Page last updated: 2024-08-21

thiazoles and Cocaine-Related Disorders

thiazoles has been researched along with Cocaine-Related Disorders in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (3.85)18.2507
2000's14 (53.85)29.6817
2010's10 (38.46)24.3611
2020's1 (3.85)2.80

Authors

AuthorsStudies
Gobin, CM; Hámor, PU; Schwendt, M1
Hadad, NA; Hiller, H; Knackstedt, LA; Krause, EG; Namba, MD; Schwendt, M; Shallcross, J; Wu, L1
Knackstedt, LA; Schwendt, M; Trantham-Davidson, HL1
Baldaia, MA; Berro, LF; Frussa-Filho, R; Hollais, AW; Longo, BM; Marinho, EA; Oliveira-Lima, AJ; Santos, R; Wuo-Silva, R1
Arreola, AC; Kimmey, BA; Pierce, RC; Schmidt, HD1
Scheyer, AF; Tseng, KY; Wolf, ME1
Kim, JH; Lawrence, AJ; Perry, CJ; Reed, F; Zbukvic, IC1
Alvarez, Jdo N; Carvalho, Rde C; Frussa-Filho, R; Fukushiro, DF; Ribeiro, LT; Ricardo, VP1
Heard, K; Krier, S; Zahniser, NR1
Anderson, SM; Famous, KR; Kumaresan, V; Pierce, RC; Schmidt, HD; Yee, J; Yuan, M1
Hao, Y; Martin-Fardon, R; Weiss, F1
Martin-Fardon, R; Weiss, F1
Kalivas, PW; Knackstedt, L; Moussawi, K; Shen, H; Wang, X1
Erdur, B; Ergin, A; Kortunay, S; Yuksel, A1
Davidson, C; Ellinwood, EH; King, GR; Lee, TH; Yu, GZ1
Dew, RE; Hughes, D1
Bloch, DA; Ciraulo, AM; Ciraulo, DA; Elkashef, A; Knapp, CM; Leiderman, DB; LoCastro, J; Montgomery, MA; Sarid-Segal, O1
Cleveland, NJ; Dewitt, CD; Heard, K1
Ciraulo, DA; Hennen, J; Jensen, JE; Ke, Y; Knapp, C; Kwak, T; Meyer, AA; Nassar, LE; Renshaw, PF; Sarid-Segal, O; Streeter, CC1
Davis, J; Goeders, NE; Grajkowska, E; Iso, Y; Johnson, KM; Kozikowski, AP; Roth, BL; Sanker, S; Tueckmantel, W; Wroblewski, JT1
Bespalov, AY; Danysz, W; Dravolina, OA1
Feng, MJ; Yan, QS; Yan, SE1
Cleveland, NR; Heard, K; Krier, S1
Hoffman, RS; Manini, AF; Pearl-Davis, MS; Wu, S1
Fishback, JA; Green, AM; Kaushal, N; Matsumoto, RR; McCurdy, CR; Mésangeau, C; Narayanan, S; Poupaert, JH; Shaikh, J; Viard, E; Xu, YT1
Fredman, SJ; Rosenbaum, JF1

Trials

2 trial(s) available for thiazoles and Cocaine-Related Disorders

ArticleYear
Efficacy screening trials of paroxetine, pentoxifylline, riluzole, pramipexole and venlafaxine in cocaine dependence.
    Addiction (Abingdon, England), 2005, Volume: 100 Suppl 1

    Topics: Adolescent; Adult; Antidepressive Agents; Benzothiazoles; Cocaine-Related Disorders; Cyclohexanols; Dopamine Agonists; Double-Blind Method; Female; Humans; Male; Middle Aged; Neuroprotective Agents; Paroxetine; Pentoxifylline; Phosphodiesterase Inhibitors; Pramipexole; Riluzole; Selective Serotonin Reuptake Inhibitors; Thiazoles; Venlafaxine Hydrochloride

2005
Prefrontal GABA levels in cocaine-dependent subjects increase with pramipexole and venlafaxine treatment.
    Psychopharmacology, 2005, Volume: 182, Issue:4

    Topics: Adult; Antidepressive Agents, Second-Generation; Antioxidants; Benzothiazoles; Cocaine-Related Disorders; Cyclohexanols; Double-Blind Method; Female; gamma-Aminobutyric Acid; Humans; Magnetic Resonance Spectroscopy; Male; Middle Aged; Nicotine; Pramipexole; Prefrontal Cortex; Protons; Retrospective Studies; Thiazoles; Time Factors; Venlafaxine Hydrochloride

2005

Other Studies

24 other study(ies) available for thiazoles and Cocaine-Related Disorders

ArticleYear
The role of glutamate mGlu5 and adenosine A2a receptor interactions in regulating working memory performance and persistent cocaine seeking in rats.
    Progress in neuro-psychopharmacology & biological psychiatry, 2020, 12-20, Volume: 103

    Topics: Adenosine A2 Receptor Antagonists; Animals; Cocaine-Related Disorders; Conditioning, Operant; Drug-Seeking Behavior; Male; Memory, Short-Term; Motor Activity; Piperidines; Psychomotor Performance; Purines; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Receptor, Metabotropic Glutamate 5; Recurrence; Self Administration; Thiazoles

2020
A novel rat model of comorbid PTSD and addiction reveals intersections between stress susceptibility and enhanced cocaine seeking with a role for mGlu5 receptors.
    Translational psychiatry, 2018, 10-05, Volume: 8, Issue:1

    Topics: Animals; Anxiety; Behavior, Animal; Brain; Cocaine; Cocaine-Related Disorders; Comorbidity; Disease Models, Animal; Drug-Seeking Behavior; Extinction, Psychological; Fear; Male; Phenotype; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Resilience, Psychological; Stress Disorders, Post-Traumatic; Stress, Psychological; Thiazoles

2018
The role of ventral and dorsal striatum mGluR5 in relapse to cocaine-seeking and extinction learning.
    Addiction biology, 2014, Volume: 19, Issue:1

    Topics: Allosteric Regulation; Analysis of Variance; Animals; Basal Ganglia; Biotinylation; Blotting, Western; Cocaine; Cocaine-Related Disorders; Cues; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Electrophysiological Phenomena; Extinction, Psychological; Infusions, Intravenous; Locomotion; Long-Term Synaptic Depression; Male; Microinjections; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Recurrence; Self Administration; Sucrose; Thiazoles

2014
Selective action of an atypical neuroleptic on the mechanisms related to the development of cocaine addiction: a pre-clinical behavioural study.
    The international journal of neuropsychopharmacology, 2014, Volume: 17, Issue:4

    Topics: Animals; Antipsychotic Agents; Aripiprazole; Behavior, Animal; Central Nervous System Sensitization; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Antagonists; Dopamine Uptake Inhibitors; Haloperidol; Male; Mice; Motor Activity; Piperazines; Quinolones; Thiazoles

2014
Group I metabotropic glutamate receptor-mediated activation of PKC gamma in the nucleus accumbens core promotes the reinstatement of cocaine seeking.
    Addiction biology, 2015, Volume: 20, Issue:2

    Topics: Animals; Benzimidazoles; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Agonists; Excitatory Amino Acid Antagonists; Glycine; Nucleus Accumbens; Phosphorylation; Protein Kinase C; Protein Kinase C beta; Protein Kinase C-alpha; Pyridines; Rats; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Resorcinols; Thiazoles

2015
A protein synthesis-dependent mechanism sustains calcium-permeable AMPA receptor transmission in nucleus accumbens synapses during withdrawal from cocaine self-administration.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Feb-19, Volume: 34, Issue:8

    Topics: Animals; Benzoates; Calcium; Cocaine-Related Disorders; Cycloheximide; Excitatory Amino Acid Antagonists; Glycine; Male; Methoxyhydroxyphenylglycol; Nucleus Accumbens; Patch-Clamp Techniques; Protein Biosynthesis; Protein Synthesis Inhibitors; Pyridines; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Self Administration; Substance Withdrawal Syndrome; Synapses; Synaptic Transmission; Thiazoles; Ventral Tegmental Area

2014
The metabotropic glutamate 5 receptor is necessary for extinction of cocaine-associated cues.
    British journal of pharmacology, 2016, Volume: 173, Issue:6

    Topics: Animals; Benzamides; Cocaine; Cocaine-Related Disorders; Conditioning, Psychological; Cues; Male; Pyrazoles; Pyridines; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Thiazoles

2016
Haloperidol (but not ziprasidone) withdrawal potentiates sensitization to the hyperlocomotor effect of cocaine in mice.
    Brain research bulletin, 2008, Sep-30, Volume: 77, Issue:2-3

    Topics: Animals; Antipsychotic Agents; Behavior, Animal; Cocaine; Cocaine-Related Disorders; Haloperidol; Humans; Male; Mice; Motor Activity; Piperazines; Schizophrenia; Substance Withdrawal Syndrome; Thiazoles

2008
Administration of ziprasidone for 10 days increases cocaine toxicity in mice.
    Human & experimental toxicology, 2008, Volume: 27, Issue:6

    Topics: Animals; Antipsychotic Agents; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug Synergism; Longevity; Male; Mice; Mice, Inbred Strains; Piperazines; Seizures; Thiazoles; Time Factors; Withholding Treatment

2008
Metabotropic glutamate receptor 5 (mGluR5) antagonists attenuate cocaine priming- and cue-induced reinstatement of cocaine seeking.
    Behavioural brain research, 2009, Sep-14, Volume: 202, Issue:2

    Topics: Animals; Catheterization; Cocaine; Cocaine-Related Disorders; Cues; Dietary Sucrose; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Extinction, Psychological; Male; Microinjections; Nucleus Accumbens; Pyridines; Rats; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Self Administration; Thiazoles

2009
Behavioral and functional evidence of metabotropic glutamate receptor 2/3 and metabotropic glutamate receptor 5 dysregulation in cocaine-escalated rats: factor in the transition to dependence.
    Biological psychiatry, 2010, Aug-01, Volume: 68, Issue:3

    Topics: Amino Acids; Analysis of Variance; Animals; Behavior, Addictive; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Depressants; Cocaine; Cocaine-Related Disorders; Dose-Response Relationship, Drug; Excitatory Amino Acid Agonists; Male; Pyridines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Reinforcement Schedule; Self Administration; Thiazoles

2010
(-)-2-oxa-4-aminobicylco[3.1.0]hexane-4,6-dicarboxylic acid (LY379268) and 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]piperidine (MTEP) similarly attenuate stress-induced reinstatement of cocaine seeking.
    Addiction biology, 2012, Volume: 17, Issue:3

    Topics: Amino Acids; Analysis of Variance; Animals; Bridged Bicyclo Compounds, Heterocyclic; Central Nervous System Stimulants; Cocaine-Related Disorders; Conditioning, Operant; Excitatory Amino Acid Antagonists; Extinction, Psychological; Male; Piperidines; Rats; Rats, Wistar; Receptors, Metabotropic Glutamate; Stress, Psychological; Thiazoles

2012
Role of mGluR5 neurotransmission in reinstated cocaine-seeking.
    Addiction biology, 2013, Volume: 18, Issue:1

    Topics: Analysis of Variance; Animals; Biotinylation; Blotting, Western; Carrier Proteins; Cocaine; Cocaine-Related Disorders; Cues; Disease Models, Animal; Dopamine Uptake Inhibitors; Drug-Seeking Behavior; Excitatory Amino Acid Agonists; Extinction, Psychological; Glycine; Homer Scaffolding Proteins; Male; Microinjections; Nucleus Accumbens; Phenylacetates; Protein Binding; Protein Transport; Pyridines; Rats, Sprague-Dawley; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Recurrence; Self Administration; Synaptic Transmission; Thiazoles

2013
Assessment of propofol, midazolam and ziprasidone, or the combinations for the prevention of acute cocaine toxicity in a mouse model.
    Environmental toxicology and pharmacology, 2013, Volume: 35, Issue:1

    Topics: Animals; Anticonvulsants; Antipsychotic Agents; Cocaine-Related Disorders; Disease Models, Animal; Dopamine Antagonists; Drug Therapy, Combination; GABA Modulators; Male; Mice; Midazolam; Piperazines; Propofol; Seizures; Serotonin Antagonists; Thiazoles

2013
Effect of daily dosing duration of direct and indirect dopamine receptor agonists: cocaine cross-tolerance following chronic regimens.
    European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology, 2002, Volume: 12, Issue:5

    Topics: Analysis of Variance; Animals; Area Under Curve; Autoreceptors; Benzothiazoles; Cocaine; Cocaine-Related Disorders; Cross-Over Studies; Dopamine Agonists; Dopamine Uptake Inhibitors; Drug Administration Schedule; Drug Interactions; Male; Motor Activity; Piperazines; Pramipexole; Psychomotor Performance; Rats; Rats, Sprague-Dawley; Thiazoles; Time Factors

2002
Acute dystonic reaction with moderate-dose ziprasidone.
    Journal of clinical psychopharmacology, 2004, Volume: 24, Issue:5

    Topics: Acute Disease; Adult; Alcoholism; Antipsychotic Agents; Cocaine-Related Disorders; Dystonic Disorders; Female; Hallucinations; Humans; Piperazines; Risk Factors; Thiazoles; Tongue Diseases; Torticollis; Violence

2004
Ziprasidone pretreatment attenuates the lethal effects of cocaine in a mouse model.
    Academic emergency medicine : official journal of the Society for Academic Emergency Medicine, 2005, Volume: 12, Issue:5

    Topics: Acute Disease; Animals; Antipsychotic Agents; Cocaine; Cocaine-Related Disorders; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Overdose; Injections, Intraperitoneal; Mice; Piperazines; Premedication; Random Allocation; Seizures; Single-Blind Method; Survival Analysis; Thiazoles; Treatment Outcome

2005
Synthesis and structure-activity relationships of 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine analogues as potent, noncompetitive metabotropic glutamate receptor subtype 5 antagonists; search for cocaine medications.
    Journal of medicinal chemistry, 2006, Feb-09, Volume: 49, Issue:3

    Topics: Allosteric Site; Animals; Cell Line; Cocaine; Cocaine-Related Disorders; Cricetinae; Cricetulus; Humans; Ligands; Male; Narcotics; Pyridines; Radioligand Assay; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Self Administration; Structure-Activity Relationship; Thiazoles

2006
Effects of group I metabotropic glutamate receptor antagonists on the behavioral sensitization to motor effects of cocaine in rats.
    Psychopharmacology, 2006, Volume: 187, Issue:4

    Topics: Analysis of Variance; Animals; Behavior, Animal; Central Nervous System Stimulants; Cocaine; Cocaine-Related Disorders; Dose-Response Relationship, Drug; Excitatory Amino Acid Antagonists; Male; Motor Activity; Pyridines; Quinolines; Rats; Rats, Wistar; Receptor, Metabotropic Glutamate 5; Receptors, Metabotropic Glutamate; Thiazoles; Time Factors

2006
RNA interference-mediated inhibition of brain-derived neurotrophic factor expression increases cocaine's cytotoxicity in cultured cells.
    Neuroscience letters, 2007, Mar-06, Volume: 414, Issue:2

    Topics: Animals; Brain; Brain-Derived Neurotrophic Factor; Cell Death; Cell Line, Tumor; Cells, Cultured; Cocaine; Cocaine-Related Disorders; Dopamine Uptake Inhibitors; Down-Regulation; Gene Expression Regulation; Humans; Neurons; Rats; Rats, Sprague-Dawley; RNA Interference; RNA, Messenger; RNA, Small Interfering; Tetrazolium Salts; Thiazoles; Transfection

2007
Ziprasidone, diazepam, or the combination for prevention of cocaine toxicity in a mouse model.
    Academic emergency medicine : official journal of the Society for Academic Emergency Medicine, 2007, Volume: 14, Issue:8

    Topics: Animals; Cocaine; Cocaine-Related Disorders; Confidence Intervals; Diazepam; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Therapy, Combination; Male; Mice; Mice, Inbred Strains; Piperazines; Random Allocation; Reference Values; Sensitivity and Specificity; Statistics, Nonparametric; Survival Rate; Thiazoles

2007
Use of antipsychotics to treat cocaine toxicity?
    Academic emergency medicine : official journal of the Society for Academic Emergency Medicine, 2008, Volume: 15, Issue:1

    Topics: Animals; Antipsychotic Agents; Cocaine; Cocaine-Related Disorders; Diazepam; Disease Models, Animal; Mice; Piperazines; Thiazoles; Treatment Outcome

2008
Conversion of a highly selective sigma-1 receptor-ligand to sigma-2 receptor preferring ligands with anticocaine activity.
    Journal of medicinal chemistry, 2008, Mar-13, Volume: 51, Issue:5

    Topics: Animals; Anticonvulsants; Brain; Cocaine; Cocaine-Related Disorders; In Vitro Techniques; Ligands; Mice; Oxazoles; Piperazines; Radioligand Assay; Rats; Receptors, sigma; Seizures; Sigma-1 Receptor; Structure-Activity Relationship; Thiazoles

2008
Pramipexole treatment for cocaine cravings.
    The American journal of psychiatry, 1999, Volume: 156, Issue:11

    Topics: Adult; Antidepressive Agents; Behavior, Addictive; Benzothiazoles; Bipolar Disorder; Cocaine-Related Disorders; Comorbidity; Diagnosis, Dual (Psychiatry); Dopamine Agonists; Drug Therapy, Combination; Humans; Lamotrigine; Male; Pramipexole; Thiazoles; Treatment Outcome; Triazines

1999