Page last updated: 2024-08-21

thiazoles and Experimental Leukemia

thiazoles has been researched along with Experimental Leukemia in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-199017 (73.91)18.7374
1990's2 (8.70)18.2507
2000's1 (4.35)29.6817
2010's3 (13.04)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Fei, F; Groffen, J; Heisterkamp, N; Kim, YM; Müschen, M; Stoddart, S1
Adamia, S; Barrett, R; Choi, HG; Deng, X; Gray, N; Griffin, JD; Kung, AL; Moreno, D; Ray, A; Weisberg, E1
Chang, CY; Chang, JY; Chang, KY; Chao, YS; Chen, CP; Chen, CT; Chen, TW; Chern, JH; Chuu, JJ; Ho, PY; Hu, CB; Huang, CL; Hwang, DR; Hwang, LL; Li, WT; Lin, CH; Lin, HL; Song, JS; Tung, FF; Wang, MH; Yeh, TK1
BURCHENAL, JH; COLEY, V; OETTGEN, HF; REPPERT, JA1
BURCHENAL, JH; COLEY, VC; KRAKOFF, IH; OETTGEN, HF; PURPLE, JR1
CIOTTI, CJ; GOLDIN, A; HUMPHREYS, SR; KAPLAN, NO; KLINE, I; VENDITTI, JM1
Cools, J; Cortes, J; Garcia-Manero, G; Gilliland, DG; Kantarjian, H; Lee, F; Lennon, PA; Manshouri, T; Quintás-Cardama, A; Tong, W; Vega, F1
Błaszczyk, B; Fiszer-Maliszewska, L; Giełdanowski, J; Kowalczyk-Bronisz, SH; Machoń, Z; Mordarski, M; Raberger, G; Wieczorek, J; Wieczorek, Z; Zimecki, M1
Bryan, GT; Ertürk, E; Headley, DB; Klopp, RG; Michie, PM1
Alvord, WG; Arthur, LO; Henderson, LE; Hewes, SM; Ott, DE1
Bryan, GT; Cohen, SM; Headley, DB1
Cheng, CC; Zee-Cheng, RK1
Bryan, GT; Cohen, SM1
Abe, T; Ohno, M1
Bonna, RL; Burns, ER; Elliot, GT; Kelly, KF; Wardlaw, TR1
Bielicki, L; Hohorst, HJ; Müller, K; Voelcker, G1
Anderson, WK; Mach, RH1
Bryan, GT; Cohen, SM; Ertürk, E3
Bryan, GT; Cohen, SM; Ertürk, E; Lower, GM1
Gutsche, W; Jungstand, W; Wohlrabe, K1
Deliwala, CV; Modi, JD; Sabnis, SS1

Other Studies

23 other study(ies) available for thiazoles and Experimental Leukemia

ArticleYear
Development of resistance to dasatinib in Bcr/Abl-positive acute lymphoblastic leukemia.
    Leukemia, 2010, Volume: 24, Issue:4

    Topics: Animals; Apoptosis; Blotting, Western; Cells, Cultured; Dasatinib; Drug Resistance, Neoplasm; Embryo, Mammalian; Fibroblasts; Fusion Proteins, bcr-abl; Humans; Leukemia, Experimental; Mice; Mice, Inbred NOD; Mice, Knockout; Mice, SCID; Phosphorylation; Precursor Cell Lymphoblastic Leukemia-Lymphoma; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Receptors, CXCR4; src-Family Kinases; Stromal Cells; Thiazoles

2010
Beneficial effects of combining a type II ATP competitive inhibitor with an allosteric competitive inhibitor of BCR-ABL for the treatment of imatinib-sensitive and imatinib-resistant CML.
    Leukemia, 2010, Volume: 24, Issue:7

    Topics: Adenosine Triphosphate; Animals; Antineoplastic Combined Chemotherapy Protocols; Benzamides; Cells, Cultured; Drug Resistance, Neoplasm; Drug Synergism; Fusion Proteins, bcr-abl; Imatinib Mesylate; Leukemia, Experimental; Mice; Piperazines; Precursor Cells, B-Lymphoid; Protein Kinase Inhibitors; Pyrimidines; Thiazoles; Xenograft Model Antitumor Assays

2010
BPR0C261 is a novel orally active antitumor agent with antimitotic and anti-angiogenic activities.
    Cancer science, 2011, Volume: 102, Issue:1

    Topics: Administration, Oral; Angiogenesis Inhibitors; Animals; Antimitotic Agents; Antineoplastic Agents; Apoptosis; Cell Cycle; Cell Line, Tumor; Dogs; Humans; Indoles; Leukemia, Experimental; Male; Mice; Mice, Inbred Strains; Microtubules; Rats; Rats, Sprague-Dawley; Thiazoles

2011
Effects of nicotinamide and related compounds on the antileukemic activity of 2-amino-1,3,4-thiadiazole.
    Cancer research, 1960, Volume: 20

    Topics: Animals; Leukemia, Experimental; Niacin; Niacinamide; Nicotinic Acids; Thiadiazoles; Thiazoles

1960
POTENTIATION OF THE ANTI-LEUKEMIC EFFECTS OF 2-AMINOTHIADIAZOLE BY ISONICOTINAMIDE AND DERIVATIVES.
    Cancer research, 1964, Volume: 24

    Topics: Amides; Animals; Antineoplastic Agents; Isonicotinic Acids; Leukemia; Leukemia L1210; Leukemia, Experimental; Mice; Niacinamide; Pharmacology; Pyridines; Research; Thiadiazoles; Thiazoles

1964
Toxicity and antileukemic effectiveness of pyridine derivatives and 1,3,4-thiadiazole derivatives in mice. Relationship to nicotinamide antagonism.
    Cancer research, 1962, Volume: 22

    Topics: Animals; Antineoplastic Agents; Leukemia, Experimental; Mice; Niacin; Niacinamide; Nicotinic Acids; Pyridines; Thiadiazoles; Thiazoles

1962
Activity of tyrosine kinase inhibitors against human NUP214-ABL1-positive T cell malignancies.
    Leukemia, 2008, Volume: 22, Issue:6

    Topics: Adaptor Proteins, Signal Transducing; Adult; Animals; Apoptosis; Benzamides; Blotting, Western; Cell Cycle; Cell Proliferation; Cell Survival; Dasatinib; Female; Humans; Imatinib Mesylate; In Situ Hybridization, Fluorescence; Leukemia-Lymphoma, Adult T-Cell; Leukemia, Experimental; Male; Mice; Mice, Inbred NOD; Mice, SCID; Nuclear Proteins; Oncogene Proteins, Fusion; Phosphorylation; Piperazines; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Reverse Transcriptase Polymerase Chain Reaction; STAT5 Transcription Factor; Thiazoles; Tumor Cells, Cultured

2008
Chemical, pharmacological and oncostatic properties of 5-(4'-hydroxybenzylidenoimino)-4, 6-diketo-4, 5, 6, 7-tetrahydropyrimidine-[4, 5-d]-3-methyl-isothiazole (compound IP-10).
    Archivum immunologiae et therapiae experimentalis, 1983, Volume: 31, Issue:5

    Topics: Animals; Antineoplastic Agents; Blood Cells; Bone Marrow; Carcinoma, Ehrlich Tumor; Cats; Central Nervous System; Chick Embryo; Dogs; Female; Guinea Pigs; Hemodynamics; Lethal Dose 50; Leukemia, Experimental; Lung Neoplasms; Male; Mass Spectrometry; Melanoma; Mice; Mice, Inbred Strains; Pyrimidinones; Rabbits; Rats; Rats, Inbred Strains; Sarcoma, Yoshida; Spectrophotometry, Infrared; Thiazoles

1983
Temporal comparisons of immune status and target organ histology in mice fed carcinogenic 5-nitrofurans and their nornitro analogs.
    Cancer research, 1981, Volume: 41, Issue:4

    Topics: Animals; Antibody Formation; Carcinogens; Diet; FANFT; Female; Furans; Immunity, Cellular; Leukemia, Experimental; Lymphoid Tissue; Mice; Mice, Inbred BALB C; Neoplasms, Experimental; Nitrofurans; Thiazoles; Time Factors; Urinary Bladder Neoplasms

1981
Inhibition of Friend virus replication by a compound that reacts with the nucleocapsid zinc finger: anti-retroviral effect demonstrated in vivo.
    Virology, 1998, Apr-10, Volume: 243, Issue:2

    Topics: Animals; Antiviral Agents; Benzothiazoles; Data Interpretation, Statistical; Friend murine leukemia virus; Leukemia, Experimental; Mice; Nucleocapsid; Retroviridae Infections; Retroviridae Proteins; Thiazoles; Tumor Virus Infections; Virus Replication; Zinc Fingers

1998
Suppression of antibody-mediated and cell-mediated murine immunity by the carcinogen N-[4-(5-nitro-2-furyl)-2-thiazolyl]acetamide.
    Cancer research, 1977, Volume: 37, Issue:4

    Topics: Animals; Antibody-Producing Cells; Carcinogens; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Graft vs Host Reaction; Immunity; Immunity, Cellular; Immunosuppressive Agents; Leukemia, Experimental; Leukemia, Lymphoid; Mice; Mice, Inbred BALB C; Neoplasms, Experimental; Nitrofurans; Thiazoles; Urinary Bladder Neoplasms

1977
Antileukemic activity of substituted ureidothiazoles, ureidothiadiazoles, and related compounds.
    Journal of medicinal chemistry, 1979, Volume: 22, Issue:1

    Topics: Animals; Antineoplastic Agents; Leukemia, Experimental; Mice; Structure-Activity Relationship; Thiadiazoles; Thiazoles; Urea

1979
Effect of p-hydroxyacetanilide, sodium sulfate, and L-methionine on the leukemogenicity of N-[4-(5-nitro-2-furyl)-2-thiazolyl]acetamide.
    Cancer research, 1978, Volume: 38, Issue:5

    Topics: Acetanilides; Animals; Carcinogens; Drug Interactions; Female; Hydrazines; Leukemia, Experimental; Leukemia, Lymphoid; Mice; Nitrofurans; Papilloma; Stomach Neoplasms; Sulfates; Thiazoles; Urinary Bladder Neoplasms

1978
Rapid colorimetric assay for the quantification of leukemia inhibitory factor (LIF) and interleukin-6 (IL-6).
    Journal of immunological methods, 1991, Dec-15, Volume: 145, Issue:1-2

    Topics: Animals; Colorimetry; Growth Inhibitors; Humans; In Vitro Techniques; Interleukin-6; Leukemia Inhibitory Factor; Leukemia, Experimental; Leukemia, Myeloid; Lymphokines; Mice; Oxidation-Reduction; Tetrazolium Salts; Thiazoles; Tumor Cells, Cultured

1991
In vitro antiproliferative activity of 2'-(2-hydroxyphenyl)-2'-thiazoline-4'-carboxylic acid and its methyl ester on L1210 and P388 murine neoplasms.
    Cancer chemotherapy and pharmacology, 1988, Volume: 21, Issue:3

    Topics: Animals; Cell Cycle; Cell Division; Depression, Chemical; Hydroxyurea; Imides; Leukemia L1210; Leukemia P388; Leukemia, Experimental; Mice; Thiazoles; Tumor Cells, Cultured

1988
Low toxicity cancer chemotherapy by suicide inactivation of DNA polymerase alpha holoenzyme: first results with new thiazolidinyl- and perhydrothiazinyl-ethyl-N-mustard-phosphamide esters.
    Journal of cancer research and clinical oncology, 1988, Volume: 114, Issue:3

    Topics: Animals; Antineoplastic Agents; DNA Polymerase II; Kinetics; Leukemia P388; Leukemia, Experimental; Mice; Nitrogen Mustard Compounds; Thiazines; Thiazoles; Thiazolidines

1988
Synthesis, chemical reactivity, and antileukemic activity of 5-substituted 6,7-bis(hydroxymethyl)pyrrolo[1,2-c]thiazole biscarbamates and the corresponding sulfoxides and sulfones.
    Journal of medicinal chemistry, 1987, Volume: 30, Issue:11

    Topics: Animals; Antineoplastic Agents; Carbamates; Leukemia P388; Leukemia, Experimental; Mice; Structure-Activity Relationship; Sulfones; Sulfoxides; Thiazoles

1987
Carcinogenicity of formic acid 2-[4-(5-nitro-2-furyl)-2-thiazolyl]-hydrazide in Swiss mice.
    Cancer research, 1970, Volume: 30, Issue:4

    Topics: Adenocarcinoma; Adenocarcinoma, Bronchiolo-Alveolar; Animals; Body Weight; Carcinogens; Carcinoma, Squamous Cell; Diet; Female; Formates; Hydrazines; Leukemia, Experimental; Liver Neoplasms; Lung Neoplasms; Mammary Neoplasms, Experimental; Mice; Neoplasm Metastasis; Neoplasms, Experimental; Nitrofurans; Skin Neoplasms; Stomach Neoplasms; Thiazoles; Uterine Neoplasms

1970
Comparative carcinogenicity in Swiss mice of N-(4-(5-nitro-2-furyl)-2-thiazolyl)acetamide and structurally related 5-nitrofurans and 4-nitrobenzenes.
    Cancer research, 1973, Volume: 33, Issue:7

    Topics: Acetamides; Animals; Carcinogens; Carcinoma, Squamous Cell; Female; Formamides; Leukemia, Experimental; Leukemia, Lymphoid; Mice; Neoplasms, Experimental; Nitrobenzenes; Nitrofurans; Papilloma; Stomach Neoplasms; Structure-Activity Relationship; Thiazoles; Thioacetamide; Urinary Bladder Neoplasms

1973
[3-step test for screening potential cancerostatics. 1. Screening program and results of the 1st step].
    Arzneimittel-Forschung, 1971, Volume: 21, Issue:3

    Topics: Animals; Antineoplastic Agents; Azo Compounds; Benzimidazoles; Carcinoma, Ehrlich Tumor; Ethers; Hydrazines; Leukemia, Experimental; Leukemia, Myeloid; Mice; Nitrogen Mustard Compounds; Purines; Sarcoma, Experimental; Thiazoles

1971
Urinary bladder carcinogenicity of N-[4-(5-nitro-2-furyl)-2-thiazolyl] formamide in female Swiss mice.
    Cancer research, 1970, Volume: 30, Issue:5

    Topics: Amides; Animals; Female; Leukemia, Experimental; Lung Neoplasms; Male; Mice; Neoplasms, Experimental; Pregnancy; Thiazoles; Urinary Bladder Neoplasms; Uterine Neoplasms

1970
Potential anticancer agents. 3. Schiff bases from benzaldehyde nitrogen mustards and aminophenylthiazoles.
    Journal of medicinal chemistry, 1970, Volume: 13, Issue:5

    Topics: Aldehydes; Amines; Animals; Antineoplastic Agents; Carcinoma 256, Walker; Chemical Phenomena; Chemistry; Leukemia L1210; Leukemia, Experimental; Nitrogen Mustard Compounds; Thiazoles

1970
Production of leukemia and stomach neoplasms in Swiss, RF, BALB-c, and C3H female mice by feeding N-[4-(5-nitro-2-furyl)-2-thiazolyl]acetamide.
    Cancer research, 1970, Volume: 30, Issue:9

    Topics: Acetates; Adenoma; Amides; Animals; Anti-Bacterial Agents; Carcinogens; Carcinoma, Squamous Cell; Diet; Female; Leukemia, Experimental; Leukemia, Lymphoid; Lung Neoplasms; Mice; Neoplasms, Experimental; Nitrofurans; Species Specificity; Stomach Neoplasms; Thiazoles

1970