thiazoles has been researched along with Malaria in 36 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 10 (27.78) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 7 (19.44) | 29.6817 |
2010's | 15 (41.67) | 24.3611 |
2020's | 4 (11.11) | 2.80 |
Authors | Studies |
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Allison, C; Arandjelovic, P; Boddey, JA; Doerflinger, M; Ebert, G; Erickson, S; Ioannidis, L; Lopaticki, S; Mackiewicz, L; O'Neill, MT; Pellegrini, M; Rajasekaran, P; Silke, J; Steel, RWJ; Yang, ASP | 1 |
Makoni, M | 1 |
Agbevo, A; Fongnikin, A; Houeto, N; N'Guessan, R; Ngufor, C; Odjo, A; Syme, T | 1 |
Celis, C; Charris, J; De Sanctis, JB; Fernandez, E; Martínez, G; Mayora, S; Mijares, M; Ramírez, H; Rodrigues, J | 1 |
Bordat, Y; Bressolle-Gomeni, F; Cerdan, R; Fraisse, L; Margout, D; Maynadier, M; Taudon, N; Tran Van Ba, C; Vial, HJ; Wein, S; Wengelnik, K | 1 |
Kumawat, MK | 1 |
Fongnikin, A; N'Guessan, R; Ngufor, C; Rowland, M | 1 |
Chung, MC; Dos Santos, JL; Ferreira, CMR; Jornada, DH; Machado, MGM; Scarim, CB | 1 |
Agossa, FR; Akinro, B; Akogbeto, MC; Akuoko, OK; Fassinou, AJYH; Koukpo, ZC; Nwangwu, UC; Odjo, EM; Padonou, GG; Salako, A; Sezonlin, M | 1 |
Bangs, MJ; Hattingh, I; Kashala, JK; Malonga, FK; Mashat, EM; Mlambo, G; Ngwej, LM | 1 |
Fuseini, G; Garcia, GA; Phiri, WP; Smith, J; von Fricken, ME | 1 |
Agumba, S; Gimnig, JE; Guyah, B; Kosgei, J; Munga, S; Ochomo, E; Ogonda, L; Ombok, M; Omondi, S | 1 |
Abramo, C; Budu, A; Butera, AP; Carmona, AK; da Silva, GR; da Silva, MG; de Almeida, HG; de Brito, CFA; de Castro, WV; de Miranda Martins, NR; de Pilla Varotti, F; de Sousa Luz, LS; de Souza Reis, V; do Nascimento, SB; Dos Santos, FV; Gazarini, ML; Guimarães, DSM; Guimarães, L; Júnior, CSN; Kemmer, VM; Maluf, SEC; Marinho, JA; Ribeiro-Viana, RM; Silva, LR; Viana, GHR | 1 |
Abong'o, B; Agossa, FR; Alyko, E; Baber, I; Coleman, S; Dabire, R; Dengela, D; Diop, A; Faye, O; Fornadel, C; Gnanguenon, V; Lucas, B; Magesa, S; Manjurano, A; Masendu, H; Okia, M; Oxborough, RM; Rakotoson, JD; Samdi, LM; Seyoum, A; Sovi, A; Varela, K; Wat'senga, F; Yihdego, Y; Yohannes, G | 1 |
Andrews, KT; Caridha, D; Chen, Y; Dow, GS; Gerena, L; Gettayacamin, M; Johnson, J; Kozikowski, AP; Li, Q; Melendez, V; Obaldia, N; Tran, TN | 1 |
Baldwin, J; Buckner, FS; Charman, S; Charman, WN; Creason, S; El Mazouni, F; Gujjar, R; Marwaha, A; Phillips, MA; Rathod, PK; Shackleford, DM; White, J; White, KL | 1 |
Bontemps, N; Bressolle, FM; Kocken, CH; Margout, D; Vial, HJ | 1 |
Alarcon, K; Boisbrun, M; Calas, M; Caldarelli, SA; Hamzé, A; Maynadier, M; Ouattara, M; Pellet, A; Peyrottes, S; Salom-Roig, X; Vial, H; Wein, S | 1 |
ASHLEY, JN; GROVE, JF | 1 |
Brun, R; Ge, JF; Ihara, M; Kaiser, M; Liu, BQ; Shi, XL; Wittlin, S | 1 |
Burrows, JN; Charman, SA; Chibale, K; Douelle, F; Feng, TS; González Cabrera, D; Nchinda, AT; Ryan, E; Waterson, D; White, KL; Wittlin, S; Witty, MJ; Wu, Q; Younis, Y | 1 |
Calas, M; Caldarelli, SA; Duckert, JF; Hamel, M; Maynadier, M; Ouattara, M; Pellet, A; Périgaud, C; Peyrottes, S; Vial, HJ; Wein, S | 1 |
Aguiar, AC; Cortopassi, WA; Figueiredo, FJ; França, TC; Krettli, AU; Meneghetti, MR; Pimentel, AS; Santos, Rde M | 1 |
NOR EL-DIN, G | 1 |
Azas, N; Darque, A; Di Giorgio, C; Galy, J; Gasquet, M; Hout, S; Robin, M; Timon-David, P | 1 |
Arnal, P; Boisbrun, M; Calas, M; Carcel, C; Hamzé, A; Maynadier, M; Rubi, E; Salom-Roig, X; Vial, H; Wein, S | 1 |
Bressolle, FM; Calas, M; Margout, D; Nicolas, O; Taudon, N; Vial, HJ; Wein, S | 1 |
Brun, R; Ihara, M; Kaiser, M; Pudhom, K; Takasu, K | 1 |
Atkinson, ER; Granchelli, FE | 1 |
Beaudoin, RL; Gentilini, M; Guillouzo, A; Landau, I; Langlois, P; Mazier, D; Mellouk, S; Miltgen, F; Stahel, E | 1 |
Lee, LG; Makler, MT; Recktenwald, D | 1 |
Bogunović-Batchelor, MV; Islip, PJ | 1 |
Roberts, EC; Shealy, YF | 1 |
Folkers, K; Friedman, MD; Porter, TH; Stotter, PL | 1 |
Aviado, DM | 1 |
Henry, DW | 1 |
3 review(s) available for thiazoles and Malaria
Article | Year |
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Thiazole Containing Heterocycles with Antimalarial Activity.
Topics: Animals; Antimalarials; Humans; Malaria; Thiazoles | 2018 |
Thiazole, thio and semicarbazone derivatives against tropical infective diseases: Chagas disease, human African trypanosomiasis (HAT), leishmaniasis, and malaria.
Topics: Animals; Chagas Disease; Drug Design; Humans; Leishmaniasis; Malaria; Protozoan Infections; Semicarbazones; Thiazoles; Thiosemicarbazones; Trypanosomiasis, African | 2019 |
Chemotherapy of Plasmodium berghei.
Topics: Animals; Anthracenes; Anti-Bacterial Agents; Anti-Infective Agents; Antimalarials; Benzene Derivatives; Cardiovascular System; Central Nervous System; Coloring Agents; Enzyme Inhibitors; Erythropoiesis; Histamine; Hormones; Malaria; Malaria, Avian; Mice; Naphthyridines; Organometallic Compounds; Plasmodium; Pteridines; Pyrimidines; Pyrroles; Quinolines; Rats; Sulfonamides; Sulfones; Thiazoles; Vitamins | 1969 |
33 other study(ies) available for thiazoles and Malaria
Article | Year |
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Targeting the Extrinsic Pathway of Hepatocyte Apoptosis Promotes Clearance of Plasmodium Liver Infection.
Topics: Administration, Oral; Animals; Apoptosis; Biological Availability; Caspase 3; Culicidae; Dipeptides; Hepatocytes; Immunity; Indoles; Inhibitor of Apoptosis Proteins; Life Cycle Stages; Liver; Malaria; Plasmodium; Protozoan Proteins; Sporozoites; Thiazoles; Tumor Necrosis Factor-alpha | 2020 |
Malaria fighters' latest chemical weapon may not last long.
Topics: Animals; Anopheles; Drug Resistance; Guanidines; Humans; Insecticides; Malaria; Neonicotinoids; Rwanda; Thiazoles | 2020 |
Efficacy of Fludora® Fusion (a mixture of deltamethrin and clothianidin) for indoor residual spraying against pyrethroid-resistant malaria vectors: laboratory and experimental hut evaluation.
Topics: Animals; Anopheles; Benin; Guanidines; Humans; Insecticide Resistance; Insecticides; Laboratories; Malaria; Mosquito Control; Mosquito Vectors; Neonicotinoids; Nitriles; Pyrethrins; Thiazoles | 2020 |
Synthesis and antimalarial and anticancer evaluation of 7-chlorquinoline-4-thiazoleacetic derivatives containing aryl hydrazide moieties.
Topics: A549 Cells; Acetic Acid; Animals; Antimalarials; Antineoplastic Agents; Apoptosis; Cell Cycle Checkpoints; Cell Survival; Disease Models, Animal; Humans; Hydrazines; Inhibitory Concentration 50; Malaria; Male; MCF-7 Cells; Mice; Mice, Inbred BALB C; Quinolines; Structure-Activity Relationship; Thiazoles | 2021 |
High Accumulation and
Topics: Animals; Antimalarials; Erythrocytes; Female; Malaria; Mice; Parasite Load; Parasitic Sensitivity Tests; Plasmodium; Spleen; Thiazoles | 2017 |
Indoor residual spraying with a mixture of clothianidin (a neonicotinoid insecticide) and deltamethrin provides improved control and long residual activity against pyrethroid resistant Anopheles gambiae sl in Southern Benin.
Topics: Animals; Anopheles; Benin; Culex; Guanidines; Housing; Humans; Insecticide Resistance; Insecticides; Malaria; Mosquito Control; Neonicotinoids; Pyrethrins; Thiazoles; World Health Organization | 2017 |
Small-scale field evaluation of the efficacy and residual effect of Fludora
Topics: Animals; Anopheles; Benin; Female; Guanidines; Insecticide Resistance; Insecticides; Malaria; Mosquito Control; Mosquito Vectors; Neonicotinoids; Nitriles; Pesticide Residues; Pyrethrins; Thiazoles | 2018 |
Indoor residual spray bio-efficacy and residual activity of a clothianidin-based formulation (SumiShield
Topics: Aerosols; Animals; Anopheles; Biological Assay; Democratic Republic of the Congo; Female; Guanidines; Insecticides; Malaria; Mosquito Control; Neonicotinoids; Survival Analysis; Thiazoles; Time Factors; Treatment Outcome | 2019 |
Evaluation of the residual effectiveness of Fludora™ fusion WP-SB, a combination of clothianidin and deltamethrin, for the control of pyrethroid-resistant malaria vectors on Bioko Island, Equatorial Guinea.
Topics: Animals; Anopheles; Equatorial Guinea; Guanidines; Humans; Insecticide Resistance; Insecticides; Islands; Malaria; Mosquito Control; Mosquito Vectors; Neonicotinoids; Nitriles; Pyrethrins; Thiazoles | 2019 |
Diagnostic dose determination and efficacy of chlorfenapyr and clothianidin insecticides against Anopheles malaria vector populations of western Kenya.
Topics: Animals; Anopheles; Dose-Response Relationship, Drug; Guanidines; Insecticides; Kenya; Lethal Dose 50; Malaria; Mosquito Control; Mosquito Vectors; Neonicotinoids; Pyrethrins; Species Specificity; Thiazoles | 2019 |
Improvement of antimalarial activity of a 3-alkylpiridine alkaloid analog by replacing the pyridine ring to a thiazole-containing heterocycle: Mode of action, mutagenicity profile, and Caco-2 cell-based permeability.
Topics: Alkaloids; Animals; Antimalarials; Caco-2 Cells; Cell Line; Cell Line, Tumor; Chloroquine; Female; Hemeproteins; Humans; Malaria; Mice; Mutagens; Permeability; Plasmodium berghei; Plasmodium falciparum; Pyridines; Thiazoles | 2019 |
Susceptibility testing of Anopheles malaria vectors with the neonicotinoid insecticide clothianidin; results from 16 African countries, in preparation for indoor residual spraying with new insecticide formulations.
Topics: Africa South of the Sahara; Animals; Anopheles; Communicable Disease Control; Guanidines; Insecticide Resistance; Insecticides; Malaria; Mosquito Control; Mosquito Vectors; Neonicotinoids; Reference Values; Thiazoles | 2019 |
Antimalarial activity of phenylthiazolyl-bearing hydroxamate-based histone deacetylase inhibitors.
Topics: Animals; Antimalarials; Aotidae; Drug Resistance; Enzyme Inhibitors; Histone Deacetylase Inhibitors; Hydroxamic Acids; In Vitro Techniques; Malaria; Malaria, Falciparum; Male; Mice; Mice, Inbred ICR; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship; Thiazoles | 2008 |
Identification of a metabolically stable triazolopyrimidine-based dihydroorotate dehydrogenase inhibitor with antimalarial activity in mice.
Topics: Administration, Oral; Animals; Antimalarials; Dihydroorotate Dehydrogenase; Humans; In Vitro Techniques; Malaria; Male; Mice; Microsomes, Liver; Models, Molecular; Oxidoreductases Acting on CH-CH Group Donors; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Pyrimidines; Structure-Activity Relationship; Thiazoles; Triazoles | 2009 |
Rapid resolution liquid chromatography-mass spectrometry determination of SAR97276 in monkey matrices. Pharmacokinetics in rhesus monkey infected by Plasmodium cynomolgi.
Topics: Animals; Antimalarials; Biological Availability; Buffers; Calibration; Chromatography, Liquid; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Drug Stability; Freezing; Half-Life; Hydrogen-Ion Concentration; Macaca mulatta; Malaria; Mass Spectrometry; Metabolic Clearance Rate; Molecular Structure; Plasmodium cynomolgi; Quality Control; Reference Standards; Reproducibility of Results; Sensitivity and Specificity; Solid Phase Extraction; Spectrometry, Mass, Electrospray Ionization; Thiazoles; Time Factors | 2009 |
Exploration of potential prodrug approach of the bis-thiazolium salts T3 and T4 for orally delivered antimalarials.
Topics: Animals; Antimalarials; Dose-Response Relationship, Drug; Malaria; Mice; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium; Prodrugs; Salts; Stereoisomerism; Structure-Activity Relationship; Thiazoles | 2010 |
Contributions to the chemistry of synthetic antimalarials; some delta-diethylamino-alpha-methylbutylamino derivatives of pyridine and thiazole.
Topics: Antimalarials; Malaria; Pyridines; Thiazoles | 1945 |
Synthesis and in vitro antiprotozoal activities of 5-phenyliminobenzo[a]phenoxazine derivatives.
Topics: Animals; Antimalarials; Antiprotozoal Agents; Drug Design; Inhibitory Concentration 50; Leishmania donovani; Malaria; Models, Chemical; Molecular Structure; Myoblasts; Oxazines; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyridinium Compounds; Rats; Structure-Activity Relationship; Thiazoles; Trypanocidal Agents; Trypanosoma brucei rhodesiense; Trypanosoma cruzi | 2011 |
Novel orally active antimalarial thiazoles.
Topics: Administration, Oral; Animals; Antimalarials; Biological Availability; Cytochrome P-450 CYP1A2 Inhibitors; Drug Interactions; Drug Resistance; Ether-A-Go-Go Potassium Channels; Humans; In Vitro Techniques; Injections, Intravenous; Malaria; Male; Mice; Microsomes; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Thiazoles | 2011 |
Disulfide prodrugs of albitiazolium (T3/SAR97276): synthesis and biological activities.
Topics: Animals; Antimalarials; Disulfides; Malaria; Mice; Plasmodium falciparum; Prodrugs; Stereoisomerism; Structure-Activity Relationship; Thiazoles | 2012 |
Antimalarial activity and mechanisms of action of two novel 4-aminoquinolines against chloroquine-resistant parasites.
Topics: Aminoquinolines; Animals; Antimalarials; Cell Line, Tumor; Chloroquine; Dose-Response Relationship, Drug; Drug Resistance; Enzyme-Linked Immunosorbent Assay; Hemeproteins; Humans; In Vitro Techniques; L-Lactate Dehydrogenase; Malaria; Mice; Models, Molecular; Molecular Structure; Plasmodium berghei; Plasmodium falciparum; Protein Binding; Protein Conformation; Tetrazolium Salts; Thiazoles | 2012 |
Recent views in treatment of malaria; a trial of a new drug (abadol).
Topics: Malaria; Thiazoles | 1951 |
Activity of benzothiazoles and chemical derivatives on Plasmodium falciparum.
Topics: Adolescent; Aged; Animals; Antimalarials; Benzothiazoles; Cell Line; Dose-Response Relationship, Drug; Drug Resistance; Female; Humans; Life Cycle Stages; Malaria; Malaria, Falciparum; Mice; Mice, Inbred BALB C; Monocytes; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Thiazoles | 2004 |
Mono- and bis-thiazolium salts have potent antimalarial activity.
Topics: Animals; Antimalarials; Female; Malaria; Mice; Plasmodium falciparum; Structure-Activity Relationship; Thiazoles | 2005 |
Pharmacological properties of a new antimalarial bisthiazolium salt, T3, and a corresponding prodrug, TE3.
Topics: Animals; Antimalarials; Bayes Theorem; Female; Injections, Intraperitoneal; Injections, Intravenous; Malaria; Mice; Models, Biological; Plasmodium; Plasmodium falciparum; Prodrugs; Rats; Rats, Sprague-Dawley; Thiazoles | 2005 |
Synthesis and antimalarial efficacy of aza-fused rhodacyanines in vitro and in the P. berghei mouse model.
Topics: Animals; Antimalarials; Aza Compounds; Cell Line; Drug Resistance; Malaria; Mice; Plasmodium berghei; Plasmodium falciparum; Pyridinium Compounds; Thiazoles | 2006 |
Antimalarials V: aminobenzothiazoles.
Topics: Animals; Antimalarials; Chickens; Malaria; Methods; Mice; Plasmodium berghei; Thiazoles | 1976 |
Iron chelators: in vitro inhibitory effect on the liver stage of rodent and human malaria.
Topics: Animals; Cells, Cultured; Deferoxamine; Dihydropyridines; Humans; Iron Chelating Agents; Liver; Malaria; Microscopy, Electron; Plasmodium falciparum; Plasmodium yoelii; Rats; Thiazoles | 1988 |
Thiazole orange: a new dye for Plasmodium species analysis.
Topics: Animals; Azure Stains; Benzothiazoles; Erythrocytes; Flow Cytometry; Fluorescent Dyes; Humans; Malaria; Plasmodium falciparum; Quinolines; Thiazoles | 1987 |
5-(Hydroxyimino)-4-methoxy-2-(pivaloylimino)thiazolidine-3 -acetamide, a reduced nitroheterocyclic derivative with potent schistosomicidal properties.
Topics: Animals; Malaria; Mice; Niridazole; Praziquantel; Schistosoma mansoni; Schistosomicides; Thiazoles | 1985 |
Folic acid analogs. Modifications in the benzene-ring region. 2. Thiazole analogs.
Topics: Animals; Carcinoma; Cell Line; Chromatography, Thin Layer; Columbidae; Enterococcus faecalis; Folic Acid; Folic Acid Antagonists; Humans; Laryngeal Neoplasms; Leukemia L1210; Liver; Magnetic Resonance Spectroscopy; Malaria; Mice; Plasmodium berghei; Structure-Activity Relationship; Thiazoles | 1972 |
Synthesis of alkyl-4,7-dioxobenzothiazoles with prophylactic antimalarial activity.
Topics: Alkanes; Animals; Antimalarials; Chickens; Malaria; Plasmodium; Thiazoles | 1973 |
Chemotherapeutic nitroheterocycles. Derivatives of 5-nitrothiazole-2-carboxaldehyde and 5-nitrothiazole-2-carboxylic acid.
Topics: Animals; Bacteria; Fungi; Malaria; Mice; Schistosomiasis; Thiazoles; Yeasts | 1969 |