thiazoles and Gastric Ulcer
thiazoles has been researched along with Gastric Ulcer in 121 studies
Research
Studies (121)
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 49 (40.50) | 18.7374 |
1990's | 33 (27.27) | 18.2507 |
2000's | 22 (18.18) | 29.6817 |
2010's | 14 (11.57) | 24.3611 |
2020's | 3 (2.48) | 2.80 |
Authors
Authors | Studies |
---|---|
Alsharif, KF; Batiha, GE; Beder, NA; Elfadadny, A; Mandour, AS; Ragab, RF; Samir, H | 1 |
Abdelmoez, AAB; Abdu-Allah, HHM; El-Awady, R; El-Shorbagi, AA; Tarazi, H | 1 |
Abd-Allah, WH; Aboregela, AM; El-Behairy, MF; Lan, P; Marzouk, AA; Shaykoon, MSA; Taher, ES | 1 |
Bird, DM; Fitzgerald, G; Guzman, DS; Lair, S; Larrat, S; Summa, NM; Troncy, E | 1 |
Fichna, J; Kordek, R; Mosinska, P; Salaga, M; Storr, M; Timmermans, JP; Zatorski, H; Zielińska, M | 1 |
Alves, D; de Oliveira, RL; Luchese, C; Pinz, MP; Reis, AS; Roehrs, JA; Sacramento, MD; Vogt, AG; Voss, GT; Wilhelm, EA | 1 |
Ansari Lari, M; Eskafian, H; Shojaee Tabrizi, A | 1 |
Farshad, S; Firoozi, MS; Jamshidzadeh, A; Kiany, S; Rahimi, HR; Rasouli, M; Taghavi, AR | 1 |
Cho, CS; Kang, YM; Kim, JH; Kim, SK; Lee, DH; Lee, SK; Lee, ST; Lee, YC; Park, SH; Park, W; Park, YW; Rew, JS; Yoo, WH | 1 |
Abdallah, MA; Amin, MM; Farghaly, TA; Masaret, GS; Muhammad, ZA | 1 |
Alam, MS; Ali, Y; Bano, S; Dhulap, A; Hamid, H; Husain, A; Kharbanda, C | 1 |
Abdel-Moty, SG; Abou-Ghadir, OM; Hussein, MA; Kafafy, AH | 1 |
Baraka, MM; El-Sabbagh, OI; Ibrahim, SM; Kothayer, H | 1 |
Date, AA; Khachane, P; Nagarsenker, MS | 2 |
Baiuomy, AR; Elmegeed, GA; Eskander, EF; Mohareb, RM; William, MG | 1 |
Bawa, S; Chawla, G; Kumar, J; Kumar, U | 1 |
Davis, EG; Kukanich, B; Vander Werf, KA | 1 |
Atilla, P; Balkan, A; Cakar, AN; Caliş, U; Gören, Z; Urgun, H; Uzbay, T | 1 |
Jain, NK; Kulkarni, SK; Singh, A | 1 |
Agarwal, SP; Baboota, S | 1 |
Bekhit, AA; Fahmy, HT | 1 |
Bazela, K; Brzozowski, T; Hahn, EG; Harsch, I; Kania, J; Konturek, PC; Konturek, SJ; Kukharsky, V; Kwiecien, S | 1 |
Dündar, Y; Küpeli, E; Noyanalpan, N; Okçelik, B; Onkol, T; Sahin, MF; Unlü, S; Yeşilada, E | 1 |
Bahekar, RH; Bhusari, KP; Chopade, RS; Khedekar, PB; Rao, AR; Umathe, SN | 1 |
de la Lastra, CA; Herrerías, JM; La Casa, C; Martín, MJ; Motilva, V; Villegas, I | 1 |
Ertan, M; Gökhan, N; Küpeli, E; Tozkoparan, B; Yeşilada, E | 1 |
Abe, M; Iida, H; Inoue, S; Okabe, S; Tanaka, J; Yuda, Y | 1 |
Mishra, DN; Vijaya Kumar, SG | 1 |
El-Fayomi, HM; El-Sadek, ME; Lashine, el-SM; Metwally, KA; Yaseen, SH | 1 |
Hane, M; Hara, S; Naito, Y; Narita, T; Okabe, N; Tani, K; Yamamoto, Y | 1 |
Becker, TL; Gambero, A; Maróstica, M; Pedrazzoli, J | 1 |
Maeno, H; Takagi, T; Takeda, M; Yashima, Y | 1 |
Barbarino, F; Brilinschi, C; Togănel, E | 1 |
Basile, M; Circosta, C; Costa De Pasquale, R; Fenech, G; Occhiuto, F; Previtera, T; Vigorita, MG | 1 |
Ando, K; Nagatomi, H | 1 |
Abignente, E; Berrino, L; de Caprariis, P; Marmo, E; Matera, MG; Sacchi, A | 1 |
Mori, H | 1 |
Abignente, E; Arena, F; De Caprariis, P; Ferreri, C; Giasi, M; Marmo, E; Ottavo, R; Rossi, F | 1 |
Amico-Roxas, M; Caruso, A; Cutuli, V; Di Pietro, E; Modica, M; Russo, F; Santagati, A; Santagati, M | 1 |
Inoue, Y; Ishikawa, H; Katsura, Y; Takasugi, H; Tomishi, T | 1 |
Czajkowski, A; Majka, J; Piotrowski, J; Slomiany, A; Slomiany, BL; Yotsumoto, F | 1 |
Ishikawa, T; Motoyama, Y; Sakai, H; Takasugi, H; Tanaka, A | 1 |
Fenech, G; Forestieri, AM; Giordano, A; Monforte, MT; Previtera, T; Vigorita, MG; Zappala, C | 1 |
Czajkowski, A; Piotrowski, J; Slomiany, A; Slomiany, BL; Yotsumoto, F | 1 |
Dohi, M; Fujisaki, J; Motoyama, Y; Namikawa, Y; Sakata, Y; Seki, J; Takasugi, H; Tanaka, A; Yoshida, K | 1 |
Ambrogi, V; D'Amico, M; de Caprariis, P; Grandolini, G; Lampa, E; Palagiano, F; Perioli, L; Rimoli, MG | 1 |
Engelhardt, G; Homma, D; Schlegel, K; Schnitzler, C; Utzmann, R | 1 |
Engelhardt, G | 1 |
Ambrogi, V; Arenare, L; De Caprariis, P; Falcone, G; Filippelli, W; Grandolini, G; Palagiano, F; Perioli, L; Rossi, F | 1 |
Forte, JG; Muto, Y; Nagao, T; Urushidani, T; Yao, X | 1 |
Bobrzynski, A; Camps, F; Fillat, O; Gedliczka, O; Herrero, E; Márquez, M; Ortiz, JA; Rembiasz, K; Torres, J | 1 |
Coltau, M; Fillat, O; Herrero, E; Márquez, M; Ortiz, JA; Puscas, C; Puscas, I; Torres, J | 1 |
Coltau, M; Fillat, O; Herrero, E; Márquez, M; Ortiz, JA; Pasca, R; Puscas, C; Puscas, I; Torres, J | 1 |
Hawkey, CJ | 2 |
Piotrowski, J; Slomiany, A; Slomiany, BL | 2 |
Engelhardt, G; Mauz, A; Pairet, M; Schierok, H; Trummlitz, G; van Ryn, J | 1 |
Demirdamar, R; Ertan, M; Kelicen, P; Krebs, B; Läge, M; Tozkoparan, B | 1 |
Forsyth, SF; Godfrey, J; Guilford, WG; Haslett, SJ | 1 |
Bornemeier, DA; Chan, K; Connor, DT; Doubleday, R; Dyer, RD; Gilbertsen, RB; Guglietta, A; Roth, BD; Schrier, DJ; Sercel, AD; Song, Y; Sorenson, RJ; Unangst, PC | 1 |
Brzozowski, T; Drozdowicz, D; Hahn, EG; Konturek, PC; Konturek, SJ; Pajdo, R; Sliwowski, Z; Stachura, J | 1 |
Demirdamar, R; Ertan, M; Ertan, R; Kelicen, P; Kilcigil, GA; Tozkoparan, B | 1 |
Arroyo, MT; Lanas, A; Sáinz, R | 1 |
Caruso, A; Cutuli, V; Mangano, N; Modica, M; Santagati, A; Santagati, M | 1 |
Brzozowski, T; Drozdowicz, D; Hahn, EG; Konturek, PC; Konturek, SJ; Pajdo, R; Ptak, A; Sliwowski, Z | 1 |
Aktay, G; Ertan, M; Tozkoparan, B; Yesilada, E | 1 |
Aktay, G; Berk, B; Ertan, M; Yesilada, E | 1 |
Caignard, DH; Chavatte, P; Espiard, JG; Lesieur, D; Poupaert, JH; Yous, S | 1 |
Ohtsuki, H; Okabe, S; Tabata, K | 1 |
Colombo, M; Márquez, M; Roberts, DJ | 1 |
Brzozowski, T; Konturek, SJ; Majka, J | 1 |
Inoue, Y; Katsura, Y; Nishino, S; Takasugi, H; Tomoi, M | 1 |
Murty, VL; Piotrowski, J; Slomiany, A; Slomiany, BL | 1 |
Caruso, A; Cutuli, V; Guccione, S; Monsù Scolaro, L; Romeo, G; Russo, F | 1 |
Bruno, M; Grassi, A; Ippen, J; Thomas, G | 1 |
Dammann, HG; Dreyer, M; Müller, P; Simon, B; Simon-Schultz, J | 1 |
Fagan, TC; Fennerty, B; Lipsy, RJ | 1 |
Battaglia, G; Bianchi Porro, G; D'Angelo, A; Da Broi, GL; Di Mario, F; Naccarato, R; Saggioro, A; Vezzadini, P | 1 |
Attaguile, G; Bousquet, E; Caruso, A; Guccione, S; Leone, MG; Romeo, G; Roxas, MA; Russo, F | 1 |
Yoshinaga, E | 1 |
Gitnick, G | 1 |
Kumadaki, Y; Nakata, H; Nakata, M; Okabe, S; Okada, M; Takeuchi, K | 1 |
Brazer, SR; Brice, RS; Garbutt, JT; Harrell, FE; Liss, CL; Pancotto, FS; Pryor, DB; Root, JK; Tyor, MP; Wildermann, NM | 1 |
Arnold, R; Beckenbach, P; Bock, H; Bormann, R; Brunner, G; Daake, H; Dammann, HG; Dietrich, K; Fuerer, M; Geiter, B | 1 |
Graham, DY; Knuff, TE; Lanza, FL; Levenson, HL; Lyon, DT; McCullough, AJ; Munsell, WP; Perozza, J; Roufail, WM; Sinar, DR | 1 |
Harvengt, C | 1 |
Miwa, T | 1 |
Kaplowitz, N; Kuhlenkamp, J; Lu, SC; Robert, A | 1 |
Barbara, L; Bianchi-Porro, G; Cheli, R; Dammann, HG; Hentschel, E; Müller, P; Paoluzzi, P; Simon, B; Walter, TA | 1 |
Barbara, L; Bianchi Porro, G; Blasi, A; Carratelli, L; Cheli, R; Corinaldesi, R; Lazzaroni, M; Mangiameli, A; Paoluzi, P; Torsoli, A | 1 |
Bianchi Porro, G | 1 |
Dammann, HG; Friedl, W; Krier, C; Müller, P; Simon, B | 1 |
Dammann, HG; Müller, P; Simon, B | 2 |
Lyon, DT | 1 |
Scarpignato, C; Tramacere, R; Zappia, L | 1 |
Dove, PA; Nielsen, ST; Schiehser, GA; Strike, DP | 1 |
Cremer, M; Dammann, HG; Keohane, PP; Mulder, H; Naccaratto, R; Sarles, H; Simon, B | 1 |
Barbara, L; Corinaldesi, R; Paparo, GF; Pasquali, R; Paternico, A; Ricci Maccarini, M; Stanghellini, V | 1 |
Goto, H; Nakazawa, S; Ozawa, T; Sugiyama, S; Takano, K | 1 |
Luskin, AT; Tomasko, MA | 1 |
Pounder, R | 1 |
Bonardelli, P; Fujita, R; Fujita, Y; Sugata, F | 1 |
Brogden, RN; Price, AH | 1 |
Imamura, Y; Oimomi, M; Yasutake, K; Yoshimura, Y | 1 |
Asano, K; Haga, K; Maruyama, Y; Osuga, K | 1 |
Evans, DC; Lin, TM; Ruffolo, RR; Warrick, MW | 1 |
Carpenter, DU; Henann, NE; Janda, SM | 1 |
Dammann, HG; Hentschel, E; Muller, P; Simon, B; Walter, TA | 2 |
Barocelli, E; Bordi, F; Impicciatore, M; Morini, G; Plazzi, PV; Silva, C | 1 |
Amico Roxas, M; Bonina, F; Caruso, A; Guerrera, F; Leone, MG; Sarvà, MC; Siracusa, MA | 1 |
Fukuda, S; Hotta, T; Itoh, H; Kawasaki, T; Komatsu, K; Kuwayama, H; Matsuo, Y; Ohsaka, Y; Seki, A | 1 |
Barthwal, JP; Bhalla, TN; Kumar, P; Pande, K; Tandon, M | 1 |
Friedmann, JC; Murphy, JR | 1 |
Kamada, T; Kawano, S; Sato, N; Takeda, M | 1 |
Kado, Y; Kumada, S; Takashima, T | 1 |
Fujimura, H; Hayashi, M; Hiramatsu, Y; Nozaki, M; Tsurumi, K | 1 |
Reviews
8 review(s) available for thiazoles and Gastric Ulcer
Article | Year |
---|---|
Pharmacology of meloxicam, a new non-steroidal anti-inflammatory drug with an improved safety profile through preferential inhibition of COX-2.
Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase Inhibitors; Disease Models, Animal; Drug Tolerance; Humans; Inflammation; Meloxicam; Mice; Rats; Stomach Ulcer; Thiazines; Thiazoles | 1996 |
The gastroenterologist's caseload: contribution of the rheumatologist.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Rheumatoid; Cyclooxygenase Inhibitors; Digestive System; Gastrointestinal Diseases; Helicobacter Infections; Helicobacter pylori; Humans; Meloxicam; Rats; Stomach Ulcer; Thiazines; Thiazoles | 1997 |
Cyclooxygenase inhibition: between the devil and the deep blue sea.
Topics: Anti-Inflammatory Agents, Non-Steroidal; Arthritis; Celecoxib; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Gastroscopy; Humans; Isoenzymes; Kidney; Lactones; Meloxicam; Membrane Proteins; Myocardial Infarction; Prostaglandin-Endoperoxide Synthases; Proton Pump Inhibitors; Pyrazoles; Randomized Controlled Trials as Topic; Stomach Ulcer; Sulfonamides; Sulfones; Thiazines; Thiazoles | 2002 |
Clinical review of histamine2 receptor antagonists.
Topics: Cimetidine; Drug Interactions; Duodenal Ulcer; Famotidine; Histamine H2 Antagonists; Humans; Nizatidine; Ranitidine; Stomach Ulcer; Thiazoles | 1990 |
Famotidine in the USA: a review of efficacy studies.
Topics: Anti-Ulcer Agents; Duodenal Ulcer; Famotidine; Gastric Acid; Gastric Juice; Histamine H2 Antagonists; Humans; Stomach Ulcer; Thiazoles | 1989 |
Histamine H2-receptor antagonists.
Topics: Animals; Clinical Trials as Topic; Duodenal Ulcer; Esophagitis, Peptic; Famotidine; Histamine H2 Antagonists; Humans; Nizatidine; Stomach Ulcer; Thiazoles | 1988 |
Nizatidine. A preliminary review of its pharmacodynamic and pharmacokinetic properties, and its therapeutic use in peptic ulcer disease.
Topics: Animals; Duodenal Ulcer; Histamine H2 Antagonists; Humans; Nizatidine; Stomach Ulcer; Thiazoles; Tissue Distribution | 1988 |
Double pylorus accompanied by gastric ulcer resistant to H2-receptor antagonist--a case report and review of the literature.
Topics: Drug Resistance; Famotidine; Female; Histamine H2 Antagonists; Humans; Middle Aged; Pylorus; Stomach Ulcer; Thiazoles | 1988 |
Trials
23 trial(s) available for thiazoles and Gastric Ulcer
Article | Year |
---|---|
Evaluation of High Dosages of Oral Meloxicam in American Kestrels ( Falco sparverius ).
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bird Diseases; Dose-Response Relationship, Drug; Falconiformes; Liver; Meloxicam; Non-alcoholic Fatty Liver Disease; Stomach Ulcer; Thiazines; Thiazoles | 2017 |
Gastroscopic Study of Meloxicam, Tramadol, and Their Combined Administration on the Development of Gastric Injuries in Dogs.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Dog Diseases; Dogs; Female; Gastroscopy; Male; Meloxicam; Stomach Ulcer; Thiazines; Thiazoles; Tramadol; Treatment Outcome | 2017 |
Preventive efficacy and safety of rebamipide in nonsteroidal anti-inflammatory drug-induced mucosal toxicity.
Topics: Adult; Aged; Alanine; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Arthritis; Butanones; Diclofenac; Double-Blind Method; Drug Administration Schedule; Gastric Mucosa; Humans; Meloxicam; Middle Aged; Misoprostol; Nabumetone; Quinolones; Stomach Ulcer; Thiazines; Thiazoles; Treatment Outcome | 2014 |
Pharmacokinetics and adverse effects of oral meloxicam tablets in healthy adult horses.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Female; Half-Life; Horse Diseases; Horses; Male; Meloxicam; Stomach Ulcer; Tablets; Thiazines; Thiazoles | 2013 |
Efficacy of ebrotidine and ranitidine in the treatment of benign gastric ulcer.
Topics: Adult; Aged; Benzenesulfonates; Double-Blind Method; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Ranitidine; Stomach Ulcer; Thiazoles | 1997 |
Studies on the protective effect of ebrotidine on experimental ulcers induced by non-steroidal anti-inflammatory drugs in healthy volunteers.
Topics: Adult; Aged; Anti-Inflammatory Agents, Non-Steroidal; Benzenesulfonates; Carbonic Anhydrases; Female; Gastric Mucosa; Histamine H2 Antagonists; Humans; Indomethacin; Male; Middle Aged; Stomach Ulcer; Thiazoles | 1997 |
Comparative study of the safety and efficacy of ebrotidine versus ranitidine and placebo in the prevention of piroxicam-induced gastroduodenal lesions.
Topics: Adult; Benzenesulfonates; Duodenal Ulcer; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Piroxicam; Ranitidine; Stomach Ulcer; Thiazoles | 1997 |
[Effective prevention of piroxicam-induced lesions of the gastric mucosa with nizatidine].
Topics: Adult; Dose-Response Relationship, Drug; Gastric Mucosa; Histamine H2 Antagonists; Humans; Male; Nizatidine; Piroxicam; Single-Blind Method; Stomach Ulcer; Thiazoles | 1990 |
Comparison of 150 mg nizatidine BID or 300 mg at bedtime, and 150 mg ranitidine BID in the treatment of gastric ulcer--an 8-week randomized, double-blind multicentre study.
Topics: Adult; Aged; Double-Blind Method; Drug Administration Schedule; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Nizatidine; Ranitidine; Stomach Ulcer; Thiazoles; Time Factors | 1990 |
Randomized, double-blind comparison of famotidine with ranitidine in treatment of acute, benign gastric ulcer disease. Community-based study coupled with a patient registry.
Topics: Clinical Trials as Topic; Double-Blind Method; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Random Allocation; Ranitidine; Registries; Stomach Ulcer; Thiazoles | 1989 |
[Treatment of acute stomach ulcer with H2 receptor antagonists. A direct therapy comparison with 300 mg nizatidine nightly and 2 times 150 mg nizatidine with twice daily 150 mg ranitidine].
Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Nizatidine; Random Allocation; Ranitidine; Stomach Ulcer; Thiazoles | 1989 |
Suppression of nocturnal acid secretion with famotidine accelerates gastric ulcer healing.
Topics: Clinical Trials as Topic; Double-Blind Method; Famotidine; Female; Gastric Acid; Histamine H2 Antagonists; Humans; Male; Middle Aged; Multicenter Studies as Topic; Random Allocation; Stomach Ulcer; Thiazoles | 1989 |
Clinical evaluation of 20 mg/day famotidine in the treatment of acute gastric mucosal lesions.
Topics: Adult; Aged; Anti-Ulcer Agents; Clinical Trials as Topic; Dose-Response Relationship, Drug; Famotidine; Gastric Mucosa; Humans; Middle Aged; Pain; Random Allocation; Stomach Ulcer; Thiazoles | 1989 |
[Accelerated healing of ulcus ventriculi by a single evening dose of famotidine. Results of an Austrian-German-Italian multicenter study].
Topics: Adolescent; Adult; Aged; Austria; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Famotidine; Female; Germany; Histamine H2 Antagonists; Humans; Italy; Male; Middle Aged; Stomach Ulcer; Thiazoles; Wound Healing | 1985 |
Famotidine (MK-208) in the treatment of gastric ulcer. Results of a multicenter double-blind controlled study.
Topics: Adolescent; Adult; Aged; Antacids; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Endoscopy; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Pain; Random Allocation; Stomach Ulcer; Thiazoles | 1985 |
Famotidine in the treatment of gastric and duodenal ulceration: overview of clinical experience.
Topics: Acute Disease; Chronic Disease; Cimetidine; Circadian Rhythm; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Duodenal Ulcer; Endoscopy; Famotidine; Gefarnate; Histamine H2 Antagonists; Humans; Ranitidine; Stomach Ulcer; Thiazoles; Time Factors | 1985 |
[I.v. famotidine versus i.v. ranitidine: intragastric pH behavior in surgical intensive care patients].
Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Critical Care; Double-Blind Method; Famotidine; Gastric Acidity Determination; Histamine H2 Antagonists; Humans; Infusions, Parenteral; Middle Aged; Peptic Ulcer Hemorrhage; Postoperative Complications; Random Allocation; Ranitidine; Stomach Ulcer; Stress, Physiological; Thiazoles | 1985 |
Efficacy and safety of famotidine in the management of benign gastric ulcers.
Topics: Adult; Clinical Trials as Topic; Famotidine; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Stomach Ulcer; Thiazoles | 1986 |
Famotidine once-a-day in the therapy of acute, benign gastric ulcer: a worldwide experience.
Topics: Acute Disease; Adult; Antacids; Double-Blind Method; Drug Administration Schedule; Famotidine; Histamine H2 Antagonists; Humans; Stomach Ulcer; Thiazoles | 1987 |
Nizatidine versus ranitidine in gastric ulcer disease. A European multicentre trial.
Topics: Adult; Aged; Aged, 80 and over; Antacids; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Female; Histamine H2 Antagonists; Humans; Male; Middle Aged; Nizatidine; Random Allocation; Ranitidine; Smoking; Stomach Ulcer; Thiazoles | 1987 |
Histamine H2-receptor antagonists.
Topics: Animals; Clinical Trials as Topic; Duodenal Ulcer; Esophagitis, Peptic; Famotidine; Histamine H2 Antagonists; Humans; Nizatidine; Stomach Ulcer; Thiazoles | 1988 |
Famotidine: proven once-a-day treatment for gastric ulcer.
Topics: Adult; Anti-Ulcer Agents; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Famotidine; Female; Humans; Male; Middle Aged; Random Allocation; Stomach Ulcer; Thiazoles | 1987 |
Famotidine: nocturnal administration for gastric ulcer healing. Results of multicenter trials in Austria and Germany.
Topics: Adolescent; Adult; Aged; Clinical Trials as Topic; Double-Blind Method; Drug Administration Schedule; Endoscopy; Famotidine; Female; Humans; Male; Middle Aged; Pain; Random Allocation; Stomach Ulcer; Thiazoles; Time Factors | 1985 |
Other Studies
91 other study(ies) available for thiazoles and Gastric Ulcer
Article | Year |
---|---|
A comparative time-dependent study of hematology, serum gastrin concentrations, and gastroscopic assessment of meloxicam-induced gastric ulceration in dogs.
Topics: Animals; Dog Diseases; Dogs; Gastrins; Gastroscopy; Hematology; Meloxicam; Stomach Ulcer; Thiazines; Thiazoles | 2021 |
Conjugation of 4-aminosalicylate with thiazolinones afforded non-cytotoxic potent in vitro and in vivo anti-inflammatory hybrids.
Topics: Administration, Oral; Aminosalicylic Acid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arachidonate 15-Lipoxygenase; Carrageenan; Cell Line, Tumor; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Dose-Response Relationship, Drug; Edema; Humans; Indomethacin; Lipoxygenase Inhibitors; Male; Molecular Docking Simulation; Molecular Structure; Rats; Rats, Wistar; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 2020 |
Design, synthesis, biological evaluation, and computational studies of novel thiazolo-pyrazole hybrids as promising selective COX-2 inhibitors: Implementation of apoptotic genes expression for ulcerogenic liability assessment.
Topics: Animals; Anti-Inflammatory Agents; Anti-Ulcer Agents; Apoptosis; Cyclooxygenase 2 Inhibitors; Dose-Response Relationship, Drug; Drug Design; Edema; Formaldehyde; Male; Models, Molecular; Molecular Structure; Pyrazoles; Rats; Rats, Wistar; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 2021 |
Highly selective CB
Topics: Animals; Anti-Ulcer Agents; Gastric Mucosa; Inflammation Mediators; Male; Mice; Mice, Inbred BALB C; Protective Agents; Receptor, Cannabinoid, CB2; Stomach Ulcer; Thiazoles; Treatment Outcome | 2017 |
7-Chloro-4-phenylsulfonyl quinoline, a new antinociceptive and anti-inflammatory molecule: Structural improvement of a quinoline derivate with pharmacological activity.
Topics: Acetic Acid; Analgesics; Animals; Anti-Inflammatory Agents; Croton Oil; Edema; Hot Temperature; Humans; Male; Meloxicam; Mice; Nociception; Pain; Quinolines; Stomach Ulcer; Thiazines; Thiazoles | 2017 |
New immunological investigations on Helicobacter pylori-induced gastric ulcer in patients.
Topics: Adolescent; Adult; Aged; Aged, 80 and over; Cell Proliferation; Cells, Cultured; Enzyme-Linked Immunosorbent Assay; Female; Helicobacter Infections; Helicobacter pylori; Humans; Interleukin-1beta; Interleukin-8; Leukocytes, Mononuclear; Male; Middle Aged; Staining and Labeling; Stomach Ulcer; Tetrazolium Salts; Thiazoles; Young Adult | 2013 |
Anti-inflammatory, Analgesic and Anti-ulcerogenic Activities of Novel bis-thiadiazoles, bis-thiazoles and bis-formazanes.
Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Dose-Response Relationship, Drug; Edema; Formazans; Male; Mice; Molecular Structure; Nociceptive Pain; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 2017 |
Novel 2,4-dichlorophenoxy acetic acid substituted thiazolidin-4-ones as anti-inflammatory agents: Design, synthesis and biological screening.
Topics: 2,4-Dichlorophenoxyacetic Acid; Animals; Anti-Inflammatory Agents; Drug Design; Rats; Rats, Wistar; Stomach Ulcer; Structure-Activity Relationship; Thiazoles; Tumor Necrosis Factor-alpha | 2017 |
Synthesis and biological activities of new substituted thiazoline-quinoline derivatives.
Topics: Acetophenones; Animals; Anti-Bacterial Agents; Anti-Inflammatory Agents, Non-Steroidal; Antifungal Agents; Edema; Fluoroquinolones; Fungi; Gatifloxacin; Gram-Negative Bacteria; Gram-Positive Bacteria; Indomethacin; Ketoconazole; Lethal Dose 50; Male; Mice; Quinolines; Rats; Stomach Ulcer; Thiazoles; Toxicity Tests, Acute | 2009 |
Synthesis of new 2,3-dihydroquinazolin-4(1H)-one derivatives for analgesic and anti-inflammatory evaluation.
Topics: Acetic Acid; Analgesics; Animals; Anti-Inflammatory Agents; Carrageenan; Chalcones; Drug Evaluation, Preclinical; Edema; Male; Mice; Molecular Structure; Pain; Pain Measurement; Pyrazoles; Quinazolinones; Rats; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 2010 |
Positively charged polymeric nanoparticles: application in improving therapeutic efficacy of meloxicam after oral administration.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Caproates; Carrageenan; Edema; Foot; Freeze Drying; Lactones; Male; Meloxicam; Nanoparticles; Particle Size; Polymers; Quaternary Ammonium Compounds; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Surface-Active Agents; Suspensions; Thiazines; Thiazoles | 2011 |
Eudragit EPO nanoparticles: application in improving therapeutic efficacy and reducing ulcerogenicity of meloxicam on oral administration.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Male; Meloxicam; Microscopy, Electron, Transmission; Nanocapsules; Nanotechnology; Particle Size; Polymethacrylic Acids; Rats; Rats, Sprague-Dawley; Solubility; Stomach Ulcer; Thiazines; Thiazoles | 2011 |
Evaluation of anti-inflammatory, anti-nociceptive, and anti-ulcerogenic activities of novel synthesized thiazolyl and pyrrolyl steroids.
Topics: Analgesics; Animals; Anti-Inflammatory Agents; Anti-Ulcer Agents; Carrageenan; Disease Models, Animal; Edema; Inflammation; Pain; Pyrroles; Rats; Rats, Sprague-Dawley; Steroids; Stomach Ulcer; Thiazoles; Ulcer | 2011 |
Syntheses and evaluation of anti-inflammatory, analgesic and ulcerogenic activities of 1,3,4-oxadiazole and 1,2,4-triazolo[3,4-b]-1,3,4-thiadiazole derivatives.
Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Female; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Mice; Oxadiazoles; Spectroscopy, Fourier Transform Infrared; Stomach Ulcer; Thiazoles | 2012 |
Evaluation of the analgesic and anti-inflammatory activities of some thiazolo[4,5-d]pyrimidines.
Topics: Acetic Acid; Analgesics, Non-Narcotic; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Edema; Gastric Mucosa; Mice; Pain; Pyrimidines; Rats; Rats, Wistar; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 2002 |
Modulation of NSAID-induced antinociceptive and anti-inflammatory effects by alpha2-adrenoceptor agonists with gastroprotective effects.
Topics: Adrenergic alpha-Agonists; Animals; Anti-Inflammatory Agents, Non-Steroidal; Clonidine; Drug Synergism; Drug Therapy, Combination; Meloxicam; Mice; Naproxen; Pain; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Stomach Ulcer; Sulfonamides; Thiazines; Thiazoles; Yohimbine | 2002 |
Meloxicam complexation with beta-cyclodextrin: influence on the anti-inflammatory and ulcerogenic activity.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; beta-Cyclodextrins; Cyclodextrins; Edema; Intestinal Mucosa; Male; Meloxicam; Rats; Rats, Wistar; Stomach Ulcer; Thiazines; Thiazoles | 2003 |
Design and synthesis of some substituted 1H-pyrazolyl-oxazolidines or 1H-pyrazolyl-thiazolidines as anti-inflammatory-antimicrobial agents.
Topics: Animals; Anti-Bacterial Agents; Anti-Infective Agents; Anti-Inflammatory Agents, Non-Steroidal; Candida albicans; Drug Design; Escherichia coli; Infusions, Parenteral; Lethal Dose 50; Male; Mice; Oxazoles; Pyrazoles; Rats; Rats, Sprague-Dawley; Staphylococcus aureus; Stomach Ulcer; Structure-Activity Relationship; Thiazoles; Toxicity Tests, Acute | 2003 |
Pioglitazone, a specific ligand of the peroxisome proliferator-activated receptor gamma reduces gastric mucosal injury induced by ischaemia/ reperfusion in rat.
Topics: Amino Acid Sequence; Animals; Cyclooxygenase 1; Cyclooxygenase 2; Gastric Mucosa; Hypoglycemic Agents; Interleukin-1; Isoenzymes; Leptin; Male; Membrane Proteins; Models, Animal; Pioglitazone; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Wistar; Receptors, Cytoplasmic and Nuclear; Reperfusion Injury; Splanchnic Circulation; Stomach Ulcer; Thiazoles; Thiazolidinediones; Transcription Factors; Tumor Necrosis Factor-alpha | 2003 |
Synthesis and analgesic and anti-inflammatory activity of some new (6-acyl-2-benzoxazolinone and 6-acyl-2-benzothiazolinone derivatives with acetic acid and propanoic acid residues.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Benzoxazoles; Edema; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Mice; Pain Measurement; Spectrophotometry, Infrared; Stomach Ulcer; Thiazoles | 2003 |
Synthesis and anti-inflammatory activity of alkyl/arylidene-2-aminobenzothiazoles and 1-benzothiazol-2-yl-3-chloro-4-substituted-azetidin-2-ones.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Azetidines; Carrageenan; Chemical Phenomena; Chemistry, Physical; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Edema; Female; Indicators and Reagents; Indomethacin; Isoenzymes; Male; Membrane Proteins; Mice; Prostaglandin-Endoperoxide Synthases; Rats; Stomach Ulcer; Thiazoles | 2003 |
Mucosal damage induced by preferential COX-1 and COX-2 inhibitors: role of prostaglandins and inflammatory response.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Cyclooxygenase Inhibitors; Dinoprostone; Dose-Response Relationship, Drug; Drug Synergism; Drug Therapy, Combination; Female; Gastric Mucosa; Gastrointestinal Hemorrhage; Hydrochloric Acid; Male; Meloxicam; Peroxidase; Piroxicam; Rats; Rats, Wistar; Stomach Ulcer; Thiazines; Thiazoles | 2004 |
Synthesis, characterization and antiinflammatory-analgesic properties of 6-(alpha-amino-4-chlorobenzyl)thiazolo [3,2-b]-1,2,4-triazol-5-ols.
Topics: Acetic Acid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Benzoquinones; Capillary Permeability; Carrageenan; Chemical Phenomena; Chemistry, Physical; Edema; Foot; Indicators and Reagents; Magnetic Resonance Spectroscopy; Male; Mice; Models, Molecular; Molecular Conformation; Naproxen; Pain; Spectroscopy, Fourier Transform Infrared; Stomach Ulcer; Structure-Activity Relationship; Thiazoles; Triazoles | 2004 |
Gastric antisecretory and anti-ulcer effect of ME3407, a new benzimidazole derivative, in rats.
Topics: Animals; Anti-Inflammatory Agents; Anti-Ulcer Agents; Aspirin; Benzimidazoles; Cysteamine; Duodenal Ulcer; Epirizole; Gastric Acid; Gastric Fistula; Gastric Mucosa; Gastrins; Histamine; Immersion; Indomethacin; Male; Pepsin A; Pylorus; Pyridines; Rats; Stomach Ulcer; Thiazoles | 2004 |
Analgesic, antiinflammatory, and ulcerogenic studies of meloxicam solid dispersion prepared with polyethylene glycol 6000.
Topics: Abdominal Pain; Acetic Acid; Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Dosage Forms; Dose-Response Relationship, Drug; Drug Compounding; Female; Gastric Mucosa; Hindlimb; Inflammation; Male; Meloxicam; Mice; Polyethylene Glycols; Rats; Rats, Wistar; Solubility; Stomach Ulcer; Thiazines; Thiazoles; Treatment Outcome | 2006 |
Non-carboxylic analogues of arylpropionic acids: synthesis, anti-inflammatory activity and ulcerogenic potential.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Flurbiprofen; Ibuprofen; Male; Naproxen; Propionates; Rats; Stomach Ulcer; Structure-Activity Relationship; Thiadiazoles; Thiazoles | 2007 |
Nonsteroidal anti-inflammatory drugs induce hypermotilinemia and disturbance of interdigestive migrating contractions in instrumented dogs.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Dogs; Duodenoscopy; Duodenum; Gastrointestinal Motility; Indomethacin; Jejunum; Male; Meloxicam; Motilin; Stomach Ulcer; Thiazines; Thiazoles | 2006 |
Effect of different cyclooxygenase inhibitors on gastric adaptive cytoprotection induced by 20% ethanol.
Topics: Animals; Celecoxib; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase Inhibitors; Cytoprotection; Diclofenac; Dinoprostone; Dose-Response Relationship, Drug; Enzyme Inhibitors; Ethanol; Gastric Acid; Gastric Mucosa; Ibuprofen; Irritants; Male; Meloxicam; Membrane Proteins; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Pyrazoles; Rats; Rats, Wistar; Stomach Ulcer; Sulfonamides; Thiazines; Thiazoles | 2007 |
Effect of a new potent H2-blocker, 3-[[[2-(diaminomethylene)amino]-4-thiazolyl]methyl]thio]-N2-sulfamoyl propionamidine (YM-11170), on gastric secretion, ulcer formation and weight of male accessory sex organs in rats.
Topics: Androgen Antagonists; Animals; Aspirin; Castration; Cimetidine; Famotidine; Gastric Juice; Gastric Mucosa; Genitalia, Male; Histamine H2 Antagonists; Male; Organ Size; Rats; Rats, Inbred Strains; Stomach Ulcer; Testosterone; Thiazoles | 1982 |
The effects of acetazolamide and of ethoxzolamide on gastric microcirculation in rats (histochemical study).
Topics: Acetazolamide; Adenosine Triphosphatases; Animals; Ethoxzolamide; Female; Gastric Mucosa; Histocytochemistry; Microcirculation; Rats; Reserpine; Stomach Ulcer; Thiazoles | 1984 |
[3,3'-bi-1,3-thiazolidine]-4,4'-dione system. I. Synthesis, conformational analysis and pharmacological activities of 2,2'-diaryl derivatives.
Topics: Analgesics; Animals; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Chemical Phenomena; Chemistry; Female; Magnetic Resonance Spectroscopy; Male; Mass Spectrometry; Mice; Molecular Conformation; Rats; Reaction Time; Spectrophotometry, Infrared; Stomach Ulcer; Temperature; Thiazoles | 1984 |
Studies on the anti-inflammatory activity and ulcerogenic adverse effect of thiazole derivatives, especially 2-amino-thiazoleacetic acid derivatives.
Topics: Acetates; Animals; Anti-Inflammatory Agents; Edema; Erythrocytes; Hemolysis; Male; Protease Inhibitors; Protein Denaturation; Rats; Rats, Inbred Strains; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 1984 |
Research on heterocyclic compounds. XIV - Imidazothiazole and imidazobenzothiazole derivatives: synthesis and antiinflammatory activity.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Chemical Phenomena; Chemistry; Imidazoles; Mice; Rats; Reaction Time; Stomach Ulcer; Thiazoles | 1983 |
[Effects of protective agents on ulcer formation].
Topics: Adult; Animals; Cimetidine; Dogs; Duodenal Ulcer; Famotidine; Gastric Juice; Gastric Mucosa; Humans; Male; Peptic Ulcer; Stomach Ulcer; Thiazoles | 1984 |
Research on heterocyclic compounds. XI. Heteroarylcarboxylic acids: preparation and antiinflammatory activity.
Topics: Analgesics; Animals; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Imidazoles; Magnetic Resonance Spectroscopy; Pyridines; Pyrimidines; Rats; Spectrophotometry, Infrared; Stomach Ulcer; Thiazoles | 1981 |
Synthesis and pharmacological properties of benzothiazole, 1,3-4-oxadiazole and 1,3,4-thiadiazole derivatives.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Benzothiazoles; Carrageenan; Edema; Lethal Dose 50; Male; Mice; Oxadiazoles; Pain Measurement; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Thiadiazoles; Thiazoles | 1994 |
Studies on antiulcer drugs. 7. 2-Guanidino-4-pyridylthiazoles as histamine H2-receptor antagonists with potent gastroprotective effects against nonsteroidal antiinflammatory drug-induced injury.
Topics: Animals; Anti-Ulcer Agents; Aspirin; Blood Flow Velocity; Dogs; Gastric Acid; Gastric Mucosa; Guanidines; Guinea Pigs; Histamine; Histamine H2 Antagonists; Indomethacin; Male; Molecular Structure; Myocardial Contraction; Rabbits; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Thiazoles | 1994 |
Gastric mucosal laminin receptor expression with ulcer healing by ebrotidine.
Topics: Amino Acid Sequence; Animals; Anti-Ulcer Agents; Benzenesulfonates; Cell Division; Cell Membrane; Gastric Mucosa; Male; Molecular Sequence Data; Rats; Rats, Sprague-Dawley; Receptors, Laminin; Stomach Ulcer; Thiazoles; Wound Healing | 1994 |
Antiplatelet agents based on cyclooxygenase inhibition without ulcerogenesis. Evaluation and synthesis of 4,5-bis(4-methoxyphenyl)-2-substituted-thiazoles.
Topics: Animals; Blood Platelets; Cyclooxygenase Inhibitors; Guinea Pigs; Male; Malondialdehyde; Molecular Structure; Piperazines; Platelet Aggregation; Platelet Aggregation Inhibitors; Rabbits; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Structure-Activity Relationship; Thiazoles; Vasodilation | 1994 |
3,3'-Bi-[1,3-thiazolidine-4-one] system. VII. Synthesis and SARS of some 2-heteroaryl derivatives with antiinflammatory and related activities.
Topics: Acetates; Acetic Acid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Carrageenan; Edema; Magnetic Resonance Spectroscopy; Male; Mice; Pain; Pain Measurement; Rats; Rats, Wistar; Spectrophotometry, Infrared; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 1994 |
Gastric mucosal EGF and PDGF receptor expression with ulcer healing by ebrotidine.
Topics: Animals; Anti-Ulcer Agents; Benzenesulfonates; ErbB Receptors; Gastric Mucosa; Male; Rats; Rats, Sprague-Dawley; Receptors, Platelet-Derived Growth Factor; Stomach Ulcer; Thiazoles | 1994 |
The anti-platelet actions of FR122047, a novel cyclooxygenase inhibitor.
Topics: Animals; Aspirin; Blood Platelets; Cyclooxygenase Inhibitors; Guinea Pigs; Humans; In Vitro Techniques; Irritants; Male; Malondialdehyde; Microsomes; Piperazines; Platelet Aggregation; Platelet Aggregation Inhibitors; Prostaglandins; Rabbits; Rats; Rats, Sprague-Dawley; Seminal Vesicles; Sheep; Stomach Ulcer; Thiazoles | 1993 |
Synthesis and pharmacological activity of imidazo[2,1-b]benzothiazole acids.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Female; Imidazoles; Magnetic Resonance Spectroscopy; Male; Mice; Molecular Conformation; Pregnancy; Rats; Stomach Ulcer; Thiazoles | 1993 |
Anti-inflammatory, analgesic, antipyretic and related properties of meloxicam, a new non-steroidal anti-inflammatory agent with favourable gastrointestinal tolerance.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Bronchial Spasm; Chemotaxis, Leukocyte; Fever; Guinea Pigs; In Vitro Techniques; Inflammation; Male; Meloxicam; Mice; Pain; Pain Measurement; Rats; Stomach Ulcer; Thiazines; Thiazoles; Uricosuric Agents | 1995 |
Synthesis and SAR study of imidazo[2,1-b]benzothiazole acids and some related compounds with anti-inflammatory and analgesic activities.
Topics: Acetates; Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Edema; Female; Imidazoles; Pain; Pain Measurement; Pregnancy; Rats; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 1996 |
ME-3407, a new antiulcer agent, inhibits acid secretion by interfering with redistribution of H(+)-K(+)-ATPase.
Topics: Acetic Acid; Androstadienes; Animals; Anti-Ulcer Agents; Cyclic AMP-Dependent Protein Kinases; Enzyme Inhibitors; Gastric Acid; H(+)-K(+)-Exchanging ATPase; In Vitro Techniques; Male; Myosin-Light-Chain Kinase; Proton Pump Inhibitors; Proton Pumps; Pyridines; Rabbits; Rats; Rats, Wistar; Stomach Ulcer; Thiazoles; Tissue Distribution; Wortmannin; Wound Healing | 1997 |
Cell cycle progression during gastric ulcer healing by ebrotidine and sucralfate.
Topics: Animals; Anti-Ulcer Agents; Benzenesulfonates; Cell Cycle; Cyclin-Dependent Kinases; Gastric Mucosa; In Vitro Techniques; Proliferating Cell Nuclear Antigen; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Sucralfate; Thiazoles | 1997 |
Differential inhibition of cyclooxygenases-1 and -2 by meloxicam and its 4'-isomer.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Cyclooxygenase Inhibitors; Dinoprostone; Humans; Isoenzymes; Male; Meloxicam; Prostaglandin-Endoperoxide Synthases; Rats; Stomach Ulcer; Thiazines; Thiazoles | 1998 |
Condensed heterocyclic compounds: synthesis and antiinflammatory activity of novel thiazolo[3,2-alpha] pyrimidines.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Edema; Female; Heterocyclic Compounds; Hindlimb; Male; Mice; Pyrimidines; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 1998 |
Endoscopy of the gastroduodenal mucosa after carprofen, meloxicam and ketoprofen administration in dogs.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carbazoles; Dogs; Endoscopy, Gastrointestinal; Gastric Mucosa; Gastrointestinal Hemorrhage; Gelatin; Ketoprofen; Meloxicam; Stomach Ulcer; Thiazines; Thiazoles | 1998 |
Synthesis, structure-activity relationships, and in vivo evaluations of substituted di-tert-butylphenols as a novel class of potent, selective, and orally active cyclooxygenase-2 inhibitors. 1. Thiazolone and oxazolone series.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Cell Line; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Edema; Gastric Mucosa; Humans; Hyperalgesia; Isoenzymes; Male; Membrane Proteins; Mice; Oxazoles; Phenols; Prostaglandin-Endoperoxide Synthases; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 1999 |
Endothelin-1, interleukin-4 and nitric oxide synthase modulators of gastric mucosal injury by indomethacin: effect of antiulcer agents.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Anti-Ulcer Agents; Apoptosis; Benzenesulfonates; Endothelin-1; Gastric Mucosa; Indomethacin; Interleukin-4; Nitric Oxide Synthase; Nitric Oxide Synthase Type III; Ranitidine; Rats; Rats, Sprague-Dawley; Sialoglycoproteins; Stomach Ulcer; Thiazoles | 1999 |
Role of prostaglandins generated by cyclooxygenase-1 and cyclooxygenase-2 in healing of ischemia-reperfusion-induced gastric lesions.
Topics: Animals; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Disease Models, Animal; Gastric Mucosa; Gastrins; Gene Expression Regulation, Enzymologic; Indomethacin; Interleukin-1; Isoenzymes; Lactones; Meloxicam; Membrane Proteins; Nitrobenzenes; Prostaglandin-Endoperoxide Synthases; Prostaglandins; Rats; Regional Blood Flow; Reperfusion Injury; Resveratrol; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stilbenes; Stomach Ulcer; Sulfonamides; Sulfones; Thiazines; Thiazoles; Time Factors | 1999 |
Synthesis and evaluation of anti-inflammatory activity of some thiazolo[3,2-b]-1,2,4-triazole-5(6H)-ones and their Michael addition products.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Edema; Female; Magnetic Resonance Spectroscopy; Male; Mice; Stomach Ulcer; Thiazoles; Triazoles | 1999 |
Prevention and healing of experimental indomethacin-induced gastric lesions: effects of ebrotidine, omeprazole and ranitidine.
Topics: Animals; Anti-Ulcer Agents; Benzenesulfonates; Disease Models, Animal; Gastric Juice; Histamine H2 Antagonists; Indomethacin; Male; Omeprazole; Ranitidine; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Thiazoles | 2000 |
Synthesis of new [1,3,4]thiadiazolo[3,2-a]thieno[2,3-d]pyrimidinone derivatives with antiinflammatory activity.
Topics: Analgesics; Animals; Anti-Inflammatory Agents, Non-Steroidal; Chemical Phenomena; Chemistry, Physical; Edema; Lethal Dose 50; Magnetic Resonance Spectroscopy; Male; Mice; Pain Measurement; Peritonitis; Pyrimidinones; Rats; Spectrophotometry, Infrared; Stomach Ulcer; Thiazoles | 2000 |
Classic NSAID and selective cyclooxygenase (COX)-1 and COX-2 inhibitors in healing of chronic gastric ulcers.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Aspirin; Chronic Disease; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Gastric Mucosa; Gastrins; Indomethacin; Interleukin-1; Isoenzymes; Lactones; Male; Meloxicam; Membrane Proteins; Nitrobenzenes; Prostaglandin-Endoperoxide Synthases; Radioimmunoassay; Rats; Rats, Wistar; Resveratrol; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Stilbenes; Stomach Ulcer; Sulfonamides; Sulfones; Thiazines; Thiazoles; Tumor Necrosis Factor-alpha | 2001 |
Synthesis of some thiazolo[3,2-b]-1,2,4-triazole-5(6H)-ones and their novel Michael addition products with anti-inflammatory activities.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Chemical Phenomena; Chemistry, Physical; Edema; Female; Magnetic Resonance Spectroscopy; Male; Mice; Spectrophotometry, Infrared; Stomach Ulcer; Thiazoles; Triazoles | 2001 |
Synthesis and pharmacological activities of some new 2-[1-(6-methoxy-2-naphthyl)ethyl]-6-(substituted)benzylidene thiazolo[3,2-b]-1,2,4-triazole-5(6H)-one derivatives.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Chromatography, Thin Layer; Cyclization; Edema; Female; Gastric Mucosa; Male; Mice; Naphthalenes; Naproxen; Stomach Ulcer; Thiazoles | 2001 |
Synthesis and pharmacological evaluation of analgesic 6-substituted 2(3H)-benzothiazolones.
Topics: Analgesics; Animals; Benzothiazoles; Drug Evaluation, Preclinical; Hyperalgesia; Mice; Pain Measurement; Stomach Ulcer; Thiazoles | 2001 |
[Irritative activity of a new anti-inflammatory agent 4-(p-chorophenyl)-2-phenyl-5-thiazoleacetic acid (CH-800) on the gastrointestinal tract in rats (author's transl)].
Topics: Acetates; Administration, Oral; Animals; Anti-Inflammatory Agents; Aspirin; Diclofenac; Digestive System; Ibuprofen; Indomethacin; Irritants; Male; Phenylbutazone; Rats; Stomach Ulcer; Thiazoles | 1979 |
Pharmacological properties of thiazolinobutazone (LAS 11 871). III. General pharmacology, ulcerogenic effects and acute toxicity.
Topics: Animals; Autonomic Nervous System; Brain; Cats; Diuresis; Female; Hemodynamics; Lethal Dose 50; Male; Mice; Motor Activity; Motor Skills; Muscle Contraction; Phenylbutazone; Rabbits; Rats; Respiration; Stomach Ulcer; Thiazoles | 1976 |
Gastroprotective and ulcer-healing activities of a new H2-receptor antagonist: ebrotidine.
Topics: Acetates; Acetic Acid; Animals; Benzenesulfonates; Epidermal Growth Factor; Ethanol; Gastric Acid; Gastric Mucosa; Gastrins; Histamine H2 Antagonists; Male; Ranitidine; Rats; Rats, Inbred Strains; Regional Blood Flow; Stomach Ulcer; Thiazoles | 1992 |
Studies on antiulcer drugs. IV. Synthesis and antiulcer activities of imidazo[1,2-a]pyridinylethylbenzothiazoles and -benzimidazoles.
Topics: Animals; Anti-Ulcer Agents; Benzimidazoles; Guinea Pigs; Histamine H2 Antagonists; In Vitro Techniques; Pyridines; Rabbits; Stomach Ulcer; Stress, Psychological; Thiazoles | 1992 |
Mechanism of ebrotidine protection against gastric mucosal injury induced by ethanol.
Topics: Animals; Benzenesulfonates; Chemical Phenomena; Chemistry, Physical; Ethanol; Gastric Mucosa; Histamine H2 Antagonists; Hydrogen; Male; Mucus; Rats; Rats, Sprague-Dawley; Stomach Ulcer; Thiazoles; Viscosity | 1992 |
Synthesis and pharmacological evaluation of pyrazolopyrimidobenzoxazole and pyrazolopyrimidobenzothiazole derivatives.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Benzoxazoles; Mice; Pyrazoles; Pyridines; Rats; Stomach Ulcer; Thiazoles | 1991 |
BAY P 1455, a thiazolylaminobenzimidazole derivative with gastroprotective properties in the rat.
Topics: Adrenalectomy; Animals; Anti-Ulcer Agents; Benzimidazoles; Cimetidine; Corticosterone; Cysteamine; Duodenal Ulcer; Ethanol; Female; Gastric Acid; Immersion; In Vitro Techniques; Indomethacin; Male; Pirenzepine; Prostaglandins E; Pylorus; Rats; Rats, Inbred Strains; Rioprostil; Stomach Ulcer; Stress, Psychological; Thiazoles | 1991 |
Synthesis and pharmacological activity of 6H-thiazolo [3',2': 1,2]-5-oxopyrimido[5,4-b]indole derivatives, a new heterocyclic ring system.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Carrageenan; Chemical Phenomena; Chemistry; Dose-Response Relationship, Drug; Edema; Exudates and Transudates; Indoles; Lethal Dose 50; Male; Mice; Psychomotor Performance; Pyrimidines; Rats; Rats, Inbred Strains; Stomach Ulcer; Thiazoles | 1990 |
[Mechanism of prevention of stress ulcer by vagotomy and famotidine: viewed from the transmucosal potential difference and histamine staining by a fluorescence histochemical method].
Topics: Animals; Famotidine; Gastric Mucosa; Histamine; Male; Membrane Potentials; Rats; Rats, Inbred Strains; Staining and Labeling; Stomach Ulcer; Stress, Physiological; Thiazoles; Vagotomy | 1986 |
[Effects of nizatidine, a new histamine H2-receptor antagonist, on gastric acid secretion and various gastric and duodenal lesions in rats: comparison with cimetidine].
Topics: Animals; Depression, Chemical; Dose-Response Relationship, Drug; Duodenal Ulcer; Gastric Acid; Histamine H2 Antagonists; Male; Nizatidine; Rats; Rats, Inbred Strains; Stomach Ulcer; Thiazoles | 1989 |
Drugs recently released in Belgium. Recombinant human erythropoietin--nizatidine.
Topics: Anemia; Erythropoietin; Histamine H2 Antagonists; Humans; Nizatidine; Recombinant Proteins; Stomach Ulcer; Thiazoles | 1989 |
Role of glutathione status in protection against ethanol-induced gastric lesions.
Topics: Acetylcysteine; Animals; Cysteamine; Ethanol; Gastric Mucosa; Glutathione; Male; Maleates; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred Strains; Stomach Ulcer; Thiazoles; Thiazolidines | 1989 |
[Famotidine. Pharmacologic and clinical profile of the new histamine H2 receptor antagonist].
Topics: Animals; Duodenal Ulcer; Famotidine; Guinea Pigs; Histamine H2 Antagonists; Humans; Kinetics; Stomach Ulcer; Thiazoles | 1986 |
Famotidine. The ACG Committee on FDA-Related Matters with primary authorship by G. Friedman. American College of Gastroenterology.
Topics: Duodenal Ulcer; Famotidine; Gastric Acid; Histamine H2 Antagonists; Humans; Recurrence; Stomach Ulcer; Thiazoles; Zollinger-Ellison Syndrome | 1987 |
Antisecretory and antiulcer effect of the H2-receptor antagonist famotidine in the rat: comparison with ranitidine.
Topics: Animals; Anti-Ulcer Agents; Duodenal Ulcer; Famotidine; Female; Gastric Emptying; Gastric Mucosa; Histamine H2 Antagonists; Male; Ranitidine; Rats; Rats, Inbred Strains; Stomach Ulcer; Thiazoles | 1987 |
Structural modification of H2-receptor antagonists provide post-H2-receptor gastric antisecretory activity.
Topics: Animals; Gastric Acid; Gastric Mucosa; Histamine H2 Antagonists; In Vitro Techniques; Phenoxypropanolamines; Rats; Rats, Inbred Strains; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 1987 |
Effects of short- and long-term administrations of famotidine and ranitidine on some pituitary, sexual and thyroid hormones.
Topics: Adult; Famotidine; Follicle Stimulating Hormone; Histamine H2 Antagonists; Humans; Luteinizing Hormone; Male; Middle Aged; Pituitary Hormones; Prolactin; Ranitidine; Stomach Ulcer; Thiazoles; Thyroid Hormones; Thyrotropin-Releasing Hormone; Time Factors | 1987 |
Effect of the H2-blocker famotidine on gastric mucosal prostaglandin levels in water immersion stress in rats.
Topics: Animals; Famotidine; Gastric Mucosa; Histamine H2 Antagonists; Immersion; Male; Phospholipases; Prostaglandins; Rats; Rats, Inbred Strains; Stomach Ulcer; Stress, Psychological; Thiazoles | 1988 |
Recurrent parotitis with H2 receptor antagonists in a patient with Sjogren's syndrome.
Topics: Cimetidine; Famotidine; Female; Histamine H2 Antagonists; Humans; Middle Aged; Parotitis; Ranitidine; Recurrence; Sjogren's Syndrome; Stomach Ulcer; Thiazoles | 1988 |
[Famotidine treatment of patients with gastric and duodenal ulcers. A comparative study with once or twice-a-day administration].
Topics: Adult; Aged; Anti-Ulcer Agents; Drug Evaluation; Duodenal Ulcer; Famotidine; Histamine H2 Antagonists; Humans; Middle Aged; Stomach Ulcer; Thiazoles; Time Factors | 1987 |
[Effect of an H+, K+-ATPase inhibitor, omeprazole (OPZ), on gastric acid secretion and gastric or duodenal lesion. Comparison with an H2-receptor antagonist, famotidine (FMD)].
Topics: Animals; Dogs; Duodenitis; Famotidine; Female; Gastric Acid; Histamine H2 Antagonists; Male; Omeprazole; Rats; Rats, Inbred Strains; Sodium-Potassium-Exchanging ATPase; Stomach Ulcer; Thiazoles | 1988 |
Actions of nizatidine on the rat uterus, dog stomach and experimentally induced gastric lesions.
Topics: Animals; Aspirin; Atropine; Dogs; Duodenum; Female; Gastrointestinal Motility; Guanidines; Guinea Pigs; Histamine; Histamine Antagonists; Ligation; Nizatidine; Pyrilamine; Rats; Stomach; Stomach Ulcer; Thiazoles; Uterus | 1986 |
Famotidine-associated mental confusion in elderly patients.
Topics: Aged; Cognition Disorders; Confusion; Famotidine; Female; Humans; Male; Stomach Ulcer; Thiazoles | 1988 |
Antipyretic activity of new compounds 4-(3-oxo-1,2-benzisothiazolin-2-yl)phenylalkanoic acids, their esters, amides and 1,1-dioxide derivatives.
Topics: Amides; Animals; Anti-Inflammatory Agents, Non-Steroidal; Bile; Body Temperature; Carboxylic Acids; Cholagogues and Choleretics; Esters; Female; Gastric Mucosa; Lethal Dose 50; Pyrogens; Rats; Rats, Inbred Strains; Stomach Ulcer; Thiazoles | 1986 |
Synthesis and analgesic antiinflammatory activities of 2-aryl-ethenyl-4-aryl-thiazole-5-acetic acids.
Topics: Acetates; Animals; Anti-Inflammatory Agents, Non-Steroidal; Behavior, Animal; Chemical Phenomena; Chemistry; Male; Mice; Rats; Rats, Inbred Strains; Stomach Ulcer; Thiazoles | 1987 |
Gastric anti-ulcer and cytoprotective properties of 2-(3,4-dimethoxyphenyl)-5-methyl-thiazolidine-4-one in rat experimental ulcers.
Topics: Acetates; Animals; Anti-Ulcer Agents; Cell Survival; Cimetidine; Ethanol; Gastric Mucosa; Indomethacin; Male; Rats; Rats, Inbred Strains; Regional Blood Flow; Stomach Ulcer; Thiazoles | 1986 |
Novel thiazolidinones as potent anti-inflammatory and analgesic agents.
Topics: Aconitine; Animals; Anti-Inflammatory Agents, Non-Steroidal; Carrageenan; Chemical Phenomena; Chemistry; Edema; Female; Gossypium; Lethal Dose 50; Male; Mice; Rats; Stomach Ulcer; Thiazoles | 1985 |
Pre-clinical toxicology of nitazoxanide--a new antiparasitic compound.
Topics: Animals; Anticestodal Agents; Blood Chemical Analysis; Body Weight; Cats; Dogs; Eye; Female; Irritants; Lethal Dose 50; Male; Mice; Mutagenicity Tests; Nitro Compounds; Organ Size; Rats; Rats, Inbred Strains; Salmonella typhimurium; Species Specificity; Stomach Ulcer; Thiazoles | 1985 |
Hemodynamics of the gastric mucosa and gastric ulceration in rats and in patients with gastric ulcer.
Topics: Animals; Blood Volume; Famotidine; Gastric Mucosa; Hemodynamics; Histamine; Humans; Microcirculation; Oxygen Consumption; Rats; Spectrophotometry; Stomach Ulcer; Stress, Physiological; Thiazoles | 1986 |
Pharmacological investigations of benzothiazoline derivatives.
Topics: Amines; Analgesics; Animals; Anti-Inflammatory Agents; Benzyl Compounds; Body Temperature; Carrageenan; Edema; Formaldehyde; Guinea Pigs; Lethal Dose 50; Male; Methylamines; Ovalbumin; Oxyphenbutazone; Phenylbutazone; Piperazines; Pyrazoles; Rats; Stomach Ulcer; Structure-Activity Relationship; Thiazoles | 1972 |
Pharmacological actions of tiaramide hydrochloride: a new anti-inflammatory drug.
Topics: Analgesics; Animals; Anti-Inflammatory Agents; Benzyl Compounds; Blood Pressure; Electrocardiography; Female; Guinea Pigs; Heart; Hemolysis; Ileum; Male; Methylamines; Mice; Piperazines; Pyrazoles; Rabbits; Rats; Respiration; Sleep; Stomach Ulcer; Thiazoles | 1972 |