D3.
Topics: Aged; Anthracenes; Dioxanes; Humans; In Vitro Techniques; JNK Mitogen-Activated Protein Kinases; Male; Muscle Contraction; Muscle, Smooth; Prostate; Protein Kinase Inhibitors; Receptors, Adrenergic, alpha-1; Thiazoles | 2012 |
Muscle cyclo-oxygenase-2 pathway contributes to the exaggerated muscle mechanoreflex in rats with congestive heart failure.
Topics: Animals; Blood Pressure; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Heart Failure; Heart Rate; Kidney; Male; Membrane Proteins; Muscle Contraction; Muscle, Skeletal; Myocardial Infarction; Piperazines; Pyrazoles; Rats; Rats, Sprague-Dawley; Reflex, Stretch; Sulfonamides; Sympathetic Nervous System; Thiazoles | 2012 |
Effects of mirabegron, a novel β3-adrenoceptor agonist, on primary bladder afferent activity and bladder microcontractions in rats compared with the effects of oxybutynin.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Female; Mandelic Acids; Muscarinic Antagonists; Muscle Contraction; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder | 2012 |
Febuxostat improves the local and remote organ changes induced by intestinal ischemia/reperfusion in rats.
Topics: Alanine Transaminase; Allopurinol; Animals; Aspartate Aminotransferases; Dose-Response Relationship, Drug; Febuxostat; Gout Suppressants; Intestinal Mucosa; Lipid Peroxidation; Lung; Male; Malondialdehyde; Muscle Contraction; Muscle, Smooth; Peroxidase; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Thiazoles; Tumor Necrosis Factor-alpha; Xanthine Dehydrogenase; Xanthine Oxidase | 2013 |
Important role of PLC-γ1 in hypoxic increase in intracellular calcium in pulmonary arterial smooth muscle cells.
Topics: Animals; Boron Compounds; Calcium; Electron Transport Complex III; Estrenes; Gene Expression; Hypoxia; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Lentivirus; Macrocyclic Compounds; Methacrylates; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Oxazoles; Phospholipase C gamma; Pulmonary Artery; Pyrrolidinones; Reactive Oxygen Species; RNA, Small Interfering; Thiazoles; Vasoconstriction | 2013 |
The novel β3-adrenoceptor agonist mirabegron reduces carbachol-induced contractile activity in detrusor tissue from patients with bladder outflow obstruction with or without detrusor overactivity.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Aged; Aged, 80 and over; Carbachol; Humans; In Vitro Techniques; Inhibitory Concentration 50; Isoproterenol; Male; Middle Aged; Muscle Contraction; Thiazoles; Urinary Bladder; Urinary Bladder Neck Obstruction; Urinary Bladder, Overactive | 2013 |
Inhibition of muscle carbonic anhydrase slows the Ca(2+) transient in rat skeletal muscle fibers.
Topics: Acetazolamide; Action Potentials; Adenosine Triphosphatases; Animals; Benzothiazoles; Calcium; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Chelating Agents; Dose-Response Relationship, Drug; Enzyme Activation; Ethoxzolamide; Female; Fura-2; In Vitro Techniques; Ion Transport; Isometric Contraction; Muscle Contraction; Muscle Fibers, Skeletal; Muscle, Skeletal; Rats; Sarcoplasmic Reticulum; Thiadiazoles; Thiazoles; Time Factors | 2002 |
New insights into the pharmacological properties of potent antiplatelet 2-amino-benzo[d]isothiazol-3-one derivatives.
Topics: Administration, Oral; Animals; Bleeding Time; Guinea Pigs; Ileum; In Vitro Techniques; Injections, Intraperitoneal; Lethal Dose 50; Male; Mice; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Peptic Ulcer; Platelet Aggregation; Platelet Aggregation Inhibitors; Pulmonary Embolism; Thiazoles | 2002 |
Effect of thiazolidinediones and metformin on LDL oxidation and aortic endothelium relaxation in diabetic GK rats.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Arteriosclerosis; Cholesterol, LDL; Chromans; Diabetes Mellitus, Type 2; Endothelium, Vascular; Hypoglycemic Agents; Isometric Contraction; Lipid Peroxidation; Lipids; Male; Metformin; Muscle Contraction; Muscle Relaxation; Oxidation-Reduction; Pioglitazone; Rats; Rats, Wistar; Thiazoles; Thiazolidinediones; Troglitazone; Vasodilator Agents | 2003 |
New thiazole derivatives as potent and selective 5-hydroxytriptamine 3 (5-HT3) receptor agonists for the treatment of constipation.
Topics: Animals; Cathartics; Cloning, Molecular; Colon; Constipation; Defecation; Ferrets; Guinea Pigs; Humans; In Vitro Techniques; Magnetic Resonance Spectroscopy; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Recombinant Proteins; Reflex; Serotonin Receptor Agonists; Thiazoles | 2003 |
Stretch-induced contractile differentiation of vascular smooth muscle: sensitivity to actin polymerization inhibitors.
Topics: Actins; Angiotensin II; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Differentiation; Culture Techniques; Cytochalasin D; Cytoskeleton; Enzyme Activation; Enzyme Inhibitors; Female; MAP Kinase Signaling System; Microfilament Proteins; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Nucleic Acid Synthesis Inhibitors; Portal Vein; Rats; Rats, Sprague-Dawley; rhoA GTP-Binding Protein; Stress, Mechanical; Thiazoles; Thiazolidines | 2003 |
Role of Rho-kinase in maintaining airway smooth muscle contractile phenotype.
Topics: Animals; Bronchodilator Agents; Cattle; Cell Division; Cells, Cultured; DNA; Enzyme Inhibitors; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Phenotype; Potassium Chloride; Protein Serine-Threonine Kinases; rho-Associated Kinases; Tetrazolium Salts; Thiazoles; Thymidine; Trachea | 2004 |
Modulation of acto-myosin contractility in skeletal muscle myoblasts uncouples growth arrest from differentiation.
Topics: Actomyosin; Animals; Antimetabolites; Azepines; Bridged Bicyclo Compounds, Heterocyclic; Bromodeoxyuridine; Cell Adhesion; Cell Cycle; Cell Cycle Proteins; Cell Differentiation; Cell Line; Cell Membrane; Cell Proliferation; Cell Separation; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Cytoskeleton; Diacetyl; DNA; Enzyme Inhibitors; Flow Cytometry; Green Fluorescent Proteins; Image Processing, Computer-Assisted; Kinetics; Mice; Microscopy, Fluorescence; Muscle Contraction; Muscle, Skeletal; Muscles; Myosin Heavy Chains; Myosin-Light-Chain Kinase; Myosins; Naphthalenes; Polymers; Resting Phase, Cell Cycle; rho GTP-Binding Proteins; rhoA GTP-Binding Protein; Signal Transduction; Thiazoles; Thiazolidines; Time Factors; Transfection; Tumor Suppressor Proteins | 2004 |
Latrunculin B increases force fluctuation-induced relengthening of ACh-contracted, isotonically shortened canine tracheal smooth muscle.
Topics: Acetylcholine; Actin Cytoskeleton; Animals; Bridged Bicyclo Compounds, Heterocyclic; Depsipeptides; Dogs; Dose-Response Relationship, Drug; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Stress, Mechanical; Thiazoles; Thiazolidines; Trachea | 2005 |
IgA immune complex blunts the contraction of cultured mesangial cells through the inhibition of protein kinase C and intracellular calcium.
Topics: Alkaloids; Angiotensin II; Animals; Benzophenanthridines; Calcium; Cell Size; Cells, Cultured; Enzyme Activators; Enzyme Inhibitors; Glomerular Mesangium; Immunoblotting; Immunoglobulin A; Ionomycin; Ionophores; Isoenzymes; Mice; Muscle Contraction; Phenanthridines; Protein Kinase C; Tetradecanoylphorbol Acetate; Tetrazolium Salts; Thiazoles | 2004 |
Microwave-assisted solvent-free synthesis of 3-[(4-substituted piperazin-1-yl)alkyl] imidazo[2,1-b][1,3]benzothiazol-2(3H)-ones as serotonin3 (5-HT3) receptor antagonists.
Topics: Animals; Chemical Phenomena; Chemistry, Physical; Chromatography, Thin Layer; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Indicators and Reagents; Microwaves; Muscle Contraction; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Spectrophotometry, Ultraviolet; Spectroscopy, Fourier Transform Infrared; Thiazoles | 2005 |
Rat airway smooth muscle cell during actin modulation: rheology and glassy dynamics.
Topics: Actins; Animals; Azepines; Biomechanical Phenomena; Bridged Bicyclo Compounds, Heterocyclic; Bucladesine; Cells, Cultured; Cross-Linking Reagents; Cytochalasin D; Genistein; Muscle Contraction; Myocytes, Smooth Muscle; Myosins; Naphthalenes; Peptides, Cyclic; Phalloidine; Rats; Rheology; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Thiazolidines; Trachea | 2005 |
Synthesis of 1,2-benzisothiazolyloxypropanolamine derivatives and investigation of their activity at beta-adrenoceptors.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; In Vitro Techniques; Molecular Structure; Muscle Contraction; Muscle, Smooth; Rats; Structure-Activity Relationship; Thiazoles | 2005 |
Rho kinase regulates fragmentation and phagocytosis of apoptotic cells.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Amides; Animals; Apoptosis; Bridged Bicyclo Compounds, Heterocyclic; Caspase Inhibitors; Caspases; Cell Membrane; Chlorocebus aethiops; COS Cells; DNA Fragmentation; Enzyme Activation; Enzyme Inhibitors; Heterocyclic Compounds, 4 or More Rings; Intracellular Signaling Peptides and Proteins; Marine Toxins; Muscle Contraction; Myosins; PC12 Cells; Phagocytosis; Protein Serine-Threonine Kinases; Protein Transport; Pyridines; Rats; rho-Associated Kinases; RNA, Small Interfering; Thiazoles; Thiazolidines | 2006 |
PPARdelta activator GW-501516 has no acute effect on glucose transport in skeletal muscle.
Topics: AMP-Activated Protein Kinases; Animals; Carrier Proteins; Glucose; Glucose Transporter Type 4; In Vitro Techniques; Ion Channels; Male; Mitochondrial Proteins; Multienzyme Complexes; Muscle Contraction; Muscle, Skeletal; p38 Mitogen-Activated Protein Kinases; Phosphorylation; PPAR delta; Protein Serine-Threonine Kinases; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Uncoupling Protein 3 | 2006 |
Benzisothiazoles and beta-adrenoceptors: synthesis and pharmacological investigation of novel propanolamine and oxypropanolamine derivatives in isolated rat tissues.
Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Synergism; Heart Atria; Ileum; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myocardial Contraction; Propanolamines; Propranolol; Rats; Thiazoles | 2005 |
Effect of (R)-2-(2-aminothiazol-4-yl)-4'-{2-[(2-hydroxy-2-phenylethyl)amino]ethyl} acetanilide (YM178), a novel selective beta3-adrenoceptor agonist, on bladder function.
Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Animals; Carbachol; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Humans; Isoproterenol; Muscle Contraction; Propanolamines; Thiazoles; Urinary Bladder | 2007 |
Urinary retention associated with ziprasidone: a case report.
Topics: Antipsychotic Agents; Diagnostic and Statistical Manual of Mental Disorders; Efferent Pathways; Female; Humans; Middle Aged; Muscle Contraction; Muscle, Smooth; Piperazines; Psychotic Disorders; Raphe Nuclei; Thiazoles; Urinary Bladder; Urinary Retention | 2008 |
Effect of selective antagonists of group I metabotropic glutamate receptors on the micturition reflex in rats.
Topics: Animals; Female; Male; Muscle Contraction; Pyrans; Pyridines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Urinary Bladder; Urination; Urodynamics | 2008 |
Species differences in the contractile response to two specific histamine H1-receptor agonists: 2-(2-pyridyl)-ethylamine and 2-(2-aminoethyl)-thiazole.
Topics: Animals; Cimetidine; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Species Specificity; Thiazoles; Vas Deferens | 1981 |
Histamine H1- and muscarinic receptor antagonist activity of cimetidine and tiotidine in the guinea pig isolated ileum.
Topics: Animals; Carbachol; Cimetidine; Guanidines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Thiazoles | 1981 |
[Racemic guanidinothiazoles with H2-antihistaminic activity. 13 H2-antihistaminics].
Topics: Animals; Chemical Phenomena; Chemistry; Guanidines; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Thiazoles | 1983 |
Vasodilator mechanism of KB-944, a new calcium antagonist.
Topics: Adenosine; Animals; Benzothiazoles; Calcium Channel Blockers; Calcium Chloride; Coronary Vessels; Diltiazem; Dogs; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Potassium; Rabbits; Thiazoles; Vasodilator Agents; Verapamil | 1982 |
Pharmacological analysis of the mechanism of action of phenthiazamine, a piscine anesthetic.
Topics: Action Potentials; Anesthetics; Animals; Calcium; Dopamine; Fishes; Ganglia, Sympathetic; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Rana catesbeiana; Thiazoles; Ureter | 1980 |
Biological properties of 3-benzyl-1,2-benzisothiazole compounds.
Topics: Acetylcholine; Animals; Guinea Pigs; Histamine; In Vitro Techniques; Muscle Contraction; Muscle Relaxants, Central; Parasympatholytics; Thiazoles | 1982 |
Effects of semotiadil fumarate (SD-3211) and its enantiomer, SD-3212, on the changes in cytosolic Ca2+ and tension caused by KCl and norepinephrine in isolated rat aortas.
Topics: Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Bepridil; Calcium; Calcium Channel Blockers; Cytosol; Diltiazem; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rats; Rats, Wistar; Stereoisomerism; Thiazoles | 1995 |
Characterization and function of histamine receptors in corpus cavernosum.
Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles | 1995 |
Increased peak oxygen consumption of trained muscle requires increased electron flux capacity.
Topics: Animals; Blood Flow Velocity; Electron Transport; Hindlimb; Methacrylates; Mitochondria, Muscle; Muscle Contraction; Muscle, Skeletal; Myofibrils; NADH Dehydrogenase; Oxygen Consumption; Perfusion; Physical Conditioning, Animal; Rats; Rats, Sprague-Dawley; Thiazoles | 1994 |
Pharmacological profile of the novel, potent and selective peptide leukotriene antagonist (E)-2,2-diethyl-3'-[2-[2-(4-isopropyl)thiazolyl]ethenyl]succinanilic acid.
Topics: Acetylcholine; Animals; Bronchodilator Agents; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Antagonists; Ileum; In Vitro Techniques; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Male; Muscle Contraction; Muscle, Smooth; Penicillin G; Pyrilamine; Thiazoles; Trachea | 1994 |
Influence of the vinyl group on the calcium antagonistic activity of analogues of Fostedil.
Topics: Animals; Aorta, Thoracic; Benzothiazoles; Calcium Channel Blockers; In Vitro Techniques; Muscle Contraction; Rabbits; Thiazoles; Vinyl Compounds | 1994 |
Effect of diacylglycerol kinase inhibitor, R59022 on cytosolic free calcium level and force development in guinea pig taenia coli.
Topics: Animals; Calcium; Colon; Guinea Pigs; Muscle Contraction; Platelet Activating Factor; Pyrimidinones; Thiazoles | 1993 |
The effect of diabetes on sexual behavior and reproductive tract function in male rats.
Topics: Animals; Body Weight; Diabetes Mellitus, Experimental; Epididymis; Male; Muscle Contraction; Muscle, Smooth; Organ Size; Piperidines; Rats; Sexual Behavior, Animal; Sperm Count; Sperm Motility; Streptozocin; Testis; Testosterone; Thiazoles; Urinary Bladder | 1993 |
The source and action of histamine in the isolated guinea-pig gallbladder.
Topics: Animals; Dimaprit; Electric Stimulation; Female; Gallbladder; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Ranitidine; Receptors, Histamine H3; Thiazoles | 1995 |
Troglitazone reduces contraction by inhibition of vascular smooth muscle cell Ca2+ currents and not endothelial nitric oxide production.
Topics: Analysis of Variance; Animals; Arteries; Calcium Channels; Chromans; Dose-Response Relationship, Drug; Hypoglycemic Agents; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Rats; Rats, Wistar; Thiazoles; Thiazolidinediones; Troglitazone | 1997 |
Structure optimization of a leukotriene D4 antagonist by combinatorial chemistry in solution.
Topics: Animals; Anti-Asthmatic Agents; Chemistry, Pharmaceutical; Guinea Pigs; Leukotriene D4; Muscle Contraction; Muscle, Smooth; Solutions; Thiazoles | 1997 |
Arachidonic acid and its metabolites are involved in the expression of morphine dependence in guinea-pig isolated ileum.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Cyclooxygenase Inhibitors; Guinea Pigs; Ileum; In Vitro Techniques; Lipoxygenase Inhibitors; Male; Masoprocol; Meloxicam; Morphine; Muscle Contraction; Naloxone; Narcotic Antagonists; Phospholipases A; Phospholipases A2; Quinacrine; Substance-Related Disorders; Thiazines; Thiazoles; Tolmetin | 1997 |
Disparate effects of antidiabetic drugs on arterial contraction.
Topics: Animals; Arteries; Blood Pressure; Glyburide; Humans; Hypoglycemic Agents; In Vitro Techniques; Insulin; Male; Metformin; Muscle Contraction; Muscle, Smooth, Vascular; Pioglitazone; Potassium Chloride; Rats; Rats, Wistar; Tail; Thiazoles; Thiazolidinediones | 1997 |
Effects of newly synthesized amino acids containing thiazole residues on electrically evoked smooth muscle contractions.
Topics: Amino Acids; Animals; Electric Stimulation; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Mice; Molecular Structure; Muscle Contraction; Muscle, Smooth; Rabbits; Rats; Rats, Wistar; Spectrophotometry, Infrared; Thiazoles | 1998 |
Antinociceptive effect of meloxicam, in neurogenic and inflammatory nociceptive models in mice.
Topics: Abdominal Muscles; Acetic Acid; Analgesics; Analgesics, Opioid; Animals; Capsaicin; Cyclooxygenase Inhibitors; Diclofenac; Formaldehyde; Inflammation; Male; Meloxicam; Mice; Morphine; Muscle Contraction; Pain; Pain Measurement; Reaction Time; Thiazines; Thiazoles | 1998 |
Histamine receptor-independent muscle relaxation elicited by a series of histamine H2-receptor agonists on the isolated guinea pig duodenum: a study into the mechanism of action.
Topics: Animals; Dimaprit; Duodenum; Electric Stimulation; Guinea Pigs; Histamine Agonists; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Structure-Activity Relationship; Thiazoles | 1998 |
In vitro pharmacologic profile of YM158, a new dual antagonist for LTD4 and TXA2 receptors.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Carbachol; Dinoprost; Guinea Pigs; Humans; In Vitro Techniques; Leukotriene Antagonists; Leukotriene D4; Male; Membrane Proteins; Muscle Contraction; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Leukotriene; Receptors, Thromboxane; Tetrazoles; Thiazoles; Trachea | 1998 |
The effects of 8-hydroxy-2-(di-n-propylamino)tetralin on the cholinergic contraction in guinea pig and human airways in vitro.
Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Bronchi; Bronchoconstriction; Capsaicin; Cholinergic Fibers; Culture Techniques; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Humans; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pindolol; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Trachea; Tropisetron | 1998 |
Effects of histamine H2 receptor agonists and antagonists on the isolated guinea pig gallbladder.
Topics: Animals; Benzothiazoles; Dopamine Agents; Famotidine; Gallbladder; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Phenoxypropanolamines; Piperidines; Pyridines; Receptors, Histamine H2; Sincalide; Thiazoles; Triazoles | 1999 |
Actin polymerization stimulated by contractile activation regulates force development in canine tracheal smooth muscle.
Topics: Acetylcholine; Actins; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cytochalasin D; Dogs; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Phosphorylation; Polymers; Thiazoles; Thiazolidines; Trachea | 1999 |
Histamine H1 receptor ligands. Part I. Novel thiazol-4-ylethanamine derivatives: synthesis and in vitro pharmacology.
Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Agonists; Ileum; In Vitro Techniques; Ligands; Male; Muscle Contraction; Muscle, Smooth; Structure-Activity Relationship; Thiazoles | 1999 |
Tracheal relaxing effects and beta2 adrenoceptor selectivity of S1319, a novel sponge-derived bronchodilator agent, in isolated guinea-pig tissues.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Benzothiazoles; Ethanolamines; Guinea Pigs; Heart Atria; In Vitro Techniques; Male; Muscle Contraction; Receptors, Adrenergic, beta-2; Thiazoles; Trachea | 1999 |
Non-imidazole histamine H3 ligands, Part 2: New 2-substituted benzothiazoles as histamine H3 antagonists.
Topics: Animals; Guinea Pigs; Histamine Antagonists; Molecular Structure; Muscle Contraction; Muscle, Smooth; Structure-Activity Relationship; Thiazoles | 1999 |
Z-338 facilitates acetylcholine release from enteric neurons due to blockade of muscarinic autoreceptors in guinea pig stomach.
Topics: Acetylcholine; Animals; Autoreceptors; Benzamides; Gastrointestinal Agents; Guinea Pigs; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptors, Muscarinic; Stomach; Thiazoles; Xenopus | 2000 |
Z-338, a newly synthetized carboxyamide derivative, stimulates gastric motility through enhancing the excitatory neurotransmission.
Topics: Animals; Benzamides; Gastrointestinal Agents; Gastrointestinal Motility; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Stomach; Thiazoles | 2000 |
Mechanisms of vasoinhibitory effect of cardioprotective agent, CP-060S, in rat aorta.
Topics: Angiotensin II; Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Arginine Vasopressin; Calcium; Calcium Channel Blockers; Cytosol; Dinoprost; Drug Interactions; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Rats; Rats, Wistar; Thiazoles; Thiazolidines; Vasoconstrictor Agents; Vasodilator Agents | 2000 |
2-Amino-Benzo[d]isothiazol-3-one derivatives: synthesis and assessment of their antiplatelet/spasmolytic effects.
Topics: Adenosine Diphosphate; Animals; Aorta; Arachidonic Acid; Benzaldehydes; Guinea Pigs; Ileum; Inhibitory Concentration 50; Male; Models, Animal; Muscle Contraction; Parasympatholytics; Platelet Aggregation; Platelet Aggregation Inhibitors; Thiazoles | 2000 |
Potential antitumor agents. Part 29(1): synthesis and potential coanthracyclinic activity of imidazo[2,1-b]thiazole guanylhydrazones.
Topics: Animals; Antineoplastic Agents; CDC2 Protein Kinase; Cell Division; Cell Survival; Guanidine; Guinea Pigs; Humans; Hydrazones; Imidazoles; Muscle Contraction; Papillary Muscles; Starfish; Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured | 2000 |
Pharmacological profile of YM-31636, a novel 5-HT3 receptor agonist, in vitro.
Topics: Acetylcholine; Action Potentials; Animals; Anthraquinones; Atrial Function; Biguanides; Binding, Competitive; Colon; Dinoprostone; Dose-Response Relationship, Drug; Guinea Pigs; Heart Atria; Humans; In Vitro Techniques; Muscle Contraction; Myocardial Contraction; Pyrroles; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Receptor Agonists; Thiazoles | 2000 |
Pseudoproline-containing analogues of morphiceptin and endomorphin-2: evidence for a cis Tyr-Pro amide bond in the bioactive conformation.
Topics: Animals; Brain; Endorphins; Guinea Pigs; Ileum; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Mice; Muscle Contraction; Muscle, Smooth; Oligopeptides; Oxazoles; Proline; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Thiazoles; Vas Deferens | 2001 |
Inhibition of muscle carbonic anhydrase increases rise and relaxation times of twitches in rat skeletal muscle fibres.
Topics: Acetazolamide; Animals; Benzolamide; Benzothiazoles; Bicarbonates; Buffers; Carbon Dioxide; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Ethoxzolamide; Female; HEPES; Hydrogen-Ion Concentration; Muscle Contraction; Muscle Fibers, Skeletal; Muscle Relaxation; Muscle, Skeletal; Rats; Rats, Inbred WF; Sarcoplasmic Reticulum; Thiadiazoles; Thiazoles | 2002 |
Oxidative capacity interacts with oxygen delivery to determine maximal O(2) uptake in rat skeletal muscles in situ.
Topics: Animals; Enzyme Inhibitors; Hindlimb; Kinetics; Methacrylates; Mitochondria, Muscle; Muscle Contraction; Muscle, Skeletal; NADH Dehydrogenase; Oxidation-Reduction; Oxygen Consumption; Perfusion; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Thiazoles | 2002 |
The effect of the selective 5-HT(3) receptor agonist on ferret gut motility.
Topics: Animals; Benzimidazoles; Colon; Defecation; Ferrets; Gastrointestinal Motility; Male; Muscle Contraction; Pyrroles; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles | 2002 |
Effect of tazolol on beta-adrenoceptors in isolated preparations of the guinea-pig and rat.
Topics: Adrenergic beta-Agonists; Animals; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Myocardial Contraction; Propanolamines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Thiazoles; Trachea | 1977 |
Analysis of the beta-receptor mediated effect on slow-contracting skeletal muscle in vitro.
Topics: Adrenergic beta-Antagonists; Animals; Dopamine; Electric Stimulation; Epinephrine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Norepinephrine; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reserpine; Terbutaline; Thiazoles; Tyramine | 1977 |
The mode of action of tiaramide hydrochloride: a new antiasthmatic drug.
Topics: Airway Resistance; Anaphylaxis; Animals; Arachidonic Acids; Benzothiazoles; Bronchodilator Agents; Guinea Pigs; Histamine Release; Humans; In Vitro Techniques; Lung; Male; Muscle Contraction; Muscle, Smooth; Piperazines; Rabbits; Thiazoles; Thromboxane A2; Trachea | 1979 |
[Pharmacological properties of dl-2-(3'-t-butylamino-2'-hydroxypropylthio)-4-(5'-carbamoyl-2'-thienyl) thiazole hydrochloride (S-596), a new beta-adrenergic blocking agent (author's transl)].
Topics: Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Blood Pressure; Chloroform; Dogs; Epinephrine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Mice; Muscle Contraction; Myocardial Contraction; Ouabain; Practolol; Propanolamines; Propranolol; Rats; Thiazoles | 1979 |
Potentiating mechanism of bradykinin action on smooth muscle by sulfhydryl compounds.
Topics: 3-Mercaptopropionic Acid; Angiotensin I; Angiotensin II; Animals; Bradykinin; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Sulfhydryl Compounds; Thiazoles; Thiazolidines; Time Factors | 1979 |
Pharmacological properties of thiazolinobutazone (LAS 11 871). III. General pharmacology, ulcerogenic effects and acute toxicity.
Topics: Animals; Autonomic Nervous System; Brain; Cats; Diuresis; Female; Hemodynamics; Lethal Dose 50; Male; Mice; Motor Activity; Motor Skills; Muscle Contraction; Phenylbutazone; Rabbits; Rats; Respiration; Stomach Ulcer; Thiazoles | 1976 |
Calcium antagonistic and binding properties of semotiadil (SD-3211), a benzothiazine derivative assessed in cerebral and coronary arteries.
Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebral Arteries; Coronary Vessels; Cytosol; Dogs; Female; In Vitro Techniques; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Radioligand Assay; Stereoisomerism; Swine; Thiazoles | 1992 |
Significant role of peptide leukotrienes (p-LTs) in the antigen-induced contractions of human and guinea pig lung parenchymas and bronchi or tracheas in vitro.
Topics: Animals; Bronchi; Cattle; Cyclooxygenase Inhibitors; Female; gamma-Globulins; Guinea Pigs; Humans; In Vitro Techniques; Indicators and Reagents; Leukotriene Antagonists; Leukotrienes; Lung; Male; Muscle Contraction; Muscle, Smooth; Penicillin G; Thiazoles; Trachea | 1992 |
Leukotriene receptors in the skin of rats differ from those of mouse skin or rat stomach strip.
Topics: Acetophenones; Animals; Capillary Permeability; Female; Mice; Mice, Inbred BALB C; Muscle Contraction; Passive Cutaneous Anaphylaxis; Rats; Rats, Wistar; Receptors, Immunologic; Receptors, Leukotriene; Skin; Species Specificity; SRS-A; Stomach; Tetrazoles; Thiazoles | 1992 |
Synthesis of 3-[(2,3-dihydro-1,1,3-trioxo-1,2-benzisothiazol-2-yl)alkyl] 1,4-dihydropyridine-3,5-dicarboxylate derivatives as calcium channel modulators.
Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Cations; Dihydropyridines; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Potassium; Rabbits; Rats; Rats, Inbred Strains; Thiazoles | 1992 |
MCI-826 is a potent and selective antagonist of peptide leukotrienes (p-LTs) and has characteristics distinctive from those of FPL 55712.
Topics: Acetylcholine; Animals; Bronchi; Chromones; Guinea Pigs; Humans; Leukotriene Antagonists; Leukotrienes; Muscle Contraction; Muscle, Smooth; Prostaglandin D2; Respiratory Physiological Phenomena; Respiratory System; SRS-A; Thiazoles; Trachea | 1992 |
Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative structure-activity relationships of substituted 4- and 5-(2-aminoethyl)thiazoles.
Topics: Animals; Atrial Function; Chemical Phenomena; Chemistry, Physical; Electrochemistry; Guinea Pigs; Heart Atria; Histamine; Ileum; Molecular Structure; Muscle Contraction; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles | 1992 |
Pharmacologic actions of Ro 24-5913, a novel antagonist of leukotriene D4.
Topics: Animals; Bronchi; Bronchoconstriction; Guinea Pigs; Humans; Leukotrienes; Male; Muscle Contraction; Muscle, Smooth; Receptors, Immunologic; Receptors, Leukotriene; SRS-A; Thiazoles; Trachea | 1991 |
4- or 5- (omega-aminoalkyl) thiazoles and derivatives; new selective H2-receptor agonists.
Topics: Amines; Animals; Atrial Function; Guanidines; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Ileum; Imidazoles; Impromidine; Molecular Structure; Muscle Contraction; Receptors, Histamine H2; Thiazoles | 1991 |
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil | 1991 |
Studies on heterocyclic compounds: 1,3-thiazolidin-4-one derivatives. V. Pharmacological activity of substituted 2-phenyl-3-(N,N-dimethylaminoprophyl)-1,3-thiazolidin-4-one .
Topics: Animals; Female; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Male; Muscle Contraction; Muscle, Smooth; Pyrilamine; Schiff Bases; Structure-Activity Relationship; Thiazoles; Thiazolidines | 1991 |
Role of phosphatidic acid in carbachol-induced contraction in guinea pig Taenia coli.
Topics: Animals; Biological Transport, Active; Calcium; Carbachol; Colon; Diacylglycerol Kinase; Diglycerides; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Phosphatidic Acids; Phosphotransferases; Pyrimidinones; Thiazoles | 1991 |
Involvement of protein kinase C in Ca(2+)-independent contraction of rat uterine smooth muscle.
Topics: Animals; Blotting, Western; Brain; Calcium; Electrophoresis, Polyacrylamide Gel; Female; In Vitro Techniques; Isoenzymes; Muscle Contraction; Muscle, Smooth; Oxytocin; Protein Kinase C; Pyrimidinones; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Thiazoles; Uterus | 1991 |
Selective implication of thromboxane A2 and PAF-acether in two guinea pig anaphylactic models.
Topics: Anaphylaxis; Animals; Antigens; Glyceryl Ethers; Guinea Pigs; Immunoglobulin E; Immunoglobulin G; In Vitro Techniques; Indomethacin; Muscle Contraction; Platelet Activating Factor; Thiazoles; Thromboxane A2; Trachea | 1990 |
Tissue selectivity of the novel calcium antagonist sesamodil fumarate in isolated smooth muscles and cardiac muscles.
Topics: Animals; Calcimycin; Calcium Channel Blockers; Diltiazem; Guinea Pigs; Heart; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Nicardipine; Nifedipine; Rabbits; Swine; Thiazoles; Verapamil | 1990 |
Ebselen inhibits contractile responses of guinea-pig parenchymal lung strips.
Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Azoles; Catechols; Cyclooxygenase Inhibitors; Guinea Pigs; Histamine; Indomethacin; Isoindoles; Isoquinolines; Lung; Male; Masoprocol; Muscle Contraction; Muscle, Smooth; Organoselenium Compounds; Piperazines; Potassium Chloride; Selenium; Thiazoles | 1990 |
Changes in capillary perfusion induced by different patterns of activity in rat skeletal muscle.
Topics: Animals; Benzothiazoles; Capillaries; Fluorescent Dyes; Male; Muscle Contraction; Muscles; Myofibrils; Rats; Rats, Inbred Strains; Regional Blood Flow; Thiazoles | 1990 |
Tentacle contraction in Heliophrya erhardi (Suctoria): the role of inositol phospholipid metabolites and cyclic nucleotides in stimulus-response coupling.
Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Chlorides; Ciliophora; Cyclic AMP; Cyclic GMP; Dibutyryl Cyclic GMP; Inositol Phosphates; Lithium; Lithium Chloride; Muscle Contraction; Pyrimidinones; Sugar Phosphates; Tetradecanoylphorbol Acetate; Thiazoles | 1988 |
The diacylglycerol kinase inhibitor, R 59022, suppresses contractility of intestinal smooth muscle.
Topics: Acetylcholine; Animals; Calcium; Diacylglycerol Kinase; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Phosphotransferases; Platelet Activating Factor; Pyrimidinones; Substance P; Thiazoles | 1989 |
R 56865 differentiates between contractile agents with respect to the nifedipine-sensitive component in the isolated rat aorta.
Topics: Angiotensin II; Animals; Aorta, Thoracic; Arginine Vasopressin; Benzothiazoles; Calcium; Calcium Channels; Cytosol; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Thiazoles | 1989 |
Pharmacological profile of 48740 R.P., a PAF-acether antagonist.
Topics: Animals; Blood Cell Count; Blood Platelets; Bronchodilator Agents; Guinea Pigs; Humans; In Vitro Techniques; Macrophages; Male; Muscle Contraction; Muscle, Smooth; N-Formylmethionine Leucyl-Phenylalanine; Perfusion; Platelet Activating Factor; Platelet Aggregation; Pulmonary Alveoli; Pyridines; Rabbits; Radioimmunoassay; Superoxides; Thiazoles; Thromboxane B2 | 1988 |
[C-2 basically substituted thiazoles with H2-antagonistic action. 21. H2-antihistaminics].
Topics: Animals; Chemical Phenomena; Chemistry; Electric Stimulation; Gastric Acid; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Inbred Strains; Thiazoles | 1985 |
Cholinergic effects of histamine-H2 receptor antagonists partly through inhibition of acetylcholinesterase.
Topics: Animals; Butyrylcholinesterase; Cholinesterase Inhibitors; Cimetidine; Famotidine; Guinea Pigs; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Ranitidine; Thiazoles | 1986 |
Direct effects of H2-receptor antagonists on airway smooth muscle and on responses mediated by H1- and H2-receptors.
Topics: Animals; Cimetidine; Famotidine; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ranitidine; Thiazoles; Trachea | 1987 |
Pharmacology of the novel H2 antagonist famotidine: in vitro studies.
Topics: Animals; Famotidine; Female; Gallbladder; Gastric Acid; Gastrointestinal Motility; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Myocardial Contraction; Rats; Thiazoles; Uterus | 1986 |
Modulation of calmodulin function and of Ca2+-induced smooth muscle contraction by the calmodulin antagonist, HT-74.
Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Anilino Naphthalenesulfonates; Animals; Benzothiazoles; Calcium; Calmodulin; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Protein Kinases; Rabbits; Sulfonamides; Thiazoles | 1986 |
PAF antagonists: different effects on platelets, neutrophils, guinea pig ileum and PAF-induced vasodilation in isolated rat lung.
Topics: Alprazolam; Angiotensin II; Animals; Blood Platelets; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Muscle Contraction; Neutrophils; Phospholipid Ethers; Platelet Activating Factor; Platelet Membrane Glycoproteins; Pulmonary Artery; Pulmonary Circulation; Rabbits; Rats; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Serotonin; SRS-A; Thiazoles; Vasodilation | 1986 |
Prostaglandins involved in contractions by angiotensin II and bradykinin of isolated dog sphincter pupillae.
Topics: Angiotensin II; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Arachidonic Acids; Bradykinin; Dinoprost; Dogs; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Prostaglandins; Pupil; Thiazoles; Thromboxane A2 | 1988 |
Different effects of R 56865 and calcium entry blockers on K+- and noradrenaline-induced contractions and 45Ca uptake in rat aorta.
Topics: Animals; Aorta; Benzothiazoles; Calcium; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Flunarizine; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Piperidines; Potassium; Rats; Rats, Inbred Strains; Thiazoles; Verapamil | 1988 |
Novel calcium antagonists. Synthesis and structure-activity relationship studies of benzothiazoline derivatives.
Topics: Animals; Blood Pressure; Calcium Channel Blockers; Chemical Phenomena; Chemistry; Guinea Pigs; Heart Conduction System; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Pulmonary Embolism; Rabbits; Rats; Rats, Inbred SHR; Structure-Activity Relationship; Thiazoles | 1988 |
Acetylene compounds of potential pharmacological value. XL. N-(tert-aminoalkynyl)-substituted 3-isothiazolidinone-1,1-dioxides and tetrahydro-1,2-thiazin-3-one-1,1-dioxides.
Topics: Animals; Anticonvulsants; Benzopyrans; Carbachol; Chemical Phenomena; Chemistry; Chromans; Cyclic S-Oxides; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Structure-Activity Relationship; Thiazines; Thiazoles | 1987 |
Selective -adrenergic myocardial stimulant.
Topics: Acetanilides; Adrenergic beta-Agonists; Amino Alcohols; Amphetamine; Animals; Blood Pressure; Dogs; Female; Heart; Heart Rate; Isoproterenol; Male; Muscle Contraction; Propylamines; Propylene Glycols; Stimulation, Chemical; Thiazoles | 1972 |
Cross tolerance to histamine by the chronic administration of histamine analogues.
Topics: Aerosols; Animals; Asthma; Blood Pressure; Body Weight; Cats; Desensitization, Immunologic; Dogs; Drug Tolerance; Ethylamines; Female; Gastric Juice; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Intestines; Muscle Contraction; Muscle, Smooth; Pyrazoles; Pyridines; Reaction Time; Stimulation, Chemical; Thiazoles | 1972 |
The mechanism of the paralysing action of tetramisole on Ascaris somatic muscle.
Topics: Acetylcholine; Animals; Anthelmintics; Ascaris; Curare; Female; Male; Membrane Potentials; Muscle Contraction; Muscles; Piperazines; Potassium; Thiazoles | 1970 |