Compounds > thiazoles
Page last updated: 2024-08-21

thiazoles and Muscle Contraction

thiazoles has been researched along with Muscle Contraction in 127 studies

Research

Studies (127)

TimeframeStudies, this research(%)All Research%
pre-199029 (22.83)18.7374
1990's38 (29.92)18.2507
2000's30 (23.62)29.6817
2010's22 (17.32)24.3611
2020's8 (6.30)2.80

Authors

AuthorsStudies
Hennenberg, M; Huang, R; Stief, CG; Strittmatter, F; Tamalunas, A; Waidelich, R1
Chess-Williams, R; Lim, I1
Clodfelder-Miller, B; McNaught, J; Ness, TJ; Su, X1
Chermansky, C; Ikeda, Y; Kanai, A; Mizoguchi, S; Singh, N; Suzuki, T; Tyagi, P; Yoshimura, N; Zabbarova, I1
Budriesi, R; Caputo, L; Cavalluzzi, MM; Corazza, I; De Salvia, MA; Franchini, C; Gualdani, R; Lentini, G; Micucci, M; Milani, G; Piarulli, M; Quintieri, L; Rosato, A; Viale, M1
Chimoto, J; Morikawa, K; Okura, T; Shiho, M; Shinozuka, K; Wakuda, H; Yamada, S1
Jung, DW; Kim, HJ; Kim, JH; Kim, SW; Lee, JH; Um, J; Williams, DR1
Deshpande, DA; Javed, E; Kambayashi, T; Lim, JM; Nayak, AP; Pan, S; Panettieri, RA; Penn, RB; Shah, SD; Sharma, P; Yadav, SK1
Kida, J; Mashimo, H; Matsuya, H; Okada, H; Sekido, N; Wakamatsu, D1
Ciotkowska, A; Gratzke, C; Hennenberg, M; Herlemann, A; Rutz, B; Sterr, CM; Stief, CG; Strittmatter, F; Wang, X; Wang, Y; Yu, Q1
Antunes, E; Bertollotto, GM; Candido, TZ; De Nucci, G; de Oliveira, MG; Kiguti, LRA; Mónica, FZ; Pupo, AS; Rojas-Moscoso, JA1
Hatanaka, T; Masuda, N; Ohtake, A; Sato, S; Someya, A; Suzuki, M; Ueshima, K; Ukai, M; Watanabe, M1
Drake, MJ; Paton, JF; Pickering, AE; Sadananda, P1
Aizawa, N; Homma, Y; Igawa, Y2
Adeoye, OO; Bouthors, V; Hubbell, MC; Pearce, WJ; Williams, JM1
Atala, A1
de Groat, WC; Reese, JN; Rogers, MJ; Roppolo, JR; Schwen, Z; Shen, B; Tai, C; Wang, J; Xiao, Z1
Calvi, P; D' Agostino, G; Maria Condino, A1
Alexandre, EC; Antunes, E; Claudino, MA; Costa, FF; da Silva, FH; de Nucci, G; Fertrin, KY; Franco-Penteado, CF; Leiria, LO; Mónica, FZ; Renno, A1
Hirayama, M; Hori, Y; Ito, K; Kawabata, Y; Kawachi, M; Matsunaga, Y; Nagahama, K; Ozaki, T; Shiraishi, Y; Takei, M; Tanaka, T1
De Wachter, S; Eastham, J; Gillespie, J; Persyn, S; Wyndaele, JJ1
Bastide, B; Cieniewski-Bernard, C; Deracinois, B; Duban-Deweer, S; Dupont, E; Krzewinski, F; Lambert, M; Richard, E1
Alexandre, EC; Antunes, E; Calmasini, FB; Candido, TZ; da Silva, CPV; da Silva, FH; de Oliveira, MG; Mónica, FZ1
Baker, DJ; Constantin, D; Constantin-Teodosiu, D; Greenhaff, PL1
Hirayama, M; Hori, Y; Inoue, N; Ito, K; Kawabata, Y; Kawachi, M; Matsunaga, Y; Nagahama, K; Ozaki, T; Takei, M; Tanaka, T; Toda, R; Yoshii, K1
Andersson, KE; Beckmann, C; Göttinger, J; Gratzke, C; Hedlund, P; Hennenberg, M; Roosen, A; Schlenker, B; Stief, CG; Strittmatter, F; Walther, S1
Gao, W; Li, J; Lu, J; Morales, A; Xing, J1
Shafik, AN1
Joseph, L; Mei, L; Song, T; Wang, YX; Yadav, VR; Zheng, YM1
Andersson, KE; Bouchelouche, K; Bouchelouche, P; Korstanje, C; Nordling, J; Svalø, J1
Gros, G; Kleinke, T; Papadopoulos, S; Wetzel, P1
Ballabeni, V; Barocelli, E; Calcina, F; Impicciatore, M; Tognolini, M; Vicini, P1
Iida, KT; Iwama, Y; Kamata, K; Kawakami, Y; Mokuno, H; Shimada, K; Shimano, H; Sone, H; Suzuki, M; Toyoshima, H; Watanabe, Y; Yamada, N1
Akuzawa, S; Imanishi, N; Ito, H; Iwaoka, K; Kazuta, K; Kiso, T; Koshio, H; Mase, T; Nagashima, SY; Ohta, M; Sakamoto, S; Tsukamoto, S1
Albinsson, S; Hellstrand, P; Malmqvist, U; Nordström, I; Swärd, K; Zeidan, A1
Gosens, R; Meurs, H; Nelemans, SA; Schaafsma, D; Zaagsma, J1
Dhawan, J; Helfman, DM1
Dowell, ML; Fredberg, JJ; Gerthoffer, WT; Halayko, AJ; Lakser, OJ; Mitchell, RW; Solway, J; Stelmack, GL1
Chen, A; Chin, TY; Chueh, SH; Jin, JS; Ka, SM; Lee, HS; Lee, WH; Lin, YF; Sheu, LF; Yao, CW1
Mahesh, R; Pandi, PV; Perumal, RV1
An, SS; Butler, JP; Fabry, B; Fredberg, JJ; Laudadio, RE; Millet, EJ1
Comini, M; Menozzi, A; Morini, G; Poli, E; Pozzoli, C2
Orlando, KA; Pittman, RN; Stone, NL1
Han, DH; Holloszy, JO; Terada, S; Wicke, S1
Maruyama, T; Matsui, T; Miyata, K; Nagase, I; Sasamata, M; Sato, S; Takasu, T; Uchida, H; Ukai, M; Yamaguchi, O1
Dowell, ML; Lakser, OJ; Mitchell, RW; Solway, J1
Certa, K; Chism, LM; Mago, R; Pinninti, NR1
Angelico, P; Clarke, DE; Farina, P; Guarneri, L; Leonardi, A; Poggesi, E; Testa, R1
Vohra, MM1
Barker, LA1
Schunack, W; Spengler, JP1
Ito, K; Kanazawa, T; Morita, T; Nose, T1
Hachisu, M; Koeda, T; Sekizawa, Y; Shitoh, K1
Impicciatore, M; Plazzi, PV; Vitali, T1
Ito, K; Ito, KM; Murakami, K; Shindo, K1
Carson, CC; Davies, MG; Hagen, PO; Kim, YC; Lee, TH1
Ogilvie, RW; Robinson, DM; Terjung, RL; Tullson, PC1
Kadowaki, S; Nakao, E; Takahashi, K; Umezu, K; Yamada, K; Yamada, N1
Baziard-Mouysset, G; Bonnafous, R; Payard, M; Stigliani, JL; Tchani, G; Tisne-Versailles, J1
Momose, K; Nobe, K; Ohata, H2
Elhilali, MM; Gagnon, C; Hassan, AA; Hassouna, MM; Taketo, T1
Davison, JS; Jennings, LJ; Lea, RW; Pozo, MJ; Salido, GM; Sharkey, KA; Singh, J1
Barazi, M; Dominguez, LJ; Igwe, R; Ram, JL; Song, J; Sowers, JR; Walsh, MF1
Maehr, H; Yang, R1
Capasso, A; Sorrentino, L1
Bourghli, M; Miller, JA; Peuler, JD; Soltis, EE; Sowers, JR; Zammam, HY1
Bocheva, A; Golovinsky, E; Stanchev, M; Todorov, S1
De Freitas, GA; Santos, AR; Vedana, EM1
Bertaccini, G; Coruzzi, G; Poli, E; Pozzoli, C; Timmerman, H1
Arakida, Y; Honda, K; Miyata, K; Ohga, K; Suwa, K; Yamada, T; Yokota, M1
De Leyn, P; Demedts, MG; Deneffe, G; Dupont, LJ; Pype, JL; Verleden, GM1
Bertaccini, G; Coppelli, G; Coruzzi, G; Poli, E; Pozzoli, C1
Gunst, SJ; Mehta, D1
Glinka, R; Timmerman, H; Walczyński, K; Zhang, MQ; Zuiderveld, OP1
Fukamachi, H; Higa, T; Miura, T; Sakakibara, M; Sindo, K; Suzuki, H; Takei, M; Ueno, A1
Guryn, R; Timmerman, H; Walczyński, K; Zuiderveld, OP1
Kaibara, M; Kurimoto, T; Ogishima, M; Taniyama, K; Ueki, S1
Ito, Y; Nakajima, T; Nawata, H1
Adachi, Y; Karaki, H; Satake, N; Sato, K; Shibata, S1
Amoretti, L; Ballabeni, V; Barocelli, E; Tognolini, M; Vicini, P1
Andreani, A; Garaliene, V; Leoni, A; Locatelli, A; Morigi, R; Rambaldi, M; Recanatini, M1
Akuzawa, S; Ito, H; Iwaoka, K; Kamato, T; Kiso, T; Miyata, K; Nagakura, Y; Naitoh, Y; Sakai, H; Suzuki, M; Yamaguchi, T; Yamano, M; Yuki, H1
Boissard, C; Chung, NN; Keller, M; Lemieux, C; Mutter, M; Patiny, L; Schiller, PW1
Gros, G; Papadopoulos, S; Wetzel, P1
Hagen, JL; Hepple, RT; Krause, DJ1
Ito, H; Iwaoka, K; Kiso, T; Miyata, K; Nagakura, Y; Yamaguchi, T1
Clark, SJ; Poyser, RH1
Waldeck, B1
Berti, F; Folco, GC; Malandrino, S; Omini, C; Sautebin, L; Viganò, T1
Aono, S; Hara, Y; Miyagishi, A; Nakatani, H; Sato, E1
Iso, T; Iwao, J; Nishimura, K; Oya, M1
Colombo, M; Márquez, M; Roberts, DJ1
Morimoto, K; Nakayama, K; Nozawa, Y; Tanaka, Y1
Horiba, M; Nabe, T; Ohata, K; Watanabe-Kohno, S; Yamamura, H; Yasui, K1
Goto, S; Inagaki, N; Koda, A; Miura, T; Nagai, H; Yoshida, K1
Alonso, S; Artalejo, CR; Cillero, J; Fau de Casa-Juana, M; García, AG; González-Morales, MA; López, MG; Santos, L; Sunkel, CE; Villarroya, M1
Horiba, M; Nabe, T; Ohata, K; Watanabe-Kohno, S; Yamamura, H1
Eriks, JC; Sterk, GJ; Timmerman, H; van der Goot, H1
Crowley, HJ; O'Donnell, M; O'Neill, N; Welton, AF; Yaremko, B1
Eriks, JC; Sterk, GJ; Timmerman, H; van Acker, SA; van der Aar, EM; van der Goot, H1
Mutafova-Yambolieva, V; Staneva-Stoytcheva, D; Todorov, S; Vassilev, P1
Calignano, A; Diurno, MV; Mazzoni, O; Piscopo, E1
Karibe, H; Oishi, K; Uchida, MK1
Bertrand, C; Landry, Y; Tschirhart, E1
Iso, T; Miyawaki, N; Nishimura, K; Yamauchi, H1
Bast, A; Leurs, R; Timmerman, H1
Egginton, S; Hargreaves, D; Hudlická, O1
Butler, RD; Evans, RL; McCrohan, CR1
Holzer, P; Lippe, IT1
Koch, P; Peters, T; Wilffert, B; Wilhelm, D1
Benveniste, J; Coëffier, E; Desquand, S; Floch, A; Lefort, J; Maridonneau-Parini, I; Randon, J; Sedivy, P; Vargaftig, BB1
Postius, S; Sattler, HJ; Schunack, W; Szelenyi, I; Trumm, KA1
Aono, M; Mizuta, K; Moriga, M; Narusawa, H1
Hashimoto, Y; Iwatsuki, N; Koga, Y1
Adami, M; Bertaccini, G; Coruzzi, G; Poli, E1
Hidaka, H; Ishikawa, T; Ito, M; Itoh, H; Kawamatsu, Y; Saitoh, M; Shin, T; Sugihara, H; Tanaka, T; Umekawa, H1
Chang, SW; Henson, PM; McMurtry, IF; Pfeffer, KD; Voelkel, NF; Worthen, SG1
Bian, K; Inatomi, A; Lu, W; Okamura, T; Toda, N1
Koch, P; Nebel, U; Peters, T; Wermelskirchen, D; Wilffert, B; Wilhelm, D1
Fujita, M; Iso, T; Iwao, J; Kato, E; Kawashima, Y; Oya, M; Tabashi, K; Yamamoto, K1
Dahlbom, R; Lindeke, B; Ringdahl, B1
Berkoz, B; Edwards, JA; Fried, JH; Halpern, O; Lewis, GS; Miller, LM; Roszkowski, AP; Strosberg, AM1
Ambrus, CM; Ambrus, JL1
Aceves, J; Erlij, D; Martínez-Marañón, R1

Reviews

1 review(s) available for thiazoles and Muscle Contraction

ArticleYear
Force fluctuation-induced relengthening of acetylcholine-contracted airway smooth muscle.
    Proceedings of the American Thoracic Society, 2008, Jan-01, Volume: 5, Issue:1

    Topics: Acetylcholine; Actin Cytoskeleton; Animals; Asthma; Bridged Bicyclo Compounds, Heterocyclic; Depsipeptides; Humans; Mitogen-Activated Protein Kinases; Muscle Contraction; Muscle, Smooth; Myosins; Stress, Mechanical; Thiazoles; Thiazolidines

2008

Other Studies

126 other study(ies) available for thiazoles and Muscle Contraction

ArticleYear
Inhibition of Full Smooth Muscle Contraction in Isolated Human Detrusor Tissues by Mirabegron Is Limited to Off-Target Inhibition of Neurogenic Contractions.
    The Journal of pharmacology and experimental therapeutics, 2022, Volume: 381, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Acetanilides; Carbachol; Endothelin-1; Female; Humans; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Receptors, Adrenergic; Thiazoles; Urinary Bladder, Overactive

2022
Mirabegron attenuates porcine ureteral contractility via α1-adrenoceptor antagonism.
    Naunyn-Schmiedeberg's archives of pharmacology, 2022, Volume: 395, Issue:7

    Topics: Acetanilides; Adrenergic beta-Antagonists; Animals; Muscle Contraction; Phenylephrine; Receptors, Adrenergic, alpha-1; Serotonin; Swine; Thiazoles

2022
Medications used to treat bladder disorders may alter effects of neuromodulation.
    Neurourology and urodynamics, 2020, Volume: 39, Issue:5

    Topics: Acetanilides; Animals; Cystitis; Electric Stimulation Therapy; Female; Mandelic Acids; Muscle Contraction; Pudendal Nerve; Rats; Rats, Sprague-Dawley; Thiazoles; Urological Agents

2020
Excitatory effect of acotiamide on rat and human bladder: Implications for underactive bladder treatment.
    Life sciences, 2020, Oct-01, Volume: 258

    Topics: Animals; Benzamides; Carbachol; Electric Stimulation; Humans; Male; Muscle Contraction; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder; Urinary Bladder, Underactive

2020
Lubeluzole: from anti-ischemic drug to preclinical antidiarrheal studies.
    Pharmacological reports : PR, 2021, Volume: 73, Issue:1

    Topics: Animals; Anti-Bacterial Agents; Antidiarrheals; Bacteria; Colon; Diarrhea; Dose-Response Relationship, Drug; Gram-Negative Bacterial Infections; Gram-Positive Bacterial Infections; Guinea Pigs; Ileum; Loperamide; Male; Microbial Sensitivity Tests; Muscle Contraction; Neuroprotective Agents; Piperidines; Quaternary Ammonium Compounds; Rats; Rats, Sprague-Dawley; Thiazoles

2021
Possible Involvement of Muscarinic Receptor Blockade in Mirabegron Therapy for Patients with Overactive Bladder.
    The Journal of pharmacology and experimental therapeutics, 2021, Volume: 377, Issue:2

    Topics: Acetanilides; Administration, Oral; Adrenergic beta-3 Receptor Agonists; Animals; Brain; Male; Muscarinic Antagonists; Muscle Contraction; Protein Binding; Rats; Rats, Sprague-Dawley; Receptors, Muscarinic; Submandibular Gland; Thiazoles; Urinary Bladder; Urinary Bladder, Overactive; Urological Agents

2021
Lithium Chloride Protects against Sepsis-Induced Skeletal Muscle Atrophy and Cancer Cachexia.
    Cells, 2021, 04-26, Volume: 10, Issue:5

    Topics: Animals; Body Weight; Cachexia; Cell Differentiation; Cell Proliferation; Culture Media, Conditioned; Glycogen Synthase Kinase 3 beta; Inflammation; Lipopolysaccharides; Lithium Chloride; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Muscle Contraction; Muscle Fibers, Skeletal; Muscle Proteins; Muscle, Skeletal; Muscular Atrophy; Neoplasms; RAW 264.7 Cells; RNA, Small Interfering; Sepsis; SKP Cullin F-Box Protein Ligases; Tetrazolium Salts; Thiazoles

2021
Diacylglycerol Kinase Inhibition Reduces Airway Contraction by Negative Feedback Regulation of Gq-Signaling.
    American journal of respiratory cell and molecular biology, 2021, Volume: 65, Issue:6

    Topics: Bronchoconstriction; Cells, Cultured; Diacylglycerol Kinase; Gene Knockdown Techniques; GTP-Binding Protein alpha Subunits, Gq-G11; Humans; Muscle Contraction; Muscle, Smooth; Pyrimidinones; Signal Transduction; Thiazoles

2021
Effects of an EP2 and EP3 Receptor Dual Agonist, ONO-8055, on a Radical Hysterectomy-Induced Underactive Bladder Model in Monkeys.
    Lower urinary tract symptoms, 2018, Volume: 10, Issue:2

    Topics: Animals; Cholinesterase Inhibitors; Disease Models, Animal; Female; Hysterectomy; Macaca fascicularis; Muscle Contraction; Pyridinium Compounds; Receptors, Prostaglandin E, EP2 Subtype; Receptors, Prostaglandin E, EP3 Subtype; Rheology; Thiazoles; Urinary Bladder, Neurogenic; Urination

2018
Inhibition of human prostate smooth muscle contraction by the LIM kinase inhibitors, SR7826 and LIMKi3.
    British journal of pharmacology, 2018, Volume: 175, Issue:11

    Topics: Actin Depolymerizing Factors; Cell Survival; Cells, Cultured; Electric Stimulation; Humans; Lim Kinases; Male; Muscle Contraction; Muscle, Smooth; Prostatic Neoplasms; Protein Kinase Inhibitors; Pyrazoles; Thiazoles

2018
Mirabegron elicits rat corpus cavernosum relaxation and increases in vivo erectile response.
    European journal of pharmacology, 2019, Sep-05, Volume: 858

    Topics: Acetanilides; Animals; Arterial Pressure; Cyclic AMP; Cyclic GMP; Gene Expression Regulation; Intracellular Space; Male; Muscle Contraction; Muscle Relaxation; Penile Erection; Penis; Rats; Rats, Wistar; Receptors, Adrenergic, beta; RNA, Messenger; Thiazoles

2019
Pharmacological profile of the selective β3-adrenoceptor agonist mirabegron in cynomolgus monkeys.
    Naunyn-Schmiedeberg's archives of pharmacology, 2013, Volume: 386, Issue:11

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; CHO Cells; Cricetulus; Cyclic AMP; Female; In Vitro Techniques; Macaca fascicularis; Muscle Contraction; Muscle, Smooth; Receptors, Adrenergic, beta-3; RNA, Messenger; Thiazoles; Urinary Bladder

2013
A functional analysis of the influence of β3-adrenoceptors on the rat micturition cycle.
    The Journal of pharmacology and experimental therapeutics, 2013, Volume: 347, Issue:2

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Female; Muscle Contraction; Perfusion; Rats; Rats, Wistar; Receptors, Adrenergic, beta-3; Thiazoles; Urinary Bladder; Urination

2013
Effects of L-arginine, mirabegron, and oxybutynin on the primary bladder afferent nerve activities synchronized with reflexic, rhythmic bladder contractions in the rat.
    Neurourology and urodynamics, 2015, Volume: 34, Issue:4

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Arginine; Electric Stimulation; Female; Mandelic Acids; Mechanotransduction, Cellular; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Nerve Fibers, Myelinated; Nerve Fibers, Unmyelinated; Neurons, Afferent; Nitric Oxide; Periodicity; Pressure; Rats, Sprague-Dawley; Reflex; Thiazoles; Time Factors; Urinary Bladder

2015
VEGF receptors mediate hypoxic remodeling of adult ovine carotid arteries.
    Journal of applied physiology (Bethesda, Md. : 1985), 2014, Oct-01, Volume: 117, Issue:7

    Topics: Animals; Carotid Arteries; Contractile Proteins; Dasatinib; Hypoxia; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Phosphorylation; Phthalazines; Pyridines; Pyrimidines; Receptors, Vascular Endothelial Growth Factor; Sheep; Thiazoles; Vascular Endothelial Growth Factor A; Vascular Remodeling

2014
Re: a functional analysis of the influence of β3-adrenoceptors on the rat micturition cycle.
    The Journal of urology, 2014, Volume: 192, Issue:1

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Female; Muscle Contraction; Receptors, Adrenergic, beta-3; Thiazoles; Urinary Bladder; Urination

2014
Role of spinal metabotropic glutamate receptor 5 in pudendal inhibition of the nociceptive bladder reflex in cats.
    American journal of physiology. Renal physiology, 2015, Apr-15, Volume: 308, Issue:8

    Topics: Acetic Acid; Action Potentials; Animals; Cats; Disease Models, Animal; Excitatory Amino Acid Antagonists; Female; Male; Muscle Contraction; Muscle, Smooth; Nerve Fibers, Unmyelinated; Neural Inhibition; Nociception; Nociceptors; Pudendal Nerve; Pyridines; Receptor, Metabotropic Glutamate 5; Reflex; Signal Transduction; Spinal Cord Injuries; Spinal Nerves; Thiazoles; Thoracic Vertebrae; Time Factors; Urinary Bladder; Urinary Bladder, Overactive; Urodynamics

2015
Involvement of β3-adrenoceptors in the inhibitory control of cholinergic activity in human bladder: Direct evidence by [(3)H]-acetylcholine release experiments in the isolated detrusor.
    European journal of pharmacology, 2015, Jul-05, Volume: 758

    Topics: Acetanilides; Acetylcholine; Adrenergic beta-3 Receptor Agonists; Aminophenols; Dose-Response Relationship, Drug; Electric Stimulation; Ethanolamines; Humans; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Propanolamines; Receptors, Adrenergic, beta-3; Sulfonamides; Thiazoles; Urinary Bladder

2015
Urinary Bladder Dysfunction in Transgenic Sickle Cell Disease Mice.
    PloS one, 2015, Volume: 10, Issue:8

    Topics: Acetanilides; Adenosine Triphosphate; Anemia, Sickle Cell; Animals; Atropine; Calcium Chloride; Carbachol; Disease Models, Animal; Diuresis; Electric Stimulation; Hemoglobin, Sickle; Humans; Isoproterenol; Mice; Mice, Inbred C57BL; Mice, Transgenic; Muscle Contraction; Muscle, Smooth; Phenylephrine; Potassium Chloride; Thiazoles; Urethra; Urinary Bladder

2015
Acotiamide Hydrochloride, a Therapeutic Agent for Functional Dyspepsia, Enhances Acetylcholine-induced Contraction via Inhibition of Acetylcholinesterase Activity in Circular Muscle Strips of Guinea Pig Stomach.
    Drug research, 2016, Volume: 66, Issue:4

    Topics: Acetylcholine; Acetylcholinesterase; Animals; Benzamides; Benzyl Compounds; Carbachol; Cholinesterase Inhibitors; Dose-Response Relationship, Drug; Drug Interactions; Dyspepsia; Guinea Pigs; In Vitro Techniques; Male; Morpholines; Muscle Contraction; Muscle, Smooth; Neostigmine; Stomach; Thiazoles

2016
The actions of isoprenaline and mirabegron in the isolated whole rat and guinea pig bladder.
    Autonomic neuroscience : basic & clinical, 2016, Volume: 198

    Topics: Acetanilides; Animals; Arecoline; Carbachol; Female; Guinea Pigs; In Vitro Techniques; Isoproterenol; Muscarinic Agonists; Muscle Contraction; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder

2016
O-GlcNAcylation is a key modulator of skeletal muscle sarcomeric morphometry associated to modulation of protein-protein interactions.
    Biochimica et biophysica acta, 2016, Volume: 1860, Issue:9

    Topics: Actinin; Acylation; Animals; Cell Line; Crystallins; Desmin; Mice; Microfilament Proteins; Muscle Contraction; Muscle Fibers, Skeletal; Muscle, Skeletal; Myofibrils; Protein Interaction Maps; Protein Processing, Post-Translational; Proteome; Pyrans; Sarcomeres; Thiazoles

2016
Long-term treatment with the beta-3 adrenoceptor agonist, mirabegron ameliorates detrusor overactivity and restores cyclic adenosine monophosphate (cAMP) levels in obese mice.
    Neurourology and urodynamics, 2017, Volume: 36, Issue:6

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Body Weight; Carbachol; Cyclic AMP; Cyclic Nucleotide Phosphodiesterases, Type 4; Male; Mice; Mice, Inbred C57BL; Mice, Obese; Muscle Contraction; Muscle, Smooth; Obesity; Thiazoles; Urinary Bladder; Urinary Bladder, Overactive; Urination

2017
PPARdelta agonism inhibits skeletal muscle PDC activity, mitochondrial ATP production and force generation during prolonged contraction.
    The Journal of physiology, 2009, Jan-15, Volume: 587, Issue:1

    Topics: Adenosine Triphosphate; Animals; Carbohydrate Metabolism; Electric Stimulation; Glucose; Lactic Acid; Male; Mitochondria, Muscle; Muscle Contraction; Muscle, Skeletal; Oxidation-Reduction; PPAR delta; Pyruvate Dehydrogenase Complex; Rats; Rats, Wistar; Thiazoles

2009
Acotiamide hydrochloride (Z-338) enhances gastric motility and emptying by inhibiting acetylcholinesterase activity in rats.
    European journal of pharmacology, 2011, Volume: 666, Issue:1-3

    Topics: Acetylcholinesterase; Animals; Benzamides; Cholinesterase Inhibitors; Clonidine; Electric Stimulation; Gastric Emptying; Male; Muscle Contraction; Rats; Rats, Sprague-Dawley; Stomach; Thiazoles

2011
Inhibition of adrenergic human prostate smooth muscle contraction by the inhibitors of c-Jun N-terminal kinase, SP600125 and BI-78D3.
    British journal of pharmacology, 2012, Volume: 166, Issue:6

    Topics: Aged; Anthracenes; Dioxanes; Humans; In Vitro Techniques; JNK Mitogen-Activated Protein Kinases; Male; Muscle Contraction; Muscle, Smooth; Prostate; Protein Kinase Inhibitors; Receptors, Adrenergic, alpha-1; Thiazoles

2012
Muscle cyclo-oxygenase-2 pathway contributes to the exaggerated muscle mechanoreflex in rats with congestive heart failure.
    Experimental physiology, 2012, Volume: 97, Issue:8

    Topics: Animals; Blood Pressure; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Heart Failure; Heart Rate; Kidney; Male; Membrane Proteins; Muscle Contraction; Muscle, Skeletal; Myocardial Infarction; Piperazines; Pyrazoles; Rats; Rats, Sprague-Dawley; Reflex, Stretch; Sulfonamides; Sympathetic Nervous System; Thiazoles

2012
Effects of mirabegron, a novel β3-adrenoceptor agonist, on primary bladder afferent activity and bladder microcontractions in rats compared with the effects of oxybutynin.
    European urology, 2012, Volume: 62, Issue:6

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Animals; Female; Mandelic Acids; Muscarinic Antagonists; Muscle Contraction; Neurons, Afferent; Rats; Rats, Sprague-Dawley; Thiazoles; Urinary Bladder

2012
Febuxostat improves the local and remote organ changes induced by intestinal ischemia/reperfusion in rats.
    Digestive diseases and sciences, 2013, Volume: 58, Issue:3

    Topics: Alanine Transaminase; Allopurinol; Animals; Aspartate Aminotransferases; Dose-Response Relationship, Drug; Febuxostat; Gout Suppressants; Intestinal Mucosa; Lipid Peroxidation; Lung; Male; Malondialdehyde; Muscle Contraction; Muscle, Smooth; Peroxidase; Rats; Rats, Sprague-Dawley; Reperfusion Injury; Thiazoles; Tumor Necrosis Factor-alpha; Xanthine Dehydrogenase; Xanthine Oxidase

2013
Important role of PLC-γ1 in hypoxic increase in intracellular calcium in pulmonary arterial smooth muscle cells.
    American journal of physiology. Lung cellular and molecular physiology, 2013, Feb-01, Volume: 304, Issue:3

    Topics: Animals; Boron Compounds; Calcium; Electron Transport Complex III; Estrenes; Gene Expression; Hypoxia; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Lentivirus; Macrocyclic Compounds; Methacrylates; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Oxazoles; Phospholipase C gamma; Pulmonary Artery; Pyrrolidinones; Reactive Oxygen Species; RNA, Small Interfering; Thiazoles; Vasoconstriction

2013
The novel β3-adrenoceptor agonist mirabegron reduces carbachol-induced contractile activity in detrusor tissue from patients with bladder outflow obstruction with or without detrusor overactivity.
    European journal of pharmacology, 2013, Jan-15, Volume: 699, Issue:1-3

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Aged; Aged, 80 and over; Carbachol; Humans; In Vitro Techniques; Inhibitory Concentration 50; Isoproterenol; Male; Middle Aged; Muscle Contraction; Thiazoles; Urinary Bladder; Urinary Bladder Neck Obstruction; Urinary Bladder, Overactive

2013
Inhibition of muscle carbonic anhydrase slows the Ca(2+) transient in rat skeletal muscle fibers.
    American journal of physiology. Cell physiology, 2002, Volume: 283, Issue:4

    Topics: Acetazolamide; Action Potentials; Adenosine Triphosphatases; Animals; Benzothiazoles; Calcium; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Chelating Agents; Dose-Response Relationship, Drug; Enzyme Activation; Ethoxzolamide; Female; Fura-2; In Vitro Techniques; Ion Transport; Isometric Contraction; Muscle Contraction; Muscle Fibers, Skeletal; Muscle, Skeletal; Rats; Sarcoplasmic Reticulum; Thiadiazoles; Thiazoles; Time Factors

2002
New insights into the pharmacological properties of potent antiplatelet 2-amino-benzo[d]isothiazol-3-one derivatives.
    Pharmacological research, 2002, Volume: 46, Issue:5

    Topics: Administration, Oral; Animals; Bleeding Time; Guinea Pigs; Ileum; In Vitro Techniques; Injections, Intraperitoneal; Lethal Dose 50; Male; Mice; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Peptic Ulcer; Platelet Aggregation; Platelet Aggregation Inhibitors; Pulmonary Embolism; Thiazoles

2002
Effect of thiazolidinediones and metformin on LDL oxidation and aortic endothelium relaxation in diabetic GK rats.
    American journal of physiology. Endocrinology and metabolism, 2003, Volume: 284, Issue:6

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Arteriosclerosis; Cholesterol, LDL; Chromans; Diabetes Mellitus, Type 2; Endothelium, Vascular; Hypoglycemic Agents; Isometric Contraction; Lipid Peroxidation; Lipids; Male; Metformin; Muscle Contraction; Muscle Relaxation; Oxidation-Reduction; Pioglitazone; Rats; Rats, Wistar; Thiazoles; Thiazolidinediones; Troglitazone; Vasodilator Agents

2003
New thiazole derivatives as potent and selective 5-hydroxytriptamine 3 (5-HT3) receptor agonists for the treatment of constipation.
    Bioorganic & medicinal chemistry, 2003, Apr-03, Volume: 11, Issue:7

    Topics: Animals; Cathartics; Cloning, Molecular; Colon; Constipation; Defecation; Ferrets; Guinea Pigs; Humans; In Vitro Techniques; Magnetic Resonance Spectroscopy; Muscle Contraction; Muscle, Smooth; Radioligand Assay; Rats; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Recombinant Proteins; Reflex; Serotonin Receptor Agonists; Thiazoles

2003
Stretch-induced contractile differentiation of vascular smooth muscle: sensitivity to actin polymerization inhibitors.
    American journal of physiology. Cell physiology, 2003, Volume: 284, Issue:6

    Topics: Actins; Angiotensin II; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cell Differentiation; Culture Techniques; Cytochalasin D; Cytoskeleton; Enzyme Activation; Enzyme Inhibitors; Female; MAP Kinase Signaling System; Microfilament Proteins; Muscle Contraction; Muscle Proteins; Muscle, Smooth, Vascular; Nucleic Acid Synthesis Inhibitors; Portal Vein; Rats; Rats, Sprague-Dawley; rhoA GTP-Binding Protein; Stress, Mechanical; Thiazoles; Thiazolidines

2003
Role of Rho-kinase in maintaining airway smooth muscle contractile phenotype.
    European journal of pharmacology, 2004, Jan-01, Volume: 483, Issue:1

    Topics: Animals; Bronchodilator Agents; Cattle; Cell Division; Cells, Cultured; DNA; Enzyme Inhibitors; Intracellular Signaling Peptides and Proteins; Isometric Contraction; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Phenotype; Potassium Chloride; Protein Serine-Threonine Kinases; rho-Associated Kinases; Tetrazolium Salts; Thiazoles; Thymidine; Trachea

2004
Modulation of acto-myosin contractility in skeletal muscle myoblasts uncouples growth arrest from differentiation.
    Journal of cell science, 2004, Aug-01, Volume: 117, Issue:Pt 17

    Topics: Actomyosin; Animals; Antimetabolites; Azepines; Bridged Bicyclo Compounds, Heterocyclic; Bromodeoxyuridine; Cell Adhesion; Cell Cycle; Cell Cycle Proteins; Cell Differentiation; Cell Line; Cell Membrane; Cell Proliferation; Cell Separation; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Cytoskeleton; Diacetyl; DNA; Enzyme Inhibitors; Flow Cytometry; Green Fluorescent Proteins; Image Processing, Computer-Assisted; Kinetics; Mice; Microscopy, Fluorescence; Muscle Contraction; Muscle, Skeletal; Muscles; Myosin Heavy Chains; Myosin-Light-Chain Kinase; Myosins; Naphthalenes; Polymers; Resting Phase, Cell Cycle; rho GTP-Binding Proteins; rhoA GTP-Binding Protein; Signal Transduction; Thiazoles; Thiazolidines; Time Factors; Transfection; Tumor Suppressor Proteins

2004
Latrunculin B increases force fluctuation-induced relengthening of ACh-contracted, isotonically shortened canine tracheal smooth muscle.
    Journal of applied physiology (Bethesda, Md. : 1985), 2005, Volume: 98, Issue:2

    Topics: Acetylcholine; Actin Cytoskeleton; Animals; Bridged Bicyclo Compounds, Heterocyclic; Depsipeptides; Dogs; Dose-Response Relationship, Drug; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Stress, Mechanical; Thiazoles; Thiazolidines; Trachea

2005
IgA immune complex blunts the contraction of cultured mesangial cells through the inhibition of protein kinase C and intracellular calcium.
    The Chinese journal of physiology, 2004, Jun-30, Volume: 47, Issue:2

    Topics: Alkaloids; Angiotensin II; Animals; Benzophenanthridines; Calcium; Cell Size; Cells, Cultured; Enzyme Activators; Enzyme Inhibitors; Glomerular Mesangium; Immunoblotting; Immunoglobulin A; Ionomycin; Ionophores; Isoenzymes; Mice; Muscle Contraction; Phenanthridines; Protein Kinase C; Tetradecanoylphorbol Acetate; Tetrazolium Salts; Thiazoles

2004
Microwave-assisted solvent-free synthesis of 3-[(4-substituted piperazin-1-yl)alkyl] imidazo[2,1-b][1,3]benzothiazol-2(3H)-ones as serotonin3 (5-HT3) receptor antagonists.
    Die Pharmazie, 2005, Volume: 60, Issue:6

    Topics: Animals; Chemical Phenomena; Chemistry, Physical; Chromatography, Thin Layer; Guinea Pigs; Ileum; Imidazoles; In Vitro Techniques; Indicators and Reagents; Microwaves; Muscle Contraction; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Spectrophotometry, Ultraviolet; Spectroscopy, Fourier Transform Infrared; Thiazoles

2005
Rat airway smooth muscle cell during actin modulation: rheology and glassy dynamics.
    American journal of physiology. Cell physiology, 2005, Volume: 289, Issue:6

    Topics: Actins; Animals; Azepines; Biomechanical Phenomena; Bridged Bicyclo Compounds, Heterocyclic; Bucladesine; Cells, Cultured; Cross-Linking Reagents; Cytochalasin D; Genistein; Muscle Contraction; Myocytes, Smooth Muscle; Myosins; Naphthalenes; Peptides, Cyclic; Phalloidine; Rats; Rheology; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Thiazolidines; Trachea

2005
Synthesis of 1,2-benzisothiazolyloxypropanolamine derivatives and investigation of their activity at beta-adrenoceptors.
    Farmaco (Societa chimica italiana : 1989), 2005, Volume: 60, Issue:10

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; In Vitro Techniques; Molecular Structure; Muscle Contraction; Muscle, Smooth; Rats; Structure-Activity Relationship; Thiazoles

2005
Rho kinase regulates fragmentation and phagocytosis of apoptotic cells.
    Experimental cell research, 2006, Jan-01, Volume: 312, Issue:1

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Actins; Amides; Animals; Apoptosis; Bridged Bicyclo Compounds, Heterocyclic; Caspase Inhibitors; Caspases; Cell Membrane; Chlorocebus aethiops; COS Cells; DNA Fragmentation; Enzyme Activation; Enzyme Inhibitors; Heterocyclic Compounds, 4 or More Rings; Intracellular Signaling Peptides and Proteins; Marine Toxins; Muscle Contraction; Myosins; PC12 Cells; Phagocytosis; Protein Serine-Threonine Kinases; Protein Transport; Pyridines; Rats; rho-Associated Kinases; RNA, Small Interfering; Thiazoles; Thiazolidines

2006
PPARdelta activator GW-501516 has no acute effect on glucose transport in skeletal muscle.
    American journal of physiology. Endocrinology and metabolism, 2006, Volume: 290, Issue:4

    Topics: AMP-Activated Protein Kinases; Animals; Carrier Proteins; Glucose; Glucose Transporter Type 4; In Vitro Techniques; Ion Channels; Male; Mitochondrial Proteins; Multienzyme Complexes; Muscle Contraction; Muscle, Skeletal; p38 Mitogen-Activated Protein Kinases; Phosphorylation; PPAR delta; Protein Serine-Threonine Kinases; Rats; Rats, Wistar; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Thiazoles; Uncoupling Protein 3

2006
Benzisothiazoles and beta-adrenoceptors: synthesis and pharmacological investigation of novel propanolamine and oxypropanolamine derivatives in isolated rat tissues.
    Archives of pharmacal research, 2005, Volume: 28, Issue:12

    Topics: Adrenergic beta-1 Receptor Antagonists; Adrenergic beta-2 Receptor Antagonists; Adrenergic beta-3 Receptor Antagonists; Adrenergic beta-Antagonists; Animals; Dose-Response Relationship, Drug; Drug Synergism; Heart Atria; Ileum; Isoproterenol; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myocardial Contraction; Propanolamines; Propranolol; Rats; Thiazoles

2005
Effect of (R)-2-(2-aminothiazol-4-yl)-4'-{2-[(2-hydroxy-2-phenylethyl)amino]ethyl} acetanilide (YM178), a novel selective beta3-adrenoceptor agonist, on bladder function.
    The Journal of pharmacology and experimental therapeutics, 2007, Volume: 321, Issue:2

    Topics: Acetanilides; Adrenergic beta-3 Receptor Agonists; Adrenergic beta-Agonists; Animals; Carbachol; CHO Cells; Cricetinae; Cricetulus; Cyclic AMP; Humans; Isoproterenol; Muscle Contraction; Propanolamines; Thiazoles; Urinary Bladder

2007
Urinary retention associated with ziprasidone: a case report.
    The Journal of clinical psychiatry, 2008, Volume: 69, Issue:3

    Topics: Antipsychotic Agents; Diagnostic and Statistical Manual of Mental Disorders; Efferent Pathways; Female; Humans; Middle Aged; Muscle Contraction; Muscle, Smooth; Piperazines; Psychotic Disorders; Raphe Nuclei; Thiazoles; Urinary Bladder; Urinary Retention

2008
Effect of selective antagonists of group I metabotropic glutamate receptors on the micturition reflex in rats.
    BJU international, 2008, Volume: 102, Issue:7

    Topics: Animals; Female; Male; Muscle Contraction; Pyrans; Pyridines; Quinolines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Urinary Bladder; Urination; Urodynamics

2008
Species differences in the contractile response to two specific histamine H1-receptor agonists: 2-(2-pyridyl)-ethylamine and 2-(2-aminoethyl)-thiazole.
    The Journal of pharmacy and pharmacology, 1981, Volume: 33, Issue:2

    Topics: Animals; Cimetidine; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Pyridines; Receptors, Histamine; Receptors, Histamine H1; Species Specificity; Thiazoles; Vas Deferens

1981
Histamine H1- and muscarinic receptor antagonist activity of cimetidine and tiotidine in the guinea pig isolated ileum.
    Agents and actions, 1981, Volume: 11, Issue:6-7

    Topics: Animals; Carbachol; Cimetidine; Guanidines; Guinea Pigs; Histamine; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Kinetics; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Thiazoles

1981
[Racemic guanidinothiazoles with H2-antihistaminic activity. 13 H2-antihistaminics].
    Arzneimittel-Forschung, 1983, Volume: 33, Issue:3

    Topics: Animals; Chemical Phenomena; Chemistry; Guanidines; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Thiazoles

1983
Vasodilator mechanism of KB-944, a new calcium antagonist.
    Arzneimittel-Forschung, 1982, Volume: 32, Issue:9

    Topics: Adenosine; Animals; Benzothiazoles; Calcium Channel Blockers; Calcium Chloride; Coronary Vessels; Diltiazem; Dogs; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Potassium; Rabbits; Thiazoles; Vasodilator Agents; Verapamil

1982
Pharmacological analysis of the mechanism of action of phenthiazamine, a piscine anesthetic.
    Journal of pharmacobio-dynamics, 1980, Volume: 3, Issue:2

    Topics: Action Potentials; Anesthetics; Animals; Calcium; Dopamine; Fishes; Ganglia, Sympathetic; Guinea Pigs; Ileum; In Vitro Techniques; Muscle Contraction; Rana catesbeiana; Thiazoles; Ureter

1980
Biological properties of 3-benzyl-1,2-benzisothiazole compounds.
    Il Farmaco; edizione scientifica, 1982, Volume: 37, Issue:10

    Topics: Acetylcholine; Animals; Guinea Pigs; Histamine; In Vitro Techniques; Muscle Contraction; Muscle Relaxants, Central; Parasympatholytics; Thiazoles

1982
Effects of semotiadil fumarate (SD-3211) and its enantiomer, SD-3212, on the changes in cytosolic Ca2+ and tension caused by KCl and norepinephrine in isolated rat aortas.
    Journal of cardiovascular pharmacology, 1995, Volume: 25, Issue:2

    Topics: Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Bepridil; Calcium; Calcium Channel Blockers; Cytosol; Diltiazem; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Potassium Chloride; Rats; Rats, Wistar; Stereoisomerism; Thiazoles

1995
Characterization and function of histamine receptors in corpus cavernosum.
    The Journal of urology, 1995, Volume: 153, Issue:2

    Topics: Acetylcholine; Animals; Cimetidine; Dimaprit; Dose-Response Relationship, Drug; Electric Stimulation; Histamine; Histamine Agonists; Histamine Antagonists; In Vitro Techniques; Male; Methylhistamines; Muscle Contraction; Papaverine; Penis; Piperidines; Pyrilamine; Rabbits; Receptors, Histamine; Thiazoles

1995
Increased peak oxygen consumption of trained muscle requires increased electron flux capacity.
    Journal of applied physiology (Bethesda, Md. : 1985), 1994, Volume: 77, Issue:4

    Topics: Animals; Blood Flow Velocity; Electron Transport; Hindlimb; Methacrylates; Mitochondria, Muscle; Muscle Contraction; Muscle, Skeletal; Myofibrils; NADH Dehydrogenase; Oxygen Consumption; Perfusion; Physical Conditioning, Animal; Rats; Rats, Sprague-Dawley; Thiazoles

1994
Pharmacological profile of the novel, potent and selective peptide leukotriene antagonist (E)-2,2-diethyl-3'-[2-[2-(4-isopropyl)thiazolyl]ethenyl]succinanilic acid.
    Arzneimittel-Forschung, 1994, Volume: 44, Issue:6

    Topics: Acetylcholine; Animals; Bronchodilator Agents; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Antagonists; Ileum; In Vitro Techniques; Leukotriene Antagonists; Leukotriene C4; Leukotriene D4; Male; Muscle Contraction; Muscle, Smooth; Penicillin G; Pyrilamine; Thiazoles; Trachea

1994
Influence of the vinyl group on the calcium antagonistic activity of analogues of Fostedil.
    Pharmaceutica acta Helvetiae, 1994, Volume: 68, Issue:3

    Topics: Animals; Aorta, Thoracic; Benzothiazoles; Calcium Channel Blockers; In Vitro Techniques; Muscle Contraction; Rabbits; Thiazoles; Vinyl Compounds

1994
Effect of diacylglycerol kinase inhibitor, R59022 on cytosolic free calcium level and force development in guinea pig taenia coli.
    Research communications in chemical pathology and pharmacology, 1993, Volume: 81, Issue:3

    Topics: Animals; Calcium; Colon; Guinea Pigs; Muscle Contraction; Platelet Activating Factor; Pyrimidinones; Thiazoles

1993
The effect of diabetes on sexual behavior and reproductive tract function in male rats.
    The Journal of urology, 1993, Volume: 149, Issue:1

    Topics: Animals; Body Weight; Diabetes Mellitus, Experimental; Epididymis; Male; Muscle Contraction; Muscle, Smooth; Organ Size; Piperidines; Rats; Sexual Behavior, Animal; Sperm Count; Sperm Motility; Streptozocin; Testis; Testosterone; Thiazoles; Urinary Bladder

1993
The source and action of histamine in the isolated guinea-pig gallbladder.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1995, Volume: 44, Issue:10

    Topics: Animals; Dimaprit; Electric Stimulation; Female; Gallbladder; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Ranitidine; Receptors, Histamine H3; Thiazoles

1995
Troglitazone reduces contraction by inhibition of vascular smooth muscle cell Ca2+ currents and not endothelial nitric oxide production.
    Diabetes, 1997, Volume: 46, Issue:4

    Topics: Analysis of Variance; Animals; Arteries; Calcium Channels; Chromans; Dose-Response Relationship, Drug; Hypoglycemic Agents; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Patch-Clamp Techniques; Rats; Rats, Wistar; Thiazoles; Thiazolidinediones; Troglitazone

1997
Structure optimization of a leukotriene D4 antagonist by combinatorial chemistry in solution.
    Bioorganic & medicinal chemistry, 1997, Volume: 5, Issue:3

    Topics: Animals; Anti-Asthmatic Agents; Chemistry, Pharmaceutical; Guinea Pigs; Leukotriene D4; Muscle Contraction; Muscle, Smooth; Solutions; Thiazoles

1997
Arachidonic acid and its metabolites are involved in the expression of morphine dependence in guinea-pig isolated ileum.
    European journal of pharmacology, 1997, Jul-09, Volume: 330, Issue:2-3

    Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Cyclooxygenase Inhibitors; Guinea Pigs; Ileum; In Vitro Techniques; Lipoxygenase Inhibitors; Male; Masoprocol; Meloxicam; Morphine; Muscle Contraction; Naloxone; Narcotic Antagonists; Phospholipases A; Phospholipases A2; Quinacrine; Substance-Related Disorders; Thiazines; Thiazoles; Tolmetin

1997
Disparate effects of antidiabetic drugs on arterial contraction.
    Metabolism: clinical and experimental, 1997, Volume: 46, Issue:10

    Topics: Animals; Arteries; Blood Pressure; Glyburide; Humans; Hypoglycemic Agents; In Vitro Techniques; Insulin; Male; Metformin; Muscle Contraction; Muscle, Smooth, Vascular; Pioglitazone; Potassium Chloride; Rats; Rats, Wistar; Tail; Thiazoles; Thiazolidinediones

1997
Effects of newly synthesized amino acids containing thiazole residues on electrically evoked smooth muscle contractions.
    Methods and findings in experimental and clinical pharmacology, 1998, Volume: 20, Issue:3

    Topics: Amino Acids; Animals; Electric Stimulation; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Mice; Molecular Structure; Muscle Contraction; Muscle, Smooth; Rabbits; Rats; Rats, Wistar; Spectrophotometry, Infrared; Thiazoles

1998
Antinociceptive effect of meloxicam, in neurogenic and inflammatory nociceptive models in mice.
    Inflammation research : official journal of the European Histamine Research Society ... [et al.], 1998, Volume: 47, Issue:7

    Topics: Abdominal Muscles; Acetic Acid; Analgesics; Analgesics, Opioid; Animals; Capsaicin; Cyclooxygenase Inhibitors; Diclofenac; Formaldehyde; Inflammation; Male; Meloxicam; Mice; Morphine; Muscle Contraction; Pain; Pain Measurement; Reaction Time; Thiazines; Thiazoles

1998
Histamine receptor-independent muscle relaxation elicited by a series of histamine H2-receptor agonists on the isolated guinea pig duodenum: a study into the mechanism of action.
    General pharmacology, 1998, Volume: 31, Issue:4

    Topics: Animals; Dimaprit; Duodenum; Electric Stimulation; Guinea Pigs; Histamine Agonists; Impromidine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Structure-Activity Relationship; Thiazoles

1998
In vitro pharmacologic profile of YM158, a new dual antagonist for LTD4 and TXA2 receptors.
    The Journal of pharmacology and experimental therapeutics, 1998, Volume: 287, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Carbachol; Dinoprost; Guinea Pigs; Humans; In Vitro Techniques; Leukotriene Antagonists; Leukotriene D4; Male; Membrane Proteins; Muscle Contraction; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandin D2; Receptors, Leukotriene; Receptors, Thromboxane; Tetrazoles; Thiazoles; Trachea

1998
The effects of 8-hydroxy-2-(di-n-propylamino)tetralin on the cholinergic contraction in guinea pig and human airways in vitro.
    American journal of respiratory and critical care medicine, 1998, Volume: 158, Issue:5 Pt 1

    Topics: 8-Hydroxy-2-(di-n-propylamino)tetralin; Acetylcholine; Animals; Bronchi; Bronchoconstriction; Capsaicin; Cholinergic Fibers; Culture Techniques; Cyclohexane Monoterpenes; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Humans; Indoles; Ketanserin; Methysergide; Muscle Contraction; Muscle, Smooth; Neuropeptides; Pindolol; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles; Trachea; Tropisetron

1998
Effects of histamine H2 receptor agonists and antagonists on the isolated guinea pig gallbladder.
    Fundamental & clinical pharmacology, 1999, Volume: 13, Issue:1

    Topics: Animals; Benzothiazoles; Dopamine Agents; Famotidine; Gallbladder; Guanidines; Guinea Pigs; Histamine; Histamine Agonists; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Phenoxypropanolamines; Piperidines; Pyridines; Receptors, Histamine H2; Sincalide; Thiazoles; Triazoles

1999
Actin polymerization stimulated by contractile activation regulates force development in canine tracheal smooth muscle.
    The Journal of physiology, 1999, Sep-15, Volume: 519 Pt 3

    Topics: Acetylcholine; Actins; Animals; Bridged Bicyclo Compounds, Heterocyclic; Cytochalasin D; Dogs; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Phosphorylation; Polymers; Thiazoles; Thiazolidines; Trachea

1999
Histamine H1 receptor ligands. Part I. Novel thiazol-4-ylethanamine derivatives: synthesis and in vitro pharmacology.
    Farmaco (Societa chimica italiana : 1989), 1999, Aug-30, Volume: 54, Issue:8

    Topics: Animals; Dose-Response Relationship, Drug; Guinea Pigs; Histamine Agonists; Ileum; In Vitro Techniques; Ligands; Male; Muscle Contraction; Muscle, Smooth; Structure-Activity Relationship; Thiazoles

1999
Tracheal relaxing effects and beta2 adrenoceptor selectivity of S1319, a novel sponge-derived bronchodilator agent, in isolated guinea-pig tissues.
    British journal of pharmacology, 1999, Volume: 128, Issue:3

    Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Animals; Atrial Function; Benzothiazoles; Ethanolamines; Guinea Pigs; Heart Atria; In Vitro Techniques; Male; Muscle Contraction; Receptors, Adrenergic, beta-2; Thiazoles; Trachea

1999
Non-imidazole histamine H3 ligands, Part 2: New 2-substituted benzothiazoles as histamine H3 antagonists.
    Archiv der Pharmazie, 1999, Volume: 332, Issue:11

    Topics: Animals; Guinea Pigs; Histamine Antagonists; Molecular Structure; Muscle Contraction; Muscle, Smooth; Structure-Activity Relationship; Thiazoles

1999
Z-338 facilitates acetylcholine release from enteric neurons due to blockade of muscarinic autoreceptors in guinea pig stomach.
    The Journal of pharmacology and experimental therapeutics, 2000, Volume: 294, Issue:1

    Topics: Acetylcholine; Animals; Autoreceptors; Benzamides; Gastrointestinal Agents; Guinea Pigs; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Receptor, Muscarinic M1; Receptor, Muscarinic M2; Receptors, Muscarinic; Stomach; Thiazoles; Xenopus

2000
Z-338, a newly synthetized carboxyamide derivative, stimulates gastric motility through enhancing the excitatory neurotransmission.
    Journal of smooth muscle research = Nihon Heikatsukin Gakkai kikanshi, 2000, Volume: 36, Issue:2

    Topics: Animals; Benzamides; Gastrointestinal Agents; Gastrointestinal Motility; Guinea Pigs; Male; Muscle Contraction; Muscle, Smooth; Stomach; Thiazoles

2000
Mechanisms of vasoinhibitory effect of cardioprotective agent, CP-060S, in rat aorta.
    European journal of pharmacology, 2000, Jul-21, Volume: 400, Issue:2-3

    Topics: Angiotensin II; Animals; Anti-Arrhythmia Agents; Aorta, Thoracic; Arginine Vasopressin; Calcium; Calcium Channel Blockers; Cytosol; Dinoprost; Drug Interactions; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Phenylephrine; Rats; Rats, Wistar; Thiazoles; Thiazolidines; Vasoconstrictor Agents; Vasodilator Agents

2000
2-Amino-Benzo[d]isothiazol-3-one derivatives: synthesis and assessment of their antiplatelet/spasmolytic effects.
    Bioorganic & medicinal chemistry, 2000, Volume: 8, Issue:9

    Topics: Adenosine Diphosphate; Animals; Aorta; Arachidonic Acid; Benzaldehydes; Guinea Pigs; Ileum; Inhibitory Concentration 50; Male; Models, Animal; Muscle Contraction; Parasympatholytics; Platelet Aggregation; Platelet Aggregation Inhibitors; Thiazoles

2000
Potential antitumor agents. Part 29(1): synthesis and potential coanthracyclinic activity of imidazo[2,1-b]thiazole guanylhydrazones.
    Bioorganic & medicinal chemistry, 2000, Volume: 8, Issue:9

    Topics: Animals; Antineoplastic Agents; CDC2 Protein Kinase; Cell Division; Cell Survival; Guanidine; Guinea Pigs; Humans; Hydrazones; Imidazoles; Muscle Contraction; Papillary Muscles; Starfish; Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured

2000
Pharmacological profile of YM-31636, a novel 5-HT3 receptor agonist, in vitro.
    European journal of pharmacology, 2000, Dec-08, Volume: 409, Issue:2

    Topics: Acetylcholine; Action Potentials; Animals; Anthraquinones; Atrial Function; Biguanides; Binding, Competitive; Colon; Dinoprostone; Dose-Response Relationship, Drug; Guinea Pigs; Heart Atria; Humans; In Vitro Techniques; Muscle Contraction; Myocardial Contraction; Pyrroles; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin; Serotonin Receptor Agonists; Thiazoles

2000
Pseudoproline-containing analogues of morphiceptin and endomorphin-2: evidence for a cis Tyr-Pro amide bond in the bioactive conformation.
    Journal of medicinal chemistry, 2001, Nov-08, Volume: 44, Issue:23

    Topics: Animals; Brain; Endorphins; Guinea Pigs; Ileum; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Mice; Muscle Contraction; Muscle, Smooth; Oligopeptides; Oxazoles; Proline; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Thiazoles; Vas Deferens

2001
Inhibition of muscle carbonic anhydrase increases rise and relaxation times of twitches in rat skeletal muscle fibres.
    Pflugers Archiv : European journal of physiology, 2002, Volume: 443, Issue:5-6

    Topics: Acetazolamide; Animals; Benzolamide; Benzothiazoles; Bicarbonates; Buffers; Carbon Dioxide; Carbonic Anhydrase Inhibitors; Carbonic Anhydrases; Ethoxzolamide; Female; HEPES; Hydrogen-Ion Concentration; Muscle Contraction; Muscle Fibers, Skeletal; Muscle Relaxation; Muscle, Skeletal; Rats; Rats, Inbred WF; Sarcoplasmic Reticulum; Thiadiazoles; Thiazoles

2002
Oxidative capacity interacts with oxygen delivery to determine maximal O(2) uptake in rat skeletal muscles in situ.
    The Journal of physiology, 2002, Jun-15, Volume: 541, Issue:Pt 3

    Topics: Animals; Enzyme Inhibitors; Hindlimb; Kinetics; Methacrylates; Mitochondria, Muscle; Muscle Contraction; Muscle, Skeletal; NADH Dehydrogenase; Oxidation-Reduction; Oxygen Consumption; Perfusion; Rats; Rats, Sprague-Dawley; Regional Blood Flow; Thiazoles

2002
The effect of the selective 5-HT(3) receptor agonist on ferret gut motility.
    Life sciences, 2002, Aug-02, Volume: 71, Issue:11

    Topics: Animals; Benzimidazoles; Colon; Defecation; Ferrets; Gastrointestinal Motility; Male; Muscle Contraction; Pyrroles; Serotonin Antagonists; Serotonin Receptor Agonists; Thiazoles

2002
Effect of tazolol on beta-adrenoceptors in isolated preparations of the guinea-pig and rat.
    The Journal of pharmacy and pharmacology, 1977, Volume: 29, Issue:10

    Topics: Adrenergic beta-Agonists; Animals; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Muscle Contraction; Myocardial Contraction; Propanolamines; Rats; Receptors, Adrenergic; Receptors, Adrenergic, beta; Thiazoles; Trachea

1977
Analysis of the beta-receptor mediated effect on slow-contracting skeletal muscle in vitro.
    The Journal of pharmacy and pharmacology, 1977, Volume: 29, Issue:9

    Topics: Adrenergic beta-Antagonists; Animals; Dopamine; Electric Stimulation; Epinephrine; Guinea Pigs; In Vitro Techniques; Isoproterenol; Male; Muscle Contraction; Norepinephrine; Propanolamines; Receptors, Adrenergic; Receptors, Adrenergic, beta; Reserpine; Terbutaline; Thiazoles; Tyramine

1977
The mode of action of tiaramide hydrochloride: a new antiasthmatic drug.
    Pharmacological research communications, 1979, Volume: 11, Issue:8

    Topics: Airway Resistance; Anaphylaxis; Animals; Arachidonic Acids; Benzothiazoles; Bronchodilator Agents; Guinea Pigs; Histamine Release; Humans; In Vitro Techniques; Lung; Male; Muscle Contraction; Muscle, Smooth; Piperazines; Rabbits; Thiazoles; Thromboxane A2; Trachea

1979
[Pharmacological properties of dl-2-(3'-t-butylamino-2'-hydroxypropylthio)-4-(5'-carbamoyl-2'-thienyl) thiazole hydrochloride (S-596), a new beta-adrenergic blocking agent (author's transl)].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1979, Volume: 75, Issue:7

    Topics: Adrenergic beta-Antagonists; Anesthetics, Local; Animals; Anti-Arrhythmia Agents; Arrhythmias, Cardiac; Blood Pressure; Chloroform; Dogs; Epinephrine; Female; Guinea Pigs; Heart Rate; In Vitro Techniques; Male; Mice; Muscle Contraction; Myocardial Contraction; Ouabain; Practolol; Propanolamines; Propranolol; Rats; Thiazoles

1979
Potentiating mechanism of bradykinin action on smooth muscle by sulfhydryl compounds.
    European journal of pharmacology, 1979, Mar-01, Volume: 54, Issue:3

    Topics: 3-Mercaptopropionic Acid; Angiotensin I; Angiotensin II; Animals; Bradykinin; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Sulfhydryl Compounds; Thiazoles; Thiazolidines; Time Factors

1979
Pharmacological properties of thiazolinobutazone (LAS 11 871). III. General pharmacology, ulcerogenic effects and acute toxicity.
    Arzneimittel-Forschung, 1976, Volume: 26, Issue:7

    Topics: Animals; Autonomic Nervous System; Brain; Cats; Diuresis; Female; Hemodynamics; Lethal Dose 50; Male; Mice; Motor Activity; Motor Skills; Muscle Contraction; Phenylbutazone; Rabbits; Rats; Respiration; Stomach Ulcer; Thiazoles

1976
Calcium antagonistic and binding properties of semotiadil (SD-3211), a benzothiazine derivative assessed in cerebral and coronary arteries.
    Journal of cardiovascular pharmacology, 1992, Volume: 20, Issue:3

    Topics: Animals; Calcium; Calcium Channel Blockers; Calcium Channels; Cerebral Arteries; Coronary Vessels; Cytosol; Dogs; Female; In Vitro Techniques; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth, Vascular; Radioligand Assay; Stereoisomerism; Swine; Thiazoles

1992
Significant role of peptide leukotrienes (p-LTs) in the antigen-induced contractions of human and guinea pig lung parenchymas and bronchi or tracheas in vitro.
    Japanese journal of pharmacology, 1992, Volume: 60, Issue:3

    Topics: Animals; Bronchi; Cattle; Cyclooxygenase Inhibitors; Female; gamma-Globulins; Guinea Pigs; Humans; In Vitro Techniques; Indicators and Reagents; Leukotriene Antagonists; Leukotrienes; Lung; Male; Muscle Contraction; Muscle, Smooth; Penicillin G; Thiazoles; Trachea

1992
Leukotriene receptors in the skin of rats differ from those of mouse skin or rat stomach strip.
    European journal of pharmacology, 1992, Oct-20, Volume: 221, Issue:2-3

    Topics: Acetophenones; Animals; Capillary Permeability; Female; Mice; Mice, Inbred BALB C; Muscle Contraction; Passive Cutaneous Anaphylaxis; Rats; Rats, Wistar; Receptors, Immunologic; Receptors, Leukotriene; Skin; Species Specificity; SRS-A; Stomach; Tetrazoles; Thiazoles

1992
Synthesis of 3-[(2,3-dihydro-1,1,3-trioxo-1,2-benzisothiazol-2-yl)alkyl] 1,4-dihydropyridine-3,5-dicarboxylate derivatives as calcium channel modulators.
    Journal of medicinal chemistry, 1992, Jun-26, Volume: 35, Issue:13

    Topics: 3-Pyridinecarboxylic acid, 1,4-dihydro-2,6-dimethyl-5-nitro-4-(2-(trifluoromethyl)phenyl)-, Methyl ester; Animals; Calcium; Calcium Channels; Cations; Dihydropyridines; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Potassium; Rabbits; Rats; Rats, Inbred Strains; Thiazoles

1992
MCI-826 is a potent and selective antagonist of peptide leukotrienes (p-LTs) and has characteristics distinctive from those of FPL 55712.
    Japanese journal of pharmacology, 1992, Volume: 60, Issue:1

    Topics: Acetylcholine; Animals; Bronchi; Chromones; Guinea Pigs; Humans; Leukotriene Antagonists; Leukotrienes; Muscle Contraction; Muscle, Smooth; Prostaglandin D2; Respiratory Physiological Phenomena; Respiratory System; SRS-A; Thiazoles; Trachea

1992
Histamine H2-receptor agonists. Synthesis, in vitro pharmacology, and qualitative structure-activity relationships of substituted 4- and 5-(2-aminoethyl)thiazoles.
    Journal of medicinal chemistry, 1992, Aug-21, Volume: 35, Issue:17

    Topics: Animals; Atrial Function; Chemical Phenomena; Chemistry, Physical; Electrochemistry; Guinea Pigs; Heart Atria; Histamine; Ileum; Molecular Structure; Muscle Contraction; Receptors, Histamine H2; Structure-Activity Relationship; Thiazoles

1992
Pharmacologic actions of Ro 24-5913, a novel antagonist of leukotriene D4.
    The Journal of pharmacology and experimental therapeutics, 1991, Volume: 259, Issue:2

    Topics: Animals; Bronchi; Bronchoconstriction; Guinea Pigs; Humans; Leukotrienes; Male; Muscle Contraction; Muscle, Smooth; Receptors, Immunologic; Receptors, Leukotriene; SRS-A; Thiazoles; Trachea

1991
4- or 5- (omega-aminoalkyl) thiazoles and derivatives; new selective H2-receptor agonists.
    Agents and actions. Supplements, 1991, Volume: 33

    Topics: Amines; Animals; Atrial Function; Guanidines; Guinea Pigs; Heart Atria; Heart Rate; Histamine; Ileum; Imidazoles; Impromidine; Molecular Structure; Muscle Contraction; Receptors, Histamine H2; Thiazoles

1991
Involvement of calcium ions in the modulation of electrically-induced rat vas deferens contractions by histaminergic drugs.
    General pharmacology, 1991, Volume: 22, Issue:4

    Topics: Animals; Calcium; Cimetidine; Dimaprit; Diphenhydramine; Electric Stimulation; Histamine; In Vitro Techniques; Male; Muscle Contraction; Rats; Receptors, Histamine H1; Receptors, Histamine H2; Thiazoles; Thiourea; Vas Deferens; Verapamil

1991
Studies on heterocyclic compounds: 1,3-thiazolidin-4-one derivatives. V. Pharmacological activity of substituted 2-phenyl-3-(N,N-dimethylaminoprophyl)-1,3-thiazolidin-4-one .
    Bollettino della Societa italiana di biologia sperimentale, 1991, Volume: 67, Issue:12

    Topics: Animals; Female; Guinea Pigs; Histamine; Histamine Antagonists; Ileum; Male; Muscle Contraction; Muscle, Smooth; Pyrilamine; Schiff Bases; Structure-Activity Relationship; Thiazoles; Thiazolidines

1991
Role of phosphatidic acid in carbachol-induced contraction in guinea pig Taenia coli.
    Research communications in chemical pathology and pharmacology, 1991, Volume: 71, Issue:1

    Topics: Animals; Biological Transport, Active; Calcium; Carbachol; Colon; Diacylglycerol Kinase; Diglycerides; Guinea Pigs; In Vitro Techniques; Muscle Contraction; Phosphatidic Acids; Phosphotransferases; Pyrimidinones; Thiazoles

1991
Involvement of protein kinase C in Ca(2+)-independent contraction of rat uterine smooth muscle.
    Biochemical and biophysical research communications, 1991, Aug-30, Volume: 179, Issue:1

    Topics: Animals; Blotting, Western; Brain; Calcium; Electrophoresis, Polyacrylamide Gel; Female; In Vitro Techniques; Isoenzymes; Muscle Contraction; Muscle, Smooth; Oxytocin; Protein Kinase C; Pyrimidinones; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Thiazoles; Uterus

1991
Selective implication of thromboxane A2 and PAF-acether in two guinea pig anaphylactic models.
    Agents and actions. Supplements, 1990, Volume: 31

    Topics: Anaphylaxis; Animals; Antigens; Glyceryl Ethers; Guinea Pigs; Immunoglobulin E; Immunoglobulin G; In Vitro Techniques; Indomethacin; Muscle Contraction; Platelet Activating Factor; Thiazoles; Thromboxane A2; Trachea

1990
Tissue selectivity of the novel calcium antagonist sesamodil fumarate in isolated smooth muscles and cardiac muscles.
    Arzneimittel-Forschung, 1990, Volume: 40, Issue:3

    Topics: Animals; Calcimycin; Calcium Channel Blockers; Diltiazem; Guinea Pigs; Heart; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Nicardipine; Nifedipine; Rabbits; Swine; Thiazoles; Verapamil

1990
Ebselen inhibits contractile responses of guinea-pig parenchymal lung strips.
    European journal of pharmacology, 1990, Apr-10, Volume: 179, Issue:1-2

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Azoles; Catechols; Cyclooxygenase Inhibitors; Guinea Pigs; Histamine; Indomethacin; Isoindoles; Isoquinolines; Lung; Male; Masoprocol; Muscle Contraction; Muscle, Smooth; Organoselenium Compounds; Piperazines; Potassium Chloride; Selenium; Thiazoles

1990
Changes in capillary perfusion induced by different patterns of activity in rat skeletal muscle.
    Microvascular research, 1990, Volume: 40, Issue:1

    Topics: Animals; Benzothiazoles; Capillaries; Fluorescent Dyes; Male; Muscle Contraction; Muscles; Myofibrils; Rats; Rats, Inbred Strains; Regional Blood Flow; Thiazoles

1990
Tentacle contraction in Heliophrya erhardi (Suctoria): the role of inositol phospholipid metabolites and cyclic nucleotides in stimulus-response coupling.
    Experimental cell research, 1988, Volume: 177, Issue:2

    Topics: 1-Methyl-3-isobutylxanthine; Animals; Bucladesine; Chlorides; Ciliophora; Cyclic AMP; Cyclic GMP; Dibutyryl Cyclic GMP; Inositol Phosphates; Lithium; Lithium Chloride; Muscle Contraction; Pyrimidinones; Sugar Phosphates; Tetradecanoylphorbol Acetate; Thiazoles

1988
The diacylglycerol kinase inhibitor, R 59022, suppresses contractility of intestinal smooth muscle.
    European journal of pharmacology, 1989, Jan-02, Volume: 159, Issue:1

    Topics: Acetylcholine; Animals; Calcium; Diacylglycerol Kinase; Female; Guinea Pigs; Histamine; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Phosphatidylinositols; Phosphotransferases; Platelet Activating Factor; Pyrimidinones; Substance P; Thiazoles

1989
R 56865 differentiates between contractile agents with respect to the nifedipine-sensitive component in the isolated rat aorta.
    Pharmacology, 1989, Volume: 39, Issue:1

    Topics: Angiotensin II; Animals; Aorta, Thoracic; Arginine Vasopressin; Benzothiazoles; Calcium; Calcium Channels; Cytosol; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Piperidines; Rats; Rats, Inbred Strains; Serotonin; Thiazoles

1989
Pharmacological profile of 48740 R.P., a PAF-acether antagonist.
    European journal of pharmacology, 1988, Jun-10, Volume: 150, Issue:3

    Topics: Animals; Blood Cell Count; Blood Platelets; Bronchodilator Agents; Guinea Pigs; Humans; In Vitro Techniques; Macrophages; Male; Muscle Contraction; Muscle, Smooth; N-Formylmethionine Leucyl-Phenylalanine; Perfusion; Platelet Activating Factor; Platelet Aggregation; Pulmonary Alveoli; Pyridines; Rabbits; Radioimmunoassay; Superoxides; Thiazoles; Thromboxane B2

1988
[C-2 basically substituted thiazoles with H2-antagonistic action. 21. H2-antihistaminics].
    Arzneimittel-Forschung, 1985, Volume: 35, Issue:3

    Topics: Animals; Chemical Phenomena; Chemistry; Electric Stimulation; Gastric Acid; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Muscle Contraction; Muscle, Smooth; Rats; Rats, Inbred Strains; Thiazoles

1985
Cholinergic effects of histamine-H2 receptor antagonists partly through inhibition of acetylcholinesterase.
    Gastroenterologia Japonica, 1986, Volume: 21, Issue:3

    Topics: Animals; Butyrylcholinesterase; Cholinesterase Inhibitors; Cimetidine; Famotidine; Guinea Pigs; Histamine H2 Antagonists; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Ranitidine; Thiazoles

1986
Direct effects of H2-receptor antagonists on airway smooth muscle and on responses mediated by H1- and H2-receptors.
    Anesthesiology, 1987, Volume: 66, Issue:2

    Topics: Animals; Cimetidine; Famotidine; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Ranitidine; Thiazoles; Trachea

1987
Pharmacology of the novel H2 antagonist famotidine: in vitro studies.
    Agents and actions, 1986, Volume: 19, Issue:3-4

    Topics: Animals; Famotidine; Female; Gallbladder; Gastric Acid; Gastrointestinal Motility; Histamine H2 Antagonists; In Vitro Techniques; Male; Muscle Contraction; Myocardial Contraction; Rats; Thiazoles; Uterus

1986
Modulation of calmodulin function and of Ca2+-induced smooth muscle contraction by the calmodulin antagonist, HT-74.
    Molecular pharmacology, 1986, Volume: 29, Issue:3

    Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Anilino Naphthalenesulfonates; Animals; Benzothiazoles; Calcium; Calmodulin; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Protein Kinases; Rabbits; Sulfonamides; Thiazoles

1986
PAF antagonists: different effects on platelets, neutrophils, guinea pig ileum and PAF-induced vasodilation in isolated rat lung.
    Prostaglandins, 1986, Volume: 32, Issue:3

    Topics: Alprazolam; Angiotensin II; Animals; Blood Platelets; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Muscle Contraction; Neutrophils; Phospholipid Ethers; Platelet Activating Factor; Platelet Membrane Glycoproteins; Pulmonary Artery; Pulmonary Circulation; Rabbits; Rats; Receptors, Cell Surface; Receptors, G-Protein-Coupled; Serotonin; SRS-A; Thiazoles; Vasodilation

1986
Prostaglandins involved in contractions by angiotensin II and bradykinin of isolated dog sphincter pupillae.
    British journal of pharmacology, 1988, Volume: 95, Issue:2

    Topics: Angiotensin II; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonic Acid; Arachidonic Acids; Bradykinin; Dinoprost; Dogs; Female; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Prostaglandins; Pupil; Thiazoles; Thromboxane A2

1988
Different effects of R 56865 and calcium entry blockers on K+- and noradrenaline-induced contractions and 45Ca uptake in rat aorta.
    European journal of pharmacology, 1988, Dec-13, Volume: 158, Issue:3

    Topics: Animals; Aorta; Benzothiazoles; Calcium; Calcium Channel Blockers; Diltiazem; Dose-Response Relationship, Drug; Flunarizine; Male; Muscle Contraction; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Piperidines; Potassium; Rats; Rats, Inbred Strains; Thiazoles; Verapamil

1988
Novel calcium antagonists. Synthesis and structure-activity relationship studies of benzothiazoline derivatives.
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:5

    Topics: Animals; Blood Pressure; Calcium Channel Blockers; Chemical Phenomena; Chemistry; Guinea Pigs; Heart Conduction System; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Pulmonary Embolism; Rabbits; Rats; Rats, Inbred SHR; Structure-Activity Relationship; Thiazoles

1988
Acetylene compounds of potential pharmacological value. XL. N-(tert-aminoalkynyl)-substituted 3-isothiazolidinone-1,1-dioxides and tetrahydro-1,2-thiazin-3-one-1,1-dioxides.
    Acta pharmaceutica Suecica, 1987, Volume: 24, Issue:4

    Topics: Animals; Anticonvulsants; Benzopyrans; Carbachol; Chemical Phenomena; Chemistry; Chromans; Cyclic S-Oxides; Guinea Pigs; Ileum; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Structure-Activity Relationship; Thiazines; Thiazoles

1987
Selective -adrenergic myocardial stimulant.
    Experientia, 1972, Nov-15, Volume: 28, Issue:11

    Topics: Acetanilides; Adrenergic beta-Agonists; Amino Alcohols; Amphetamine; Animals; Blood Pressure; Dogs; Female; Heart; Heart Rate; Isoproterenol; Male; Muscle Contraction; Propylamines; Propylene Glycols; Stimulation, Chemical; Thiazoles

1972
Cross tolerance to histamine by the chronic administration of histamine analogues.
    Research communications in chemical pathology and pharmacology, 1972, Volume: 3, Issue:2

    Topics: Aerosols; Animals; Asthma; Blood Pressure; Body Weight; Cats; Desensitization, Immunologic; Dogs; Drug Tolerance; Ethylamines; Female; Gastric Juice; Gastric Mucosa; Guinea Pigs; Histamine; In Vitro Techniques; Intestines; Muscle Contraction; Muscle, Smooth; Pyrazoles; Pyridines; Reaction Time; Stimulation, Chemical; Thiazoles

1972
The mechanism of the paralysing action of tetramisole on Ascaris somatic muscle.
    British journal of pharmacology, 1970, Volume: 38, Issue:3

    Topics: Acetylcholine; Animals; Anthelmintics; Ascaris; Curare; Female; Male; Membrane Potentials; Muscle Contraction; Muscles; Piperazines; Potassium; Thiazoles

1970