Page last updated: 2024-09-03

sb 204070a and Muscle Contraction

sb 204070a has been researched along with Muscle Contraction in 8 studies

Research

Studies (8)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (50.00)18.2507
2000's4 (50.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Karaki, S; Kuwahara, A; Mitsui, R; Ono, S2
Bingham, S; Ellis, ES; Gaster, LM; Joiner, GF; King, FD; Sanger, GJ; Sutton, JM; Wardle, KA; Wyman, PA1
Bingham, S; Gaster, L; King, BF; Rushant, B; Sanger, GJ; Smith, MI1
Ellis, ES; Gaster, LM; Jennings, AJ; Joiner, GF; King, FD; Mulholland, KR; Rahman, SK; Starr, S; Wardle, KA; Wyman, PA1
Briejer, MR; Schuurkes, JA1
Naylor, RJ; Tuladhar, BR; Womack, MD1
Bosmans, JP; Briejer, MR; Heylen, L; Jurzak, M; Leysen, JE; Prins, NH; Schuurkes, JA; Van Daele, P1

Other Studies

8 other study(ies) available for sb 204070a and Muscle Contraction

ArticleYear
Neural and non-neural mediation of propionate-induced contractile responses in the rat distal colon.
    Neurogastroenterology and motility, 2005, Volume: 17, Issue:4

    Topics: Acetates; Anesthetics, Local; Animals; Atropine; Butyrates; Colon; Cyclooxygenase Inhibitors; Dioxanes; Dose-Response Relationship, Drug; Enteric Nervous System; Fatty Acids, Volatile; Intestinal Mucosa; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Piperidines; Piroxicam; Propionates; Rats; Receptors, Serotonin; Serotonin Antagonists

2005
Muscarinic and 5-HT4 receptors participate in the regulation of the frequency of spontaneous contractions of the longitudinal muscle in rat distal colon.
    Biomedical research (Tokyo, Japan), 2005, Volume: 26, Issue:4

    Topics: Animals; Atropine; Colon; Dioxanes; Gastrointestinal Motility; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists

2005
N-[(1-butyl-4-piperidinyl)methyl]-3,4dihydro-2H-[1,3]oxazino[3,2- a]indole10-carboxamide hydrochloride: the first potent and selective 5-HT4 receptor antagonist amide with oral activity.
    Journal of medicinal chemistry, 1995, Nov-24, Volume: 38, Issue:24

    Topics: Administration, Oral; Animals; Dioxanes; Dogs; Guinea Pigs; Indoles; Muscle Contraction; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Structure-Activity Relationship; Sulfonamides

1995
Antagonism by SB 204070 of 5-HT-evoked contractions in the dog stomach: an in-vivo model of 5-HT4 receptor function.
    The Journal of pharmacy and pharmacology, 1995, Volume: 47, Issue:3

    Topics: 4-Aminobenzoic Acid; Animals; Atropine; Dioxanes; Dogs; Dose-Response Relationship, Drug; Drug Interactions; Gastric Mucosa; Gastrointestinal Motility; Granisetron; Injections, Intravenous; Ketanserin; Male; Methiothepin; Methysergide; Muscle Contraction; Muscle, Smooth; para-Aminobenzoates; Piperidines; Random Allocation; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Stomach

1995
(1-Butyl-4-piperidinyl)methyl 8-amino-7-chloro-1,4-benzodioxane-5-carboxylate hydrochloride: a highly potent and selective 5-HT4 receptor antagonist derived from metoclopramide.
    Journal of medicinal chemistry, 1993, Dec-10, Volume: 36, Issue:25

    Topics: Animals; Dioxanes; Guinea Pigs; Metoclopramide; Muscle Contraction; Piperidines; Receptors, Serotonin; Serotonin Antagonists; Structure-Activity Relationship

1993
5-HT3 and 5-HT4 receptors and cholinergic and tachykininergic neurotransmission in the guinea-pig proximal colon.
    European journal of pharmacology, 1996, Jul-18, Volume: 308, Issue:2

    Topics: Animals; Biphenyl Compounds; Colon; Dioxanes; Dose-Response Relationship, Drug; Drug Interactions; Female; Granisetron; Guinea Pigs; In Vitro Techniques; Interneurons; Male; Motor Neurons; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Piperidines; Receptors, Neurokinin-1; Receptors, Serotonin; Serotonin; Serotonin Receptor Agonists

1996
Pharmacological characterization of the 5-HT receptor-mediated contraction in the mouse isolated ileum.
    British journal of pharmacology, 2000, Volume: 131, Issue:8

    Topics: Animals; Atropine; Dioxanes; Dose-Response Relationship, Drug; Female; Granisetron; Ileum; In Vitro Techniques; Indoles; Ketanserin; Male; Mice; Muscle Contraction; Ondansetron; Piperidines; Receptors, Serotonin; Ritanserin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Tetrodotoxin; Tropanes; Tropisetron

2000
The in vitro pharmacological profile of prucalopride, a novel enterokinetic compound.
    European journal of pharmacology, 2001, Jun-29, Volume: 423, Issue:1

    Topics: Acetylcholine; Animals; Benzofurans; Binding, Competitive; Carbachol; Cell Line; CHO Cells; Colon; Cricetinae; Dioxanes; Dogs; Dose-Response Relationship, Drug; Electric Stimulation; Esophagus; Female; Gallbladder; Gastrointestinal Agents; Granisetron; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Indoles; Indomethacin; Male; Motilin; Muscle Contraction; Piperidines; Rabbits; Rats; Rats, Wistar; Receptors, Cholecystokinin; Receptors, Dopamine D2; Receptors, Dopamine D4; Receptors, Gastrointestinal Hormone; Receptors, Neuropeptide; Receptors, Serotonin; Serotonin; Serotonin Antagonists; Serotonin Receptor Agonists; Sincalide; Stomach; Sulfonamides; Vasodilator Agents

2001