Page last updated: 2024-08-24

sulofenur and Adenocarcinoma

sulofenur has been researched along with Adenocarcinoma in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Aikins, J; Crowell, TA; Grossman, CS; Harper, RW; Howbert, JJ; Kramer, KE; Poore, GA; Rieder, BJ; Rinzel, SM; Tao, EV1
Cheshire, PJ; Grindey, GB; Houghton, JA; Houghton, PJ; Lutz, L; Myers, L; Toth, J1
Berezesky, IK; Boder, GB; Jain, PT; Phelps, PC; Trump, BF1
Boder, GB; Grindey, GB; Houghton, PJ; Sosinski, J; Thakar, JH1
Germain, GS; Harwood, FC; Houghton, PJ; Sosinski, J; Thakar, JH1
Houghton, JA; Houghton, PJ1
Coleman, R; Hatty, S; Kamthan, A; Peters, B; Scarffe, JH; Smyth, JF; Walling, J1
Alberts, DS; Fossella, FV; Hardy, J; Haynes, TR; Lippman, SM; O'Brien, M; Seitz, DE; Taylor, CW; Wiltshaw, E; Wolen, RL1
Bailey, FC; Germain, GS; Grindey, GB; Houghton, JA; Houghton, PJ; Witt, BC1

Reviews

1 review(s) available for sulofenur and Adenocarcinoma

ArticleYear
Antitumor diarylsulfonylureas: novel agents with unfulfilled promise.
    Investigational new drugs, 1996, Volume: 14, Issue:3

    Topics: Adenocarcinoma; Adult; Animals; Antineoplastic Agents; Benzofurans; Child; Clinical Trials, Phase I as Topic; Colonic Neoplasms; Drug Resistance, Multiple; Humans; Phenylurea Compounds; Sulfonylurea Compounds; Transplantation, Heterologous

1996

Trials

2 trial(s) available for sulofenur and Adenocarcinoma

ArticleYear
A phase II study of sulofenur (LY186641) in gastric cancer.
    Anti-cancer drugs, 1992, Volume: 3, Issue:4

    Topics: Adenocarcinoma; Adult; Aged; Antineoplastic Agents; Esophageal Neoplasms; Female; Humans; Male; Middle Aged; Stomach Neoplasms; Sulfonylurea Compounds

1992
Hypoprothrombinemia from coadministration of sulofenur (LY 186641) and warfarin: report of three cases.
    Investigational new drugs, 1991, Volume: 9, Issue:4

    Topics: Adenocarcinoma; Antineoplastic Combined Chemotherapy Protocols; Drug Evaluation; Drug Interactions; Female; Humans; Hypoprothrombinemias; Lung Neoplasms; Middle Aged; Ovarian Neoplasms; Sulfonylurea Compounds; Warfarin

1991

Other Studies

6 other study(ies) available for sulofenur and Adenocarcinoma

ArticleYear
Novel agents effective against solid tumors: the diarylsulfonylureas. Synthesis, activities, and analysis of quantitative structure-activity relationships.
    Journal of medicinal chemistry, 1990, Volume: 33, Issue:9

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Chemical Phenomena; Chemistry; Humans; Lymphoma, Non-Hodgkin; Male; Mice; Mice, Inbred BALB C; Mice, Inbred C57BL; Mice, Inbred DBA; Multiple Myeloma; Rats; Rats, Inbred Strains; Structure-Activity Relationship; Sulfonylurea Compounds; Tumor Cells, Cultured

1990
Efficacy of sulofenur and a second generation diarylsulfonylurea, N-[5-(2,3-dihydrobenzofuryl)sulfonyl]-N'-(3,4-dichlorophenyl)urea (LY295501), against colon adenocarcinoma xenografts.
    Anti-cancer drugs, 1995, Volume: 6, Issue:2

    Topics: Adenocarcinoma; Animals; Antineoplastic Agents; Benzofurans; Colonic Neoplasms; Female; Humans; Mice; Mice, Inbred CBA; Neoplasm Transplantation; Phenylurea Compounds; Sulfonylurea Compounds; Transplantation, Heterologous

1995
Sulofenur cytotoxicity and changes in cytosolic calcium and mitochondrial membrane potential in human colon adenocarcinoma cell lines.
    Cancer letters, 1995, Jan-06, Volume: 88, Issue:1

    Topics: Adenocarcinoma; Calcium; Cell Death; Cell Survival; Colonic Neoplasms; Cytosol; Dose-Response Relationship, Drug; Humans; In Vitro Techniques; Membrane Potentials; Microscopy, Electron; Mitochondria; Sulfonylurea Compounds; Tumor Cells, Cultured

1995
Characterization of the intracellular distribution and binding in human adenocarcinoma cells of N-(4-azidophenylsulfonyl)-N'-(4-chlorophenyl)urea (LY219703), a photoaffinity analogue of the antitumor diarylsulfonylurea sulofenur.
    Biochemical pharmacology, 1995, Mar-01, Volume: 49, Issue:5

    Topics: Adenocarcinoma; Affinity Labels; Antineoplastic Agents; Cell-Free System; Drug Resistance; Humans; Mitochondria; Photochemistry; Subcellular Fractions; Sulfonylurea Compounds; Tumor Cells, Cultured

1995
Proliferation-dependent and -independent cytotoxicity by antitumor diarylsulfonylureas. Indication of multiple mechanisms of drug action.
    Biochemical pharmacology, 1993, May-25, Volume: 45, Issue:10

    Topics: Adenocarcinoma; Antineoplastic Agents; Apoptosis; Cell Death; Cell Division; DNA Damage; DNA, Neoplasm; Drug Resistance; Humans; Kinetics; Neoplasms, Experimental; Nucleosomes; Sulfonylurea Compounds; Tumor Cells, Cultured

1993
N-(5-indanylsulfonyl)-N'-(4-chlorophenyl)urea, a novel agent equally cytotoxic to nonproliferating human colon adenocarcinoma cells.
    Cancer research, 1990, Jan-15, Volume: 50, Issue:2

    Topics: Adenocarcinoma; Antineoplastic Agents; Blood Physiological Phenomena; Cell Division; Cell Survival; Colonic Neoplasms; Culture Media; Humans; Serum Albumin; Sulfonylurea Compounds; Tumor Cells, Cultured

1990