Page last updated: 2024-09-05

sch 58261 and Anochlesia

sch 58261 has been researched along with Anochlesia in 6 studies

Research

Studies (6)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (83.33)29.6817
2010's1 (16.67)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chen, L; Engber, T; Grant, D; Hetu, G; Huang, C; Jin, X; Kumaravel, G; Peng, B; Petter, RC; Phadke, D; Reilly, J; Smits, G; Tam, S; Vu, CB; Zhang, J1
Engber, T; Huang, C; Jin, X; Kumaravel, G; Pan, D; Peng, B; Petter, RC; Phadke, D; Reilly, J; Sha, L; Tam, S; Vu, CB1
Bohnert, T; Chang, H; Engber, TM; Ensinger, CL; Huang, C; Kumaravel, G; Peng, H; Petter, RC; Sha, L; Van Vlijmen, H; Vu, CB; Wang, J; Whalley, ET; Yao, G1
Chang, H; Conlon, PR; Engber, TM; Haque, S; Kiesman, WF; Kumaravel, G; Petter, RC; Sha, L; Wang, J; Whalley, ET; Yao, G1
Engber, T; Grant, D; Hetu, G; Huang, C; Jin, X; Kumaravel, G; Pan, D; Peng, B; Petter, RC; Phadke, D; Reilly, J; Smits, G; Tam, S; Vu, CB1
Barodia, SK; Luthra, PM; Mishra, CB; Prakash, A; Senthil Kumar, JB1

Other Studies

6 other study(ies) available for sch 58261 and Anochlesia

ArticleYear
Piperazine derivatives of [1,2,4]triazolo[1,5-a][1,3,5]triazine as potent and selective adenosine A2a receptor antagonists.
    Journal of medicinal chemistry, 2004, Aug-12, Volume: 47, Issue:17

    Topics: Adenosine A2 Receptor Antagonists; Administration, Oral; Animals; Antiparkinson Agents; Biological Availability; Brain; Catalepsy; Heterocyclic Compounds, 2-Ring; In Vitro Techniques; Male; Mice; Parkinsonian Disorders; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Adenosine A2A; Structure-Activity Relationship; Triazines; Triazoles

2004
Studies on adenosine A2a receptor antagonists: comparison of three core heterocycles.
    Bioorganic & medicinal chemistry letters, 2004, Oct-04, Volume: 14, Issue:19

    Topics: Adenosine A2 Receptor Antagonists; Animals; Antiparkinson Agents; Catalepsy; Mice; Pyrimidines; Structure-Activity Relationship; Triazoles

2004
Novel bicyclic piperazine derivatives of triazolotriazine and triazolopyrimidines as highly potent and selective adenosine A2A receptor antagonists.
    Journal of medicinal chemistry, 2004, Dec-02, Volume: 47, Issue:25

    Topics: Adenosine A2 Receptor Antagonists; Administration, Oral; Animals; Catalepsy; Disease Models, Animal; Drug Stability; In Vitro Techniques; Male; Mice; Microsomes, Liver; Molecular Structure; Parkinson Disease; Piperazines; Pyrimidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Stereoisomerism; Structure-Activity Relationship; Triazines; Triazoles

2004
Synthesis of alkyne derivatives of a novel triazolopyrazine as A(2A) adenosine receptor antagonists.
    Bioorganic & medicinal chemistry letters, 2005, Feb-01, Volume: 15, Issue:3

    Topics: Adenosine A2 Receptor Antagonists; Administration, Oral; Alkynes; Animals; Catalepsy; Cerebral Cortex; Disease Models, Animal; Mice; Oxidopamine; Parkinson Disease; Pyrazines; Rats; Structure-Activity Relationship; Triazoles

2005
Novel diamino derivatives of [1,2,4]triazolo[1,5-a][1,3,5]triazine as potent and selective adenosine A2a receptor antagonists.
    Journal of medicinal chemistry, 2005, Mar-24, Volume: 48, Issue:6

    Topics: Adenosine A2 Receptor Antagonists; Administration, Oral; Animals; Antiparkinson Agents; Binding, Competitive; Biological Availability; Catalepsy; Cerebral Cortex; Combinatorial Chemistry Techniques; Diamines; In Vitro Techniques; Male; Mice; Pyrrolidines; Radioligand Assay; Rats; Rats, Sprague-Dawley; Stereoisomerism; Triazines; Triazoles

2005
Novel 8-(furan-2-yl)-3-substituted thiazolo [5,4-e][1,2,4] triazolo[1,5-c] pyrimidine-2(3H)-thione derivatives as potential adenosine A(2A) receptor antagonists.
    Bioorganic & medicinal chemistry, 2010, Apr-01, Volume: 18, Issue:7

    Topics: Adenosine A2 Receptor Antagonists; Animals; Antipsychotic Agents; Catalepsy; Cell Line; Cell Membrane; Chromatography, Thin Layer; Computer Simulation; Crystallography, X-Ray; Cyclic AMP; Drug Evaluation, Preclinical; Dyskinesia, Drug-Induced; Haloperidol; Humans; Magnetic Resonance Spectroscopy; Male; Mice; Models, Molecular; Motor Activity; Protein Binding; Pyrimidines; Radioligand Assay; Structure-Activity Relationship; Thiones

2010