Page last updated: 2024-08-24

setoperone and Schizophrenia

setoperone has been researched along with Schizophrenia in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19902 (15.38)18.7374
1990's6 (46.15)18.2507
2000's5 (38.46)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Kapur, S; Mamo, D; Mann, S; Papatheodorou, G; Remington, G; Shammi, CM; Therrien, F1
Ansari, MS; Dawant, B; Jayathilake, K; Kessler, RM; Li, R; Meltzer, HY; Riccardi, P1
Graff, A; Kapur, S; Mamo, D; Mizrahi, R; Romeyer, F; Shammi, CM1
Houle, S; Jones, C; Kapur, S; McKay, G; Remington, G; Zipursky, R1
Attar-Levy, D; Martinot, JL; Monnet, F; Paillère-Martinot, ML; Recassens, C; Trichard, C1
Attar-Levy, D; Blin, J; Feline, A; Martinot, JL; Paillère-Martinot, ML; Trichard, C1
DaSilva, J; Houle, S; Jones, C; Kapur, S; Remington, G; Wilson, AA; Zipursky, RB1
Brown, GM; DaSilva, J; Houle, S; Jones, C; Kapur, S; Lewis, R; Wilson, AA; Zipursky, RB1
Kapur, S; Remington, G; Zipursky, RB1
Liddle, PF; Ngan, ET; Ruth, TJ; Yatham, LN1
Hussey, D; Kapur, S; Kecojevic, A; Lewis, R; Meyer, JH; Tauscher, J; Verhoeff, NP; Zipursky, RB1
Gelders, YG1
Ceulemans, DL; Gelders, YG; Hoppenbrouwers, ML; Janssen, PA; Reyntjens, AJ1

Trials

5 trial(s) available for setoperone and Schizophrenia

ArticleYear
A PET study of dopamine D2 and serotonin 5-HT2 receptor occupancy in patients with schizophrenia treated with therapeutic doses of ziprasidone.
    The American journal of psychiatry, 2004, Volume: 161, Issue:5

    Topics: Adult; Antipsychotic Agents; Brain; Corpus Striatum; Drug Administration Schedule; Female; Humans; Male; Piperazines; Psychotic Disorders; Pyrimidinones; Raclopride; Receptors, Dopamine D2; Receptors, Serotonin, 5-HT2; Schizophrenia; Thiazoles; Tomography, Emission-Computed

2004
Occupancy of striatal and extrastriatal dopamine D2/D3 receptors by olanzapine and haloperidol.
    Neuropsychopharmacology : official publication of the American College of Neuropsychopharmacology, 2005, Volume: 30, Issue:12

    Topics: Adult; Antipsychotic Agents; Benzamides; Benzodiazepines; Brain Chemistry; Corpus Striatum; Dopamine Antagonists; Female; Haloperidol; Humans; Image Processing, Computer-Assisted; Male; Middle Aged; Olanzapine; Positron-Emission Tomography; Pyrimidinones; Pyrrolidines; Radiopharmaceuticals; Receptor, Serotonin, 5-HT2A; Receptors, Dopamine D3; Schizophrenia; Serotonin Antagonists

2005
Differential effects of aripiprazole on D(2), 5-HT(2), and 5-HT(1A) receptor occupancy in patients with schizophrenia: a triple tracer PET study.
    The American journal of psychiatry, 2007, Volume: 164, Issue:9

    Topics: Adult; Antipsychotic Agents; Aripiprazole; Basal Ganglia; Basal Ganglia Diseases; Carbon Radioisotopes; Caudate Nucleus; Cerebral Cortex; Dopamine D2 Receptor Antagonists; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fluorine Radioisotopes; Humans; Male; Piperazines; Positron-Emission Tomography; Psychotic Disorders; Putamen; Pyridines; Pyrimidinones; Quinolones; Raclopride; Receptor, Serotonin, 5-HT1A; Receptors, Dopamine; Receptors, Dopamine D2; Schizophrenia; Serotonin 5-HT1 Receptor Agonists; Treatment Outcome

2007
5-HT2 and D2 receptor occupancy of olanzapine in schizophrenia: a PET investigation.
    The American journal of psychiatry, 1998, Volume: 155, Issue:7

    Topics: Adult; Antipsychotic Agents; Benzodiazepines; Carbon Radioisotopes; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fluorine Radioisotopes; Humans; Male; Olanzapine; Pirenzepine; Prolactin; Pyrimidinones; Raclopride; Receptors, Dopamine D2; Receptors, Serotonin; Salicylamides; Schizophrenia; Tomography, Emission-Computed; Treatment Outcome

1998
Thymosthenic agents, a novel approach in the treatment of schizophrenia.
    The British journal of psychiatry. Supplement, 1989, Issue:5

    Topics: Brain; Butyrophenones; Humans; Isoxazoles; Piperidines; Pyrimidinones; Randomized Controlled Trials as Topic; Receptors, Serotonin; Risperidone; Ritanserin; Schizophrenia; Schizophrenic Psychology; Serotonin Antagonists

1989

Other Studies

8 other study(ies) available for setoperone and Schizophrenia

ArticleYear
PET evidence that loxapine is an equipotent blocker of 5-HT2 and D2 receptors: implications for the therapeutics of schizophrenia.
    The American journal of psychiatry, 1997, Volume: 154, Issue:11

    Topics: Adult; Cerebellum; Corpus Striatum; Dopamine Antagonists; Female; Fluorine Radioisotopes; Humans; Loxapine; Male; Pyrimidinones; Raclopride; Receptors, Dopamine D2; Receptors, Serotonin; Salicylamides; Schizophrenia; Tomography, Emission-Computed

1997
Binding of antipsychotic drugs to cortical 5-HT2A receptors: a PET study of chlorpromazine, clozapine, and amisulpride in schizophrenic patients.
    The American journal of psychiatry, 1998, Volume: 155, Issue:4

    Topics: Adolescent; Adult; Amisulpride; Animals; Antipsychotic Agents; Cerebral Cortex; Chlorpromazine; Clozapine; Dose-Response Relationship, Drug; Drug Administration Schedule; Female; Fluorine Radioisotopes; Humans; Male; Pyrimidinones; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Schizophrenia; Sulpiride; Tomography, Emission-Computed

1998
No serotonin 5-HT2A receptor density abnormality in the cortex of schizophrenic patients studied with PET.
    Schizophrenia research, 1998, May-04, Volume: 31, Issue:1

    Topics: Adult; Cell Count; Cerebral Cortex; Female; Functional Laterality; Humans; Male; Pyrimidinones; Receptors, Serotonin; Schizophrenia; Tomography, Emission-Computed

1998
Serotonin 5-HT2 receptors in schizophrenia: a PET study using [18F]setoperone in neuroleptic-naive patients and normal subjects.
    The American journal of psychiatry, 1999, Volume: 156, Issue:1

    Topics: Antipsychotic Agents; Brain Chemistry; Cerebral Cortex; Contrast Media; Fluorine Radioisotopes; Humans; Prefrontal Cortex; Pyrimidinones; Receptors, Serotonin; Schizophrenia; Tomography, Emission-Computed

1999
Clinical and theoretical implications of 5-HT2 and D2 receptor occupancy of clozapine, risperidone, and olanzapine in schizophrenia.
    The American journal of psychiatry, 1999, Volume: 156, Issue:2

    Topics: Adult; Antipsychotic Agents; Benzodiazepines; Carbon Radioisotopes; Clozapine; Drug Administration Schedule; Female; Fluorine Radioisotopes; Humans; Male; Middle Aged; Olanzapine; Pirenzepine; Pyrimidinones; Raclopride; Receptors, Dopamine D2; Receptors, Serotonin; Risperidone; Salicylamides; Schizophrenia; Tomography, Emission-Computed

1999
Decreased serotonin 2A receptor densities in neuroleptic-naive patients with schizophrenia: A PET study using [(18)F]setoperone.
    The American journal of psychiatry, 2000, Volume: 157, Issue:6

    Topics: Adolescent; Adult; Antipsychotic Agents; Brain; Female; Fluorine Radioisotopes; Frontal Lobe; Humans; Male; Pyrimidinones; Radionuclide Imaging; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Schizophrenia

2000
A voxel-by-voxel analysis of [18F]setoperone PET data shows no substantial serotonin 5-HT(2A) receptor changes in schizophrenia.
    Psychiatry research, 2000, Oct-30, Volume: 99, Issue:3

    Topics: Adult; Age Factors; Analysis of Variance; Brain; Case-Control Studies; Contrast Media; Female; Fluorine Radioisotopes; Humans; Male; Psychiatric Status Rating Scales; Pyrimidinones; Receptor, Serotonin, 5-HT2A; Receptors, Serotonin; Schizophrenia; Schizophrenic Psychology; Serotonin Antagonists; Tomography, Emission-Computed

2000
Effect of serotonin antagonism in schizophrenia: a pilot study with setoperone.
    Psychopharmacology, 1985, Volume: 85, Issue:3

    Topics: Adult; Aged; Basal Ganglia Diseases; Female; Humans; Male; Middle Aged; Pilot Projects; Psychiatric Status Rating Scales; Pyrimidinones; Schizophrenia; Serotonin Antagonists

1985