quinuclidines has been researched along with Muscle Contraction in 82 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 27 (32.93) | 18.7374 |
1990's | 26 (31.71) | 18.2507 |
2000's | 24 (29.27) | 29.6817 |
2010's | 5 (6.10) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Costa, AM; Galatioto, GP; Gravina, GL; Martella, O; Ronchi, P; Vicentini, C | 1 |
Atorino, G; Aviello, G; Borrelli, F; Capasso, R; Pagano, E; Romano, B | 1 |
Ballarín, M; Balsa, D; Cabellos, J; Davalillo, S; Fernández, A; Lagunas, C; Pérez-Del-Pulgar, S; Salcedo, C | 1 |
Belmonte, K; Blaney, FE; Burman, M; Dufour, J; Foley, JJ; Lainé, DI; Luttmann, MA; McCleland, B; Neipp, C; Palovich, MR; Salmon, M; Thomas, S; Underwood, B; Webb, EF; Widdowson, KL | 1 |
Chen, SJ; Liao, Z; Meng, XM; Mo, ZJ; Xiao, HT; Yan, XY | 1 |
Miyata, K; Ohtake, A; Sasamata, M; Sato, S | 1 |
Colucci, M; Di Giannuario, A; Maione, F; Mascolo, N; Mastriota, M; Palmery, M; Perretti, M; Pieretti, S; Severini, C | 1 |
Akino, H; Aoki, Y; Ito, H; Nagase, K; Tanase, K; Yokoyama, O | 1 |
Chess-Williams, R; Moro, C; Uchiyama, J | 1 |
Chai, W; Chan, KY; Danser, AH; de Maeyer, JH; de Vries, R; MaassenVanDenBrink, A; Saxena, PR; Schuurkes, JA; van den Bogeardt, AJ; Villalón, CM | 1 |
Honda, K; Ikeda, K; Kobayashi, S; Miyata, K; Suzuki, M; Takeuchi, M; Yamada, T | 1 |
Hirano, K; Kanaide, H; Naito, S; Nishimura, J; Takahashi, R | 1 |
De Swert, KO; Joos, GF; Leclere, PG; Lefebvre, RA; Pauwels, RA; Tournoy, KG | 1 |
Depoortere, I; Peeters, TL; Thielemans, L; Thijs, T | 1 |
Shea-Donohue, T; Zhao, A | 1 |
Capparelli, A; Mulè, F; Pizzuti, R; Vergnolle, N | 1 |
Ikeda, K; Naito, R; Okamoto, Y; Takeuchi, M; Toyoshima, A; Yonetoku, Y | 1 |
Chen, HZ; Cui, YY; Feng, JM; Wu, XJ; Zhu, L | 1 |
Bianchetti, A; Croci, T; Di Marzo, V; Di Palo, S; Ferla, G; Guagnini, F; Matias, I; Mukenge, S; Valenti, M | 1 |
Amato, A; Faussone-Pellegrini, MS; Mulè, F; Serio, R; Vannucchi, MG | 1 |
Hatanaka, T; Miyata, K; Noguchi, Y; Ohtake, A; Okutsu, H; Saitoh, C; Sasamata, M; Sato, S; Suzuki, M; Ukai, M; Yuyama, H | 1 |
Inadome, A; Maeda, Y; Masunaga, K; Murakami, S; Satoji, Y; Sugiyama, Y; Ueda, S; Yoshida, M | 1 |
Barlow, RB; Scott, NC; Stephenson, RP | 1 |
Ehler, FJ; Jenden, DJ; Ringdahl, B | 1 |
Jenden, DJ; Jope, RS; Ringdahl, B | 1 |
Jedrych, Z | 1 |
Eikenburg, BE; Johnson, LR; Seidel, ER; Woods, J | 1 |
Johnson, LR; Seidel, ER | 1 |
Lambrecht, G | 1 |
Croci, T; Emonds-Alt, X; Le Fur, G; Manara, L | 1 |
Giuliani, S; Lecci, A; Maggi, CA; Meini, S | 1 |
Andersson, KE; Ishizuka, O; Mattiasson, A | 1 |
Gabelt, BT; Kaufman, PL; Poyer, JF | 1 |
Bonhaus, DW; Clark, R; Eglen, RM; Jakeman, L; Leung, E; Loury, D; Parnes, H; Whiting, RL; Wong, EH | 1 |
Hisaki, M; Kodama, I; Matsushita, T; Ohta, Y; Sakamoto, H; Satake, N; Shibata, S; Zhou, Q | 1 |
Maggi, CA; Meini, S | 1 |
Flügel, C; Kaufman, PL; Poyer, JF | 1 |
Giuliani, S; Maggi, CA | 2 |
Giuliani, S; Maggi, CA; Zagorodnyuk, V | 1 |
Criscuoli, M; Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M | 1 |
Hammer, R; Walland, A | 1 |
Bartolini, A; Bellucci, C; Dei, S; Galeotti, N; Ghelardini, C; Gualtieri, F | 1 |
Giorgio, RD; Giuliani, S; Lecci, A; Maggi, CA; Tramontana, M | 1 |
Aronstam, R; Buccafusco, J; Canney, DJ; Doukas, PH; Gattu, M; Massakowski, C; Zhang, M | 1 |
Angelucci, D; Büchler, MW; Di Mola, FF; Di Sebastiano, P; Friess, H; Grossi, L; Innocenti, P; Marzio, L | 1 |
Hacksell, U; Johansson, G; Nilsson, BM; Nilvebrant, L; Nordvall, G; Sundquist, S | 1 |
Chen, JS; Tian, J; Wei, EQ; Zhang, WP | 1 |
Buljubasich, S; Lau, WA; Pennefather, JN; Ventura, S | 1 |
Alfaro, MJ; Benhamú, B; López-Rodríguez, ML; Martín, MI; Morcillo, MJ; Orensanz, L; Tejada, ID | 1 |
Mustafa, S; Oriowo, MA | 1 |
Giuliani, S; Lecci, A; Maggi, CA; Meini, S; Santicioli, P; Tramontana, M | 1 |
Coupar, IM; Kerr, KP; Mitchelson, F | 1 |
Holzer, P; Shahbazian, A | 1 |
Carr, MJ; Schechter, NM; Undem, BJ | 1 |
Coupar, IM; Kerr, KP; Thai, B | 1 |
Arisawa, H; Fujise, N; Fukui, K; Masunaga, H | 1 |
Furness, JB; Kumano, K; Kunze, WA; Larsson, H; Murr, E; Vogalis, F | 1 |
Mann, TA; Villani, FJ; Wefer, EA | 1 |
Cohen, S; Snape, WJ; Sullivan, MA | 1 |
Aronstam, RS; Eldefrawi, ME; Triggle, DJ | 1 |
Gaginella, TS; Rimele, TJ; Rogers, WA | 1 |
Carson, S; Godwin, S; Kato, G; Massoulié, J | 1 |
Hata, T; Kita, T; Noguchi, Y; Takeyasu, K; Uchida, S; Yoshida, H | 1 |
Hong, E | 1 |
Barlow, RB; Casy, AF | 1 |
Cohen, S; Maayani, S; Sokolovsky, M; Srebrenik, S; Weinstein, H | 1 |
Eglen, RM; Ford, AP; Harris, GC; Pfister, JR; Whiting, RL; Wong, EH | 1 |
Gitter, BD; Howbert, JJ; Nixon, JA; Regoli, D; Rouissi, N; Waters, DC | 1 |
Harada, M; Hidaka, K; Konishi, T; Tamura, T; Terai, M; Tsukamoto, S; Usuda, S; Wanibuchi, F | 1 |
Abreu, M; Audia, VH; Kachur, JF; Kaiser, C; McPherson, DW; Rzeszotarski, WJ; Sturm, B; Weitzberg, M | 1 |
Brotcke, TP; Longhurst, PA | 1 |
Hsu, CT; Hyman, PE; Kao, HW; Ringer, MJ; Snape, WJ; Tomomasa, T | 1 |
Chen, SQ; Dan, ZY; Geng, RL; Yu, ST | 1 |
Cohen, S; Fisher, A; Rubinstein, R | 1 |
Bajgar, J; Bielavský, J; Fusek, J; Herink, J; Hrdina, V; Patocka, J | 1 |
Tarakhovskii, ML | 1 |
Abramson, FB; Barlow, RB; Franks, FM; Pearson, JD | 1 |
Lambrecht, G; Mutschler, E | 1 |
Durant, RC; Friess, SL; Hudak, WV; Martin, HL | 1 |
Dresse, A; Van Dorsser, W | 1 |
Belleau, B; Cox, B; Robinson, JB | 1 |
1 review(s) available for quinuclidines and Muscle Contraction
Article | Year |
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The forefront for novel therapeutic agents based on the pathophysiology of lower urinary tract dysfunction: ameliorative effect of solifenacin succinate (Vesicare), a bladder-selective antimuscarinic agent, on overactive bladder symptoms, especially urgen
Topics: Adenosine Triphosphate; Afferent Pathways; Animals; Disease Models, Animal; Humans; Muscarinic Antagonists; Muscle Contraction; Quinuclidines; Rats; Receptors, Muscarinic; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder, Overactive | 2010 |
2 trial(s) available for quinuclidines and Muscle Contraction
Article | Year |
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Urodynamic parameters after solifenacin treatment in men with overactive bladder symptoms and detrusor underactivity.
Topics: Aged; Humans; Male; Middle Aged; Muscarinic Antagonists; Muscle Contraction; Perception; Prospective Studies; Quality of Life; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Time Factors; Treatment Outcome; Urinary Bladder; Urinary Bladder, Overactive; Urodynamics | 2009 |
Colonic myoelectrical activity in irritable-bowel syndrome. Effect of eating and anticholinergics.
Topics: Administration, Oral; Adult; Aged; Clinical Trials as Topic; Colon; Colonic Diseases, Functional; Eating; Electrophysiology; Gastrointestinal Motility; Humans; Middle Aged; Muscle Contraction; Parasympatholytics; Quinuclidines | 1978 |
79 other study(ies) available for quinuclidines and Muscle Contraction
Article | Year |
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Inhibitory effect of quercetin on rat trachea contractility in vitro.
Topics: Adrenergic alpha-Antagonists; Adrenergic beta-Antagonists; Animals; Antioxidants; Benzamides; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Phentolamine; Piperidines; Propranolol; Quercetin; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Trachea | 2009 |
In vivo and in vitro pharmacological characterization of SVT-40776, a novel M3 muscarinic receptor antagonist, for the treatment of overactive bladder.
Topics: Animals; Atrial Function; Benzhydryl Compounds; Benzofurans; Carbamates; Cresols; Guinea Pigs; In Vitro Techniques; Male; Mice; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder | 2009 |
Discovery of novel 1-azoniabicyclo[2.2.2]octane muscarinic acetylcholine receptor antagonists.
Topics: Animals; Benzhydryl Compounds; Biological Availability; Bronchi; Bronchoconstriction; Bronchodilator Agents; Calcium; CHO Cells; Cricetinae; Cricetulus; Humans; In Vitro Techniques; Mice; Models, Molecular; Muscle Contraction; Muscle, Smooth; Quinuclidines; Radioligand Assay; Rats; Receptor, Muscarinic M3; Structure-Activity Relationship | 2009 |
Characterization of the effect of penehyclidine hydrochloride on muscarinic receptor subtypes mediating the contraction of guinea-pig isolated gastrointestinal smooth muscle.
Topics: Acetylcholine; Animals; Atropine; Cyclic AMP; Dose-Response Relationship, Drug; Female; Gastrointestinal Tract; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Quinuclidines; Radioligand Assay; Receptor, Muscarinic M2; Receptor, Muscarinic M3 | 2009 |
Guinea pig ileum motility stimulation elicited by N-formyl-Met-Leu-Phe (fMLF) involves neurotransmitters and prostanoids.
Topics: Animals; Atropine; Cyclooxygenase 2 Inhibitors; Cyclooxygenase Inhibitors; Dinoprostone; Gastrointestinal Motility; Gastrointestinal Transit; Guinea Pigs; Ileum; Lower Gastrointestinal Tract; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth; N-Formylmethionine Leucyl-Phenylalanine; Neurokinin-1 Receptor Antagonists; Neurotransmitter Agents; Oligopeptides; Piperidines; Piroxicam; Prostaglandins; Quinuclidines; Tetrodotoxin; Thiophenes; Upper Gastrointestinal Tract | 2011 |
Co-administration of an α(1) -blocker improves the efficacy and safety of antimuscarinic agents in rats with detrusor overactivity.
Topics: Adrenergic alpha-1 Receptor Antagonists; Analysis of Variance; Animals; Disease Models, Animal; Diterpenes; Drug Therapy, Combination; Female; Infarction, Middle Cerebral Artery; Muscarinic Antagonists; Muscle Contraction; Organ Size; Quinuclidines; Rats; Rats, Sprague-Dawley; Solifenacin Succinate; Statistics, Nonparametric; Sulfonamides; Tamsulosin; Tetrahydroisoquinolines; Urinary Bladder; Urinary Bladder, Overactive | 2011 |
Urothelial/lamina propria spontaneous activity and the role of M3 muscarinic receptors in mediating rate responses to stretch and carbachol.
Topics: Animals; Atropine; Benzhydryl Compounds; Benzofurans; Carbachol; Cresols; Diamines; Mandelic Acids; Mucous Membrane; Muscarinic Antagonists; Muscle Contraction; Phenylpropanolamine; Piperidines; Pirenzepine; Pyrrolidines; Quinuclidines; Receptor, Muscarinic M3; Solifenacin Succinate; Stress, Mechanical; Swine; Tetrahydroisoquinolines; Tolterodine Tartrate; Urinary Bladder; Urothelium | 2011 |
Inotropic effects of prokinetic agents with 5-HT(4) receptor agonist actions on human isolated myocardial trabeculae.
Topics: 5-Methoxytryptamine; Adolescent; Adult; Aged; Benzofurans; Calcium Channels; Child; Cisapride; Female; Gastrointestinal Agents; Heart Atria; Heart Ventricles; Humans; Indoles; Male; Middle Aged; Muscle Contraction; Myocardium; Pyridines; Quinuclidines; Receptors, Serotonin, 5-HT4; Serotonin; Serotonin 5-HT4 Receptor Agonists; Serotonin Antagonists; Sulfonamides; Young Adult | 2012 |
M(3) receptor antagonism by the novel antimuscarinic agent solifenacin in the urinary bladder and salivary gland.
Topics: Animals; Benzofurans; Bradycardia; Calcium; Carbachol; Cells, Cultured; Cytosol; Dose-Response Relationship, Drug; Female; Guinea Pigs; Humans; In Vitro Techniques; Isoquinolines; Kinetics; Male; Mandelic Acids; Mice; Mice, Inbred BALB C; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Pyrrolidines; Quinuclidines; Rats; Receptor, Muscarinic M3; Receptors, Muscarinic; Salivary Glands; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder | 2002 |
The mechanisms for tachykinin-induced contractions of the rabbit corpus cavernosum.
Topics: Animals; Benzamides; Calcium; Dose-Response Relationship, Drug; Glycopeptides; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Penis; Permeability; Piperidines; Quinuclidines; Rabbits; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Type C Phospholipases | 2002 |
Modulatory role of tachykinin NK1 receptor in cholinergic contraction of mouse trachea.
Topics: Animals; Atropine; Chromatography, High Pressure Liquid; Electric Stimulation; Mice; Mice, Knockout; Muscle Contraction; Parasympathetic Nervous System; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Stereoisomerism; Substance P; Synaptic Transmission; Tetrodotoxin; Trachea | 2003 |
Mechanisms involved in the loss of excitatory post-stimulus responses by inflammation.
Topics: Adenosine Triphosphate; Animals; Colitis; Cyclooxygenase Inhibitors; Electric Stimulation; Female; In Vitro Techniques; Indomethacin; Male; Methiothepin; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase; Piperidines; Purinergic P2 Receptor Antagonists; Quinuclidines; Rabbits; Serotonin Antagonists; Substance P; Suramin; Trinitrobenzenesulfonic Acid | 2003 |
PAR-2 agonists induce contraction of murine small intestine through neurokinin receptors.
Topics: Animals; Benzamides; Capsaicin; Female; Intestine, Small; Mice; Mice, Inbred BALB C; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin-1 Receptor Antagonists; Oligopeptides; Piperidines; Quinuclidines; Receptor, PAR-2; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Thrombin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Substance P; Tetrodotoxin; Trypsin | 2003 |
Evidence for the presence of functional protease activated receptor 4 (PAR4) in the rat colon.
Topics: Animals; Atropine; Benzamides; Capsaicin; Colitis; Colon; Dose-Response Relationship, Drug; Gastrointestinal Motility; Immunohistochemistry; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Oligopeptides; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Receptors, Thrombin; Reverse Transcriptase Polymerase Chain Reaction; RNA, Messenger; Tetrodotoxin | 2004 |
Synthesis and antimuscarinic properties of quinuclidin-3-yl 1,2,3,4-tetrahydroisoquinoline-2-carboxylate derivatives as novel muscarinic receptor antagonists.
Topics: Animals; Female; Models, Molecular; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Quinuclidines; Radioligand Assay; Rats; Rats, Wistar; Receptor, Muscarinic M3; Saliva; Solifenacin Succinate; Stereoisomerism; Structure-Activity Relationship; Tetrahydroisoquinolines; Urinary Bladder; Urinary Incontinence | 2005 |
Aceclidine and pilocarpine interact differently with muscarinic receptor in isolated rabbit iris muscle.
Topics: Animals; Carbachol; Iris; Muscarinic Agonists; Muscle Contraction; Muscle, Smooth; Pilocarpine; Quinuclidines; Rabbits; Receptors, Muscarinic | 2006 |
Neural contractions in colonic strips from patients with diverticular disease: role of endocannabinoids and substance P.
Topics: Adrenergic beta-Agonists; Adrenergic beta-Antagonists; Aged; Arachidonic Acids; Benzoxazines; Cannabinoid Receptor Modulators; Case-Control Studies; Colon; Diverticulum; Endocannabinoids; Female; Glycerides; Humans; Imidazoles; Isoproterenol; Male; Middle Aged; Morpholines; Muscle Contraction; Muscle, Smooth; Naphthalenes; Neurokinin-1 Receptor Antagonists; Piperidines; Polyunsaturated Alkamides; Propanolamines; Pyrazoles; Quinuclidines; Rimonabant; Substance P; Tetrodotoxin | 2006 |
Altered tachykinergic influence on gastric mechanical activity in mdx mice.
Topics: Animals; Benzamides; Disease Models, Animal; Enzyme Inhibitors; Gastrointestinal Motility; Immunohistochemistry; Male; Manometry; Mice; Mice, Inbred mdx; Muscle Contraction; Muscle Tonus; Muscle, Smooth; Muscular Dystrophy, Duchenne; Neurokinin-1 Receptor Antagonists; NG-Nitroarginine Methyl Ester; Nitric Oxide Synthase Type I; Organ Culture Techniques; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Stomach; Tachykinins | 2006 |
Pharmacological characterization of a new antimuscarinic agent, solifenacin succinate, in comparison with other antimuscarinic agents.
Topics: Animals; Atropine; Benzhydryl Compounds; Benzilates; Benzofurans; Binding, Competitive; Carbachol; CHO Cells; Cholinergic Agonists; Cresols; Cricetinae; Cricetulus; Dose-Response Relationship, Drug; In Vitro Techniques; Male; Mandelic Acids; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; N-Methylscopolamine; Phenylpropanolamine; Pyrrolidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Rats, Wistar; Receptors, Muscarinic; Solifenacin Succinate; Tetrahydroisoquinolines; Tolterodine Tartrate; Transfection; Urinary Bladder; Urinary Bladder, Overactive; Urination | 2007 |
Pharmacological effects of solifenacin on human isolated urinary bladder.
Topics: Aged; Calcium Chloride; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; Female; Humans; In Vitro Techniques; Male; Microdialysis; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Potassium Chloride; Quinuclidines; Solifenacin Succinate; Tetrahydroisoquinolines; Urinary Bladder | 2008 |
The affinity and efficacy of onium salts on the frog rectus abdominis.
Topics: Acetylcholine; Animals; Anura; In Vitro Techniques; Muscle Contraction; Pyridinium Compounds; Pyrrolidines; Quinuclidines; Tetraethylammonium Compounds | 1967 |
Muscarinic activity and receptor binding of the enantiomers of aceclidine and its methiodide.
Topics: Analgesics; Animals; Body Temperature; Brain; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Mice; Muscle Contraction; Muscle, Smooth; Oxotremorine; Parasympathomimetics; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic; Stereoisomerism | 1982 |
Inhibition of high affinity choline transport by stereoisomers of some 3-quinuclidinol derivatives.
Topics: Animals; Anura; Biological Transport; Brain; Choline; In Vitro Techniques; Mice; Muscle Contraction; Quinuclidines; Rats; Stereoisomerism | 1984 |
Cholinolytic activity of 3-hydroxyquinuclidyl-1-phenyl-1-cyclohexyl-1-carboxylate hydrochloride (ANC-821).
Topics: Acetylcholine; Animals; Atropine; Bronchi; Electrocardiography; In Vitro Techniques; Male; Mice; Muscle Contraction; Oxotremorine; Parasympatholytics; Pilocarpine; Quinuclidines; Rats; Rats, Inbred Strains | 1983 |
Muscarinic cholinergic receptors in the piebald mouse model for Hirschsprung's disease.
Topics: Animals; Cecum; Colon; Female; Hirschsprung Disease; In Vitro Techniques; Intestine, Large; Kinetics; Male; Mice; Muscle Contraction; Muscle, Smooth; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Rectum | 1983 |
Contraction and [3H]QNB binding in collagenase isolated fundic smooth muscle cells.
Topics: Acetylcholine; Animals; Atropine; Guinea Pigs; Kinetics; Male; Muscle Contraction; Muscle, Smooth; Ouabain; Oxotremorine; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic; Scopolamine; Stomach | 1983 |
[Structure- and conformation-activity relationship of heterocyclic acetylcholine analogs. 13. Cholinergic properties of tertiary and quaternary 4-acetoxyquinuclidines].
Topics: Animals; Cholinesterase Inhibitors; Guinea Pigs; In Vitro Techniques; Molecular Conformation; Muscle Contraction; Muscle, Smooth; Nicotine; Parasympathomimetics; Quinuclidines; Structure-Activity Relationship | 1982 |
In vitro characterization of the non-peptide tachykinin NK1 and NK2-receptor antagonists, SR140333 and SR48968 in different rat and guinea-pig intestinal segments.
Topics: Animals; Atropine; Benzamides; Duodenum; Esophagus; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Piperidines; Quinuclidines; Rats; Receptors, Tachykinin; Substance P | 1995 |
Pharmacological analysis of the local and reflex responses to bradykinin on rat urinary bladder motility in vivo.
Topics: Adrenergic beta-Antagonists; Animals; Bradykinin; Capsaicin; Dose-Response Relationship, Drug; Indoles; Indomethacin; Injections, Spinal; Isoindoles; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Quinuclidines; Rats; Rats, Wistar; Reflex; Substance P; Urinary Bladder | 1995 |
Tachykinin effects on bladder activity in conscious normal rats.
Topics: Administration, Intravesical; Animals; Benzamides; Female; Indoles; Injections, Intra-Arterial; Isoindoles; Muscle Contraction; Muscle, Smooth; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Substance P; Urinary Bladder; Urination | 1995 |
The effect of muscarinic agonists and selective receptor subtype antagonists on the contractile response of the isolated rhesus monkey ciliary muscle.
Topics: Animals; Carbachol; Ciliary Body; Dose-Response Relationship, Drug; In Vitro Techniques; Macaca mulatta; Muscarinic Agonists; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Oxotremorine; Piperidines; Pirenzepine; Quinuclidines | 1994 |
The interaction of RS 25259-197, a potent and selective antagonist, with 5-HT3 receptors, in vitro.
Topics: Animals; Autoradiography; Binding, Competitive; Brain; Guinea Pigs; Ileum; In Vitro Techniques; Isoquinolines; Mice; Muscle Contraction; Muscle, Smooth; Myenteric Plexus; Palonosetron; Quinuclidines; Quipazine; Radioligand Assay; Rats; Receptors, Serotonin; Serotonin Antagonists; Stereoisomerism; Structure-Activity Relationship | 1995 |
Vasoinhibitory effects of NC 1005 and NC 1006, new synthesized antiarrhythmic agents, in isolated rat aorta.
Topics: Aniline Compounds; Animals; Anti-Arrhythmia Agents; Aorta; Calcium; Cyclic AMP; Endothelium; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth, Vascular; Phenylephrine; Potassium Chloride; Quinuclidines; Rats; Rats, Wistar | 1994 |
Evidence for a capsaicin-sensitive, tachykinin-mediated, component in the NANC contraction of the rat urinary bladder to nerve stimulation.
Topics: Adenosine Triphosphate; Animals; Atropine; Capsaicin; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tachykinins; Urinary Bladder | 1994 |
Age does not affect contractile responses of the isolated rhesus monkey ciliary muscle to muscarinic agonists.
Topics: Aging; Animals; Atropine; Carbachol; Cells, Cultured; Ciliary Body; Culture Media; Ganglionic Stimulants; Macaca mulatta; Muscle Contraction; Muscles; Quinuclidines | 1993 |
Role of tachykinins as excitatory mediators of NANC contraction in the circular muscle of rat small intestine.
Topics: Animals; Calcium Channel Blockers; Duodenum; Electric Stimulation; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Nifedipine; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Tachykinins | 1995 |
Evidence that tachykinin NK2 receptors modulate resting tone in the rat isolated small intestine.
Topics: Analysis of Variance; Animals; Benzamides; Electric Stimulation; Evoked Potentials; Intestine, Small; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Neurokinin A; Oligopeptides; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Tachykinin | 1996 |
Sequential activation of the triple excitatory transmission to the circular muscle of guinea-pig colon.
Topics: 4-Aminopyridine; Animals; Atropine; Colon; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Membrane Potentials; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Physalaemin; Piperidines; Quinuclidines; Receptors, Neurokinin-2; Stereoisomerism; Synaptic Transmission; Time Factors | 1997 |
MEN 11,420, a peptide tachykinin NK2 receptor antagonist, reduces motor responses induced by the intravesical administration of capsaicin in vivo.
Topics: Animals; Capsaicin; Hexamethonium; Male; Muscle Contraction; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Tachykinin; Urinary Bladder | 1997 |
Muscarinic contraction in isolated guinea-pig trachea and antagonism by noradrenaline.
Topics: Animals; Bucladesine; Female; Guinea Pigs; In Vitro Techniques; Male; Muscarinic Agonists; Muscle Contraction; Norepinephrine; Quinuclidines; Trachea | 1997 |
In vitro characterization of a novel, potent and selective M3 antagonist.
Topics: Animals; Atrial Function; CHO Cells; Cricetinae; Female; Guinea Pigs; Heart Atria; Ileum; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Quinuclidines; Rabbits; Receptors, Muscarinic; Transfection; Uterine Contraction; Vas Deferens | 1997 |
The role of tachykinin NK1 and NK2 receptors in atropine-resistant colonic propulsion in anaesthetized guinea-pigs.
Topics: Anesthesia; Animals; Apamin; Atropine; Benzamides; Colon; Guinea Pigs; Hexamethonium; Male; Models, Biological; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Peptides, Cyclic; Peristalsis; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2 | 1998 |
Characterization of ethyl (3-quinuclidinyl) acetate (EQA) as a ligand for acetylcholine receptors.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Behavior, Animal; Cerebral Cortex; Evaluation Studies as Topic; Ligands; Male; Mecamylamine; Muscle Contraction; Muscle, Smooth; Nicotinic Antagonists; Quinuclidines; Radioligand Assay; Rats; Rats, Wistar; Receptors, Nicotinic | 1998 |
SR140333, a substance P receptor antagonist, influences morphological and motor changes in rat experimental colitis.
Topics: Animals; Colitis; Colon; Inflammation; Male; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Stereoisomerism; Substance P; Trinitrobenzenesulfonic Acid | 1999 |
Quinuclidin-2-ene-based muscarinic antagonists.
Topics: Animals; Cerebral Cortex; Guinea Pigs; Heart; Molecular Structure; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Myocardium; Parotid Gland; Quinuclidines; Radioligand Assay; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship; Urinary Bladder | 1995 |
Effect of SR-140333, a neurokinin-1 receptor antagonist, on airway reactivity to methacholine in sedated rats.
Topics: Albuterol; Animals; Atropine; Female; In Vitro Techniques; Male; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Respiration; Trachea | 1997 |
An immunohistochemical and pharmacological study of tachykinins in the rat and guinea-pig prostate glands.
Topics: Animals; Atropine; Benzamides; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Immunohistochemistry; In Vitro Techniques; Male; Muscle Contraction; Neurokinin A; Peptide Fragments; Piperidines; Prostate; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Neurokinin-2; Substance P; Tachykinins | 1999 |
Benzimidazole derivatives. 2. Synthesis and structure-activity relationships of new azabicyclic benzimidazole-4-carboxylic acid derivatives with affinity for serotoninergic 5-HT(3) receptors.
Topics: Animals; Benzimidazoles; Cell Membrane; Cerebral Cortex; Electric Stimulation; Guinea Pigs; Ileum; Male; Molecular Structure; Muscle Contraction; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Serotonin; Receptors, Serotonin, 5-HT3; Serotonin Antagonists; Structure-Activity Relationship | 1999 |
Inhibitory effect of capsaicin on cholinergic transmission in ovine airways: evidence for non-cholinergic contractions.
Topics: Acetylcholine; Animals; Capsaicin; Carbachol; Dose-Response Relationship, Drug; Electric Stimulation; In Vitro Techniques; Lung; Muscle Contraction; Muscle, Smooth; Neural Inhibition; Neurokinin-1 Receptor Antagonists; Neuromuscular Junction; Peptides, Cyclic; Quinuclidines; Receptors, Drug; Receptors, Neurokinin-2; Serotonin; Sheep; Substance P; Synaptic Transmission; Trachea | 1999 |
Tachykinin-mediated effect of nociceptin in the rat urinary bladder in vivo.
Topics: Administration, Topical; Animals; Ganglia, Autonomic; Male; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Nociceptin; Opioid Peptides; Peptides, Cyclic; Piperidines; Quinuclidines; Rats; Rats, Wistar; Receptors, Neurokinin-2; Tachykinins; Urinary Bladder; Urination | 2000 |
Tachykinins play a minor role in mediating the third phase of the contractile response to vagal nerve stimulation of the guinea-pig oesophagus.
Topics: Animals; Benzamides; Electric Stimulation; Esophagus; Guinea Pigs; In Vitro Techniques; Indoles; Isoindoles; Male; Muscle Contraction; Neurokinin-1 Receptor Antagonists; Piperidines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Receptors, Tachykinin; Vagus Nerve | 2000 |
Differences in circular muscle contraction and peristaltic motor inhibition caused by tachykinin NK1 receptor agonists in the guinea-pig small intestine.
Topics: Adenosine Triphosphate; Animals; Enzyme Inhibitors; Female; Guinea Pigs; Intestine, Small; Male; Motor Neurons; Muscle Contraction; Muscle, Smooth; Neurokinin A; NG-Nitroarginine Methyl Ester; Nitric Oxide; Nitric Oxide Synthase; Peptide Fragments; Peristalsis; Piperidines; Purinergic P2 Receptor Antagonists; Pyrrolidonecarboxylic Acid; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Sincalide; Spasm; Substance P; Suramin; Tetrodotoxin | 2000 |
Trypsin-induced, neurokinin-mediated contraction of guinea pig bronchus.
Topics: Animals; Benzamides; Bronchoconstriction; Capsaicin; Chymases; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Neurokinin-1 Receptor Antagonists; Oligopeptides; Piperidines; Quinuclidines; Receptor, PAR-1; Receptor, PAR-2; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Thrombin; Serine Endopeptidases; Tachykinins; Thrombin; Trachea; Trypsin; Tryptases | 2000 |
Tachykinin-induced contraction of the guinea-pig isolated oesophageal mucosa is mediated by NK(2) receptors.
Topics: Animals; Benzamides; Captopril; Dose-Response Relationship, Drug; Esophagus; Guinea Pigs; In Vitro Techniques; Mucous Membrane; Muscle Contraction; Neurokinin A; Neurokinin B; Neurokinin-1 Receptor Antagonists; Peptide Fragments; Piperidines; Protease Inhibitors; Quinolines; Quinuclidines; Receptors, Neurokinin-1; Receptors, Neurokinin-2; Receptors, Neurokinin-3; Substance P; Tachykinins; Thiorphan | 2000 |
General pharmacological profile of the novel muscarinic receptor agonist SNI-2011, a drug for xerostomia in Sjögren's syndrome. 2nd communication: effects on somatic nervous system and on autonomic nervous system and smooth muscle.
Topics: Anesthetics; Animals; Autonomic Nervous System; Catecholamines; Cats; Guinea Pigs; Histamine Antagonists; Male; Mice; Mice, Inbred ICR; Muscarinic Agonists; Muscle Contraction; Muscle Relaxants, Central; Muscle, Smooth; Muscle, Smooth, Vascular; Neuromuscular Junction; Nictitating Membrane; Peripheral Nervous System; Pupil; Quinuclidines; Rabbits; Rats; Rats, Inbred F344; Rats, Wistar; Sjogren's Syndrome; Thiophenes; Xerostomia | 2002 |
Sensitization of enteric reflexes in the rat colon in vitro.
Topics: Animals; Area Under Curve; Carbachol; Cholinergic Agonists; Colon; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Female; Gastrointestinal Motility; Granisetron; Hexamethonium; In Vitro Techniques; Indomethacin; Male; Muscle Contraction; Neurons, Afferent; Nicotinic Antagonists; Piperidines; Quinuclidines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Receptors, Tachykinin; Serotonin Antagonists; Time Factors | 2002 |
Tricyclic quinuclidylidenes as potential antihistamine-bronchodilating agents.
Topics: Aerosols; Animals; Bronchodilator Agents; Dyspnea; Guinea Pigs; Histamine; Histamine H1 Antagonists; Lung; Muscle Contraction; Quinuclidines | 1975 |
Structural and stereochemical requirements for muscarinic receptor binding.
Topics: Animals; Binding, Competitive; Brain; Chemical Phenomena; Chemistry; Guinea Pigs; Ileum; In Vitro Techniques; Kinetics; Male; Molecular Conformation; Muscle Contraction; Muscle, Smooth; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Stereoisomerism; Structure-Activity Relationship | 1979 |
Characterization of muscarinic cholinergic receptors in the lower esophageal sphincter of the cat: binding of [3H]quinuclidinyl benzilate.
Topics: Animals; Atropine; Bethanechol Compounds; Cats; Esophagogastric Junction; Female; Kinetics; Male; Muscle Contraction; Quinuclidines; Quinuclidinyl Benzilate; Receptors, Cholinergic; Receptors, Muscarinic | 1979 |
Biochemical studies on muscarinic receptors.
Topics: Acetylcholine; Alkylating Agents; Animals; Atropine; Binding, Competitive; Brain; Carbachol; Cattle; Choline; Dexetimide; Kinetics; Ligands; Muscle Contraction; Muscle, Smooth; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Muscarinic; Solubility; Subcellular Fractions | 1977 |
Decrease in muscarinic acetylcholine receptors in the small intestine of mice subjected to repeated cold stress.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Brain; Cold Temperature; In Vitro Techniques; Intestine, Small; Male; Mice; Muscle Contraction; Muscle, Smooth; Parasympatholytics; Quinuclidines; Receptors, Cholinergic; Receptors, Muscarinic; Stress, Physiological | 1978 |
On the adrenergic neuron blocking activity of 1-methyl-3-keto-4-phenylquinuclidinium bromide (MA540) during acute and chronic administration.
Topics: Animals; Cats; Drug Tolerance; Electric Stimulation; Female; Guanethidine; Hypertension; Ileum; Male; Muscle Contraction; Muscle, Smooth; Nictitating Membrane; Norepinephrine; Quinuclidines; Rabbits; Sympathetic Nervous System; Sympatholytics; Tyramine | 1976 |
Inversion of stereospecificity by methylation of compounds acting at acetylcholine receptors.
Topics: Acetylcholine; Animals; Anura; Guinea Pigs; Ileum; In Vitro Techniques; Methylation; Molecular Conformation; Muscle Contraction; Muscle, Smooth; Muscles; Quinuclidines; Rana temporaria; Receptors, Cholinergic; Stereoisomerism; Structure-Activity Relationship | 1975 |
A theoretical and experimental study of the semirigid cholinergic agonist 3-acetoxyquinuclidine.
Topics: Acetylcholinesterase; Animals; Binding Sites; Butyrylcholinesterase; Chemical Phenomena; Chemistry; Energy Transfer; Erythrocytes; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Mice; Models, Structural; Molecular Conformation; Muscle Contraction; Muscle, Smooth; Optical Rotation; Parasympathomimetics; Pupil; Quantum Theory; Quinuclidines | 1975 |
The action of (+/-)L-660,863 [(+/-)3-(3-amino-1,2,4-oxadiazole-5-yl)-quinuclidine] at muscarinic receptor subtypes in vitro.
Topics: Animals; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Oxadiazoles; Quinuclidines; Radioligand Assay; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Uterine Contraction | 1992 |
Selectivity and specificity of new, non-peptide, quinuclidine antagonists of substance P.
Topics: Angiotensin II; Animals; Blood Vessels; Bradykinin; Cell Line; Guinea Pigs; Humans; Muscle Contraction; Norepinephrine; Quinuclidines; Rabbits; Rats; Rats, Inbred Strains; Receptors, Neurokinin-1; Receptors, Neurotransmitter; Substance P | 1991 |
Pharmacological studies on novel muscarinic agonists, 1-oxa-8-azaspiro[4.5]decane derivatives, YM796 and YM954.
Topics: Animals; Avoidance Learning; Hippocampus; Hydrolysis; Hypothermia; Ileum; In Vitro Techniques; Male; Mice; Mice, Inbred ICR; Muscle Contraction; Muscle, Smooth; Parasympathomimetics; Phosphatidylinositols; Quinuclidines; Rats; Rats, Inbred Strains; Receptors, Muscarinic; Scopolamine; Spiro Compounds; Succinimides; Thiophenes; Tremor | 1990 |
Synthesis of some 3-(1-azabicyclo[2.2.2]octyl) 3-amino-2-hydroxy-2-phenylpropionates: profile of antimuscarinic efficacy and selectivity.
Topics: Animals; Bridged Bicyclo Compounds; Bridged-Ring Compounds; Carbachol; Chemical Phenomena; Chemistry; Guinea Pigs; Ileum; Lactates; Male; Molecular Structure; Muscle Contraction; Myocardial Contraction; Parasympatholytics; Phenylpropionates; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Rats; Receptors, Muscarinic; Vas Deferens | 1990 |
Effects of castration and diabetes mellitus on cholinergic responsiveness and muscarinic receptors in the rat vas deferens.
Topics: Animals; Atropine; Binding Sites; Carbachol; Diabetes Mellitus, Experimental; Male; Muscle Contraction; Muscle, Smooth; Orchiectomy; Potassium Chloride; Quinuclidines; Quinuclidinyl Benzilate; Rats; Rats, Inbred BB; Rats, Inbred Strains; Receptors, Muscarinic; Vas Deferens | 1989 |
[3H]QNB binding and contraction of rabbit colonic smooth muscle cells.
Topics: Animals; Atropine; Bethanechol; Bethanechol Compounds; Binding, Competitive; Cell Count; Colon; Kinetics; Male; Microbial Collagenase; Muscle Contraction; Muscle, Smooth; Phenethylamines; Pirenzepine; Quinuclidines; Quinuclidinyl Benzilate; Rabbits; Receptors, Cholinergic | 1987 |
[Studies on the synthesis and neuromuscular-blocking activity of symmetrical bis-and poly-quaternary derivatives of quinuclidine and tropine].
Topics: Animals; Diaphragm; Muscle Contraction; Neuromuscular Blocking Agents; Quinuclidines; Rats; Tropanes | 1987 |
Antihistaminic properties of AF-14, an experimental quinuclidine derivative: discrimination between two histaminergic sites in both guinea-pig ileum and bladder.
Topics: Animals; Atropine; Guinea Pigs; Histamine; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neostigmine; Parasympatholytics; Quinuclidines; Receptors, Histamine; Urinary Bladder | 1985 |
Pharmacology of 1, 2, 3, 4-tetrahydro-9-amino-acridine.
Topics: Acetylcholinesterase; Acridines; Allosteric Regulation; Amines; Animals; Benzilates; Binding Sites; Cholinesterase Inhibitors; Cholinesterases; Depression, Chemical; Gastrointestinal Motility; Heart; Heart Rate; In Vitro Techniques; Kinetics; Muscle Contraction; Physostigmine; Quinuclidines; Rats; Stimulation, Chemical; Tubocurarine | 1974 |
Role of sulfhydryl groups in the mechanism of uterine contraction in response to stimulation of cholinergic and serotoninergic receptors.
Topics: Animals; Barium; Cadmium; Chlorpromazine; Female; Morphine; Muscle Contraction; Procaine; Quinuclidines; Rats; Receptors, Cholinergic; Receptors, Drug; Serotonin; Stimulation, Chemical; Sulfhydryl Compounds; Uterus | 1974 |
Relationships between chemical structure and affinity for postganglionic acetylcholine receptors of the guinea-pig ileum.
Topics: Acetylcholine; Amino Alcohols; Animals; Atropine; Autonomic Fibers, Postganglionic; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; In Vitro Techniques; Mathematics; Methylation; Molecular Conformation; Muscle Contraction; Parasympathomimetics; Piperidines; Pyrrolidines; Quinuclidines; Receptors, Cholinergic; Structure-Activity Relationship | 1974 |
[Structure- and conformation-activity relationships of cyclic acetylcholine analogs of the piperidine and quinuclidine series].
Topics: Acetylcholine; Animals; Dose-Response Relationship, Drug; Esters; Guinea Pigs; Ileum; Molecular Conformation; Muscle Contraction; Piperidines; Quinuclidines; Receptors, Cholinergic; Structure-Activity Relationship | 1974 |
Comparative blocking actions of methylated 3-quinuclidinyl and 3-tropinyl residues in cholinergic systems.
Topics: Animals; Cats; Dose-Response Relationship, Drug; Electric Stimulation; Evoked Potentials; Ganglia, Autonomic; Muscle Contraction; Muscles; Parasympathetic Nervous System; Quinuclidines; Tropanes | 1973 |
[Comparative effects of various antidepressants on the response to noradrenaline of the deferent canal and the arterial pressure, and the response to 5-hydroxytryptamine of the rat uterus].
Topics: Amitriptyline; Animals; Antidepressive Agents; Blood Pressure; Carotid Arteries; Clomipramine; Dibenzazepines; Dose-Response Relationship, Drug; Drug Interactions; Female; Imipramine; In Vitro Techniques; Male; Muscle Contraction; Norepinephrine; Orphenadrine; Quinuclidines; Rats; Serotonin; Uterus; Vas Deferens | 1974 |
3-acetoxyquinuclidine methiodide. Resolution, absolute configuration, and stereospecificity of interaction with the acetylcholine binding sites.
Topics: Acetylcholine; Acetylcholinesterase; Animals; Atropine; Binding Sites; Chemical Phenomena; Chemistry; Erythrocytes; Guinea Pigs; Ileum; Iodides; Kinetics; Muscle Contraction; Parasympathomimetics; Quinuclidines; Stereoisomerism | 1969 |