Page last updated: 2024-08-21

thiazoles and Malaria, Falciparum

thiazoles has been researched along with Malaria, Falciparum in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (45.45)29.6817
2010's6 (54.55)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abdulla, S; Bonkian, LN; Bouyou-Akotet, M; Cantalloube, C; Djeriou, E; Held, J; Kreidenweiss, A; Kremsner, PG; Mordmüller, B; Nahum, A; Ogutu, B; Salazar, CLO; Sié, A; Siribie, M; Sirima, SB; Supan, C; Tinto, H1
Bordat, Y; Fraisse, L; Maynadier, M; Perez, J; Peyrottes, S; Tran Van Ba, C; Vial, HJ; Wein, S1
Boisson, A; Chantelauze, H; Fraisse, L; Penarete-Vargas, DM; Peyrottes, S; Urbach, S; Vial, HJ1
Andrews, KT; Caridha, D; Chen, Y; Dow, GS; Gerena, L; Gettayacamin, M; Johnson, J; Kozikowski, AP; Li, Q; Melendez, V; Obaldia, N; Tran, TN1
Boykin, DW; Branowska, D; Brun, R; Farahat, AA; Kumar, A; Liu, Y; Wenzler, T; Wilson, WD1
Clark, MA; Ferrer, P; Hand, CC; Rienhoff, HY; Sullivan, DJ; Tripathi, AK1
Chibale, K; Gordon, R; Paquet, T; Waterson, D; Witty, MJ1
Azas, N; Darque, A; Di Giorgio, C; Galy, J; Gasquet, M; Hout, S; Robin, M; Timon-David, P1
Brun, R; Ihara, M; Inoue, H; Kaiser, M; Kasai, K; Pudhom, K; Takasu, K; Terauchi, H1
Biagini, GA; Boudou, F; Bray, PG; Calas, M; Dubremetz, JF; Precigout, E; Richier, E; Vial, HJ; Ward, SA; Wein, S1
Chemaly, SM; Chen, CT; van Zyl, RL1

Trials

1 trial(s) available for thiazoles and Malaria, Falciparum

ArticleYear
Safety and efficacy of the choline analogue SAR97276 for malaria treatment: results of two phase 2, open-label, multicenter trials in African patients.
    Malaria journal, 2017, 05-04, Volume: 16, Issue:1

    Topics: Adolescent; Adult; Africa South of the Sahara; Antimalarials; Child; Child, Preschool; Cohort Studies; Female; Humans; Incidence; Infant; Malaria, Falciparum; Male; Middle Aged; Plasmodium falciparum; Thiazoles; Treatment Outcome; Young Adult

2017

Other Studies

10 other study(ies) available for thiazoles and Malaria, Falciparum

ArticleYear
New insight into the mechanism of accumulation and intraerythrocytic compartmentation of albitiazolium, a new type of antimalarial.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:9

    Topics: Antimalarials; Babesia; Cell Membrane; Drug Resistance; Erythrocytes; Humans; Malaria, Falciparum; Plasmodium falciparum; Proton-Motive Force; Thiazoles

2014
A chemical proteomics approach for the search of pharmacological targets of the antimalarial clinical candidate albitiazolium in Plasmodium falciparum using photocrosslinking and click chemistry.
    PloS one, 2014, Volume: 9, Issue:12

    Topics: Animals; Antimalarials; Binding, Competitive; Click Chemistry; Cross-Linking Reagents; Diacylglycerol Cholinephosphotransferase; Endoplasmic Reticulum; Humans; Malaria, Falciparum; Models, Chemical; Molecular Structure; Plasmodium falciparum; Protein Binding; Proteome; Proteomics; Protozoan Proteins; Thiazoles; trans-Golgi Network

2014
Antimalarial activity of phenylthiazolyl-bearing hydroxamate-based histone deacetylase inhibitors.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:10

    Topics: Animals; Antimalarials; Aotidae; Drug Resistance; Enzyme Inhibitors; Histone Deacetylase Inhibitors; Hydroxamic Acids; In Vitro Techniques; Malaria; Malaria, Falciparum; Male; Mice; Mice, Inbred ICR; Plasmodium; Plasmodium berghei; Plasmodium falciparum; Structure-Activity Relationship; Thiazoles

2008
Synthesis and antiprotozoal activity of 2,5-bis[amidinoaryl]thiazoles.
    Bioorganic & medicinal chemistry, 2010, May-15, Volume: 18, Issue:10

    Topics: Administration, Oral; Animals; Antimalarials; Antiprotozoal Agents; Disease Models, Animal; DNA, Protozoan; Drug Stability; Malaria, Falciparum; Mice; Parasitic Sensitivity Tests; Pentamidine; Plasmodium falciparum; Rats; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2010
Antimalarial iron chelator, FBS0701, shows asexual and gametocyte Plasmodium falciparum activity and single oral dose cure in a murine malaria model.
    PloS one, 2012, Volume: 7, Issue:5

    Topics: Animals; Antimalarials; Disease Models, Animal; Ethyl Ethers; Iron Chelating Agents; Malaria, Falciparum; Mice; Parasitemia; Plasmodium falciparum; Thiazoles; Treatment Outcome

2012
Antimalarial aminothiazoles and aminopyridines from phenotypic whole-cell screening of a SoftFocus(®) library.
    Future medicinal chemistry, 2012, Volume: 4, Issue:18

    Topics: Aminopyridines; Animals; Antimalarials; Databases, Pharmaceutical; Drug Resistance; Humans; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship; Thiazoles

2012
Activity of benzothiazoles and chemical derivatives on Plasmodium falciparum.
    Parasitology, 2004, Volume: 129, Issue:Pt 5

    Topics: Adolescent; Aged; Animals; Antimalarials; Benzothiazoles; Cell Line; Dose-Response Relationship, Drug; Drug Resistance; Female; Humans; Life Cycle Stages; Malaria; Malaria, Falciparum; Mice; Mice, Inbred BALB C; Monocytes; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Thiazoles

2004
Synthesis of three classes of rhodacyanine dyes and evaluation of their in vitro and in vivo antimalarial activity.
    Bioorganic & medicinal chemistry, 2006, Dec-15, Volume: 14, Issue:24

    Topics: Animals; Antimalarials; Cells, Cultured; Chloroquine; Coloring Agents; Drug Resistance; Malaria, Falciparum; Male; Mice; Mice, Inbred ICR; Myoblasts, Skeletal; Plasmodium berghei; Plasmodium falciparum; Pyridinium Compounds; Rats; Thiazoles

2006
Potent antihematozoan activity of novel bisthiazolium drug T16: evidence for inhibition of phosphatidylcholine metabolism in erythrocytes infected with Babesia and Plasmodium spp.
    Antimicrobial agents and chemotherapy, 2006, Volume: 50, Issue:10

    Topics: Animals; Antimalarials; Antiprotozoal Agents; Babesia; Babesiosis; Erythrocytes; Hemolysis; Humans; Malaria, Falciparum; Phosphatidylcholines; Plasmodium falciparum; Thiazoles

2006
Naturally occurring cobalamins have antimalarial activity.
    Journal of inorganic biochemistry, 2007, Volume: 101, Issue:5

    Topics: Animals; Antimalarials; Hemeproteins; Humans; Malaria, Falciparum; Plasmodium falciparum; Tetrazolium Salts; Thiazoles; Vitamin B 12

2007