Page last updated: 2024-08-21

thiazoles and Experimental Mammary Neoplasms

thiazoles has been researched along with Experimental Mammary Neoplasms in 42 studies

Research

Studies (42)

TimeframeStudies, this research(%)All Research%
pre-199015 (35.71)18.7374
1990's4 (9.52)18.2507
2000's9 (21.43)29.6817
2010's11 (26.19)24.3611
2020's3 (7.14)2.80

Authors

AuthorsStudies
Fu, A; Huang, R; Liang, J; Tang, M; Wang, L; Zhou, J1
Cai, Y; Gao, X; Shuai, Q; Sun, X; Xu, J; Xu, Z; Zhu, F1
Chen, B; Chen, T; Duan, Y; Han, D; Li, C; Li, Y; Liang, Y; Liu, Y; Song, X; Wang, L; Wang, X; Yang, Q; Zhang, H; Zhang, N; Zhao, W1
Bradshaw, C; Flecknell, P; Lee, CCS; Lofgren, J; Miller, AL; Roughan, J1
Cheung, P; Kakit, C; Kiess, N; Parsons, R; Pegno, S; Poulikakos, PI; Schmidt, H; Stratikopoulos, EE; Szabolcs, M; Wu, X1
Brunton, VG; Carragher, NO; Creedon, H; Evans, TR; Gusterson, B; Karim, SA; Morton, JP; Muller, WJ; Patel, H; Sansom, OJ1
Fant, ME; Glazer, RI; Kallakury, B; Kopelovich, L; Lu, J; Umans, R; Upadhyay, G; Xiao, J; Yin, Y; Yuan, H1
Bailey, ST; Clark, K; Damrauer, JS; Darr, D; Diehn, M; Fan, C; Hadzic, T; Jeong, Y; Jin, J; Kim, WY; Lee, CY; Levine, RL; Miller, CR; Murphy, L; Perou, CM; Troester, MA; Zhou, B1
Beristain, AG; Chang, MC; Di Grappa, MA; Joshi, PA; Khokha, R; Kirschner, LS; Molyneux, SD; Pomroy, NC; Privé, GG; Pujana, MA1
Aly, H; Attia, SM; Bahashwan, SA; El-Beshbishy, HA; Ghobara, MM; Hassan, MH1
Krop, IE; Lin, NU; Liu, P; Roberts, TM; Spangle, JM; Von, T; Wang, Q; Winer, EP; Zhao, JJ1
Bansal, N; Bosch, A; Cubedo, E; Farias, E; Fishel, M; Jones, JW; Kane, M; Leibovitch, B; Pereira, L; Pierzchalski, K; Waxman, S; Yu, J; Zelent, A1
Chamberlin, R; Chen, PL; Lau, J; Lee, WH; Qiu, XL; Wu, G; Zhou, L; Zhu, J1
Batlle, A; Battah, S; Casas, A; Di Venosa, G; Dobbin, P; Fukuda, H; MacRobert, AJ; Rodriguez, L1
Egleston, BL; Golemis, EA; Izumchenko, E; Klein-Szanto, AJ; Singh, MK; Wolfson, M1
Forinash, KD; Lawrence, NJ; Martin, MP; Patel, RA; Pireddu, R; Schönbrunn, E; Sebti, SM; Sun, N; Sun, Y1
Alley, MC; Bibby, MC; Bradshaw, TD; Cooper, PA; Donohue, S; Double, JA; Fichtner, I; Sausville, EA; Stevens, MF; Stinson, SF; Tomaszewjski, JE1
Brugge, JS; Daley, GQ; Koh, EY; Leder, P; Lu, Y; Martin, SS; Michelman, M; Pinkas, J; Reginato, MJ; Ridgeway, AG1
Bai, R; Dettin, LE; Glazer, RI; Kopelovich, L; Kopleovich, L; Kozikowski, AP; Russell, RG; Wei, ZL; Yin, Y1
Kumar, P; McEwan, AJ; McQuarrie, SA; Wiebe, LI; Zhou, A1
Bryan, GT; Croft, WA; Wang, CY1
Bryan, GT; Ertürk, E; Swaminathan, S1
Mroczkowski, Z; Rockwell, S; Rupp, WD1
Baruchel, S; Batist, G; Farah, R; Jamali, M; Wang, T1
Batist, G; Carystinos, GD; Chen, X1
Fujishita, T; Kobayashi, M; Mizushima, Y; Oosaki, R; Sassa, K1
Koeffler, HP; Mehta, RG; Patel, MK; Williamson, E1
Beauchamp, BK; Ding, I; Fenton, BM; Okunieff, P; Paoni, SF1
Bruwiere, H; Dillen, L; Floren, W; Janicot, M; Janssen, B; Moelans, P; Sanz, G; van der Leede, BJ; van Dun, J; Van Ginckel, R; Van Heusden, J; Van Hove, C; Venet, M; Willemsens, G; Wouters, W1
Rockwell, S1
Dixon, B; Furr, BJ; Jordan, VC; Prestwich, G1
Joss, U; Schieweck, K; Schmidt-Ruppin, KH1
Müller, MR; Twentyman, PR; Wright, KA1
Coley, HM; Twentyman, PR; Workman, P1
Ip, MM; Schenkel, L; Sylvester, PW1
Bryan, GT; Cohen, SM; Ertürk, E2
Atassi, SA; Bryan, GT; Cohen, SM; Ertürk, E; Price, JM; Yoshida, O1
Van Belle, H1
Bryan, GT; Cohen, SM; Ertürk, E; Price, JM1
Bryan, GT; Cohen, SM; Crovetti, AJ; Ertürk, E; Morris, JE; Price, JM; Von Esch, AM1
Gabryel, P; Kasprzak, K; Malejka, D1

Reviews

1 review(s) available for thiazoles and Experimental Mammary Neoplasms

ArticleYear
Potential for selective modulation of glutathione in cancer chemotherapy.
    Chemico-biological interactions, 1998, Apr-24, Volume: 111-112

    Topics: Animals; Buthionine Sulfoximine; Cell Communication; Drug Resistance; Enzyme Inhibitors; Female; Gap Junctions; Glutamate-Cysteine Ligase; Glutathione; Humans; Mammary Neoplasms, Experimental; Neoplasms; Prodrugs; Pyroglutamate Hydrolase; Pyrrolidonecarboxylic Acid; Rats; Thiazoles; Thiazolidines

1998

Other Studies

41 other study(ies) available for thiazoles and Experimental Mammary Neoplasms

ArticleYear
Design and development of novel fasudil derivatives as potent antibreast cancer agent that improves intestinal flora and intestinal barrier function in rats.
    Chemical biology & drug design, 2021, Volume: 98, Issue:6

    Topics: 1-(5-Isoquinolinesulfonyl)-2-Methylpiperazine; Animals; Antineoplastic Agents; Breast Neoplasms; Colon; Drug Screening Assays, Antitumor; Female; Gastrointestinal Microbiome; Humans; Lipid Peroxidation; Mammary Neoplasms, Experimental; MCF-7 Cells; Rats, Sprague-Dawley; rho-Associated Kinases; Thiazoles

2021
Tumor-targeting peptide functionalized PEG-PLA micelles for efficient drug delivery.
    Biomaterials science, 2020, Apr-15, Volume: 8, Issue:8

    Topics: Animals; Antineoplastic Agents, Phytogenic; Cell Survival; Coumarins; Drug Delivery Systems; Drug Liberation; Female; Humans; Mammary Neoplasms, Experimental; MCF-7 Cells; Mice, Inbred ICR; Micelles; Paclitaxel; Peptides; Polyethylene Glycols; Spheroids, Cellular; Thiazoles; Tumor Burden

2020
Fatostatin in Combination with Tamoxifen Induces Synergistic Inhibition in ER-Positive Breast Cancer.
    Drug design, development and therapy, 2020, Volume: 14

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Breast Neoplasms; Cell Line, Tumor; Cell Movement; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Female; Humans; Injections, Intraperitoneal; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Mice, Nude; Pyridines; Receptors, Estrogen; Structure-Activity Relationship; Tamoxifen; Thiazoles

2020
Analgesics promote welfare and sustain tumour growth in orthotopic 4T1 and B16 mouse cancer models.
    Laboratory animals, 2018, Volume: 52, Issue:4

    Topics: Analgesics; Animal Welfare; Animals; Breast Neoplasms; Buprenorphine; Cell Line, Tumor; Disease Models, Animal; Female; Lung Neoplasms; Mammary Neoplasms, Experimental; Melanoma, Experimental; Meloxicam; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Neoplasm Metastasis; Pain; Thiazines; Thiazoles; Xenograft Model Antitumor Assays

2018
Mouse ER+/PIK3CA
    Oncogene, 2019, Volume: 38, Issue:1

    Topics: Aniline Compounds; Animals; Antineoplastic Agents, Hormonal; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Apoptosis Regulatory Proteins; Bcl-2-Like Protein 11; BH3 Interacting Domain Death Agonist Protein; Cell Line, Tumor; Class I Phosphatidylinositol 3-Kinases; Cocarcinogenesis; Drug Resistance, Neoplasm; Drug Screening Assays, Antitumor; Drug Synergism; Estradiol; Estrogen Receptor alpha; Female; Fulvestrant; Gene Expression Regulation, Neoplastic; Gene Knock-In Techniques; Mammary Neoplasms, Experimental; Mice; Mice, Nude; Mutation, Missense; Neoplasm Proteins; Neoplasms, Hormone-Dependent; Neuropeptides; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Sulfonamides; Thiazoles

2019
Dasatinib inhibits mammary tumour development in a genetically engineered mouse model.
    The Journal of pathology, 2013, Volume: 230, Issue:4

    Topics: Administration, Oral; Animals; Antineoplastic Agents; beta Catenin; Breast Neoplasms; Cadherins; Cell Differentiation; Cell Line, Tumor; Cell Movement; Cell Proliferation; Dasatinib; Dose-Response Relationship, Drug; Drug Administration Schedule; Enhancer Elements, Genetic; Female; Gene Expression Regulation, Neoplastic; Genes, erbB-2; Integrases; Lactoglobulins; Mammary Neoplasms, Experimental; Mice; Mice, Inbred C57BL; Mice, Knockout; Mice, Transgenic; Neoplasm Invasiveness; Protein Kinase Inhibitors; PTEN Phosphohydrolase; Pyrimidines; Signal Transduction; src-Family Kinases; Thiazoles; Time Factors

2013
PPARδ induces estrogen receptor-positive mammary neoplasia through an inflammatory and metabolic phenotype linked to mTOR activation.
    Cancer research, 2013, Jul-15, Volume: 73, Issue:14

    Topics: Animals; Carcinogenesis; Carcinoma, Ductal; Epithelium; Female; Gene Expression; Genes, erbB-2; Inflammation; Inflammatory Breast Neoplasms; Mammary Neoplasms, Experimental; Metabolomics; Mice; Mice, Transgenic; Phenotype; PPAR delta; Proto-Oncogene Proteins c-akt; Receptors, Estrogen; Receptors, Progesterone; Thiazoles; TOR Serine-Threonine Kinases

2013
Erythropoietin promotes breast tumorigenesis through tumor-initiating cell self-renewal.
    The Journal of clinical investigation, 2014, Volume: 124, Issue:2

    Topics: Animals; Breast Neoplasms; Carcinogenesis; Cell Line, Tumor; Cell Proliferation; Cell Transformation, Neoplastic; Disease Progression; Disease-Free Survival; Endothelial Cells; Erythropoietin; Female; Gene Expression Regulation; Humans; Hypoxia; Mammary Neoplasms, Experimental; Mice; Neoplasm Transplantation; Neoplastic Stem Cells; Recurrence; Signal Transduction; Tetrazolium Salts; Thiazoles; Time Factors

2014
PKA signaling drives mammary tumorigenesis through Src.
    Oncogene, 2015, Feb-26, Volume: 34, Issue:9

    Topics: Androstadienes; Animals; Cell Line; Cell Proliferation; Cell Transformation, Neoplastic; Cyclic AMP-Dependent Protein Kinase RIalpha Subunit; Dasatinib; Epithelial Cells; Female; Humans; Mammary Glands, Animal; Mammary Neoplasms, Experimental; Mice; Phosphorylation; Pyrimidines; Signal Transduction; src-Family Kinases; Thiazoles; Wortmannin

2015
Modulatory effects of meloxicam on cardiotoxicity and antitumor activity of doxorubicin in mice.
    Cancer chemotherapy and pharmacology, 2014, Volume: 74, Issue:3

    Topics: Animals; Antibiotics, Antineoplastic; Caspase 3; Catalase; Cyclooxygenase 2 Inhibitors; Dinoprostone; Doxorubicin; Female; Glutathione; Glutathione Peroxidase; Heart Diseases; L-Lactate Dehydrogenase; Lipid Peroxidation; Mammary Neoplasms, Experimental; Meloxicam; Mice; Myocardium; Organ Size; Superoxide Dismutase; Thiazines; Thiazoles

2014
PI3K-p110α mediates resistance to HER2-targeted therapy in HER2+, PTEN-deficient breast cancers.
    Oncogene, 2016, 07-07, Volume: 35, Issue:27

    Topics: Animals; Breast Neoplasms; Cell Line, Tumor; Cell Survival; Class I Phosphatidylinositol 3-Kinases; Drug Resistance, Neoplasm; Female; Humans; Lapatinib; Mammary Neoplasms, Experimental; Mice, Knockout; Molecular Targeted Therapy; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-akt; PTEN Phosphohydrolase; Quinazolines; Receptor, ErbB-2; Signal Transduction; Thiazoles; Tumor Burden; Xenograft Model Antitumor Assays

2016
Blocking the PAH2 domain of Sin3A inhibits tumorigenesis and confers retinoid sensitivity in triple negative breast cancer.
    Oncotarget, 2016, Jul-12, Volume: 7, Issue:28

    Topics: Animals; Antineoplastic Agents; Benzoates; Carcinogenesis; Cell Line, Tumor; Female; Humans; Indoles; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Receptors, Retinoic Acid; Repressor Proteins; Sin3 Histone Deacetylase and Corepressor Complex; Tetrahydronaphthalenes; Thiazoles; Triple Negative Breast Neoplasms

2016
Small molecule targeting the Hec1/Nek2 mitotic pathway suppresses tumor cell growth in culture and in animal.
    Cancer research, 2008, Oct-15, Volume: 68, Issue:20

    Topics: Animals; Antineoplastic Agents; Benzamides; Cell Line, Tumor; Cell Proliferation; Cytoskeletal Proteins; Female; Humans; Indoles; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Mitosis; Neoplasm Transplantation; NIMA-Related Kinases; Nuclear Proteins; Protein Serine-Threonine Kinases; Signal Transduction; Thiazoles; Transplantation, Heterologous; Valerates

2008
Sustained and efficient porphyrin generation in vivo using dendrimer conjugates of 5-ALA for photodynamic therapy.
    Journal of controlled release : official journal of the Controlled Release Society, 2009, Apr-17, Volume: 135, Issue:2

    Topics: Adenocarcinoma; Aminolevulinic Acid; Animals; Cell Line, Tumor; Cell Survival; Coloring Agents; Dendrimers; Dose-Response Relationship, Drug; Injections, Subcutaneous; Male; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Molecular Structure; Molecular Weight; Photochemotherapy; Photosensitizing Agents; Porphyrins; Protoporphyrins; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles; Time Factors; Xenograft Model Antitumor Assays

2009
Enhanced genetic instability and dasatinib sensitivity in mammary tumor cells lacking NEDD9.
    Cancer research, 2010, Nov-01, Volume: 70, Issue:21

    Topics: Adaptor Proteins, Signal Transducing; Animals; Aurora Kinases; Blotting, Western; Cell Adhesion; Cell Cycle; Cell Movement; Cell Proliferation; Dasatinib; Embryo, Mammalian; Female; Fibroblasts; Flow Cytometry; Fluorescent Antibody Technique; Lung Neoplasms; Mammary Glands, Animal; Mammary Neoplasms, Experimental; Mammary Tumor Virus, Mouse; Mice; Mice, SCID; NIH 3T3 Cells; Protein Kinase Inhibitors; Protein Serine-Threonine Kinases; Protein-Tyrosine Kinases; Proto-Oncogene Proteins c-akt; Pyrimidines; src-Family Kinases; Thiazoles; Xenograft Model Antitumor Assays

2010
RKI-1447 is a potent inhibitor of the Rho-associated ROCK kinases with anti-invasive and antitumor activities in breast cancer.
    Cancer research, 2012, Oct-01, Volume: 72, Issue:19

    Topics: Animals; Antineoplastic Agents; Binding Sites; Blotting, Western; Breast Neoplasms; Cell Line, Tumor; Cell Movement; Crystallography, X-Ray; Cytoskeleton; Humans; Mammary Neoplasms, Experimental; Mice; Mice, Transgenic; Models, Molecular; Molecular Structure; Neoplasm Invasiveness; NIH 3T3 Cells; Protein Binding; Protein Kinase Inhibitors; Protein Structure, Tertiary; rho-Associated Kinases; Substrate Specificity; Thiazoles; Tumor Burden; Urea

2012
Preclinical evaluation of amino acid prodrugs of novel antitumor 2-(4-amino-3-methylphenyl)benzothiazoles.
    Molecular cancer therapeutics, 2002, Volume: 1, Issue:4

    Topics: Amino Acids; Aniline Compounds; Animals; Antineoplastic Agents; Benzothiazoles; Blotting, Western; Cell Division; Cytochrome P-450 CYP1A1; Dogs; Dose-Response Relationship, Drug; Drug Evaluation, Preclinical; Female; Humans; Male; Mammary Neoplasms, Experimental; Mice; Mice, Nude; Ovarian Neoplasms; Prodrugs; Rats; Rats, Sprague-Dawley; Thiazoles; Tumor Cells, Cultured; Xenograft Model Antitumor Assays

2002
A cytoskeleton-based functional genetic screen identifies Bcl-xL as an enhancer of metastasis, but not primary tumor growth.
    Oncogene, 2004, Jun-03, Volume: 23, Issue:26

    Topics: Animals; bcl-X Protein; Breast Neoplasms; Bridged Bicyclo Compounds, Heterocyclic; Cytoskeleton; Genetic Techniques; Genetic Vectors; Humans; Mammary Neoplasms, Experimental; MAP Kinase Kinase 1; Mice; Mitogen-Activated Protein Kinase Kinases; Neoplasm Metastasis; Proto-Oncogene Proteins c-bcl-2; Thiazoles; Thiazolidines

2004
Peroxisome proliferator-activated receptor delta and gamma agonists differentially alter tumor differentiation and progression during mammary carcinogenesis.
    Cancer research, 2005, May-01, Volume: 65, Issue:9

    Topics: Animals; Anticarcinogenic Agents; Carcinoma, Adenosquamous; Carcinoma, Ductal; Carcinoma, Squamous Cell; Cell Differentiation; Disease Progression; Female; Gene Expression Profiling; Mammary Neoplasms, Experimental; Mice; Oxazoles; PPAR delta; PPAR gamma; Thiazoles; Tyrosine

2005
[131I]Iodoazomycin arabinoside for low-dose-rate isotope radiotherapy: radiolabeling, stability, long-term whole-body clearance and radiation dosimetry estimates in mice.
    Nuclear medicine and biology, 2005, Volume: 32, Issue:6

    Topics: Animals; Cell Hypoxia; Cell Proliferation; Female; Humans; Iodine Radioisotopes; Mammary Neoplasms, Experimental; Metabolic Clearance Rate; Mice; Mice, Inbred BALB C; Nitroimidazoles; Radioimmunotherapy; Radiometry; Radiopharmaceuticals; Radiotherapy Dosage; Tetrazolium Salts; Thiazoles; Tissue Distribution; Tumor Cells, Cultured

2005
Tumor production in germ-free rats fed 5-nitrofurans.
    Cancer letters, 1984, Volume: 21, Issue:3

    Topics: Animals; Biotransformation; Carcinogens; FANFT; Female; Germ-Free Life; Intestines; Mammary Neoplasms, Experimental; Neoplasms, Experimental; Nitrofurans; Nitrofurantoin; Rats; Rats, Inbred Strains; Thiazoles

1984
Mutagenicity, carcinogenicity, distribution, and nitroreduction of 4-(5-nitro-2-furyl)thiazole in the rat.
    Cancer research, 1981, Volume: 41, Issue:7

    Topics: Animals; Carcinogens; Chromatography, High Pressure Liquid; Diet; FANFT; Feces; Female; Gas Chromatography-Mass Spectrometry; Liver Neoplasms; Mammary Neoplasms, Experimental; Mutagens; Nitrofurans; Rats; Salmonella typhimurium; Stomach Neoplasms; Thiazoles; Tissue Distribution

1981
Evaluation of 2-amino-5-nitrothiazole as a hypoxic cell radiosensitizer.
    Radiation research, 1982, Volume: 90, Issue:3

    Topics: Animals; Cells, Cultured; Drug Evaluation; Escherichia coli; Female; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Radiation-Sensitizing Agents; Thiazoles

1982
In vivo selective modulation of tissue glutathione in a rat mammary carcinoma model.
    Biochemical pharmacology, 1995, Oct-26, Volume: 50, Issue:9

    Topics: Animals; Antimetabolites, Antineoplastic; Bone Marrow; Buthionine Sulfoximine; Drug Synergism; Female; Glutathione; Kidney; Liver; Mammary Neoplasms, Experimental; Methionine Sulfoximine; Pyrrolidonecarboxylic Acid; Rats; Rats, Inbred F344; Thiazoles; Thiazolidines; Tumor Cells, Cultured

1995
Therapeutic effect of clarithromycin on a transplanted tumor in rats.
    Antimicrobial agents and chemotherapy, 1999, Volume: 43, Issue:1

    Topics: Adenocarcinoma; Animals; Chromium Radioisotopes; Clarithromycin; Collagenases; Coloring Agents; Cytotoxicity, Immunologic; Humans; Interleukin-6; Male; Mammary Neoplasms, Experimental; Matrix Metalloproteinase 9; Neoplasm Transplantation; Rats; Rats, Inbred F344; Spleen; Tetrazolium Salts; Thiazoles; Transforming Growth Factor beta; Tumor Cells, Cultured; Tumor Necrosis Factor-alpha

1999
A ligand of peroxisome proliferator-activated receptor gamma, retinoids, and prevention of preneoplastic mammary lesions.
    Journal of the National Cancer Institute, 2000, Mar-01, Volume: 92, Issue:5

    Topics: 9,10-Dimethyl-1,2-benzanthracene; Animals; Anticarcinogenic Agents; Antineoplastic Agents; Carcinogens; Chromans; Estradiol; Female; Ligands; Mammary Glands, Animal; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Organ Culture Techniques; Precancerous Conditions; Progesterone; Receptors, Cytoplasmic and Nuclear; Receptors, Retinoic Acid; Retinoic Acid Receptor alpha; Retinoic Acid Receptor gamma; Retinoid X Receptors; Retinoids; Thiazoles; Thiazolidinediones; Transcription Factors; Tretinoin; Troglitazone

2000
Characterization of the effects of antiangiogenic agents on tumor pathophysiology.
    American journal of clinical oncology, 2001, Volume: 24, Issue:5

    Topics: Angiogenesis Inhibitors; Animals; Celecoxib; Cell Hypoxia; Cyclooxygenase 2; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Etanidazole; Hydrocarbons, Fluorinated; Image Processing, Computer-Assisted; Immunohistochemistry; Isoenzymes; Mammary Neoplasms, Experimental; Meloxicam; Mice; Mice, Inbred C3H; Models, Animal; Neovascularization, Pathologic; Prostaglandin-Endoperoxide Synthases; Pyrazoles; Sulfonamides; Thiazines; Thiazoles

2001
Inhibition of all-TRANS-retinoic acid metabolism by R116010 induces antitumour activity.
    British journal of cancer, 2002, Feb-12, Volume: 86, Issue:4

    Topics: Animals; Antineoplastic Agents; Benzothiazoles; Breast Neoplasms; Cell Division; Chromatography, High Pressure Liquid; Cytochrome P-450 Enzyme Inhibitors; Cytochrome P-450 Enzyme System; Dose-Response Relationship, Drug; Female; Humans; Imidazoles; Mammary Neoplasms, Experimental; Mice; Mice, Inbred Strains; Mixed Function Oxygenases; Retinoic Acid 4-Hydroxylase; Reverse Transcriptase Polymerase Chain Reaction; Thiazoles; Tretinoin; Tumor Cells, Cultured

2002
Cytotoxic and radiosensitizing effects of hypoxic cell sensitizers on EMT6 mouse mammary tumour cells in vivo and in vitro.
    The British journal of cancer. Supplement, 1978, Volume: 3

    Topics: Animals; Cell Survival; In Vitro Techniques; Lethal Dose 50; Mammary Neoplasms, Experimental; Mice; Mice, Inbred BALB C; Nitroimidazoles; Oxygen; Pyrroles; Radiation-Sensitizing Agents; Thiazoles

1978
The mode of action of the antitumour agent GP 48,989 in the rat.
    European journal of cancer, 1979, Volume: 15, Issue:5

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Castration; Female; Luteinizing Hormone; Mammary Neoplasms, Experimental; Neoplasm Transplantation; Ovary; Random Allocation; Rats; Receptors, Estrogen; Tamoxifen; Thiazoles; Time Factors; Transplantation, Homologous; Uterus

1979
Regression of "hormone-independent" DMBA-induced mammary carcinomas in response to GP 48989 and its effects on hormone receptors.
    Oncology, 1976, Volume: 33, Issue:5-6

    Topics: 9,10-Dimethyl-1,2-benzanthracene; Adenofibroma; Animals; Benz(a)Anthracenes; Carcinoma; Castration; Cytoplasm; Estradiol; Female; Mammary Neoplasms, Experimental; Rats; Receptors, Estrogen; Thiazoles; Thiazolidines

1976
Differential properties of cisplatin and tetraplatin with respect to cytotoxicity and perturbation of cellular glutathione levels.
    Cancer chemotherapy and pharmacology, 1991, Volume: 28, Issue:4

    Topics: Animals; Antineoplastic Agents; Cell Line; Cisplatin; Coloring Agents; Drug Resistance; Drug Screening Assays, Antitumor; Glutathione; Mammary Neoplasms, Experimental; Mice; Organoplatinum Compounds; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1991
Identification of anthracyclines and related agents that retain preferential activity over adriamycin in multidrug-resistant cell lines, and further resistance modification by verapamil and cyclosporin A.
    Cancer chemotherapy and pharmacology, 1989, Volume: 24, Issue:5

    Topics: Animals; Antibiotics, Antineoplastic; Carcinoma, Small Cell; Cell Line; Coloring Agents; Cyclosporins; Doxorubicin; Drug Resistance; Drug Screening Assays, Antitumor; Female; Humans; Lung Neoplasms; Mammary Neoplasms, Experimental; Mice; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured; Verapamil

1989
Antitumor efficacy in rats of CGP 19984, a thiazolidinedione derivative that inhibits luteinizing hormone secretion.
    Cancer research, 1986, Volume: 46, Issue:4 Pt 1

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Castration; Corticosterone; Female; Luteinizing Hormone; Male; Mammary Neoplasms, Experimental; Neoplasms, Hormone-Dependent; Prolactin; Prostatic Neoplasms; Rats; Rats, Inbred F344; Testosterone; Thiazoles; Thiazolidines

1986
Carcinogenicity of N-[4-(5-nitro-2-furyl)-2-thiazolyl] acetamide in female rats.
    Cancer research, 1970, Volume: 30, Issue:4

    Topics: Acetamides; Adenocarcinoma; Adenocarcinoma, Bronchiolo-Alveolar; Adenofibroma; Animals; Carcinogens; Carcinoma, Squamous Cell; Carcinoma, Transitional Cell; Chemical Phenomena; Chemistry; Female; Fibroma; Fibrosarcoma; Intestinal Neoplasms; Kidney Neoplasms; Liver Neoplasms; Lung Neoplasms; Lymphoma, Non-Hodgkin; Mammary Neoplasms, Experimental; Neoplasm Metastasis; Neoplasm Transplantation; Neoplasms, Experimental; Nitrofurans; Rats; Salivary Gland Neoplasms; Skin Neoplasms; Splenic Neoplasms; Thiazoles; Time Factors; Transplantation, Homologous

1970
Carcinogenicity of formic acid 2-[4-(5-nitro-2-furyl)-2-thiazolyl]-hydrazide in Swiss mice.
    Cancer research, 1970, Volume: 30, Issue:4

    Topics: Adenocarcinoma; Adenocarcinoma, Bronchiolo-Alveolar; Animals; Body Weight; Carcinogens; Carcinoma, Squamous Cell; Diet; Female; Formates; Hydrazines; Leukemia, Experimental; Liver Neoplasms; Lung Neoplasms; Mammary Neoplasms, Experimental; Mice; Neoplasm Metastasis; Neoplasms, Experimental; Nitrofurans; Skin Neoplasms; Stomach Neoplasms; Thiazoles; Uterine Neoplasms

1970
Comparative urinary and gallbladder carcinogenicity of N-(4-(5-nitro-2-furyl)-2-thiazolyl)formamide and N-(4-(5-nitro-2-furyl)-2-thiazolyl)acetamide in the dog.
    Journal of the National Cancer Institute, 1970, Volume: 45, Issue:3

    Topics: Acetamides; Adenocarcinoma; Adenocarcinoma, Scirrhous; Adenofibroma; Animals; Carcinogens; Carcinoma, Transitional Cell; Dogs; Female; Formamides; Gallbladder; Gallbladder Neoplasms; Kidney Neoplasms; Mammary Neoplasms, Experimental; Neoplasms, Experimental; Nitrofurans; Thiazoles; Ureteral Neoplasms; Urinary Bladder Neoplasms; Urogenital Neoplasms; Urogenital System

1970
Kinetics and inhibition of alkaline phosphatases from canine tissues.
    Biochimica et biophysica acta, 1972, Nov-10, Volume: 289, Issue:1

    Topics: Alkaline Phosphatase; Animals; Anthelmintics; Autoanalysis; Bone and Bones; Dogs; Escherichia coli; Ethanolamines; Female; Hydrogen-Ion Concentration; Imidazoles; Intestines; Kidney; Kinetics; Liver; Magnesium; Mammary Neoplasms, Experimental; Nitrophenols; Organ Specificity; Osmolar Concentration; Placenta; Pregnancy; Structure-Activity Relationship; Thiazoles

1972
Comparative carcinogenicity in the rat of 2-hydrazinothiazoles with nitrofuryl, nitrophenyl, or aminophenyl substituents in the 4-position.
    Cancer research, 1970, Volume: 30, Issue:4

    Topics: Adenocarcinoma; Adenofibroma; Animals; Body Weight; Carcinogens; Chemical Phenomena; Chemistry; Diet; Female; Hydrazines; Lung Neoplasms; Lymphoma, Non-Hodgkin; Mammary Neoplasms, Experimental; Neoplasm Metastasis; Neoplasms, Experimental; Nitrobenzenes; Nitrofurans; Rats; Salivary Gland Neoplasms; Splenic Neoplasms; Thiazoles

1970
Comparative carcinogenicity of formic acid 2-[4-(5-nitro-2-furyl)-2-thiazolyl]hydrazide and related chemicals in the rat.
    Journal of the National Cancer Institute, 1971, Volume: 47, Issue:2

    Topics: Animals; Carcinogens; Female; Formates; Furans; Hydrazines; Kidney Neoplasms; Liver Neoplasms; Male; Mammary Neoplasms, Experimental; Mice; Neoplasms, Experimental; Nitrofurans; Rats; Semicarbazides; Thiazoles

1971
Autoradiographic evaluation of the distribution of N,N'-bis(thiazole)-2,7-fluorene-disulphonamide-35S in organs of rats.
    Nature, 1965, Jun-19, Volume: 206, Issue:990

    Topics: Animals; Autoradiography; Carcinoma 256, Walker; Fluorenes; In Vitro Techniques; Kidney; Liver; Male; Mammary Neoplasms, Experimental; Rats; Spleen; Sulfonamides; Sulfur Isotopes; Thiazoles

1965