Page last updated: 2024-08-21

thiazoles and Leukemia, Myeloid

thiazoles has been researched along with Leukemia, Myeloid in 30 studies

Research

Studies (30)

TimeframeStudies, this research(%)All Research%
pre-19902 (6.67)18.7374
1990's12 (40.00)18.2507
2000's11 (36.67)29.6817
2010's5 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Congleton, J; MacDonald, R; Malavasi, F; Shen, M; Yen, A1
Albitar, M; Bornmann, W; Estrov, Z; Faderl, S; Harris, D; Hazan-Halevy, I; Kantarjian, HM; Liu, Z; Maxwell, D; Pal, A; Peng, Z; Van, Q1
Tojo, A1
Arceci, R; Blanchard, EG; Cayre, YE; Corey, SJ; Futami, M; Guerrouahen, BS; Kanerva, J; Kornblau, SM; Lee, FY; Nwawka, K; Robinson, LJ; Vaklavas, C; Whichard, ZL; Wieder, E1
Gao, LP; Liu, JJ; Liu, Q; Wei, HL; Yi, J; Zhao, HS1
Congleton, J; MacDonald, R; Yen, A1
Blum, W; Caligiuri, M; Croce, CM; Garzon, R; Kauffman, M; Klisovic, R; Marcucci, G; Na, C; Ranganathan, P; Santhanam, R; Shacham, S; Walker, A; Yu, X1
Kato, Y; Kawaguchi, M; Koshimura, K; Murakami, Y; Tanaka, J; Tsumori, M1
Eppinger, E; Meinhardt, G; Schmidmaier, R1
Creutzig, U; Hählen, K; Harbott, J; Huismans, DR; Kaspers, GJ; Pieters, R; Slater, RM; Veerman, AJ; Zimmermann, M; Zwaan, CM1
Chan, AS; Chen, J; Cheng, CH; Cheng, GY; Chui, CH; Kok, SH; Lam, WS; Lau, FY; Tang, JC; Tang, WK; Wong, RS1
Bold, G; Furet, P; Guagnano, V; Meyer, T; Roesel, J1
Cheng, YC; Huang, MJ; Lin, S; Liu, CR; Liu, HE1
Kim, DK; Kim, JH; Lee, HJ; Yoon, MJ1
Ainoon, O; Cheong, SK; Fazlina, N; Hamidah, H; Hamidah, NH; Jamal, R; Maha, A; Zarina, AL; Zulkifli, SZ1
Efferth, T; Fabry, U; Glatte, P; Osieka, R1
Beelen, RH; Broekhoven, MG; Langenhuijsen, MM; Ossenkoppele, GJ; van de Loosdrecht, AA1
Yu, D; Yu, LL1
Elgie, AW; Sargent, JM; Taylor, CG; Williamson, C1
Borg, AG; Burgess, R; Fisher, A; Grey, M; Wood, P; Yin, JA1
Alton, P; Elgie, AW; Noordhuis, P; Peters, GJ; Sargent, JM; Taylor, CG; Williamson, CJ1
Kiriyama, Y; Nochi, H; Sakurada, Y; Sugimura, A; Tamoto, K; Tokumitsu, Y; Tsuchiya, H; Ui, M1
Asou, H; Elstner, E; Kamada, N; Koeffler, HP; Kubota, T; Verbeek, W; Williamson, E1
Bagchi, D; Bagchi, M; Stohs, SJ1
Kass, L1
Abe, T; Ohno, M1
Glasebrook, AL; Hatfield, SM; Rodgers, GH; Roehm, NW1
Bazill, GW; Dexter, TM1
Lalezari, I; Schwartz, EL1
Gutsche, W; Jungstand, W; Wohlrabe, K1

Reviews

1 review(s) available for thiazoles and Leukemia, Myeloid

ArticleYear
[Clinical use of tyrosine kinase inhibitors for treatment of myeloid leukemias].
    Nihon rinsho. Japanese journal of clinical medicine, 2009, Volume: 67, Issue:10

    Topics: Antineoplastic Agents; Benzamides; Clinical Trials as Topic; Dasatinib; Drug Design; fms-Like Tyrosine Kinase 3; Humans; Imatinib Mesylate; Leukemia, Myeloid; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Thiazoles

2009

Other Studies

29 other study(ies) available for thiazoles and Leukemia, Myeloid

ArticleYear
Phosphorylation of c-Cbl and p85 PI3K driven by all-trans retinoic acid and CD38 depends on Lyn kinase activity.
    Cellular signalling, 2014, Volume: 26, Issue:7

    Topics: Adaptor Proteins, Signal Transducing; ADP-ribosyl Cyclase 1; Antineoplastic Agents; Cell Differentiation; Cell Line, Tumor; Class Ia Phosphatidylinositol 3-Kinase; Dasatinib; HL-60 Cells; Humans; Leukemia, Myeloid; Membrane Glycoproteins; Phosphatidylinositol 3-Kinases; Phosphoproteins; Phosphorylation; Protein Binding; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-cbl; Proto-Oncogene Proteins c-vav; Pyrimidines; src-Family Kinases; Thiazoles; Tretinoin

2014
Kit inhibitor APcK110 induces apoptosis and inhibits proliferation of acute myeloid leukemia cells.
    Cancer research, 2009, May-01, Volume: 69, Issue:9

    Topics: Acute Disease; Apoptosis; Benzamides; Caspases; Cell Growth Processes; Cell Survival; Dasatinib; Drug Screening Assays, Antitumor; Humans; Imatinib Mesylate; Leukemia, Myeloid; Mutation; Oncogene Protein v-akt; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-kit; Pyrazoles; Pyridines; Pyrimidines; STAT3 Transcription Factor; Stem Cell Factor; Thiazoles

2009
Dasatinib inhibits the growth of molecularly heterogeneous myeloid leukemias.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2010, Feb-15, Volume: 16, Issue:4

    Topics: Cell Cycle; Cell Line, Tumor; Cell Proliferation; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Dasatinib; Humans; Leukemia, Myeloid; Proto-Oncogene Proteins c-kit; Pyrimidines; src-Family Kinases; Thiazoles

2010
Inhibition of thioredoxin reductase by auranofin induces apoptosis in adriamycin-resistant human K562 chronic myeloid leukemia cells.
    Die Pharmazie, 2011, Volume: 66, Issue:6

    Topics: Antibiotics, Antineoplastic; Antirheumatic Agents; Apoptosis; Auranofin; Caspase 3; Cell Survival; Coloring Agents; Doxorubicin; Drug Resistance, Neoplasm; Enzyme Inhibitors; Flow Cytometry; Humans; K562 Cells; Leukemia, Myeloid; Tetrazolium Salts; Thiazoles; Thioredoxin-Disulfide Reductase

2011
Src inhibitors, PP2 and dasatinib, increase retinoic acid-induced association of Lyn and c-Raf (S259) and enhance MAPK-dependent differentiation of myeloid leukemia cells.
    Leukemia, 2012, Volume: 26, Issue:6

    Topics: Antineoplastic Agents; Blotting, Western; Cell Cycle; Cell Differentiation; Dasatinib; Extracellular Signal-Regulated MAP Kinases; Flow Cytometry; Humans; Immunoprecipitation; Leukemia, Myeloid; Mitogen-Activated Protein Kinases; Phosphorylation; Protein Kinase Inhibitors; Protein Kinases; Proto-Oncogene Proteins c-raf; Pyrimidines; RNA, Small Interfering; Signal Transduction; src-Family Kinases; Thiazoles; Tretinoin; Tumor Cells, Cultured

2012
Preclinical activity of a novel CRM1 inhibitor in acute myeloid leukemia.
    Blood, 2012, Aug-30, Volume: 120, Issue:9

    Topics: Acrylamides; Acrylates; Acute Disease; Adult; Aged; Aged, 80 and over; Animals; Antineoplastic Agents; Apoptosis; Blotting, Western; Cell Differentiation; Cell Line, Tumor; Cell Nucleus; Cell Proliferation; Drug Evaluation, Preclinical; Exportin 1 Protein; Female; fms-Like Tyrosine Kinase 3; Humans; Kaplan-Meier Estimate; Karyopherins; Leukemia, Myeloid; Mice; Mice, Inbred NOD; Mice, SCID; Middle Aged; Receptors, Cytoplasmic and Nuclear; Thiazoles; Triazoles; Tumor Suppressor Protein p53; Xenograft Model Antitumor Assays; Young Adult

2012
Cytotoxic effect of nitric oxide on human hematological malignant cells.
    Acta biochimica Polonica, 2002, Volume: 49, Issue:1

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Agents; Female; Humans; Leukemia, Myeloid; Lymphoma; Male; Nitric Oxide; Nitric Oxide Donors; Nitroprusside; Tetrazolium Salts; Thiazoles

2002
Effect of novel modulators of protein kinase C activity upon chemotherapy-induced differentiation and apoptosis in myeloid leukemic cells.
    Anti-cancer drugs, 2002, Volume: 13, Issue:7

    Topics: Antineoplastic Agents; Apoptosis; CD11c Antigen; CD4 Antigens; Cell Cycle; Cell Differentiation; Diacylglycerol Kinase; Enzyme Activators; Enzyme Inhibitors; Farnesol; Flow Cytometry; Genes, fos; Genes, jun; Humans; Immunoblotting; Isoenzymes; Leukemia, Myeloid; Naphthalenes; Oncogene Protein p21(ras); Piperidines; Protein Kinase C; Pyrimidinones; Quinazolines; Quinazolinones; Sulfonamides; Thiazoles; Triazoles; Tumor Cells, Cultured

2002
Cellular drug resistance in childhood acute myeloid leukemia is related to chromosomal abnormalities.
    Blood, 2002, Nov-01, Volume: 100, Issue:9

    Topics: Acute Disease; Adolescent; Antibiotics, Antineoplastic; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Child; Child, Preschool; Chromosome Aberrations; Chromosome Inversion; Chromosomes, Human; Cladribine; Cytarabine; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Etoposide; Female; Humans; Infant; Leukemia, Myeloid; Male; Neoplastic Stem Cells; Recurrence; Remission Induction; Tetrazolium Salts; Thiazoles; Translocation, Genetic; Trisomy

2002
Mechanistic insight into a novel synthetic cantharidin analogue in a leukaemia model.
    International journal of molecular medicine, 2006, Volume: 18, Issue:2

    Topics: Adult; Animals; Antineoplastic Agents; Bone Marrow Cells; Cantharidin; Cell Cycle; Cell Line, Tumor; Cells, Cultured; Enzyme Inhibitors; Female; Humans; In Situ Nick-End Labeling; Insecta; Leukemia, Myeloid; Male; Mitochondria; Thiazoles

2006
Aromatic interactions with phenylalanine 691 and cysteine 828: a concept for FMS-like tyrosine kinase-3 inhibition. Application to the discovery of a new class of potential antileukemia agents.
    Journal of medicinal chemistry, 2006, Jul-27, Volume: 49, Issue:15

    Topics: Acute Disease; Adenosine Triphosphate; Antineoplastic Agents; Binding Sites; Cell Line, Tumor; Cysteine; fms-Like Tyrosine Kinase 3; Humans; Leukemia, Myeloid; Models, Molecular; Mutation; Phenylalanine; Protein Structure, Tertiary; Thiazoles

2006
A small-molecule c-Myc inhibitor, 10058-F4, induces cell-cycle arrest, apoptosis, and myeloid differentiation of human acute myeloid leukemia.
    Experimental hematology, 2006, Volume: 34, Issue:11

    Topics: Acute Disease; Antineoplastic Agents; Apoptosis; Basic-Leucine Zipper Transcription Factors; Cell Cycle; Cell Differentiation; Cell Line, Tumor; Cell Proliferation; Cyclin-Dependent Kinase Inhibitor p21; Cyclin-Dependent Kinase Inhibitor p27; Dimerization; Down-Regulation; Drug Screening Assays, Antitumor; G1 Phase; HL-60 Cells; Humans; Leukemia, Myeloid; Myeloid Cells; Proto-Oncogene Proteins c-myc; Resting Phase, Cell Cycle; Structure-Activity Relationship; Thiazoles; U937 Cells; Up-Regulation

2006
Extracellular ATP induces apoptotic signaling in human monocyte leukemic cells, HL-60 and F-36P.
    Archives of pharmacal research, 2006, Volume: 29, Issue:11

    Topics: Adenosine Triphosphate; Annexins; Apoptosis; Calcium; Caspases; Cell Cycle; Cell Line, Tumor; Cell Proliferation; Colorimetry; Flow Cytometry; HL-60 Cells; Humans; Leukemia, Myeloid; Receptors, Purinergic P2; Receptors, Purinergic P2Y2; Signal Transduction; Tetrazolium Salts; Thiazoles

2006
Expression of multidrug resistance (MDR) proteins and in vitro drug resistance in acute leukemias.
    Hematology (Amsterdam, Netherlands), 2007, Volume: 12, Issue:1

    Topics: Acute Disease; Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B; Cell Survival; Child; Child, Preschool; Coloring Agents; Cytarabine; Daunorubicin; Drug Resistance, Multiple; Drug Resistance, Neoplasm; Female; Humans; Infant; Inhibitory Concentration 50; Leukemia; Leukemia, Myeloid; Male; Methylphenazonium Methosulfate; Middle Aged; Neoplasm Proteins; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Recurrence; Staining and Labeling; Tetrazolium Salts; Thiazoles; Treatment Outcome; Tumor Cells, Cultured

2007
Expression of apoptosis-related oncoproteins and modulation of apoptosis by caffeine in human leukemic cells.
    Journal of cancer research and clinical oncology, 1995, Volume: 121, Issue:11

    Topics: Apoptosis; Caffeine; Carboplatin; Cluster Analysis; Coloring Agents; Daunorubicin; Drug Resistance, Neoplasm; Flow Cytometry; G2 Phase; Gamma Rays; Gene Expression Regulation, Leukemic; Glutathione; GTP-Binding Proteins; HL-60 Cells; Humans; Immunohistochemistry; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Leukemia, Myeloid, Acute; Leukemia, Promyelocytic, Acute; Lymphoma, Non-Hodgkin; Multivariate Analysis; Oncogene Proteins v-fos; Proto-Oncogene Proteins; Proto-Oncogene Proteins c-bcl-2; Radiation Tolerance; ras Proteins; S Phase; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Tumor Suppressor Protein p53

1995
A tetrazolium-based colorimetric MTT assay to quantitate human monocyte mediated cytotoxicity against leukemic cells from cell lines and patients with acute myeloid leukemia.
    Journal of immunological methods, 1994, Sep-14, Volume: 174, Issue:1-2

    Topics: Acute Disease; Colorimetry; Cytotoxicity, Immunologic; Humans; Immunity, Cellular; Immunologic Techniques; In Vitro Techniques; Leukemia, Myeloid; Monocytes; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1994
Optimal conditions of chemotherapeutic sensitivity in K562 cell line using tetrazolium dye assay.
    Zhongguo yao li xue bao = Acta pharmacologica Sinica, 1993, Volume: 14, Issue:2

    Topics: Antineoplastic Agents; Coloring Agents; Drug Screening Assays, Antitumor; Humans; Leukemia, Myeloid; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1993
An in vitro study of blast cell metabolism in acute myeloid leukaemia using the MTT assay.
    Leukemia research, 1996, Volume: 20, Issue:5

    Topics: Acute Disease; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Division; Cell Size; Drug Resistance, Multiple; Drug Screening Assays, Antitumor; Humans; Individuality; Leukemia, Myeloid; Reproducibility of Results; Tetrazolium Salts; Thiazoles

1996
Effect on cell kill of addition of multidrug resistance modifiers cyclosporin A and PSC 833 to cytotoxic agents in acute myeloid leukaemia.
    Leukemia research, 1997, Volume: 21, Issue:9

    Topics: Acute Disease; Adolescent; Adult; Aged; Antibiotics, Antineoplastic; ATP Binding Cassette Transporter, Subfamily B, Member 1; Biological Transport; Cell Survival; Coloring Agents; Cyclosporine; Cyclosporins; Cytarabine; Daunorubicin; Drug Resistance, Neoplasm; Drug Synergism; Etoposide; Female; Humans; Idarubicin; Leukemia, Myeloid; Male; Middle Aged; Mitoxantrone; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1997
Modulation of resistance to ara-C by bryostatin in fresh blast cells from patients with AML.
    Leukemia research, 1998, Volume: 22, Issue:4

    Topics: Acute Disease; Antineoplastic Agents; Arabinofuranosylcytosine Triphosphate; Bryostatins; Cell Death; Cytarabine; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Humans; Lactones; Leukemia, Myeloid; Leukocytes, Mononuclear; Macrolides; Tetrazolium Salts; Thiazoles

1998
Troglitazone suppresses cell growth of myeloid leukemia cell lines by induction of p21WAF1/CIP1 cyclin-dependent kinase inhibitor.
    Biochemical and biophysical research communications, 1999, Aug-11, Volume: 261, Issue:3

    Topics: Antineoplastic Agents; Cell Cycle; Cell Division; Chromans; Cyclin-Dependent Kinase Inhibitor p21; Cyclins; DNA; Enzyme Inhibitors; Flow Cytometry; Gene Expression; Humans; Hypereosinophilic Syndrome; Leukemia, Myeloid; Leukemia, Myelomonocytic, Acute; Leukemia, Myelomonocytic, Chronic; RNA, Messenger; Thiazoles; Thiazolidinediones; Troglitazone; Tumor Cells, Cultured

1999
Growth inhibition of myeloid leukemia cells by troglitazone, a ligand for peroxisome proliferator activated receptor gamma, and retinoids.
    International journal of oncology, 1999, Volume: 15, Issue:5

    Topics: Alitretinoin; Antineoplastic Agents; Antioxidants; Cell Cycle; Cell Differentiation; Cell Division; Chromans; DNA-Binding Proteins; HL-60 Cells; Humans; Leukemia, Myeloid; Receptors, Cytoplasmic and Nuclear; Superoxides; Thiazoles; Thiazolidinediones; Transcription Factors; Tretinoin; Troglitazone; Tumor Cells, Cultured; U937 Cells

1999
Chromium (VI)-induced oxidative stress, apoptotic cell death and modulation of p53 tumor suppressor gene.
    Molecular and cellular biochemistry, 2001, Volume: 222, Issue:1-2

    Topics: Animals; Apoptosis; Carcinogens; Cell Line; Chromium; Cytochrome c Group; DNA Fragmentation; Female; Flow Cytometry; Gene Expression Regulation; Humans; Hydroxyl Radical; K562 Cells; Leukemia, Myeloid; Lipid Peroxidation; Macrophages; Mice; Mice, Inbred C57BL; Mice, Knockout; Microscopy, Confocal; Oxidation-Reduction; Oxidative Stress; Superoxides; Tetrazolium Salts; Thiazoles; Tumor Suppressor Protein p53

2001
Basic blue 54: a new colorant for monocytes.
    Biotechnic & histochemistry : official publication of the Biological Stain Commission, 1992, Volume: 67, Issue:1

    Topics: Azo Compounds; Chromatin; Cytoplasm; Humans; Leukemia, Myelogenous, Chronic, BCR-ABL Positive; Leukemia, Myeloid; Leukemia, Myelomonocytic, Acute; Leukocytes; Monocytes; Neutrophils; Staining and Labeling; Thiazoles

1992
Rapid colorimetric assay for the quantification of leukemia inhibitory factor (LIF) and interleukin-6 (IL-6).
    Journal of immunological methods, 1991, Dec-15, Volume: 145, Issue:1-2

    Topics: Animals; Colorimetry; Growth Inhibitors; Humans; In Vitro Techniques; Interleukin-6; Leukemia Inhibitory Factor; Leukemia, Experimental; Leukemia, Myeloid; Lymphokines; Mice; Oxidation-Reduction; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1991
An improved colorimetric assay for cell proliferation and viability utilizing the tetrazolium salt XTT.
    Journal of immunological methods, 1991, Sep-13, Volume: 142, Issue:2

    Topics: Animals; Cell Division; Cell Survival; Colorimetry; Coloring Agents; Concanavalin A; Dose-Response Relationship, Drug; In Vitro Techniques; Interleukin-2; Interleukin-4; Leukemia, Myeloid; Mast Cells; Methylphenazonium Methosulfate; Mice; Spleen; T-Lymphocytes; Tetrazolium Salts; Thiazoles; Vitamin K

1991
Role of endocytosis in the action of ether lipids on WEHI-3B, HL60, and FDCP-mix A4 cells.
    Cancer research, 1990, Dec-01, Volume: 50, Issue:23

    Topics: Animals; Antineoplastic Agents; Azepines; Cell Survival; Chloroquine; Diltiazem; Drug Synergism; Endocytosis; Furans; Humans; Hydroxyzine; In Vitro Techniques; Leukemia, Myeloid; Mice; Nifedipine; Phospholipid Ethers; Platelet Activating Factor; Pyridines; Quinidine; Quinine; Sodium Fluoride; Thiazoles; Triazoles; Verapamil

1990
Synthesis and antineoplastic activity of 5-aryl-2,3-dihydropyrrolo[2,1-b]thiazole-6,7-dimethanol 6,7-bis(isopropylcarbamates).
    Journal of medicinal chemistry, 1988, Volume: 31, Issue:7

    Topics: Carbamates; Cell Division; Cell Survival; Chemical Phenomena; Chemistry; Colonic Neoplasms; Humans; Leukemia, Myeloid; Neoplasms; Pyrroles; Structure-Activity Relationship; Thiazoles; Tumor Cells, Cultured

1988
[3-step test for screening potential cancerostatics. 1. Screening program and results of the 1st step].
    Arzneimittel-Forschung, 1971, Volume: 21, Issue:3

    Topics: Animals; Antineoplastic Agents; Azo Compounds; Benzimidazoles; Carcinoma, Ehrlich Tumor; Ethers; Hydrazines; Leukemia, Experimental; Leukemia, Myeloid; Mice; Nitrogen Mustard Compounds; Purines; Sarcoma, Experimental; Thiazoles

1971