Page last updated: 2024-08-21

thiazoles and African Sleeping Sickness

thiazoles has been researched along with African Sleeping Sickness in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19902 (20.00)18.7374
1990's0 (0.00)18.2507
2000's1 (10.00)29.6817
2010's6 (60.00)24.3611
2020's1 (10.00)2.80

Authors

AuthorsStudies
Comini, MA; Franco, J; Scarone, L1
Chung, MC; Dos Santos, JL; Ferreira, CMR; Jornada, DH; Machado, MGM; Scarim, CB1
Erath, J; Ferrins, L; Gillingwater, K; Leed, SE; Mehta, N; Mensa-Wilmot, K; Pollastri, MP; Rodriguez, A; Sciotti, RJ; Sharma, A; Tanghe, S; Thomas, SM1
Ding, Q; Ge, J; Jiang, Z; Liu, D; Luo, P; Peng, Y1
Behera, R; Edwards, P; Guyett, PJ; Karver, CE; Mensa-Wilmot, K; Patel, G; Pollastri, MP; Roncal, NE; Sullenberger, C1
Engman, L; Gustafsson, TN; Gustavsson, AL; Holmgren, A; Johansson, HA; Kumar, S; Lu, J; Rottenberg, ME; Sjöberg, B; Tjernberg, A; Vodnala, SK1
Barrett, MP; Bradley, B; Kennedy, PG; Rodgers, J; Stone, TW1
Boykin, DW; Branowska, D; Brun, R; Farahat, AA; Kumar, A; Liu, Y; Wenzler, T; Wilson, WD1
Cerami, A; Ulrich, P1
Roffey, P; Verge, JP1

Reviews

1 review(s) available for thiazoles and African Sleeping Sickness

ArticleYear
Thiazole, thio and semicarbazone derivatives against tropical infective diseases: Chagas disease, human African trypanosomiasis (HAT), leishmaniasis, and malaria.
    European journal of medicinal chemistry, 2019, Jan-15, Volume: 162

    Topics: Animals; Chagas Disease; Drug Design; Humans; Leishmaniasis; Malaria; Protozoan Infections; Semicarbazones; Thiazoles; Thiosemicarbazones; Trypanosomiasis, African

2019

Other Studies

9 other study(ies) available for thiazoles and African Sleeping Sickness

ArticleYear
Novel distamycin analogues that block the cell cycle of African trypanosomes with high selectivity and potency.
    European journal of medicinal chemistry, 2020, Mar-01, Volume: 189

    Topics: Animals; Cell Cycle; Distamycins; Female; Macrophages; Mice; Mice, Inbred BALB C; Thiazoles; Trypanocidal Agents; Trypanosoma; Trypanosoma brucei brucei; Trypanosomiasis, African

2020
Anilinoquinoline based inhibitors of trypanosomatid proliferation.
    PLoS neglected tropical diseases, 2018, Volume: 12, Issue:11

    Topics: Animals; Antiprotozoal Agents; Cell Proliferation; Chagas Disease; Female; Humans; Leishmania; Leishmaniasis; Mice; Thiazoles; Trypanosoma brucei brucei; Trypanosoma cruzi; Trypanosomiasis, African

2018
Synthesis of 2-Arylbenzothiazole and 2-Arylthiazole Derivatives via a Ru-Catalyzed
    The Journal of organic chemistry, 2019, 10-18, Volume: 84, Issue:20

    Topics: Benzothiazoles; Catalysis; Humans; Molecular Structure; Nitrates; Ruthenium; Stereoisomerism; Thiazoles; Trypanocidal Agents; Trypanosomiasis, African

2019
Kinase scaffold repurposing for neglected disease drug discovery: discovery of an efficacious, lapatinib-derived lead compound for trypanosomiasis.
    Journal of medicinal chemistry, 2013, May-23, Volume: 56, Issue:10

    Topics: Animals; Cell Cycle; Cell Line, Tumor; Cell Survival; Coloring Agents; Drug Design; Drug Discovery; ErbB Receptors; Humans; Indicators and Reagents; Lapatinib; Morpholines; Neglected Diseases; Phosphotransferases; Quinazolines; Structure-Activity Relationship; Tetrazolium Salts; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2013
Ebsulfur is a benzisothiazolone cytocidal inhibitor targeting the trypanothione reductase of Trypanosoma brucei.
    The Journal of biological chemistry, 2013, Sep-20, Volume: 288, Issue:38

    Topics: Animals; Male; Mice; NADH, NADPH Oxidoreductases; Platelet Aggregation Inhibitors; Protozoan Proteins; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2013
Kynurenine pathway inhibition reduces central nervous system inflammation in a model of human African trypanosomiasis.
    Brain : a journal of neurology, 2009, Volume: 132, Issue:Pt 5

    Topics: Animals; Blood-Brain Barrier; Central Nervous System Protozoal Infections; Female; Inhibitory Concentration 50; Kynurenine; Mice; Mice, Inbred Strains; Pentamidine; Signal Transduction; Sulfonamides; Thiazoles; Time Factors; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2009
Synthesis and antiprotozoal activity of 2,5-bis[amidinoaryl]thiazoles.
    Bioorganic & medicinal chemistry, 2010, May-15, Volume: 18, Issue:10

    Topics: Administration, Oral; Animals; Antimalarials; Antiprotozoal Agents; Disease Models, Animal; DNA, Protozoan; Drug Stability; Malaria, Falciparum; Mice; Parasitic Sensitivity Tests; Pentamidine; Plasmodium falciparum; Rats; Stereoisomerism; Structure-Activity Relationship; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2010
Potential antitrypanosomal agents. 1,N2-Disubstituted 2-amino-5-hydroxy-4-methylnaphtho[1,2-d]thiazolium salts and related compounds.
    Journal of medicinal chemistry, 1982, Volume: 25, Issue:6

    Topics: Animals; Chemical Phenomena; Chemistry; Female; Mice; Rats; Thiazoles; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

1982
Antiprotozoal Thiazoles. 2-(5-Nitro-2-thienyl)thiazoles.
    Journal of medicinal chemistry, 1975, Volume: 18, Issue:8

    Topics: Administration, Oral; Animals; Chagas Disease; Injections, Intraperitoneal; Lethal Dose 50; Mice; Nitro Compounds; Thiazoles; Thiophenes; Trypanocidal Agents; Trypanosomiasis, African

1975