thiazoles has been researched along with African Sleeping Sickness in 10 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 2 (20.00) | 18.7374 |
1990's | 0 (0.00) | 18.2507 |
2000's | 1 (10.00) | 29.6817 |
2010's | 6 (60.00) | 24.3611 |
2020's | 1 (10.00) | 2.80 |
Authors | Studies |
---|---|
Comini, MA; Franco, J; Scarone, L | 1 |
Chung, MC; Dos Santos, JL; Ferreira, CMR; Jornada, DH; Machado, MGM; Scarim, CB | 1 |
Erath, J; Ferrins, L; Gillingwater, K; Leed, SE; Mehta, N; Mensa-Wilmot, K; Pollastri, MP; Rodriguez, A; Sciotti, RJ; Sharma, A; Tanghe, S; Thomas, SM | 1 |
Ding, Q; Ge, J; Jiang, Z; Liu, D; Luo, P; Peng, Y | 1 |
Behera, R; Edwards, P; Guyett, PJ; Karver, CE; Mensa-Wilmot, K; Patel, G; Pollastri, MP; Roncal, NE; Sullenberger, C | 1 |
Engman, L; Gustafsson, TN; Gustavsson, AL; Holmgren, A; Johansson, HA; Kumar, S; Lu, J; Rottenberg, ME; Sjöberg, B; Tjernberg, A; Vodnala, SK | 1 |
Barrett, MP; Bradley, B; Kennedy, PG; Rodgers, J; Stone, TW | 1 |
Boykin, DW; Branowska, D; Brun, R; Farahat, AA; Kumar, A; Liu, Y; Wenzler, T; Wilson, WD | 1 |
Cerami, A; Ulrich, P | 1 |
Roffey, P; Verge, JP | 1 |
1 review(s) available for thiazoles and African Sleeping Sickness
Article | Year |
---|---|
Thiazole, thio and semicarbazone derivatives against tropical infective diseases: Chagas disease, human African trypanosomiasis (HAT), leishmaniasis, and malaria.
Topics: Animals; Chagas Disease; Drug Design; Humans; Leishmaniasis; Malaria; Protozoan Infections; Semicarbazones; Thiazoles; Thiosemicarbazones; Trypanosomiasis, African | 2019 |
9 other study(ies) available for thiazoles and African Sleeping Sickness
Article | Year |
---|---|
Novel distamycin analogues that block the cell cycle of African trypanosomes with high selectivity and potency.
Topics: Animals; Cell Cycle; Distamycins; Female; Macrophages; Mice; Mice, Inbred BALB C; Thiazoles; Trypanocidal Agents; Trypanosoma; Trypanosoma brucei brucei; Trypanosomiasis, African | 2020 |
Anilinoquinoline based inhibitors of trypanosomatid proliferation.
Topics: Animals; Antiprotozoal Agents; Cell Proliferation; Chagas Disease; Female; Humans; Leishmania; Leishmaniasis; Mice; Thiazoles; Trypanosoma brucei brucei; Trypanosoma cruzi; Trypanosomiasis, African | 2018 |
Synthesis of 2-Arylbenzothiazole and 2-Arylthiazole Derivatives via a Ru-Catalyzed
Topics: Benzothiazoles; Catalysis; Humans; Molecular Structure; Nitrates; Ruthenium; Stereoisomerism; Thiazoles; Trypanocidal Agents; Trypanosomiasis, African | 2019 |
Kinase scaffold repurposing for neglected disease drug discovery: discovery of an efficacious, lapatinib-derived lead compound for trypanosomiasis.
Topics: Animals; Cell Cycle; Cell Line, Tumor; Cell Survival; Coloring Agents; Drug Design; Drug Discovery; ErbB Receptors; Humans; Indicators and Reagents; Lapatinib; Morpholines; Neglected Diseases; Phosphotransferases; Quinazolines; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 2013 |
Ebsulfur is a benzisothiazolone cytocidal inhibitor targeting the trypanothione reductase of Trypanosoma brucei.
Topics: Animals; Male; Mice; NADH, NADPH Oxidoreductases; Platelet Aggregation Inhibitors; Protozoan Proteins; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 2013 |
Kynurenine pathway inhibition reduces central nervous system inflammation in a model of human African trypanosomiasis.
Topics: Animals; Blood-Brain Barrier; Central Nervous System Protozoal Infections; Female; Inhibitory Concentration 50; Kynurenine; Mice; Mice, Inbred Strains; Pentamidine; Signal Transduction; Sulfonamides; Thiazoles; Time Factors; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 2009 |
Synthesis and antiprotozoal activity of 2,5-bis[amidinoaryl]thiazoles.
Topics: Administration, Oral; Animals; Antimalarials; Antiprotozoal Agents; Disease Models, Animal; DNA, Protozoan; Drug Stability; Malaria, Falciparum; Mice; Parasitic Sensitivity Tests; Pentamidine; Plasmodium falciparum; Rats; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 2010 |
Potential antitrypanosomal agents. 1,N2-Disubstituted 2-amino-5-hydroxy-4-methylnaphtho[1,2-d]thiazolium salts and related compounds.
Topics: Animals; Chemical Phenomena; Chemistry; Female; Mice; Rats; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African | 1982 |
Antiprotozoal Thiazoles. 2-(5-Nitro-2-thienyl)thiazoles.
Topics: Administration, Oral; Animals; Chagas Disease; Injections, Intraperitoneal; Lethal Dose 50; Mice; Nitro Compounds; Thiazoles; Thiophenes; Trypanocidal Agents; Trypanosomiasis, African | 1975 |