Page last updated: 2024-08-26

sr141716 and Muscle Relaxation

sr141716 has been researched along with Muscle Relaxation in 10 studies

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (40.00)18.2507
2000's4 (40.00)29.6817
2010's2 (20.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Beaumont, H; Boeckxstaens, G; Carlsson, A; Jensen, J; Lehmann, A; Ruth, M1
Blondeau, K; Boecxstaens, V; Farré, R; Gasbarrini, A; Scarpellini, E; Tack, J; Vos, R1
Altun, A; Bagcivan, I; Durmus, N; Kaya, T; Sarac, B; Sencan, M; Turan, M1
Blackshaw, LA; Brändén, L; Carlsson, A; Jensen, J; Lehmann, A; Nygren, E; Smid, SD1
Abe, T; Arisaka, O; Morimoto, H; Yamada, Y; Yoshihara, S1
Campbell, WB; Edgemond, WS; Hillard, CJ; Pratt, PF1
Hiley, CR; White, R1
Bukoski, RD; Ishioka, N1
Chaytor, AT; Evans, WH; Griffith, TM; Martin, PE; Randall, MD1
Chapnick, BM; Howlett, AC; Mukhopadhyay, S1

Trials

2 trial(s) available for sr141716 and Muscle Relaxation

ArticleYear
Effect of delta9-tetrahydrocannabinol, a cannabinoid receptor agonist, on the triggering of transient lower oesophageal sphincter relaxations in dogs and humans.
    British journal of pharmacology, 2009, Volume: 156, Issue:1

    Topics: Adult; Animals; Cannabinoid Receptor Agonists; Deglutition; Dogs; Dose-Response Relationship, Drug; Double-Blind Method; Dronabinol; Esophageal Sphincter, Lower; Female; Gastroesophageal Reflux; Humans; Hydrogen-Ion Concentration; Male; Middle Aged; Muscle Relaxation; Piperidines; Postprandial Period; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Species Specificity; Young Adult

2009
Effect of rimonabant on oesophageal motor function in man.
    Alimentary pharmacology & therapeutics, 2011, Volume: 33, Issue:6

    Topics: Adult; Epidemiologic Methods; Esophageal Sphincter, Lower; Esophagus; Female; Gastrointestinal Agents; Gastrointestinal Motility; Humans; Hydrogen-Ion Concentration; Male; Muscle Relaxation; Piperidines; Postprandial Period; Pyrazoles; Receptor, Cannabinoid, CB1; Rimonabant; Young Adult

2011

Other Studies

8 other study(ies) available for sr141716 and Muscle Relaxation

ArticleYear
Effects of cannabinoid agonists on sheep sphincter of oddi in vitro.
    Pancreatology : official journal of the International Association of Pancreatology (IAP) ... [et al.], 2011, Volume: 11, Issue:4

    Topics: Analgesics; Animals; Arachidonic Acids; Benzoxazines; Camphanes; Cannabinoid Receptor Agonists; Cannabinoids; Carbachol; Cyclic GMP; Male; Morpholines; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; NG-Nitroarginine Methyl Ester; Organ Culture Techniques; Piperidines; Pyrazoles; Rimonabant; Sheep; Sphincter of Oddi

2011
Cannabinoid receptor agonism inhibits transient lower esophageal sphincter relaxations and reflux in dogs.
    Gastroenterology, 2002, Volume: 123, Issue:4

    Topics: Analgesics; Animals; Benzoxazines; Dogs; Esophagogastric Junction; Female; Ferrets; GABA-B Receptor Agonists; Gastroesophageal Reflux; Ligands; Male; Mechanoreceptors; Morpholines; Muscle Relaxation; Naphthalenes; Neurons, Afferent; Piperidines; Pyrazoles; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Vagus Nerve

2002
Cannabinoid receptor agonists inhibit sensory nerve activation in guinea pig airways.
    American journal of respiratory and critical care medicine, 2004, Nov-01, Volume: 170, Issue:9

    Topics: Analysis of Variance; Animals; Benzoxazines; Camphanes; Cannabinoid Receptor Antagonists; Disease Models, Animal; Electric Stimulation; Guinea Pigs; Male; Morpholines; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Naphthalenes; Neurokinin A; Piperidines; Probability; Pyrazoles; Respiratory Muscles; Rimonabant; Sensitivity and Specificity; Sensory Receptor Cells

2004
N-arachidonylethanolamide relaxation of bovine coronary artery is not mediated by CB1 cannabinoid receptor.
    The American journal of physiology, 1998, Volume: 274, Issue:1

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Animals; Arachidonic Acids; Biotransformation; Cannabinoids; Cattle; Cells, Cultured; Coronary Vessels; Endocannabinoids; Endothelium, Vascular; Ethanolamines; In Vitro Techniques; Isometric Contraction; Muscle Relaxation; Muscle Tonus; Muscle, Smooth, Vascular; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rats; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Vasodilation

1998
The actions of the cannabinoid receptor antagonist, SR 141716A, in the rat isolated mesenteric artery.
    British journal of pharmacology, 1998, Volume: 125, Issue:4

    Topics: Animals; Benzimidazoles; Calcium; Cannabinoids; Carbachol; Cromakalim; Dose-Response Relationship, Drug; Drug Interactions; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Methoxamine; Muscle Relaxation; Muscle, Smooth, Vascular; Penicillamine; Piperidines; Potassium Channels; Pyrazoles; Rats; Rats, Wistar; Rimonabant

1998
A role for N-arachidonylethanolamine (anandamide) as the mediator of sensory nerve-dependent Ca2+-induced relaxation.
    The Journal of pharmacology and experimental therapeutics, 1999, Volume: 289, Issue:1

    Topics: Animals; Arachidonic Acids; Calcium Signaling; Cannabinoids; Endocannabinoids; In Vitro Techniques; Isometric Contraction; Male; Mesenteric Arteries; Muscle Relaxation; Muscle, Smooth, Vascular; Neurons, Afferent; Neurotransmitter Agents; Norepinephrine; Pinacidil; Piperidines; Polyunsaturated Alkamides; Potassium Channel Blockers; Pyrazoles; Rats; Rats, Wistar; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Vasoconstrictor Agents

1999
The endothelial component of cannabinoid-induced relaxation in rabbit mesenteric artery depends on gap junctional communication.
    The Journal of physiology, 1999, Oct-15, Volume: 520 Pt 2

    Topics: Acetylcholine; Animals; Arachidonic Acids; Benzofurans; Cannabinoid Receptor Modulators; Cannabinoids; COS Cells; Endocannabinoids; Gap Junctions; Glycyrrhetinic Acid; Indomethacin; Isoquinolines; Male; Mesenteric Artery, Superior; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Phenylephrine; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rabbits; Receptors, Cannabinoid; Receptors, Drug; Rimonabant

1999
Anandamide-induced vasorelaxation in rabbit aortic rings has two components: G protein dependent and independent.
    American journal of physiology. Heart and circulatory physiology, 2002, Volume: 282, Issue:6

    Topics: Animals; Aorta; Arachidonic Acids; Cannabinoids; Capsaicin; Endocannabinoids; Endothelium, Vascular; Enzyme Inhibitors; Gap Junctions; GTP-Binding Proteins; Male; Muscle Relaxation; Muscle, Smooth, Vascular; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Pertussis Toxin; Piperidines; Polyunsaturated Alkamides; Pyrazoles; Rabbits; Receptors, Calcitonin Gene-Related Peptide; Receptors, Cannabinoid; Receptors, Drug; Rimonabant; Virulence Factors, Bordetella

2002