Page last updated: 2024-08-21

thiazoles and Leukemia

thiazoles has been researched along with Leukemia in 77 studies

Research

Studies (77)

TimeframeStudies, this research(%)All Research%
pre-19906 (7.79)18.7374
1990's7 (9.09)18.2507
2000's36 (46.75)29.6817
2010's25 (32.47)24.3611
2020's3 (3.90)2.80

Authors

AuthorsStudies
Bielawska, A; Bielawski, K; Czarnomysy, R; Finiuk, N; Gzella, A; Holota, S; Ivasechko, I; Kashchak, N; Khyluk, D; Klyuchivska, O; Lesyk, D; Lesyk, R; Roszczenko, P; Senkiv, J; Stoika, R; Yushyn, I1
Cherniienko, A; Finiuk, N; Klyuchivska, O; Lesyk, R; Lozynskyi, A; Manko, N; Senkiv, J; Stoika, R; Yushyn, I; Zelisko, N1
Jasek-Gajda, E; Jasińska, M; Jurkowska, H; Lis, GJ; Litwin, JA1
Das, T; Dash, J; Debnath, M; Dutta, D; Paul, R1
Hattori, Y; Kato, J; Kohashi, S; Matsuki, E; Matsushita, M; Mori, T; Okamoto, S; Tonegawa, K1
Baldwin, AS; Christopherson, RI; Cooper, MJ; Cox, NJ; Dewar, BJ; Duncan, JS; Frye, SV; Ghose Roy, S; Graves, LM; Jin, J; Johnson, GL; Jones, LS; Kuan, PF; Nguyen, TA; Richards, KL; Smalley, DM; Whittle, MC; Zimmerman, EI1
Jozwiak, Z; Laroche-Clary, A; Marszalek, I; Matusiak, A; Robert, J; Szwed, M1
Brüning, A; Gafiuc, D; Mylonas, I; Weiß, M1
Bertomeu, T; Bucur, O; Dewar, R; Goganau, I; Khosravi-Far, R; Pennarun, B; Petrescu, SM; Stancu, AL1
Hu, R; Liao, A; Liu, Z; Wang, H; Wang, X; Yang, W; Zhang, J; Zhao, C1
Faiz, SA; Jimenez, CA; Sahay, S1
Asmussen, J; Craik, CS; Jun, YW; Seo, D; Shah, N; Tajon, CA1
Ding, N; Feng, L; Ping, L; Shi, Y; Song, Y; Zheng, X; Zhu, J1
Stone, RM; Wolach, O1
Birgens, H; Brown, Pde N; Dalseg, AM; Dufva, IH; Hasselbalch, HC; Jensen, MK; Vangsted, A1
Chen, SH; Chen, YJ; Chen, YY; Hsu, ML; Huang, WP; Lee, JJ; Lin, CP; Shieh, HR; Tseng, YJ; Yang, YC1
Lohiya, NK; Pal, R; Talwar, GP; Vishwakarma, R; Vyas, HK1
Chen, B; Guo, D; Hu, H; Li, X; Wang, X; Wu, C1
Bailly, C; Baldeyrou, B; Beauchard, A; Besson, T; Chérouvrier, JR; Domon, L; Jaunet, A; Lansiaux, A; Murillo, L; Picot, L; Thiéry, V1
Horiike, S; Kobayashi, T; Kuroda, J; Matsumoto, Y; Mizutani, S; Ohshiro, M; Sasaki, N; Shimazaki, C; Shimura, Y; Taniwaki, M; Tsutsumi, Y; Uchiyama, H; Yamamoto, M1
Chen, CT; Chung, JG; Hsu, YM; Huang, SP; Ip, SW; Lin, JG; Lin, JP; Wu, CC; Wu, PP; Yang, JS; Yu, FS1
Chen, Y; Jing, YX; Qi, SN; Song, LJ1
Lasho, T; Pardanani, A; Tefferi, A1
Kavitha, CV; Prasanna, DS; Raghavan, SC; Ranganatha, SR; Rangappa, KS; Vinaya, K1
Cai, Q; Ding, K; Feng, Y; Gan, J; Li, X; Lu, X; Luo, K; Ren, X; Tu, Z; Wan, J; Wang, D; Yingxue, L; Zhang, F; Zhang, Z1
Bensdorf, K; Cai, X; Cao, P; Gust, R; Huang, W; Li, Z; Liu, W; Qi, F; Qian, H; Wellner, A; Zhang, H; Zhou, J1
Einsele, H; Ekblom, M; Gostick, E; Koechel, C; Kreutzman, A; Ladell, K; Melo, T; Mustjoki, S; Porkka, K; Price, DA; Seggewiss, R; Stenke, L1
Akbarzadeh, T; Bu, Y; Fallah-Tafti, A; Foroumadi, A; Hangauer, DG; Parang, K; Shafiee, A; Shirazi, AN; Tiwari, R1
Cowell, JK; Qin, H; Ren, M; Ren, R; Tidwell, J1
Agrawal, S; Furlong, MT; Hawthorne, D; Krueger, L; Lago, M; Stouffer, B; Unger, S1
Einsele, H; Hassold, N; Kempf, K; Seggewiss-Bernhardt, R; Seystahl, K; Urlaub, D; Watzl, C; Wischhusen, J; Zekl, M1
Harada, H; Harada, Y; Imagawa, J; Matsumoto, K; Morita, K; Tanaka, H1
Dingermann, T; Marschalek, R; Zündorf, I1
Gaston, K; Jayaraman, PS; Noy, P1
Chauvier, D; Kegelaer, G; Manfait, M; Morjani, H1
Akutsu, M; Furukawa, Y; Izumi, T; Kano, Y; Ohmine, K; Tsunoda, S1
Martin-Kleiner, I1
Cai, RB; Chen, XS; Fang, TL; Guo, GL1
Liu, XP; Narla, RK; Uckun, FM1
Lyubchenko, TA; Wurth, GA; Zweifach, A1
Abe, A; Emi, N; Kanbe, E; Kawabe, T; Saito, H; Towatari, M1
Boranić, M; Gabrilovac, J; Kusec, R; Martin-Kleiner, I1
BURCHENAL, JH; COLEY, VC; KRAKOFF, IH; OETTGEN, HF; PURPLE, JR1
Batorsky, R; Keller, KA; Kim, KS; Kimball, SD; Lee, FY; Lu, S; Misra, RN; Mulheron, JG; Sack, JS; Tokarski, JS; Webster, KR; Williams, DK; Xiao, HY1
Broekhuizen, AJ; Creutzig, U; Gibson, B; Hubeek, I; Kaspers, GJ; Peters, GJ; Schouten van Meeteren, AY; Talianidis, I; van Wering, ER1
D'Cruz, OJ; Tai, HL; Uckun, FM1
Benyumov, AO; Downs, S; Dumezb, D; Grigoriants, OO; Tibbles, HE; Uckun, FM; Vassilev, AO; Venkatachalam, TK1
Conrad, DM; Hoskin, DW; Mader, JS; Salsman, J1
Morachevskaya, EA; Negulyaev, YA; Staruschenko, A1
Aninat, C; Fardel, O; Le Vee, M; Sparfel, L; Van Grevenynghe, J1
Amirghofran, Z; Azadmehr, A; Bahmani, M; Javidnia, K1
Anuchapreeda, S; Chanarat, P; Limtrakul, P; Sittipreechacharn, S; Thanarattanakorn, P1
Böttger, S; Low, B; Walker, C1
Güzel, O; Salman, A1
Akgün-Dar, K; Atasever, B; Carin, M; Kiliçaslan-Ayna, T; Kuruca, SE; Meriçli, F; Seyhan, VG; Turan, N1
Ainoon, O; Cheong, SK; Fazlina, N; Hamidah, H; Hamidah, NH; Jamal, R; Maha, A; Zarina, AL; Zulkifli, SZ1
Scorilas, A; Thomadaki, H; Tsiapalis, CM1
Hampton, T1
Bergmann, L; Esser, R; Glienke, W; Koehl, U; Maute, L; Milz, E1
Chen, GQ; Wang, LS; Wu, YL; Yu, Y1
Esser, R; Kalaäoui, RE; Klingebiel, T; Kloess, S; Koehl, U; Kreuter, J; Lehrnbecher, T; Munkelt, D; Schubert, R; Schwabe, D; Wehner, S; Zimmermann, SY1
Lei, P; Li, W; Shao, J; Shen, G; Wang, X; Yang, J; Ye, Q; Zhang, Y; Zhu, H1
Notario, A; Ranghetti, L; Stanziale, D; Torriani, A; Vitti, MP1
Blagosklonny, MV; Neckers, LM1
Tan, BK; Wong, KT1
Efferth, T; Fabry, U; Osieka, R1
Liu, J; Wei, D; Zhang, C; Zhang, P; Zhao, Z1
Ahmed, N; Berridge, MV1
Cinatl, J; Kreuter, J; Langer, K; Matousek, J; Michaelis, M; Schwabe, D; Slavik, T; Vogel, JU1
Capone, F; Chimirri, A; Grimaudo, S; Monforte, AM; Poretto, F; Raimondi, MV; Simoni, D; Tolomeo, M1
Jiang, B; Li, CM; Li, ML; Lin, ZW; Mei, SX; Na, Z; Niu, XM; Sun, HD; Yang, H1
Fujii, Y; Hongo, T1
Duke, M; Goh, TS; Kirkpatrick, DL1
Borghi, G; Bravi, M; Broglia, M; Guerra, G; Notario, A; Torriani, A1
Baguley, BC; Finlay, GJ; Wilson, WR1
Deliwala, CV; Modi, JD; Sabnis, SS1
Rice, LM; Scott, KR1

Reviews

4 review(s) available for thiazoles and Leukemia

ArticleYear
Pleural effusions in acute and chronic leukemia and myelodysplastic syndrome.
    Current opinion in pulmonary medicine, 2014, Volume: 20, Issue:4

    Topics: Acute Disease; Biopsy; Bone Marrow; Chronic Disease; Dasatinib; Humans; Leukemia; Myelodysplastic Syndromes; Pleura; Pleural Effusion; Prognosis; Protein Kinase Inhibitors; Pyrimidines; Thiazoles

2014
[Novel medical treatment modalities in hematology].
    Ugeskrift for laeger, 2008, Jun-09, Volume: 170, Issue:24

    Topics: Aminoglycosides; Anemia, Hemolytic; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antibodies, Monoclonal, Murine-Derived; Antineoplastic Agents; Benzamides; Benzoates; Boronic Acids; Bortezomib; Carbazoles; Carrier Proteins; Cyclophosphamide; Dasatinib; Furans; Gemtuzumab; Hematologic Diseases; Humans; Hydrazines; Imatinib Mesylate; Immunologic Factors; Indoles; Lenalidomide; Leukemia; Leukemia, Lymphocytic, Chronic, B-Cell; Leukemia, Myeloid, Acute; Lymphoma; Multiple Myeloma; Myelodysplastic Syndromes; Piperazines; Purpura, Thrombocytopenic; Pyrazines; Pyrazoles; Pyrimidines; Receptors, Fc; Recombinant Fusion Proteins; Rituximab; Thalidomide; Thiazoles; Thrombopoietin; Vidarabine

2008
[Leukemia: A highly malignant disease].
    Pharmazie in unserer Zeit, 2012, Volume: 41, Issue:3

    Topics: Animals; Antineoplastic Agents; Benzamides; Dasatinib; Disease Models, Animal; History, 19th Century; Humans; Imatinib Mesylate; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Philadelphia Chromosome; Piperazines; Pyrimidines; Thiazoles; Tretinoin

2012
Leukemia, an effective model for chemical biology and target therapy.
    Acta pharmacologica Sinica, 2007, Volume: 28, Issue:9

    Topics: Antineoplastic Agents; Apoptosis; Arsenic Trioxide; Arsenicals; Benzamides; Dasatinib; Growth Inhibitors; Humans; Imatinib Mesylate; Leukemia; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Promyelocytic, Acute; Oxides; Piperazines; Protein Kinase Inhibitors; Pyrimidines; Thiazoles; Tretinoin

2007

Trials

1 trial(s) available for thiazoles and Leukemia

ArticleYear
A validated LC-MS/MS assay for the simultaneous determination of the anti-leukemic agent dasatinib and two pharmacologically active metabolites in human plasma: application to a clinical pharmacokinetic study.
    Journal of pharmaceutical and biomedical analysis, 2012, Jan-25, Volume: 58

    Topics: Antineoplastic Agents; Calibration; Chromatography, Liquid; Dasatinib; Humans; Leukemia; Pyrimidines; Reference Standards; Reproducibility of Results; Sensitivity and Specificity; Solid Phase Extraction; Spectrometry, Mass, Electrospray Ionization; Tandem Mass Spectrometry; Thiazoles

2012

Other Studies

72 other study(ies) available for thiazoles and Leukemia

ArticleYear
Development of Novel Pyridine-Thiazole Hybrid Molecules as Potential Anticancer Agents.
    Molecules (Basel, Switzerland), 2022, Sep-21, Volume: 27, Issue:19

    Topics: Antineoplastic Agents; Benzoic Acid; Cell Line, Tumor; Cell Proliferation; DNA; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Esters; Humans; Leukemia; Molecular Structure; Neoplasms; Pyridines; Structure-Activity Relationship; Thiazoles

2022
Thiopyrano[2,3-d]thiazole structures as promising scaffold with anticancer potential.
    Chemico-biological interactions, 2022, Dec-01, Volume: 368

    Topics: Animals; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Glioblastoma; HEK293 Cells; Humans; Leukemia; Mammals; Mice; Reactive Oxygen Species; Thiazoles

2022
Combination of ERK2 inhibitor VX-11e and voreloxin synergistically enhances anti-proliferative and pro-apoptotic effects in leukemia cells.
    Apoptosis : an international journal on programmed cell death, 2019, Volume: 24, Issue:11-12

    Topics: Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Cell Cycle Checkpoints; Cell Proliferation; Cyclin-Dependent Kinase Inhibitor p21; Dose-Response Relationship, Drug; Drug Synergism; Humans; K562 Cells; Leukemia; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Mitogen-Activated Protein Kinase 3; Naphthyridines; NF-kappa B; Signal Transduction; Thiazoles

2019
G4 Sensing Pyridyl-Thiazole Polyamide Represses c-KIT Expression in Leukemia Cells.
    Chemistry (Weinheim an der Bergstrasse, Germany), 2021, Jun-10, Volume: 27, Issue:33

    Topics: G-Quadruplexes; Humans; Leukemia; Ligands; Nylons; Promoter Regions, Genetic; Proto-Oncogene Mas; Thiazoles

2021
Detection of leukemia associated antigen-specific cytotoxic T cells in a patient with Philadelphia chromosome-positive leukemia during treatment with dasatinib.
    Leukemia & lymphoma, 2014, Volume: 55, Issue:3

    Topics: Antigens, Neoplasm; Antineoplastic Agents; Dasatinib; Epitopes, T-Lymphocyte; Humans; Leukemia; Male; Middle Aged; Philadelphia Chromosome; Protein Kinase Inhibitors; Pyrimidines; T-Lymphocytes, Cytotoxic; Thiazoles; Treatment Outcome

2014
Application of multiplexed kinase inhibitor beads to study kinome adaptations in drug-resistant leukemia.
    PloS one, 2013, Volume: 8, Issue:6

    Topics: Benzamides; Cell Line; Cell Survival; Chromatography, Affinity; Dasatinib; Drug Resistance, Neoplasm; Fusion Proteins, bcr-abl; Humans; Imatinib Mesylate; Immunoblotting; Leukemia; NF-kappa B; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; src-Family Kinases; Thiazoles

2013
Transferrin as a drug carrier: Cytotoxicity, cellular uptake and transport kinetics of doxorubicin transferrin conjugate in the human leukemia cells.
    Toxicology in vitro : an international journal published in association with BIBRA, 2014, Volume: 28, Issue:2

    Topics: Algorithms; Antibiotics, Antineoplastic; Biological Transport, Active; Cell Line, Tumor; Cell Survival; Coloring Agents; Doxorubicin; Drug Carriers; Flow Cytometry; Humans; K562 Cells; Kinetics; Leukemia; Lymphocytes; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Spectrometry, Mass, Matrix-Assisted Laser Desorption-Ionization; Tetrazolium Salts; Thiazoles; Transferrin

2014
Borrelidin has limited anti-cancer effects in bcl-2 overexpressing breast cancer and leukemia cells and reveals toxicity in non-malignant breast epithelial cells.
    Journal of applied toxicology : JAT, 2014, Volume: 34, Issue:10

    Topics: Adenosine Triphosphate; Antibiotics, Antineoplastic; Blotting, Western; Breast; Breast Neoplasms; Cell Line, Tumor; Epithelial Cells; Fatty Alcohols; Female; Genes, bcl-2; Human Umbilical Vein Endothelial Cells; Humans; Leukemia; Tetrazolium Salts; Thiazoles

2014
Combination of bortezomib and mitotic inhibitors down-modulate Bcr-Abl and efficiently eliminates tyrosine-kinase inhibitor sensitive and resistant Bcr-Abl-positive leukemic cells.
    PloS one, 2013, Volume: 8, Issue:10

    Topics: Benzamides; Boronic Acids; Bortezomib; Caspases; Cell Death; Cell Line, Tumor; Dasatinib; Down-Regulation; Drug Resistance, Neoplasm; Drug Synergism; Enzyme Activation; Fusion Proteins, bcr-abl; Heterocyclic Compounds, 2-Ring; Humans; Imatinib Mesylate; JNK Mitogen-Activated Protein Kinases; Leukemia; Mitosis; Models, Biological; p38 Mitogen-Activated Protein Kinases; Paclitaxel; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Pteridines; Pyrazines; Pyrimidines; Signal Transduction; STAT5 Transcription Factor; Thiazoles

2013
Methylation of SFRP5 is related to multidrug resistance in leukemia cells.
    Cancer gene therapy, 2014, Volume: 21, Issue:2

    Topics: Adaptor Proteins, Signal Transducing; Analysis of Variance; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; beta Catenin; Blotting, Western; Cell Line, Tumor; DNA Methylation; Doxorubicin; Drug Resistance, Multiple; Eye Proteins; Gene Expression Regulation, Neoplastic; Humans; Inhibitory Concentration 50; Leukemia; Membrane Proteins; Real-Time Polymerase Chain Reaction; Reverse Transcriptase Polymerase Chain Reaction; Tetrazolium Salts; Thiazoles; Wnt Signaling Pathway

2014
Sensitive and selective plasmon ruler nanosensors for monitoring the apoptotic drug response in leukemia.
    ACS nano, 2014, Sep-23, Volume: 8, Issue:9

    Topics: Apoptosis; Caspase 3; Dasatinib; Enzyme Assays; Gold; Humans; K562 Cells; Leukemia; Nanoparticles; Nanotechnology; Proteomics; Pyrimidines; Silicon Dioxide; Thiazoles

2014
Thiamet-G-mediated inhibition of O-GlcNAcase sensitizes human leukemia cells to microtubule-stabilizing agent paclitaxel.
    Biochemical and biophysical research communications, 2014, Oct-24, Volume: 453, Issue:3

    Topics: beta-N-Acetylhexosaminidases; Humans; Jurkat Cells; Leukemia; Microtubules; Paclitaxel; Phosphorylation; Pyrans; tau Proteins; Thiazoles

2014
How I treat mixed-phenotype acute leukemia.
    Blood, 2015, Apr-16, Volume: 125, Issue:16

    Topics: Acute Disease; Antineoplastic Combined Chemotherapy Protocols; B-Lymphocytes; Biomarkers, Tumor; Chromosome Aberrations; Combined Modality Therapy; Dasatinib; Flow Cytometry; Fusion Proteins, bcr-abl; Humans; Immunophenotyping; Leukemia; Middle Aged; Myeloid Cells; Pyrimidines; Stem Cell Transplantation; T-Lymphocytes; Thiazoles; Transplantation, Homologous

2015
Platonin induces autophagy-associated cell death in human leukemia cells.
    Autophagy, 2009, Volume: 5, Issue:2

    Topics: Amino Acid Chloromethyl Ketones; Autophagy; Caspases; Cell Cycle; Cell Differentiation; Cell Line, Tumor; Cell Membrane; Cell Proliferation; Cell Survival; Cytoplasm; Diploidy; Humans; Leukemia; Membrane Potential, Mitochondrial; Microtubule-Associated Proteins; Mitochondria; Monocytes; Thiazoles; Time Factors; Vacuoles

2009
Selective killing of leukemia and lymphoma cells ectopically expressing hCGbeta by a conjugate of curcumin with an antibody against hCGbeta subunit.
    Oncology, 2009, Volume: 76, Issue:2

    Topics: Aged; Antigens, CD; Antigens, Differentiation, Myelomonocytic; Cell Separation; Chorionic Gonadotropin, beta Subunit, Human; Curcumin; Drug Design; Female; Humans; Leukemia; Leukemia, Myeloid, Acute; Leukocytes, Mononuclear; Lymphoma; Male; Middle Aged; Sialic Acid Binding Ig-like Lectin 3; Tetrazolium Salts; Thiazoles; U937 Cells

2009
Study on the enhanced cellular uptake effect of daunorubicin on leukemia cells mediated via functionalized nickel nanoparticles.
    Biomedical materials (Bristol, England), 2009, Volume: 4, Issue:2

    Topics: Antineoplastic Agents; Biocompatible Materials; Cell Line, Tumor; Daunorubicin; Electrochemistry; Humans; K562 Cells; Leukemia; Metal Nanoparticles; Microscopy, Atomic Force; Microscopy, Fluorescence; Nanotechnology; Nickel; Permeability; Tetrazolium Salts; Thiazoles

2009
Synthesis and antitumoral activity of novel thiazolobenzotriazole, thiazoloindolo[3,2-c]quinoline and quinolinoquinoline derivatives.
    European journal of medicinal chemistry, 2009, Volume: 44, Issue:10

    Topics: Animals; Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; DNA; DNA Topoisomerases, Type I; Female; Humans; Indoles; Leukemia; Quinolines; Thiazoles; Topoisomerase I Inhibitors; Triazoles

2009
Allogenic bone marrow transplantation with fludarabine/busulfan16 conditioning regimen and dasatinib maintenance therapy for elderly Philadelphia-positive acute/advanced leukemia patients.
    Leukemia research, 2010, Volume: 34, Issue:4

    Topics: Acute Disease; Aged; Antineoplastic Combined Chemotherapy Protocols; Bone Marrow Transplantation; Busulfan; Chemotherapy, Adjuvant; Dasatinib; Humans; Immunosuppressive Agents; Leukemia; Male; Philadelphia Chromosome; Pyrimidines; Thiazoles; Transplantation Conditioning; Transplantation, Homologous; Vidarabine

2010
Diallyl sulfide inhibits murine WEHI-3 leukemia cells in BALB/c mice in vitro and in vivo.
    Human & experimental toxicology, 2009, Volume: 28, Issue:12

    Topics: Allyl Compounds; Animals; Antineoplastic Agents, Phytogenic; Cell Line, Tumor; Cell Survival; Coloring Agents; Dose-Response Relationship, Drug; Fluorescent Antibody Technique; Indicators and Reagents; Leukemia; Liver; Male; Membrane Proteins; Mice; Mice, Inbred BALB C; Neoplasm Transplantation; Spleen; Sulfides; Tetrazolium Salts; Thiazoles

2009
Reversal of mdr1-mediated multidrug resistance in human leukemia cells by a new spin-labeled derivative of podophyllotoxin.
    Die Pharmazie, 2010, Volume: 65, Issue:2

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; ATP Binding Cassette Transporter, Subfamily B; ATP Binding Cassette Transporter, Subfamily B, Member 1; Blotting, Western; Cell Division; Cell Line, Tumor; DNA Fragmentation; DNA, Neoplasm; Down-Regulation; Drug Resistance, Neoplasm; Electrophoresis, Agar Gel; Flow Cytometry; G2 Phase; Humans; K562 Cells; Leukemia; Podophyllotoxin; Spin Labels; Tetrazolium Salts; Thiazoles

2010
Inhibition of JAK-STAT signaling by TG101348: a novel mechanism for inhibition of KITD816V-dependent growth in mast cell leukemia cells.
    Leukemia, 2010, Volume: 24, Issue:7

    Topics: Cell Proliferation; Cells, Cultured; Dasatinib; Drug Synergism; Humans; Janus Kinase 2; Leukemia; Mast Cells; Mutation; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-kit; Pyrimidines; Pyrrolidines; Signal Transduction; STAT5 Transcription Factor; Sulfonamides; Thiazoles

2010
Synthesis and identification of a new class of antileukemic agents containing 2-(arylcarboxamide)-(S)-6-amino-4,5,6,7-tetrahydrobenzo[d]thiazole.
    European journal of medicinal chemistry, 2010, Volume: 45, Issue:11

    Topics: Cell Line, Tumor; Humans; Leukemia; Magnetic Resonance Spectroscopy; Spectrometry, Mass, Electrospray Ionization; Spectrophotometry, Infrared; Structure-Activity Relationship; Thiazoles

2010
Hybrid compounds as new Bcr/Abl inhibitors.
    Bioorganic & medicinal chemistry letters, 2011, Apr-01, Volume: 21, Issue:7

    Topics: Cell Line, Tumor; Drug Screening Assays, Antitumor; Fusion Proteins, bcr-abl; Humans; Leukemia; Models, Molecular; Structure-Activity Relationship; Thiazoles

2011
Synthesis and biological activities of 2-amino-thiazole-5-carboxylic acid phenylamide derivatives.
    Archiv der Pharmazie, 2011, Volume: 344, Issue:7

    Topics: Amides; Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Combinatorial Chemistry Techniques; Dasatinib; Female; HT29 Cells; Humans; Inhibitory Concentration 50; Leukemia; Pyrimidines; Structure-Activity Relationship; Thiazoles

2011
Expansion of highly differentiated CD8+ T-cells or NK-cells in patients treated with dasatinib is associated with cytomegalovirus reactivation.
    Leukemia, 2011, Volume: 25, Issue:10

    Topics: Adult; Aged; Apoptosis; Base Sequence; CD8-Positive T-Lymphocytes; Cell Differentiation; Cell Division; Cytomegalovirus; Dasatinib; DNA Primers; Female; Flow Cytometry; Humans; Killer Cells, Natural; Leukemia; Male; Middle Aged; Protein Kinase Inhibitors; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Virus Activation

2011
Thiazolyl N-benzyl-substituted acetamide derivatives: synthesis, Src kinase inhibitory and anticancer activities.
    European journal of medicinal chemistry, 2011, Volume: 46, Issue:10

    Topics: Acetamides; Animals; Antineoplastic Agents; Breast Neoplasms; Cell Line, Tumor; Cell Proliferation; Colonic Neoplasms; Female; Humans; Inhibitory Concentration 50; Leukemia; Mice; Morpholines; NIH 3T3 Cells; Protein Kinase Inhibitors; Pyridines; src-Family Kinases; Structure-Activity Relationship; Thiazoles

2011
Src activation plays an important key role in lymphomagenesis induced by FGFR1 fusion kinases.
    Cancer research, 2011, Dec-01, Volume: 71, Issue:23

    Topics: 3T3 Cells; Animals; Cell Death; Cell Growth Processes; Cell Line, Tumor; Cell Transformation, Neoplastic; Cells, Cultured; Dasatinib; DNA-Binding Proteins; Female; Humans; Leukemia; Lymphoma, B-Cell; Lymphoma, T-Cell; Membrane Proteins; Mice; Mice, Inbred BALB C; Oncogene Proteins, Fusion; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-bcr; Pyrimidines; Receptor, Fibroblast Growth Factor, Type 1; Signal Transduction; src-Family Kinases; Thiazoles; Transcription Factors; Translocation, Genetic

2011
Enhancement of natural killer cell effector functions against selected lymphoma and leukemia cell lines by dasatinib.
    International journal of cancer, 2012, Sep-15, Volume: 131, Issue:6

    Topics: Apoptosis; Calcium; Cell Line, Tumor; Cytokines; Cytotoxicity, Immunologic; Dasatinib; GPI-Linked Proteins; Granzymes; Histocompatibility Antigens Class I; HLA-E Antigens; Humans; Killer Cells, Natural; Leukemia; Lymphoma; Lysosomal-Associated Membrane Protein 1; Lysosomal-Associated Membrane Protein 2; Necrosis; NK Cell Lectin-Like Receptor Subfamily K; Protein Kinase Inhibitors; Pyrimidines; Receptors, IgG; Thiazoles

2012
A sharp fluctuation in peripheral blood cells shortly after dasatinib administration.
    International journal of hematology, 2012, Volume: 96, Issue:2

    Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Blood Cells; Blood Platelets; Cell Adhesion Molecules; Dasatinib; Humans; Leukemia; Leukocyte Count; Leukocytes; Middle Aged; Platelet Count; Protein Kinase Inhibitors; Pyrimidines; Thiazoles; Time Factors

2012
Dasatinib inhibits leukaemic cell survival by decreasing PRH/Hhex phosphorylation resulting in increased repression of VEGF signalling genes.
    Leukemia research, 2012, Volume: 36, Issue:11

    Topics: Antineoplastic Agents; Blotting, Western; Cell Line, Tumor; Cell Survival; Dasatinib; Gene Expression Regulation, Neoplastic; Homeodomain Proteins; Humans; Leukemia; Phosphorylation; Polymerase Chain Reaction; Pyrimidines; Signal Transduction; Thiazoles; Transcription Factors; Vascular Endothelial Growth Factor A

2012
Reversal of multidrug resistance-associated protein-mediated daunorubicin resistance by camptothecin.
    Journal of pharmaceutical sciences, 2002, Volume: 91, Issue:8

    Topics: Antibiotics, Antineoplastic; Antineoplastic Agents, Phytogenic; Breast Neoplasms; Camptothecin; Cell Line; Cell Nucleus; Chemokines, CC; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Flow Cytometry; Fluorescent Antibody Technique; Gene Expression Regulation, Neoplastic; Humans; Leukemia; Microscopy, Confocal; Reverse Transcriptase Polymerase Chain Reaction; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2002
Schedule-dependent synergism and antagonism between methotrexate and cytarabine against human leukemia cell lines in vitro.
    Leukemia, 2002, Volume: 16, Issue:9

    Topics: Antineoplastic Combined Chemotherapy Protocols; Cell Cycle; Cytarabine; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Screening Assays, Antitumor; Drug Synergism; Humans; Leukemia; Methotrexate; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2002
The effect of opioid agonists of delta-class DSLET, mu-class DAMGO, kappa-class U-69593 and an opioid antagonist, naloxone, on MTT activity of NALM-1 leukemic cells.
    Biomedicine & pharmacotherapy = Biomedecine & pharmacotherapie, 2002, Volume: 56, Issue:9

    Topics: Benzeneacetamides; Cell Division; Cell Survival; Colorimetry; DNA Fragmentation; Enkephalin, Ala(2)-MePhe(4)-Gly(5)-; Enkephalin, Leucine; Humans; Leukemia; Naloxone; Narcotic Antagonists; Pyrrolidines; Receptors, Opioid, delta; Receptors, Opioid, kappa; Receptors, Opioid, mu; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2002
[Development of MTS/pms colorimetric assay in the proliferation of leukemic cells].
    Zhongguo shi yan xue ye xue za zhi, 2002, Volume: 10, Issue:5

    Topics: Cell Division; Colorimetry; Formazans; HL-60 Cells; Humans; K562 Cells; Leukemia; Methylphenazonium Methosulfate; Tetrazolium Salts; Thiazoles

2002
Organic phenyl arsonic acid compounds with potent antileukemic activity.
    Bioorganic & medicinal chemistry letters, 2003, Feb-10, Volume: 13, Issue:3

    Topics: Antineoplastic Agents; Arsenicals; Cell Lineage; Genes, p53; Humans; Leukemia; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2003
The actin cytoskeleton and cytotoxic T lymphocytes: evidence for multiple roles that could affect granule exocytosis-dependent target cell killing.
    The Journal of physiology, 2003, Mar-15, Volume: 547, Issue:Pt 3

    Topics: Actin Cytoskeleton; Antibodies, Monoclonal; Antineoplastic Agents; Bridged Bicyclo Compounds, Heterocyclic; Calcium; CD3 Complex; Cell Membrane; Cell Movement; Depsipeptides; Exocytosis; Humans; Leukemia; Lymphoma, B-Cell; Membrane Glycoproteins; Peptides, Cyclic; Perforin; Pore Forming Cytotoxic Proteins; Signal Transduction; T-Lymphocytes, Cytotoxic; Thiazoles; Thiazolidines; Tumor Cells, Cultured

2003
DR1-like element in human topoisomerase IIalpha gene involved in enhancement of etoposide-induced apoptosis by PPARgamma ligand.
    Experimental hematology, 2003, Volume: 31, Issue:4

    Topics: Antigens, Neoplasm; Apoptosis; Chromans; DNA Topoisomerases, Type II; DNA-Binding Proteins; Electrophoretic Mobility Shift Assay; Etoposide; Flow Cytometry; Gene Expression; Humans; Jurkat Cells; Leukemia; Ligands; Mutagenesis; Phosphoproteins; Promoter Regions, Genetic; Prostaglandin D2; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoid X Receptors; Thiazoles; Thiazolidinediones; Topoisomerase II Inhibitors; Transcription Factors; Transfection; Troglitazone; Tumor Cells, Cultured

2003
Methionine enkephalin suppresses metabolic activity of a leukemic cell line (NALM-1) and enhances CD10 expression.
    International immunopharmacology, 2003, Volume: 3, Issue:5

    Topics: Cell Line, Tumor; DNA, Complementary; Enkephalin, Methionine; Humans; Leukemia; Neprilysin; Protease Inhibitors; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles; Thiorphan

2003
POTENTIATION OF THE ANTI-LEUKEMIC EFFECTS OF 2-AMINOTHIADIAZOLE BY ISONICOTINAMIDE AND DERIVATIVES.
    Cancer research, 1964, Volume: 24

    Topics: Amides; Animals; Antineoplastic Agents; Isonicotinic Acids; Leukemia; Leukemia L1210; Leukemia, Experimental; Mice; Niacinamide; Pharmacology; Pyridines; Research; Thiadiazoles; Thiazoles

1964
Synthesis and biological activity of N-aryl-2-aminothiazoles: potent pan inhibitors of cyclin-dependent kinases.
    Bioorganic & medicinal chemistry letters, 2004, Jun-07, Volume: 14, Issue:11

    Topics: Animals; Antineoplastic Agents; Cell Line, Tumor; Cell Survival; Cyclin-Dependent Kinases; Enzyme Inhibitors; Inhibitory Concentration 50; Leukemia; Mice; Neoplasms, Experimental; Protein Binding; Structure-Activity Relationship; Thiazoles; Treatment Outcome

2004
Immunocytochemical detection of deoxycytidine kinase in pediatric malignancies in relation to in vitro cytarabine sensitivity.
    Nucleosides, nucleotides & nucleic acids, 2004, Volume: 23, Issue:8-9

    Topics: Antimetabolites, Antineoplastic; Brain; Brain Neoplasms; Cell Line, Tumor; Coloring Agents; Cytarabine; Deoxycytidine Kinase; Drug Resistance, Neoplasm; Humans; Immunohistochemistry; Leukemia; Neoplasms; Retinoblastoma; Tetrazolium Salts; Thiazoles

2004
Antileukemic activity and cellular metabolism of the aryl phosphate derivative of bromo-methoxy zidovudine (compound WHI-07).
    Arzneimittel-Forschung, 2005, Volume: 55, Issue:1

    Topics: Animals; Antimetabolites, Antineoplastic; Biotransformation; Carboxylic Ester Hydrolases; Cell Division; Cell Line, Tumor; Cell Survival; Cholinesterase Inhibitors; Dideoxynucleotides; Drug Resistance, Multiple; Embryo, Nonmammalian; Glutathione; Humans; Leukemia; Nucleosides; Paraoxon; Rhodamine 123; Subcellular Fractions; Tetrazolium Salts; Thiazoles; Thymidine Monophosphate; Tumor Stem Cell Assay; Zebrafish; Zidovudine

2005
Anti-proliferative and anti-leukemic activity of DDE46 (compound WHI-07), a novel bromomethoxylated arylphosphate derivative of zidovudine, and related compounds. Studies using human acute lymphoblastic leukemia cells and the zebrafish model.
    Arzneimittel-Forschung, 2005, Volume: 55, Issue:2

    Topics: Animals; Antineoplastic Agents; Apoptosis; Caspase Inhibitors; Cell Proliferation; Dideoxynucleotides; Drug Screening Assays, Antitumor; Humans; Jurkat Cells; Leukemia; Magnetic Resonance Spectroscopy; Nephelometry and Turbidimetry; Prodrugs; Tetrazolium Salts; Thiazoles; Thymidine Monophosphate; Tubulin; Zebrafish; Zidovudine

2005
Bovine lactoferricin selectively induces apoptosis in human leukemia and carcinoma cell lines.
    Molecular cancer therapeutics, 2005, Volume: 4, Issue:4

    Topics: Animals; Annexin A5; Anti-Bacterial Agents; Antioxidants; Apoptosis; Carcinoma; Caspase 2; Caspase 3; Caspase 9; Caspases; Cattle; Cell Line, Tumor; Cell Survival; DNA Fragmentation; Dose-Response Relationship, Drug; Endothelial Cells; Enzyme Activation; Enzyme Inhibitors; Fibroblasts; Humans; Immunoblotting; Jurkat Cells; Lactoferrin; Leukemia; Lymphocytes; Membrane Potentials; Microscopy, Electron; Mitochondria; Oligopeptides; Phosphatidylserines; Reactive Oxygen Species; Tetrazolium Salts; Thiazoles; Time Factors

2005
Actin cytoskeleton disassembly affects conductive properties of stretch-activated cation channels in leukaemia cells.
    Biochimica et biophysica acta, 2005, May-15, Volume: 1669, Issue:1

    Topics: Actins; Bridged Bicyclo Compounds, Heterocyclic; Cytochalasin D; Cytoskeleton; Humans; Ion Channels; K562 Cells; Leukemia; Microtubules; Thiazoles; Thiazolidines

2005
Potent inhibition of carcinogen-bioactivating cytochrome P450 1B1 by the p53 inhibitor pifithrin alpha.
    Carcinogenesis, 2006, Volume: 27, Issue:3

    Topics: Apoptosis; Aryl Hydrocarbon Hydroxylases; Benzo(a)pyrene; Benzothiazoles; Breast Neoplasms; Carcinogens; Cytochrome P-450 CYP1A1; Cytochrome P-450 CYP1A2; Cytochrome P-450 CYP1B1; Humans; Leukemia; Macrophages; Microsomes, Liver; Protein Isoforms; Thiazoles; Toluene; Tumor Cells, Cultured; Tumor Suppressor Protein p53

2006
Induction of apoptosis in leukemia cell lines by Linum persicum and Euphorbia cheiradenia.
    Journal of cancer research and clinical oncology, 2006, Volume: 132, Issue:7

    Topics: Anticarcinogenic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Colorimetry; Coloring Agents; DNA Fragmentation; Dose-Response Relationship, Drug; Euphorbia; Flax; Flow Cytometry; HeLa Cells; Humans; Jurkat Cells; K562 Cells; Leukemia; Phytotherapy; Plant Extracts; Tetrazolium Salts; Thiazoles

2006
Inhibitory effect of curcumin on WT1 gene expression in patient leukemic cells.
    Archives of pharmacal research, 2006, Volume: 29, Issue:1

    Topics: Adolescent; Antineoplastic Agents; Cell Line, Tumor; Child; Child, Preschool; Curcumin; Electrophoresis, Polyacrylamide Gel; Female; Gene Expression Regulation, Neoplastic; Genes, Wilms Tumor; Humans; Infant; K562 Cells; Leukemia; Male; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrazolium Salts; Thiazoles

2006
Mortalin-based cytoplasmic sequestration of p53 in a nonmammalian cancer model.
    The American journal of pathology, 2006, Volume: 168, Issue:5

    Topics: Animals; Cytosol; Disease Models, Animal; Hemocytes; HSP70 Heat-Shock Proteins; Immunohistochemistry; Immunoprecipitation; Leukemia; Molecular Sequence Data; Mya; Neoplasms; Pyridines; Subcellular Fractions; Thiazoles; Tumor Suppressor Protein p53

2006
Synthesis, antimycobacterial and antitumor activities of new (1,1-dioxido-3-oxo-1,2-benzisothiazol-2(3H)-yl)methyl N,N-disubstituted dithiocarbamate/O-alkyldithiocarbonate derivatives.
    Bioorganic & medicinal chemistry, 2006, Dec-01, Volume: 14, Issue:23

    Topics: Anti-Bacterial Agents; Antineoplastic Agents; Carbonates; Carboxylic Acids; Carcinoma, Non-Small-Cell Lung; Cell Line, Tumor; Drug Screening Assays, Antitumor; Female; Humans; Inhibitory Concentration 50; Leukemia; Male; Microbial Sensitivity Tests; Mycobacterium tuberculosis; Ovarian Neoplasms; Saccharin; Structure-Activity Relationship; Thiazoles; Thiocarbamates

2006
Cytotoxic effects of leaf, stem and root extracts of Nerium oleander on leukemia cell lines and role of the p-glycoprotein in this effect.
    Journal of experimental therapeutics & oncology, 2006, Volume: 6, Issue:1

    Topics: ATP Binding Cassette Transporter, Subfamily B, Member 1; Cardenolides; Cell Line, Tumor; Dose-Response Relationship, Drug; HL-60 Cells; Humans; K562 Cells; Leukemia; Nerium; Phytotherapy; Plant Extracts; Plant Leaves; Plant Roots; Plant Stems; Tetrazolium Salts; Thiazoles

2006
Expression of multidrug resistance (MDR) proteins and in vitro drug resistance in acute leukemias.
    Hematology (Amsterdam, Netherlands), 2007, Volume: 12, Issue:1

    Topics: Acute Disease; Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Cell Survival; Child; Child, Preschool; Coloring Agents; Cytarabine; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Infant; Inhibitory Concentration 50; Leukemia; Leukemia, Myeloid; Male; Methylphenazonium Methosulfate; Middle Aged; Neoplasm Proteins; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Recurrence; Staining and Labeling; Tetrazolium Salts; Thiazoles; Treatment Outcome; Tumor Cells, Cultured

2007
The effect of the polyadenylation inhibitor cordycepin on human Molt-4 and Daudi leukaemia and lymphoma cell lines.
    Cancer chemotherapy and pharmacology, 2008, Volume: 61, Issue:4

    Topics: Antineoplastic Agents; Blotting, Western; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Deoxyadenosines; DNA Fragmentation; Flow Cytometry; Fluorescent Dyes; Humans; Image Processing, Computer-Assisted; Indoles; Leukemia; Lymphoma; Membrane Potentials; Mitochondria; Necrosis; Polynucleotide Adenylyltransferase; Tetrazolium Salts; Thiazoles

2008
Cancer agents show first-line potential.
    JAMA, 2007, Jul-25, Volume: 298, Issue:4

    Topics: Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Arsenic Trioxide; Arsenicals; Bevacizumab; Dasatinib; Humans; Kidney Neoplasms; Leukemia; Oxides; Pyrimidines; Thiazoles

2007
Effective treatment of leukemic cell lines with wt1 siRNA.
    Leukemia, 2007, Volume: 21, Issue:10

    Topics: Apoptosis; Cell Line, Tumor; Cell Proliferation; Flow Cytometry; Genes, Wilms Tumor; Genetic Therapy; HL-60 Cells; Humans; K562 Cells; Leukemia; Proto-Oncogene Proteins c-bcl-2; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Time Factors; Transfection

2007
Cytotoxic effects of treosulfan and busulfan against leukemic cells of pediatric patients.
    Cancer chemotherapy and pharmacology, 2008, Volume: 62, Issue:5

    Topics: Antineoplastic Agents; Antineoplastic Agents, Alkylating; Apoptosis; Busulfan; Caspase 3; Cell Line, Tumor; Child; Dose-Response Relationship, Drug; Flow Cytometry; Humans; Killer Cells, Natural; Leukemia; Stem Cells; T-Lymphocytes; Tetrazolium Salts; Thiazoles; Vidarabine

2008
Antisense RNA of survivin gene inhibits the proliferation of leukemia cells and sensitizes leukemia cell line to taxol-induced apoptosis.
    Journal of Huazhong University of Science and Technology. Medical sciences = Hua zhong ke ji da xue xue bao. Yi xue Ying De wen ban = Huazhong keji daxue xuebao. Yixue Yingdewen ban, 2008, Volume: 28, Issue:1

    Topics: Antineoplastic Agents, Phytogenic; Apoptosis; Cell Line, Tumor; Cell Nucleus; Cell Proliferation; Flow Cytometry; HL-60 Cells; Humans; Inhibitor of Apoptosis Proteins; Inhibitory Concentration 50; Leukemia; Microtubule-Associated Proteins; Neoplasm Proteins; Paclitaxel; RNA, Antisense; Survivin; Tetrazolium Salts; Thiazoles

2008
Drugs affecting the hormonal receptors of normal and leukaemic peripheral leucocytes.
    International journal of tissue reactions, 1984, Volume: 6, Issue:5

    Topics: Estradiol; Estriol; Flurbiprofen; Humans; Hydrocortisone; In Vitro Techniques; Leukemia; Leukocytes; Receptors, Steroid; Testosterone; Theophylline; Thiazoles; Thiazolidines

1984
Cytostatic and cytotoxic activity of sex steroids against human leukemia cell lines.
    Cancer letters, 1994, Jan-30, Volume: 76, Issue:2-3

    Topics: Androgens; Antineoplastic Agents; Diethylstilbestrol; Estrogens; Glucocorticoids; Gonadal Steroid Hormones; Humans; Leukemia; Neoplasms, Hormone-Dependent; Progesterone; Steroids; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1994
In vitro cytotoxicity and immunomodulating property of Rhaphidophora korthalsii.
    Journal of ethnopharmacology, 1996, Volume: 52, Issue:1

    Topics: Adenocarcinoma; Adjuvants, Immunologic; Animals; Antineoplastic Agents, Phytogenic; Carcinoma, Squamous Cell; Cell Division; Colonic Neoplasms; Coloring Agents; Concanavalin A; Dose-Response Relationship, Drug; Female; Humans; Leukemia; Leukemia P388; Lymphocyte Activation; Mice; Mice, Inbred BALB C; Nasopharyngeal Neoplasms; Plant Extracts; Plant Lectins; Plants, Medicinal; Spleen; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Water

1996
Apoptosis and resistance to daunorubicin in human leukemic cells.
    Leukemia, 1997, Volume: 11, Issue:7

    Topics: Antibiotics, Antineoplastic; Apoptosis; Daunorubicin; Drug Resistance; Humans; Leukemia; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1997
[Improved MTT colorimetric assay for NKC activity].
    Hua xi yi ke da xue xue bao = Journal of West China University of Medical Sciences = Huaxi yike daxue xuebao, 1996, Volume: 27, Issue:2

    Topics: Adult; Colorimetry; Coloring Agents; Cytotoxicity, Immunologic; Humans; Killer Cells, Natural; Leukemia; Tetrazolium Salts; Thiazoles

1996
N-glycosylation of glucose transporter-1 (Glut-1) is associated with increased transporter affinity for glucose in human leukemic cells.
    Leukemia research, 1999, Volume: 23, Issue:4

    Topics: 3-O-Methylglucose; Cell Division; Deoxyglucose; Glucose; Glucose Transporter Type 1; Glycosylation; HL-60 Cells; Humans; K562 Cells; Leukemia; Monosaccharide Transport Proteins; Tetrazolium Salts; Thiazoles; Tunicamycin; U937 Cells

1999
Bovine seminal ribonuclease attached to nanoparticles made of polylactic acid kills leukemia and lymphoma cell lines in vitro.
    Anti-cancer drugs, 2000, Volume: 11, Issue:5

    Topics: Animals; Antineoplastic Agents; Apoptosis; Cattle; Cell Division; Dose-Response Relationship, Drug; Drug Carriers; Endoribonucleases; Fibroblasts; Humans; Lactic Acid; Leukemia; Lymphoma; Male; Mice; Mice, Inbred ICR; Microspheres; Polyesters; Polymers; Spermatozoa; Testis; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2000
Apoptotic effects of thiazolobenzimidazole derivatives on sensitive and multidrug resistant leukaemic cells.
    European journal of cancer (Oxford, England : 1990), 2001, Volume: 37, Issue:1

    Topics: Antineoplastic Agents; Apoptosis; Benzimidazoles; Caspase Inhibitors; Cell Cycle; Drug Resistance, Multiple; Drug Resistance, Neoplasm; fas Receptor; HL-60 Cells; Humans; Leukemia; Thiazoles

2001
Abietane diterpenoids from Coleus xanthanthus.
    Journal of natural products, 2002, Volume: 65, Issue:5

    Topics: Antineoplastic Agents, Phytogenic; Diterpenes; Drug Screening Assays, Antitumor; Drugs, Chinese Herbal; Humans; Lamiaceae; Leukemia; Molecular Conformation; Molecular Structure; Nuclear Magnetic Resonance, Biomolecular; Plants, Medicinal; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

2002
In vitro chemosensitivity of lymphoblasts at relapse in childhood leukemia using the MTT assay.
    International journal of hematology, 1991, Volume: 54, Issue:3

    Topics: Acute Disease; Antineoplastic Agents; Child; Colorimetry; Drug Resistance; Drug Screening Assays, Antitumor; Humans; Leukemia; Neoplasm Recurrence, Local; Neoplastic Stem Cells; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1991
Chemosensitivity testing of fresh human leukemia cells using both a dye exclusion assay and a tetrazolium dye (MTT) assay.
    Leukemia research, 1990, Volume: 14, Issue:5

    Topics: Antineoplastic Agents; Cell Survival; Coloring Agents; Drug Screening Assays, Antitumor; Humans; Leukemia; Predictive Value of Tests; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1990
The influence of thyroid hormones on colony growth of peripheral CFU-GM from normal and leukemic subjects.
    Tumori, 1988, Oct-31, Volume: 74, Issue:5

    Topics: Cells, Cultured; Flurbiprofen; Granulocytes; Hematopoietic Stem Cells; Humans; Leukemia; Monocytes; Thiazoles; Thiazolidines; Thyroid Hormones

1988
Comparison of in vitro activity of cytotoxic drugs towards human carcinoma and leukaemia cell lines.
    European journal of cancer & clinical oncology, 1986, Volume: 22, Issue:6

    Topics: Aminoacridines; Amsacrine; Antineoplastic Agents; Cell Count; Cell Line; Cell Survival; Colonic Neoplasms; Humans; Kinetics; Leukemia; Tetrazolium Salts; Thiazoles

1986
Potential anticancer agents. Nitrogen mustards of aminophenylthiazoles.
    Journal of medicinal chemistry, 1971, Volume: 14, Issue:9

    Topics: Animals; Antineoplastic Agents; Benzene Derivatives; Benzyl Compounds; Carcinoma 256, Walker; Chlorine; Ethers; Ethylamines; Leukemia; Leukemia L1210; Nitrogen Mustard Compounds; Structure-Activity Relationship; Thiazoles; Toluene

1971
Imidothiazoles.
    Journal of medicinal chemistry, 1968, Volume: 11, Issue:1

    Topics: Acids; Adenocarcinoma; Animals; Carcinoma; Culture Techniques; Imides; Leukemia; Leukemia L1210; Melanoma; Methods; Mice; Sarcoma 180; Thiazoles

1968