tamsulosin has been researched along with Muscle Contraction in 58 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 0 (0.00) | 18.7374 |
1990's | 17 (29.31) | 18.2507 |
2000's | 24 (41.38) | 29.6817 |
2010's | 16 (27.59) | 24.3611 |
2020's | 1 (1.72) | 2.80 |
Authors | Studies |
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Cheung, P; Evangelisto, M; Jolliffe, L; Kuo, GH; Murray, WV; Prouty, C; Pulito, V; Varga, S; Wang, J | 1 |
Amorim, AC; Antunes, E; Britto-Júnior, J; Campos, R; da Silva-Filho, WP; De Nucci, G; Fregonesi, A; Monica, FZ; Moraes, MEA; Moraes, MO | 1 |
Chakrabarty, B; Ellem, SJ; Exintaris, B; Frydenberg, M; Lawrentschuk, N; Lee, SN; Middendorff, R; Papargiris, M; Risbridger, GP; Ryan, A; Wittmer, B | 1 |
Egawa, S; Furuta, A; Igarashi, T; Koike, Y; Suzuki, Y; Yoshimura, N | 1 |
Hakozaki, A; Miyoshi, K; Noma, T; Orimoto, N; Sasaki, E; Tsukihara, H; Yoshida, S | 1 |
Campbell, A; Chapple, CR; Chess-Williams, R; Davis, BJ; Naylor, AL; Sellers, DJ; Sillar, D | 1 |
Fujimura, M; Fukui, T; Oka, M; Oyama, T; Yoshifuji, M; Yoshinaga, R | 1 |
Chakrabarty, B; Dey, A; Exintaris, B; Lam, M; Ventura, S | 1 |
Whan Lee, J; Young Lee, M; Young Seo, I | 1 |
Hayashi, T; Matsuoka, K; Nakamura, K; Takeya, M | 1 |
Acevedo, A; Ciotkowska, A; Gratzke, C; Hennenberg, M; Herlemann, A; Kan, A; Rutz, B; Stief, CG; Strittmatter, F; Tamalunas, A; Wang, Y; Wiemer, N; Yu, Q | 1 |
Aswathaman, K; Gopalakrishnan, G; Kekre, NS; Rajpathy, J; Sinha, M; Subramani, S | 1 |
Anisuzzaman, AS; Morishima, S; Muramatsu, I; Myagmar, BE; Rodrigo, MC; Simpson, PC; Suzuki, F; Tanaka, T; Yoshiki, H | 1 |
Kawatani, M; Momota, Y; Nimura, T; Wang, X; Yanase, H | 1 |
Anand, N; Chugh, A; Gupta, JB; Gupta, S; Hegde, LG; Jain, S; Malhotra, S; Nanda, K; Naruganahalli, KS; Ray, A; Sinha, N; Tiwari, A | 1 |
Yokoyama, O | 1 |
de Almeida Kiguti, LR; Pupo, AS | 1 |
Akino, H; Aoki, Y; Ito, H; Nagase, K; Tanase, K; Yokoyama, O | 1 |
Allona, A; Angulo, J; Cuevas, P; Fernández, A; La Fuente, JM; Moncada, I; Sáenz de Tejada, I | 1 |
Goseki, T; Ishikawa, H; Mashimo, K; Nemoto, N; Ogasawara, S; Shimizu, K; Taguchi, Y; Yago, K | 1 |
Botto, H; Camparo, P; Gilles, N; Guérard, M; Guilloteau, V; Lluel, P; Maiga, A; Palea, S; Rekik, M; Rischmann, P; Rouget, C | 1 |
Benigni, F; Buono, R; Fossati, N; Hedlund, P; Montorsi, F; Rigatti, P; Villa, L | 1 |
Ashitomi, K; Hatano, T; Miyazato, M; Nishijima, S; Ogawa, Y; Sugaya, K | 1 |
Kontani, H; Shiraoya, C | 1 |
Ameda, K; Kakizaki, H; Kobayashi, S; Koyanagi, T; Shibata, T; Tanaka, H | 1 |
Fujimoto, K; Fukui, Y; Hirao, Y; Hirayama, A; Matsumoto, Y; Samma, S; Yamaguchi, A | 1 |
Alexandre, L; Allard, J; Bernabe, J; Droupy, S; Giuliano, F | 1 |
Haferkamp, A; Knapp, PA; Kyburz, T; Reitz, A; Schurch, B; Wefer, B | 1 |
Dessi, C; Marchese, G; Mongeau, R; Pani, L; Ruiu, S; Tambaro, S | 1 |
Alvarez, S; Andersen, L; Bouchelouche, K; Bouchelouche, P; Nordling, J | 1 |
Bae, JH; Jung, PB; Lee, JG | 1 |
Miyata, K; Noguchi, Y; Ohtake, A; Okutsu, H; Saitoh, C; Sasamata, M; Sato, S; Sonoda, R; Ukai, M; Yuyama, H | 1 |
Benson, JS; Jones, AW; Magliola, L; Troxel, SA | 1 |
Hatanaka, T; Matsushima, H; Miyata, K; Ohtake, A; Sasamata, M; Sato, S; Suzuki, M | 1 |
An, LM; Chen, IJ; Chou, YH; Huang, CH; Liu, CM; Lo, YC; Wu, BN; Wu, WJ | 1 |
Akino, H; Aoki, Y; Ito, H; Miwa, Y; Oyama, N; Yokoyama, O | 1 |
Fujimori, A; Koakutsu, A; Miyata, K; Ohtake, A; Sanagi, M; Sasamata, M; Sato, S; Sudoh, K; Ukai, M; Yuyama, H | 1 |
Drescher, P; Eckert, RE; Madsen, PO | 1 |
Breslin, D; Chou, TC; Felsen, D; Fields, DW; Kane, M; Marion, DN; Vaughan, ED | 1 |
Chapple, CR; Chess-Williams, R; Furukawa, K; Rosario, DJ; Smith, DJ; Uchiyama, T | 1 |
Chalmers, DH; Kenny, BA; Miller, AM; Naylor, AM; O'Connell, J; Williamson, IJ | 1 |
Chen, J; Chueh, SC; Guh, JH; Ko, FN; Lai, MK; Teng, CM | 1 |
Black, JW; Shankley, NP; Van der Graaf, PH | 1 |
Akiyama, K; Hora, M; Iizuka, K; Kitazawa, M; Kurashina, Y; Masuda, N; Matsuzawa, A; Murata, S; Nakamura, S; Ujiie, A; Yamagishi, R | 1 |
Akiyama, K; Ishida, N; Kawabe, K; Moriyama, N; Murata, S; Taniguchi, J; Yamazaki, S | 1 |
Bischoff, A; Chen, H; Michel, MC; Philipp, T; Schäfers, RF; Wambach, G | 1 |
Hattori, K; Makara, Y; Maruyama, K; Nagatomo, T; Ohnuki, T; Suzuki, M; Tsuchiya, M; Watanabe, K | 1 |
Muramatsu, I; Okada, K; Taniguchi, T | 1 |
Hiraoka, Y; Kato, H; Morikawa, K; Muramatsu, I; Nagata, O; Ohmura, T; Oshita, M; Taniguchi, T; Watanabe, Y | 1 |
Kim, SC; Lee, MY; Lim, SW; Seo, KK | 1 |
Muramatsu, I; Murata, S; Taniguchi, T | 1 |
Aisaka, K; Kanada, A; Muramatsu, I; Okaya, Y; Suzuki, Y | 1 |
Aisaka, K; Kawabe, K; Moriyama, N; Nishimatsu, H; Okaya, Y; Suzuki, Y | 1 |
Chin, C; Lau, WA; Pennefather, JN; Story, ME; Ventura, S | 1 |
Akiyama, K; Muramatsu, I; Murata, S; Okada, K; Takahashi, M; Taniguchi, T | 1 |
Ahmed, H; Aisaka, K; Akiyama, K; Fukasawa, R; Kitamura, T; Moriyama, N; Nishimatsu, H; Suzuki, Y; Tanaka, Y; Tatemichi, S | 1 |
Cheung, P; Evangelisto, M; Jolliffe, L; Kuo, GH; Murray, WV; Prouty, C; Pulito, V; Shaw, C; Varga, S | 1 |
Agnello, G; Amadesi, S; Borea, PA; Daniele, C; Geppetti, P; Spisani, L; Turini, A; Varani, K; Zamboni, P | 1 |
1 trial(s) available for tamsulosin and Muscle Contraction
Article | Year |
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Urodynamic effects of alpha1-blocker tamsulosin on voiding dysfunction in patients with neurogenic bladder.
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Aged, 80 and over; Female; Humans; Male; Middle Aged; Muscle Contraction; Pressure; Sex Factors; Sulfonamides; Tamsulosin; Treatment Outcome; Urinary Bladder, Neurogenic; Urination Disorders; Urodynamics | 2003 |
57 other study(ies) available for tamsulosin and Muscle Contraction
Article | Year |
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Design, synthesis, and structure-activity relationships of phthalimide-phenylpiperazines: a novel series of potent and selective alpha(1)(a)-adrenergic receptor antagonists.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Drug Design; Humans; Male; Muscle Contraction; Phthalimides; Piperazines; Prostatic Hyperplasia; Radioligand Assay; Rats; Rats, Long-Evans; Receptors, Adrenergic, alpha-1; Structure-Activity Relationship; Vasoconstriction | 2000 |
6-nitrodopamine is a major endogenous modulator of human vas deferens contractility.
Topics: Adrenergic Antagonists; Amitriptyline; Animals; Antidepressive Agents, Tricyclic; Carbamazepine; Chromatography, Liquid; Desipramine; Dopamine; Doxazosin; Epinephrine; Humans; Male; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nitric Oxide; Norepinephrine; Prazosin; Rats; Receptors, Adrenergic; Tamsulosin; Tandem Mass Spectrometry; Vas Deferens | 2022 |
Age Related Differences in Responsiveness to Sildenafil and Tamsulosin are due to Myogenic Smooth Muscle Tone in the Human Prostate.
Topics: Adrenergic alpha-1 Receptor Antagonists; Aged; Aging; Humans; Male; Middle Aged; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Phosphodiesterase 5 Inhibitors; Prostate; Sildenafil Citrate; Tamsulosin | 2017 |
Effects of combined treatment of tadalafil and tamsulosin on bladder dysfunction via the inhibition of afferent nerve activities in a rat model of bladder outlet obstruction.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Blood Pressure; Drug Therapy, Combination; Female; Muscle Contraction; Muscle, Smooth; Phosphodiesterase 5 Inhibitors; Rats; Sulfonamides; Tadalafil; Tamsulosin; Urinary Bladder; Urinary Bladder Neck Obstruction; Urodynamics | 2018 |
Therapeutic effect of TAC-302, a cyclohexenoic fatty alcohol derivative, on bladder denervation-related storage and voiding dysfunctions in rats.
Topics: Adrenergic alpha-Antagonists; Animals; Cyclohexenes; Denervation; Fatty Alcohols; Female; Immunohistochemistry; Muscle Contraction; Rats; Rats, Sprague-Dawley; Tamsulosin; Urethral Obstruction; Urinary Bladder; Urinary Bladder Neck Obstruction; Urination; Urodynamics; Urological Agents | 2018 |
α
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Humans; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Penile Erection; Penis; Prazosin; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin | 2018 |
Comparison of the Effects of Tadalafil and α
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Ejaculation; Electric Stimulation; Indoles; Male; Muscle Contraction; Naphthalenes; Phosphodiesterase 5 Inhibitors; Piperazines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Seminal Vesicles; Tadalafil; Tamsulosin; Vas Deferens | 2019 |
Tamsulosin modulates, but does not abolish the spontaneous activity in the guinea pig prostate gland.
Topics: Adrenergic alpha-1 Receptor Antagonists; Aging; Animals; Electrophysiological Phenomena; Guinea Pigs; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Prostate; Sulfonamides; Tamsulosin | 2015 |
In-vitro study on ureteral smooth muscle contractility with tamsulosin, nifedipine, and terpene mixture (Rowatinex®).
Topics: Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Nifedipine; Rabbits; Sulfonamides; Tamsulosin; Terpenes; Ureter; Vasodilator Agents | 2015 |
Effects of Silodosin and Tamsulosin on the Seminal Vesicle Contractile Response.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Guinea Pigs; Indoles; Male; Muscle Contraction; Seminal Vesicles; Sulfonamides; Tamsulosin | 2016 |
Non-Adrenergic, Tamsulosin-Insensitive Smooth Muscle Contraction is Sufficient to Replace α
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Adrenergic alpha-1 Receptor Antagonists; Cells, Cultured; Endothelins; Humans; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Prostate; Prostatic Hyperplasia; Statistics as Topic; Sulfonamides; Tamsulosin; Vasoconstrictor Agents | 2017 |
An in vitro study on human ureteric smooth muscle with the alpha1-adrenoceptor subtype blocker, tamsulosin.
Topics: Adrenergic alpha-Antagonists; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Sulfonamides; Tamsulosin; Ureter | 2008 |
Identification of alpha 1L-adrenoceptor in mice and its abolition by alpha 1A-adrenoceptor gene knockout.
Topics: Animals; Cerebral Cortex; Female; In Vitro Techniques; Indoles; Male; Mice; Mice, Inbred C57BL; Mice, Knockout; Muscle Contraction; Norepinephrine; Prazosin; Prostate; Radioligand Assay; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tritium; Vas Deferens | 2008 |
The involvement of urothelial alpha1A adrenergic receptor in controlling the micturition reflex.
Topics: Administration, Intravesical; Adrenergic alpha-Antagonists; Animals; Female; Humans; Indoles; Male; Muscle Contraction; Norepinephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Reflex; Sulfonamides; Tamsulosin; Urinary Bladder; Urination; Urodynamics; Urothelium | 2008 |
RBx 6198: a novel alpha1-adrenoceptor antagonist for the treatment of benign prostatic hyperplasia.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; CHO Cells; Cricetinae; Cricetulus; Dogs; Humans; Injections, Intravenous; Male; Muscle Contraction; Phenylephrine; Phthalimides; Piperazines; Prostate; Prostatic Hyperplasia; Protein Binding; Radioligand Assay; Rats; Rats, Wistar; Spleen; Sulfonamides; Tamsulosin | 2009 |
Pharmacological and genetic analysis of mechanisms underlying detrusor overactivity in rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Afferent Pathways; Animals; Benzhydryl Compounds; Brain; Cerebral Infarction; Cresols; Cyclooxygenase 2; Dinoprostone; Disease Models, Animal; Dose-Response Relationship, Drug; Early Growth Response Protein 1; Excitatory Amino Acid Antagonists; Muscarinic Antagonists; Muscle Contraction; Nerve Fibers, Unmyelinated; Neuronal Plasticity; Phenylpropanolamine; Proto-Oncogene Proteins c-fos; Rats; Rats, Sprague-Dawley; Receptors, AMPA; Receptors, N-Methyl-D-Aspartate; Receptors, Prostaglandin E; Receptors, Prostaglandin E, EP1 Subtype; RNA, Messenger; Sulfonamides; Tamsulosin; Time Factors; Tolterodine Tartrate; Transcription, Genetic; Urinary Bladder; Urinary Bladder, Overactive | 2010 |
Investigation of the effects of α1-adrenoceptor antagonism and L-type calcium channel blockade on ejaculation and vas deferens and seminal vesicle contractility in vitro.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Calcium Channel Blockers; Calcium Channels, L-Type; Dihydropyridines; Dose-Response Relationship, Drug; Ejaculation; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Seminal Vesicles; Sulfonamides; Tamsulosin; Vas Deferens | 2012 |
Co-administration of an α(1) -blocker improves the efficacy and safety of antimuscarinic agents in rats with detrusor overactivity.
Topics: Adrenergic alpha-1 Receptor Antagonists; Analysis of Variance; Animals; Disease Models, Animal; Diterpenes; Drug Therapy, Combination; Female; Infarction, Middle Cerebral Artery; Muscarinic Antagonists; Muscle Contraction; Organ Size; Quinuclidines; Rats; Rats, Sprague-Dawley; Solifenacin Succinate; Statistics, Nonparametric; Sulfonamides; Tamsulosin; Tetrahydroisoquinolines; Urinary Bladder; Urinary Bladder, Overactive | 2011 |
Tadalafil enhances the inhibitory effects of tamsulosin on neurogenic contractions of human prostate and bladder neck.
Topics: Adrenergic alpha-1 Receptor Antagonists; Carbolines; Electric Stimulation; Humans; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Nitric Oxide Donors; Nitroprusside; Phosphodiesterase 5 Inhibitors; Prostate; Prostatic Hyperplasia; Sulfonamides; Tadalafil; Tamsulosin; Urinary Bladder | 2012 |
Effects of tamsulosin and silodosin on isolated albino and pigmented rabbit iris dilators: possible mechanism of intraoperative floppy-iris syndrome.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Animals; Dose-Response Relationship, Drug; Indoles; Intraoperative Complications; Iris; Iris Diseases; Male; Melanins; Muscle Contraction; Muscle Hypotonia; Muscle, Smooth; Phenylephrine; Pigment Epithelium of Eye; Rabbits; Receptors, Adrenergic, alpha-1; Sulfonamides; Syndrome; Tamsulosin | 2012 |
Effects of ρ-Da1a a peptidic α(1) (A) -adrenoceptor antagonist in human isolated prostatic adenoma and anaesthetized rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Aged; Anesthesia; Animals; Blood Pressure; Chlorocebus aethiops; COS Cells; Elapid Venoms; Epinephrine; Humans; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Peptides; Phenylephrine; Prostate; Prostatic Hyperplasia; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Urethra | 2013 |
Effects by silodosin on the partially obstructed rat ureter in vivo and on human and rat isolated ureters.
Topics: Adrenergic alpha-1 Receptor Antagonists; Animals; Arterial Pressure; Dose-Response Relationship, Drug; Humans; Indoles; Male; Muscle Contraction; Prazosin; Rats; Rats, Sprague-Dawley; Species Specificity; Sulfonamides; Tamsulosin; Ureter; Ureteral Obstruction | 2013 |
Effects of intrathecal injection of tamsulosin and naftopidil, alpha-1A and -1D adrenergic receptor antagonists, on bladder activity in rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Efferent Pathways; Female; Hypogastric Plexus; Injections, Spinal; Male; Muscle Contraction; Muscle, Smooth; Naphthalenes; Parasympathetic Nervous System; Piperazines; Prostatic Hyperplasia; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Spinal Cord; Sulfonamides; Tamsulosin; Urinary Bladder | 2002 |
Method for simultaneous recording of the prostatic contractile and urethral pressure responses in anesthetized rats and the effects of tamsulosin.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Clonidine; Electric Stimulation; Male; Muscle Contraction; Muscle, Smooth; Phenylephrine; Pressure; Prostate; Rats; Rats, Wistar; Sulfonamides; Tamsulosin; Urethra | 2002 |
Alpha-blocker test: alternative to pressure-flow study of bladder outlet obstruction and detrusor contractility in patients without an enlarged prostate.
Topics: Adrenergic alpha-Antagonists; Aged; Aged, 80 and over; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Sulfonamides; Tamsulosin; Urinary Bladder Neck Obstruction; Urodynamics | 2004 |
A comparison of the effects of tamsulosin and alfuzosin on neurally evoked increases in bladder neck and seminal vesicle pressure in rats.
Topics: Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Ejaculation; Evoked Potentials; Male; Muscle Contraction; Pressure; Quinazolines; Rats; Rats, Wistar; Seminal Vesicles; Sulfonamides; Tamsulosin; Urinary Bladder | 2004 |
The effect of tamsulosin on the resting tone and the contractile behaviour of the female urethra: a functional urodynamic study in healthy women.
Topics: Adrenergic alpha-Antagonists; Adult; Electromagnetic Phenomena; Female; Humans; Lumbosacral Plexus; Muscle Contraction; Physical Stimulation; Sulfonamides; Tamsulosin; Urethra; Urodynamics | 2004 |
Evaluation of tamsulosin and alfuzosin activity in the rat vas deferens: relevance to ejaculation delays.
Topics: Adrenergic alpha-Antagonists; Animals; Dose-Response Relationship, Drug; Ejaculation; Electric Stimulation; Epididymis; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Quinazolines; Rats; Rats, Sprague-Dawley; Sulfonamides; Tamsulosin; Vas Deferens; Vasoconstrictor Agents | 2005 |
Increased contractile response to phenylephrine in detrusor of patients with bladder outlet obstruction: effect of the alpha1A and alpha1D-adrenergic receptor antagonist tamsulosin.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Aged; Humans; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Phenylephrine; Sulfonamides; Tamsulosin; Urinary Bladder Neck Obstruction | 2005 |
The effects of alpha-adrenoceptor antagonists on the urethral perfusion pressure of the female rat.
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Doxazosin; Female; Male; Muscle Contraction; Muscle, Smooth; Phentolamine; Pressure; Rats; Rats, Sprague-Dawley; Sulfonamides; Tamsulosin; Urethra; Urinary Bladder Neck Obstruction | 2005 |
Effect of tamsulosin on spontaneous bladder contraction in conscious rats with bladder outlet obstruction: comparison with effect on intraurethral pressure.
Topics: Animals; Dose-Response Relationship, Drug; Female; Muscle Contraction; Pressure; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Urinary Bladder; Urinary Bladder Neck Obstruction | 2006 |
Physiologic effect of nifedipine and tamsulosin on contractility of distal ureter.
Topics: Adrenergic alpha-Antagonists; Animals; In Vitro Techniques; Muscle Contraction; Nifedipine; Sulfonamides; Swine; Tamsulosin; Ureter; Vasodilator Agents | 2006 |
Relationship between the functional effect of tamsulosin and its concentration in lower urinary tract tissues in dogs.
Topics: Administration, Oral; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Area Under Curve; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Half-Life; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth; Phenylephrine; Prostate; Sulfonamides; Tamsulosin; Treatment Outcome; Urethra; Urinary Bladder; Urodynamics | 2007 |
cGMP-enhancing- and alpha1A/alpha1D-adrenoceptor blockade-derived inhibition of Rho-kinase by KMUP-1 provides optimal prostate relaxation and epithelial cell anti-proliferation efficacy.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Adrenergic alpha-Antagonists; Animals; Blotting, Western; Cell Proliferation; Cyclic AMP; Cyclic GMP; Cyclic GMP-Dependent Protein Kinases; Cyclic Nucleotide Phosphodiesterases, Type 5; Drug Synergism; Epithelial Cells; Humans; In Vitro Techniques; Intracellular Signaling Peptides and Proteins; Male; Muscle Contraction; Muscle, Smooth; Piperazines; Piperidines; Prostate; Protein Serine-Threonine Kinases; Purines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha; rho-Associated Kinases; Sildenafil Citrate; Sulfonamides; Sulfones; Tamsulosin; Xanthines | 2007 |
Antimuscarinic drug inhibits detrusor overactivity induced by topical application of prostaglandin E2 to the urethra with a decrease in urethral pressure.
Topics: Administration, Intravesical; Administration, Topical; Adrenergic alpha-Antagonists; Animals; Atropine; Benzilates; Calcium Channel Blockers; Cholinergic Antagonists; Dinoprostone; Disease Models, Animal; Female; Injections, Intra-Arterial; Muscarinic Antagonists; Muscle Contraction; omega-Conotoxins; Oxytocics; Pressure; Rats; Rats, Sprague-Dawley; Sulfonamides; Tamsulosin; Treatment Outcome; Urethra; Urinary Bladder; Urinary Bladder, Overactive; Verapamil | 2007 |
In vitro and in vivo effects of endothelin-1 and YM598, a selective endothelin ET A receptor antagonist, on the lower urinary tract.
Topics: Acetylcholine; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Drug Synergism; Endothelin A Receptor Antagonists; Endothelin-1; Heart Rate; In Vitro Techniques; Injections, Intra-Arterial; Injections, Intravenous; Male; Molecular Structure; Muscle Contraction; Muscle, Smooth; Phenylephrine; Prostate; Pyrimidines; Rabbits; Receptor, Endothelin B; Sulfonamides; Tamsulosin; Urethra; Urinary Bladder; Viper Venoms | 2008 |
Role of intracellular Ca2+ stores in smooth muscle contractions of the guinea pig vas deferens.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Calcium Channels; Guinea Pigs; Humans; In Vitro Techniques; Intracellular Fluid; Male; Models, Biological; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenylephrine; Prazosin; Prostatic Hyperplasia; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Vas Deferens | 1993 |
Medical management of benign prostatic hyperplasia: a canine model comparing the in vivo efficacy of alpha-1 adrenergic antagonists in the prostate.
Topics: Adrenergic alpha-Antagonists; Animals; Dogs; Dose-Response Relationship, Drug; Epinephrine; Male; Muscle Contraction; Phenoxybenzamine; Prazosin; Prostate; Prostatic Hyperplasia; Receptors, Adrenergic, alpha; Sulfonamides; Tamsulosin | 1993 |
Alpha 1A-adrenoceptor-mediated contractile responses of the human vas deferens.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Adult; Binding, Competitive; Calcium; Clonidine; Extracellular Space; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Phenylephrine; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Vas Deferens | 1995 |
Evaluation of the pharmacological selectivity profile of alpha 1 adrenoceptor antagonists at prostatic alpha 1 adrenoceptors: binding, functional and in vivo studies.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Doxazosin; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Phenylephrine; Prazosin; Pressure; Prostate; Quinazolines; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin | 1996 |
Inhibition by tamsulosin of tension responses of human hyperplastic prostate to electrical field stimulation.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aged; Calcium Channel Blockers; Electric Stimulation; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Nifedipine; Norepinephrine; Phenylephrine; Potassium; Prazosin; Prostate; Prostatic Hyperplasia; Sulfonamides; Tamsulosin | 1996 |
Analysis of the effects of alpha 1-adrenoceptor antagonists on noradrenaline-mediated contraction of rat small mesenteric artery.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Analysis of Variance; Animals; Benzazepines; Dopamine Antagonists; Dose-Response Relationship, Drug; Male; Mesenteric Arteries; Muscle Contraction; Norepinephrine; Phenylephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin | 1996 |
Effect of KMD-3213, an alpha 1a-adrenoceptor-selective antagonist, on the contractions of rabbit prostate and rabbit and rat aorta.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Indoles; Male; Muscle Contraction; Muscle, Smooth; Phenylephrine; Prostate; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin | 1996 |
KMD-3213, a novel alpha1A-adrenoceptor antagonist, potently inhibits the functional alpha1-adrenoceptor in human prostate.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Indoles; Male; Muscle Contraction; Norepinephrine; Prazosin; Prostate; Prostatectomy; Prostatic Hyperplasia; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin | 1997 |
Vasoconstriction of rat renal interlobar arteries by noradrenaline and neuropeptide Y.
Topics: Adrenergic alpha-Antagonists; Animals; Calcium; Dose-Response Relationship, Drug; Kidney Tubules, Distal; Kidney Tubules, Proximal; Male; Muscle Contraction; Muscle, Smooth, Vascular; Neuropeptide Y; Norepinephrine; Prazosin; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Renal Artery; Sulfonamides; Sympathetic Nervous System; Tamsulosin; Vasoconstriction; Yohimbine | 1997 |
Discrimination of alpha1-adrenoceptor subtypes in rat aorta and prostate.
Topics: Acetonitriles; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Clonidine; Dioxanes; Dose-Response Relationship, Drug; Male; Muscle Contraction; Muscle, Smooth; Nifedipine; Piperazines; Prazosin; Prostate; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Vasoconstriction; Vasodilator Agents | 1998 |
Tamsulosin: alpha1-adrenoceptor subtype-selectivity and comparison with terazosin.
Topics: Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Binding, Competitive; Dogs; Dose-Response Relationship, Drug; Humans; Male; Muscle Contraction; Norepinephrine; Prazosin; Prostate; Rabbits; Rats; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin | 1998 |
Binding and functional characterization of alpha1-adrenoceptor subtypes in the rat prostate.
Topics: Acetonitriles; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Binding, Competitive; Dioxanes; Dose-Response Relationship, Drug; In Vitro Techniques; Kinetics; Male; Muscle Contraction; Norepinephrine; Oxymetazoline; Piperazines; Prazosin; Prostate; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Tritium | 1999 |
Comparison of relaxation responses of cavernous and trigonal smooth muscles from rabbits by alpha1-adrenoceptor antagonists; prazosin, terazosin, doxazosin, and tamsulosin.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Doxazosin; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Prazosin; Rabbits; Sulfonamides; Tamsulosin | 1999 |
Pharmacological analysis of the novel, selective alpha1-adrenoceptor antagonist, KMD-3213, and its suitability as a tritiated radioligand.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Arteries; COS Cells; Dogs; In Vitro Techniques; Indoles; Ligands; Male; Muscle Contraction; Muscle, Smooth, Vascular; Prazosin; Radioligand Assay; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Sulfonamides; Tamsulosin; Tritium | 1999 |
Effect of JTH-601, a novel alpha1-adrenoceptor antagonist, on the function of lower urinary tract and blood pressure.
Topics: Adrenergic alpha-Antagonists; Anesthesia; Animals; Blood Pressure; Consciousness; Cresols; Hypotension, Orthostatic; In Vitro Techniques; Male; Muscle Contraction; Prazosin; Prostate; Rabbits; Sulfonamides; Tamsulosin; Urethra; Urinary Bladder; Urinary Tract Physiological Phenomena; Vas Deferens | 1999 |
Age-related change of the role of alpha1L-adrenoceptor in canine urethral smooth muscle.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Aging; Animals; Autoradiography; Binding, Competitive; Cresols; Dogs; Dose-Response Relationship, Drug; Female; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Parity; Phentolamine; Phenylephrine; Prazosin; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin; Urethra; Vasoconstrictor Agents | 1999 |
alpha(1L)-adrenoceptors mediate noradrenaline-induced contractions of the guinea-pig prostate stroma.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Dioxanes; Dose-Response Relationship, Drug; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Prazosin; Prostate; Receptors, Adrenergic, alpha-1; Sulfonamides; Tamsulosin | 1999 |
Tissue selectivity of KMD-3213, an alpha(1)-adrenoreceptor antagonist, in human prostate and vasculature.
Topics: Adrenergic alpha-Antagonists; Aorta; Binding, Competitive; Blood Vessels; Culture Techniques; Humans; Indoles; Male; Mesenteric Arteries; Muscle Contraction; Prazosin; Prostate; Radioligand Assay; Sulfonamides; Tamsulosin | 2000 |
Contractile properties of urethral smooth muscles of young and aged female dogs: morphological and pharmacological aspects.
Topics: Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Aging; Animals; Autoradiography; Dogs; Female; Muscle Contraction; Muscle, Smooth; Norepinephrine; Phenylephrine; Prazosin; Sulfonamides; Tamsulosin; Urethra | 2000 |
Design, synthesis and biological evaluation of pyridine-phenylpiperazines: a novel series of potent and selective alpha1a-adrenergic receptor antagonist.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Binding, Competitive; Blood Pressure; Combinatorial Chemistry Techniques; Dogs; Dose-Response Relationship, Drug; Humans; Kinetics; Male; Models, Animal; Muscle Contraction; Piperazines; Prostate; Protein Binding; Pyridines; Rats; Rats, Long-Evans; Receptors, Adrenergic, alpha-1; Stereoisomerism; Structure-Activity Relationship; Sulfonamides; Tamsulosin; Vasoconstrictor Agents | 2000 |
Comparison of prazosin, terazosin and tamsulosin: functional and binding studies in isolated prostatic and vascular human tissues.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Dose-Response Relationship, Drug; Female; Humans; Kinetics; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Prostate; Receptors, Adrenergic, alpha-1; Renal Artery; Saphenous Vein; Sulfonamides; Tamsulosin; Umbilical Veins | 2001 |