Page last updated: 2024-09-03

tafenoquine and Malaria, Falciparum

tafenoquine has been researched along with Malaria, Falciparum in 24 studies

Research

Studies (24)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (4.17)18.2507
2000's10 (41.67)29.6817
2010's9 (37.50)24.3611
2020's4 (16.67)2.80

Authors

AuthorsStudies
Fidock, DA; Flannery, EL; Winzeler, EA1
Iyer, PS; Kannan, M; Khan, FR; Raichurkar, AV1
Attaher, O; Bousema, T; Bradley, J; Diallo, M; Dicko, A; Dicko, OM; Drakeley, C; Issiaka, D; Keita, S; Lanke, K; Maguiraga, SO; Mahamar, A; McCall, MBB; Niambele, SM; Sacko, A; Samake, S; Sanogo, K; Sinaba, Y; Smit, MJ; Stone, W; Ter Heine, R; Traore, SF1
White, NJ1
Abd-Rahman, AN; Barber, BE; Birrell, GW; Edstein, MD; Leelasena, I; Llewellyn, S; Marquart, L; McCarthy, JS; Moehrle, JJ; Potter, AJ; Sahai, N; Shanks, GD; Webster, R; Wesche, D1
Contreras-Mancilla, J; Delgado-Ratto, C; Fernandez-Miñope, C; Ferrucci, HR; Gamboa, D; Llanos-Cuentas, A; Van Geertruyden, JP1
Dow, G; Smith, B1
Berman, J; Dobbin, C; Dow, GS; Marquart, L; McCarthy, JS; Read, LT; Reid, M; Smith, B; West, L1
Berman, JD1
Dow, GS; McCarthy, WF; Reid, M; Shanks, GD; Smith, B; Tang, D1
Dow, GS; Hetzell, B; Lin, G; Liu, J; McCarthy, WF; Smith, B; Tang, D; Thieling, S1
Kaewpruk, N; Mungthin, M; Sitthichot, N; Suwandittakul, N; Tan-ariya, P; Ward, SA1
Gbotosho, GO; Happi, CT; Okuboyejo, TM; Sowunmi, A1
Adjuik, M; Baird, JK; Binka, FN; Franke, ED; Fryauff, DJ; Hale, BR; Hoffman, SL; Horton, J; Koram, KA; Nkrumah, F; Oduro, AR; Owusu-Agyei, S; Prescott, WR; Ritchie, TL1
Peters, W; Robinson, BL; Stewart, LB1
Brewer, TG; Cherdchu, C; Eamsila, C; Edstein, MD; Jarasrumgsichol, P; Khaewsathien, P; Rieckmann, KH; Sangkharomya, S; Sasiprapha, T; Supakalin, P; Tang, DB; Walsh, DS1
Prajakwong, S; Sirichaisinthop, J; Vollnberg, A; Wernsdorfer, G; Wernsdorfer, WH; Wiedermann, G1
Czarnecki, E; Fusai, T; Koeck, JL; Kombila, M; Mamfoumbi, MM; Mosnier, J; Pradines, B; Rogier, C; Sokhna, C; Spiegel, A; Tall, A; Trape, JF1
Crockett, M; Kain, KC1
Brueckner, RP; Coster, T; Schuster, BG; Shmuklarsky, M; Wesche, DL1
Borrmann, S; Dangelmaier, O; Faucher, JF; Horton, J; Kremsner, PG; Lell, B; Missinou, MA1
Eamsila, C; Edstein, MD; Kitchener, S; Nasveld, PE; Rieckmann, KH; Sasiprapha, T; Walsh, DS1
Aleman, GM; Braitman, D; Brueckner, R; Horton, J; Klotz, FW; Ohrt, C; Oloo, AJ; Shanks, GD1

Reviews

4 review(s) available for tafenoquine and Malaria, Falciparum

ArticleYear
Using genetic methods to define the targets of compounds with antimalarial activity.
    Journal of medicinal chemistry, 2013, Oct-24, Volume: 56, Issue:20

    Topics: Animals; Anopheles; Antimalarials; Drug Resistance; Genetic Association Studies; Genome, Protozoan; Humans; Malaria, Falciparum; Molecular Targeted Therapy; Plasmodium falciparum

2013
The blood schizonticidal activity of tafenoquine makes an essential contribution to its prophylactic efficacy in nonimmune subjects at the intended dose (200 mg).
    Malaria journal, 2017, 05-19, Volume: 16, Issue:1

    Topics: Aminoquinolines; Animals; Antimalarials; Half-Life; Humans; Malaria, Falciparum; Malaria, Vivax; Plasmodium falciparum; Plasmodium vivax; Schizonts

2017
Tafenoquine: a promising new antimalarial agent.
    Expert opinion on investigational drugs, 2007, Volume: 16, Issue:5

    Topics: Aminoquinolines; Animals; Antimalarials; Humans; Malaria, Falciparum; Malaria, Vivax; Recurrence; Treatment Outcome

2007
Malaria prophylaxis/radical cure: recent experiences of the Australian Defence Force.
    Medecine tropicale : revue du Corps de sante colonial, 2001, Volume: 61, Issue:1

    Topics: Aminoquinolines; Antimalarials; Australia; Controlled Clinical Trials as Topic; Endemic Diseases; Humans; Malaria; Malaria, Falciparum; Malaria, Vivax; Military Personnel; Primaquine

2001

Trials

9 trial(s) available for tafenoquine and Malaria, Falciparum

ArticleYear
Single low-dose tafenoquine combined with dihydroartemisinin-piperaquine to reduce Plasmodium falciparum transmission in Ouelessebougou, Mali: a phase 2, single-blind, randomised clinical trial.
    The Lancet. Microbe, 2022, Volume: 3, Issue:5

    Topics: Aminoquinolines; Animals; Artemisinins; Humans; Malaria; Malaria, Falciparum; Mali; Piperazines; Plasmodium falciparum; Quinolines; Single-Blind Method

2022
Blood Schizonticidal Activity and Safety of Tafenoquine When Administered as Chemoprophylaxis to Healthy, Nonimmune Participants Followed by Blood Stage Plasmodium falciparum Challenge: A Randomized, Double-blind, Placebo-controlled Phase 1b Study.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2019, 07-18, Volume: 69, Issue:3

    Topics: Adult; Aminoquinolines; Antimalarials; Chemoprevention; Double-Blind Method; Female; Healthy Volunteers; Humans; Malaria, Falciparum; Male; Parasitemia; Placebos; Plasmodium falciparum; Schizonts; Young Adult

2019
Summary of anti-malarial prophylactic efficacy of tafenoquine from three placebo-controlled studies of residents of malaria-endemic countries.
    Malaria journal, 2015, Nov-26, Volume: 14

    Topics: Adolescent; Adult; Africa; Aminoquinolines; Antimalarials; Chemoprevention; Double-Blind Method; Female; Humans; Malaria, Falciparum; Male; Mefloquine; Middle Aged; Placebos; Treatment Outcome; Young Adult

2015
A randomized, double-blind, placebo-controlled, dose-ranging trial of tafenoquine for weekly prophylaxis against Plasmodium falciparum.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2003, Mar-01, Volume: 36, Issue:5

    Topics: Adult; Aged; Aminoquinolines; Animals; Antimalarials; Chemoprevention; Double-Blind Method; Female; Humans; Malaria, Falciparum; Male; Middle Aged; Plasmodium falciparum; Treatment Outcome

2003
Efficacy of monthly tafenoquine for prophylaxis of Plasmodium vivax and multidrug-resistant P. falciparum malaria.
    The Journal of infectious diseases, 2004, Oct-15, Volume: 190, Issue:8

    Topics: Administration, Oral; Aminoquinolines; Animals; Antimalarials; Double-Blind Method; Drug Administration Schedule; Drug Resistance, Multiple; Follow-Up Studies; Humans; Malaria, Falciparum; Malaria, Vivax; Military Personnel; Plasmodium falciparum; Thailand; Treatment Outcome

2004
Prophylaxis of Plasmodium falciparum infection in a human challenge model with WR 238605, a new 8-aminoquinoline antimalarial.
    Antimicrobial agents and chemotherapy, 1998, Volume: 42, Issue:5

    Topics: Adult; Aminoquinolines; Animals; Antimalarials; Double-Blind Method; Female; Humans; Malaria, Falciparum; Male; Plasmodium falciparum

1998
Malaria chemoprophylaxis with tafenoquine: a randomised study.
    Lancet (London, England), 2000, Jun-10, Volume: 355, Issue:9220

    Topics: Adolescent; Adult; Aminoquinolines; Antimalarials; Child; Dose-Response Relationship, Drug; Double-Blind Method; Drug Administration Schedule; Female; Gabon; Humans; Malaria, Falciparum; Male; Phenanthrenes

2000
Malaria prophylaxis/radical cure: recent experiences of the Australian Defence Force.
    Medecine tropicale : revue du Corps de sante colonial, 2001, Volume: 61, Issue:1

    Topics: Aminoquinolines; Antimalarials; Australia; Controlled Clinical Trials as Topic; Endemic Diseases; Humans; Malaria; Malaria, Falciparum; Malaria, Vivax; Military Personnel; Primaquine

2001
A new primaquine analogue, tafenoquine (WR 238605), for prophylaxis against Plasmodium falciparum malaria.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2001, Dec-15, Volume: 33, Issue:12

    Topics: Adolescent; Adult; Aminoquinolines; Animals; Antimalarials; Chemoprevention; Double-Blind Method; Female; Humans; Malaria, Falciparum; Male; Middle Aged; Plasmodium falciparum; Treatment Outcome

2001

Other Studies

12 other study(ies) available for tafenoquine and Malaria, Falciparum

ArticleYear
Synthesis and in vitro evaluation of novel 8-aminoquinoline-pyrazolopyrimidine hybrids as potent antimalarial agents.
    Bioorganic & medicinal chemistry letters, 2015, Mar-01, Volume: 25, Issue:5

    Topics: Aminoquinolines; Antimalarials; Humans; Malaria, Falciparum; Molecular Docking Simulation; Parasitic Sensitivity Tests; Plasmodium falciparum; Pyrazoles; Pyrimidines; Structure-Activity Relationship

2015
The Antimalarial Activity of Tafenoquine in Falciparum Malaria.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2023, 06-08, Volume: 76, Issue:11

    Topics: Aminoquinolines; Antimalarials; Healthy Volunteers; Humans; Malaria, Falciparum; Plasmodium falciparum

2023
Characterizing the Blood-Stage Antimalarial Activity of Tafenoquine in Healthy Volunteers Experimentally Infected With Plasmodium falciparum.
    Clinical infectious diseases : an official publication of the Infectious Diseases Society of America, 2023, 06-08, Volume: 76, Issue:11

    Topics: Adult; Antimalarials; Artemether; Artemether, Lumefantrine Drug Combination; Australia; Healthy Volunteers; Humans; Malaria, Falciparum; Parasitemia; Plasmodium falciparum

2023
Towards one standard treatment for uncomplicated Plasmodium falciparum and Plasmodium vivax malaria: Perspectives from and for the Peruvian Amazon.
    International journal of infectious diseases : IJID : official publication of the International Society for Infectious Diseases, 2021, Volume: 105

    Topics: Adult; Aminoquinolines; Artemisinins; Female; Humans; Malaria, Falciparum; Malaria, Vivax; Peru; Plasmodium falciparum; Plasmodium vivax; Prevalence; Primaquine; Reference Standards

2021
Approval of Tafenoquine for Malaria Chemoprophylaxis.
    The American journal of tropical medicine and hygiene, 2019, Volume: 100, Issue:6

    Topics: Aminoquinolines; Antimalarials; Australia; Chemoprevention; Child; Contraindications, Drug; Drug Administration Schedule; Drug Approval; Female; Fetus; Glucosephosphate Dehydrogenase Deficiency; Hemoglobins; Humans; Malaria, Falciparum; Methemoglobin; Pregnancy; Psychotic Disorders; United States

2019
A retrospective analysis of the protective efficacy of tafenoquine and mefloquine as prophylactic anti-malarials in non-immune individuals during deployment to a malaria-endemic area.
    Malaria journal, 2014, Feb-06, Volume: 13

    Topics: Aminoquinolines; Antimalarials; Australia; Chemoprevention; Endemic Diseases; Humans; Incidence; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Military Personnel; Retrospective Studies; Timor-Leste; Travel; Treatment Outcome; United States

2014
PFMDR1 POLYMORPHISMS INFLUENCE ON IN VITRO SENSITIVITY OF THAI PLASMODIUM FALCIPARUM ISOLATES TO PRIMAQUINE, SITAMAQUINE AND TAFENOQUINE.
    The Southeast Asian journal of tropical medicine and public health, 2016, Volume: 47, Issue:3

    Topics: Aminoquinolines; Antimalarials; Humans; Malaria, Falciparum; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Primaquine; Thailand

2016
Risk factors for gametocyte carriage in uncomplicated falciparum malaria in children before and after artemisinin-based combination treatments.
    Chemotherapy, 2011, Volume: 57, Issue:6

    Topics: Adolescent; Aminoquinolines; Antimalarials; Artemisinins; Child; Child, Preschool; Drug Therapy, Combination; Female; Follow-Up Studies; Humans; Infant; Malaria, Falciparum; Male; Risk Factors

2011
The chemotherapy of rodent malaria. LXI. Drug combinations to impede the selection of drug resistance, part 4: the potential role of 8-aminoquinolines.
    Annals of tropical medicine and parasitology, 2003, Volume: 97, Issue:3

    Topics: Aminoquinolines; Animals; Antimalarials; Chloroquine; Disease Models, Animal; Drug Resistance; Drug Therapy, Combination; Malaria; Malaria, Falciparum; Malaria, Vivax; Mefloquine; Mice; Plasmodium berghei; Plasmodium chabaudi; Plasmodium yoelii; Primaquine; Time Factors

2003
Molecule of the month. Tafenoquine succinate.
    Drug news & perspectives, 2003, Volume: 16, Issue:4

    Topics: Aminoquinolines; Antimalarials; Drug Administration Schedule; Humans; Malaria, Falciparum; Randomized Controlled Trials as Topic

2003
In-vitro interaction of tafenoquine and chloroquine in Plasmodium falciparum from northwestern Thailand.
    Wiener klinische Wochenschrift, 2003, Volume: 115 Suppl 3

    Topics: Adolescent; Adult; Aminoquinolines; Animals; Antimalarials; Cell Proliferation; Chloroquine; Dose-Response Relationship, Drug; Drug Combinations; Drug Evaluation; Humans; Malaria, Falciparum; Plasmodium falciparum; Species Specificity; Thailand

2003
In vitro activity of tafenoquine against the asexual blood stages of Plasmodium falciparum isolates from Gabon, Senegal, and Djibouti.
    Antimicrobial agents and chemotherapy, 2006, Volume: 50, Issue:9

    Topics: Aminoquinolines; Animals; Antimalarials; Djibouti; Gabon; Humans; Malaria, Falciparum; Plasmodium falciparum; Senegal

2006