Page last updated: 2024-08-17

quinoxalines and Carcinoma, Transitional Cell

quinoxalines has been researched along with Carcinoma, Transitional Cell in 26 studies

Research

Studies (26)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (3.85)29.6817
2010's4 (15.38)24.3611
2020's21 (80.77)2.80

Authors

AuthorsStudies
Claiborne, RT; Tsan, GL1
Avadhani, A; De Porre, P; Dosne, AG; Goeyvaerts, N; Li, LY; O'Hagan, A; Ouellet, D; Perez Ruixo, JJ; Valade, E1
Akapame, S; Burgess, EF; Duran, I; Fleming, MT; García-Donas, J; Huddart, RA; Joshi, M; Loriot, Y; Mellado, B; Monga, M; Necchi, A; O'Hagan, A; Park, SH; Rezazadeh Kalebasty, A; Santiago-Walker, AE; Siefker-Radtke, AO; Tagawa, ST; Varlamov, S; Zakharia, Y1
Loriot, Y; Siefker-Radtke, AO1
Cosmai, L; Franza, A; Giannatempo, P; Pirovano, M1
Belal, F; El-Enany, N; Elawady, T; Khedr, A1
Arai, S; Fujizuka, Y; Kato, M; Koike, H; Maeno, Y; Matsui, H; Miyazawa, Y; Ohtsu, A; Sawada, T; Sekine, Y; Suzuki, K1
Chang, SS1
Bellmunt, J; Montazeri, K1
Kolesar, JM; Myint, ZW; Roubal, K1
Grülllich, C1
Burgess, M; English, A; Hartmann, A; Major, C; Sweeney, M; Wang, S1
Galsky, MD; Patel, V; Qin, Q1
Amir, M; Javed, S; Qureshi, MA1
Ertl, IE; Ilijazi, D; Loriot, Y; Mostafaei, H; Shariat, SF1
Bagby, S; Bortoletti, C; D'Angelo, A; Galli, IC; Roviello, G1
Montazeri, K; Sonpavde, G1
Bossaer, JB; Weaver, A1
Bansal, P; Dwivedi, DK; Goyal, S; Gupta, V; Hatwal, D; Maithani, M; Sharma, P1
Hubert, P; Loriot, Y; Selmani, Z; Thiery-Vuillemin, A1
Kim, HS; Seo, HK1
Markham, A1
He, S; Li, X; Martin, DT; Tian, Y; Weiss, RM1
Burki, TK1
Bastaros, JM; Carles, J; de Castro, AM; Maldonado, X; Morales-Barrera, R; Morote, J; Racca, F; Suárez, C; Valverde, C1
Archer, CL; Haas, GP; Jones, RF; Morse, P; Shirai, T; Wang, CY1

Reviews

12 review(s) available for quinoxalines and Carcinoma, Transitional Cell

ArticleYear
Erdafitinib in locally advanced/metastatic urothelial carcinoma with certain
    Future oncology (London, England), 2022, Volume: 18, Issue:19

    Topics: Carcinoma, Transitional Cell; Humans; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Urinary Bladder Neoplasms

2022
Erdafitinib for the treatment of metastatic bladder cancer.
    Expert review of clinical pharmacology, 2020, Volume: 13, Issue:1

    Topics: Animals; Carcinoma, Transitional Cell; Humans; Neoplasm Metastasis; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 2; Receptor, Fibroblast Growth Factor, Type 3; Urinary Bladder Neoplasms

2020
Erdafitinib: A novel therapy for FGFR-mutated urothelial cancer.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2020, Feb-19, Volume: 77, Issue:5

    Topics: Antineoplastic Agents; Carcinoma, Transitional Cell; Humans; Progression-Free Survival; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 2; Receptor, Fibroblast Growth Factor, Type 3; Urinary Bladder Neoplasms

2020
[High response rates for erdafitinib in patients with FGFR-mutated urothelial carcinoma following failure of platinum-based chemotherapy].
    Der Urologe. Ausg. A, 2020, Volume: 59, Issue:4

    Topics: Carcinoma, Transitional Cell; Humans; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Treatment Outcome; Urologic Neoplasms; Urothelium

2020
Urothelial carcinoma: the development of FGFR inhibitors in combination with immune checkpoint inhibitors.
    Expert review of anticancer therapy, 2020, Volume: 20, Issue:6

    Topics: Antineoplastic Combined Chemotherapy Protocols; Carcinoma, Transitional Cell; Drug Development; Humans; Immune Checkpoint Inhibitors; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 3; Signal Transduction; Urinary Bladder Neoplasms

2020
Fibroblast growth factor receptors across urothelial carcinoma landscape.
    Current opinion in urology, 2020, Volume: 30, Issue:4

    Topics: Antineoplastic Agents; Carcinoma, Transitional Cell; Humans; Neoplasm Recurrence, Local; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 3; Receptors, Fibroblast Growth Factor; Treatment Outcome; Urinary Bladder Neoplasms; Urologic Neoplasms

2020
Overview of the clinical use of erdafitinib as a treatment option for the metastatic urothelial carcinoma: where do we stand.
    Expert review of clinical pharmacology, 2020, Volume: 13, Issue:10

    Topics: Administration, Oral; Adult; Antineoplastic Agents; Apoptosis; Carcinoma, Transitional Cell; Disease Progression; Humans; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Urinary Bladder Neoplasms

2020
Salvage systemic therapy for metastatic urothelial carcinoma: an unmet clinical need.
    Expert review of anticancer therapy, 2021, Volume: 21, Issue:3

    Topics: Antibodies, Monoclonal; Biomarkers, Tumor; Carcinoma, Transitional Cell; Humans; Immune Checkpoint Inhibitors; Molecular Targeted Therapy; Neoplasm Metastasis; Pyrazoles; Quinoxalines; Salvage Therapy; Survival Rate; Urinary Bladder Neoplasms

2021
Fibroblast growth factor receptor (FGFR) inhibitors: A review of a novel therapeutic class.
    Journal of oncology pharmacy practice : official publication of the International Society of Oncology Pharmacy Practitioners, 2021, Volume: 27, Issue:3

    Topics: Bile Duct Neoplasms; Carcinoma, Transitional Cell; Cholangiocarcinoma; Clinical Trials as Topic; Humans; Morpholines; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Pyrroles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 2; Receptor, Fibroblast Growth Factor, Type 3

2021
Erdafitinib as a Novel and Advanced Treatment Strategy of Metastatic Urothelial Carcinoma.
    Anti-cancer agents in medicinal chemistry, 2021, Volume: 21, Issue:18

    Topics: Antineoplastic Agents; Carcinoma, Transitional Cell; Cell Proliferation; Drug Screening Assays, Antitumor; Humans; Pyrazoles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 3; Urinary Bladder Neoplasms

2021
Emerging treatments for bacillus Calmette-Guérin-unresponsive non-muscle-invasive bladder cancer.
    Investigative and clinical urology, 2021, Volume: 62, Issue:4

    Topics: Adjuvants, Immunologic; Administration, Intravesical; Antineoplastic Agents; BCG Vaccine; Carcinoma, Transitional Cell; Clinical Trials as Topic; Genes, Viral; Genetic Therapy; Humans; Hyperthermia; Immune Checkpoint Inhibitors; Immunoconjugates; Organ Sparing Treatments; Photochemotherapy; Pyrazoles; Quinoxalines; Retreatment; Treatment Failure; Urinary Bladder Neoplasms

2021
Targeting fibroblast growth factor receptors and immune checkpoint inhibitors for the treatment of advanced bladder cancer: New direction and New Hope.
    Cancer treatment reviews, 2016, Volume: 50

    Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Carcinoma, Transitional Cell; Humans; Ipilimumab; Nivolumab; Phenylurea Compounds; Piperazines; Pyrazoles; Pyridines; Pyrimidines; Quinolines; Quinoxalines; Receptors, Fibroblast Growth Factor; Urinary Bladder Neoplasms

2016

Trials

3 trial(s) available for quinoxalines and Carcinoma, Transitional Cell

ArticleYear
Exposure-response analyses of erdafitinib in patients with locally advanced or metastatic urothelial carcinoma.
    Cancer chemotherapy and pharmacology, 2022, Volume: 89, Issue:2

    Topics: Aged; Carcinoma, Transitional Cell; Dose-Response Relationship, Drug; Female; Humans; Male; Middle Aged; Progression-Free Survival; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Receptors, Fibroblast Growth Factor; Survival Rate; Urinary Bladder Neoplasms

2022
Efficacy and safety of erdafitinib in patients with locally advanced or metastatic urothelial carcinoma: long-term follow-up of a phase 2 study.
    The Lancet. Oncology, 2022, Volume: 23, Issue:2

    Topics: Aged; Carcinoma, Transitional Cell; Central Serous Chorioretinopathy; ErbB Receptors; Follow-Up Studies; Humans; Middle Aged; Mutation; Neoplasm Metastasis; Pyrazoles; Quinoxalines; Urinary Bladder Neoplasms

2022
Erdafitinib for advanced urothelial carcinoma.
    The Lancet. Oncology, 2019, Volume: 20, Issue:9

    Topics: Carcinoma, Transitional Cell; Drug-Related Side Effects and Adverse Reactions; Humans; Mutation; Progression-Free Survival; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 2; Receptor, Fibroblast Growth Factor, Type 3; Urologic Neoplasms; Urothelium

2019

Other Studies

11 other study(ies) available for quinoxalines and Carcinoma, Transitional Cell

ArticleYear
Case Report: Erdafitinib-induced Central Serous Chorioretinopathy.
    Optometry and vision science : official publication of the American Academy of Optometry, 2022, 01-01, Volume: 99, Issue:1

    Topics: Aged, 80 and over; Carcinoma, Transitional Cell; Central Serous Chorioretinopathy; Female; Humans; Male; Protein Kinase Inhibitors; Pyrazoles; Quality of Life; Quinoxalines; Receptors, Fibroblast Growth Factor; United States; Urinary Bladder Neoplasms

2022
Erdafitinib for locally advanced or metastatic urothelial carcinoma.
    American journal of health-system pharmacy : AJHP : official journal of the American Society of Health-System Pharmacists, 2022, 05-24, Volume: 79, Issue:11

    Topics: Carcinoma, Transitional Cell; Humans; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Urinary Bladder Neoplasms

2022
Utility of Kolliphor RH 40 in micellar sensitized fluorescence of the novel tyrosine kinase inhibitor "Erdafitinib": Application to human plasma.
    Spectrochimica acta. Part A, Molecular and biomolecular spectroscopy, 2022, Oct-05, Volume: 278

    Topics: Carcinoma, Transitional Cell; Humans; Micelles; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Solvents; Spectrometry, Fluorescence; Urinary Bladder Neoplasms

2022
Fibroblast growth factor receptor inhibitor erdafitinib promotes Mcl-1 degradation and synergistically induces apoptosis with Bcl-xL/Bcl-2 inhibitor in urothelial cancer cells.
    Biochemical and biophysical research communications, 2022, 11-05, Volume: 628

    Topics: Antineoplastic Agents; Apoptosis; Apoptosis Regulatory Proteins; bcl-X Protein; Carcinoma, Transitional Cell; Cell Line, Tumor; Humans; Myeloid Cell Leukemia Sequence 1 Protein; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-bcl-2; Pyrazoles; Quinoxalines; Receptors, Fibroblast Growth Factor

2022
Re: Erdafitinib in Locally Advanced or Metastatic Urothelial Carcinoma.
    The Journal of urology, 2020, Volume: 203, Issue:2

    Topics: Carcinoma, Transitional Cell; Humans; Pyrazoles; Quinoxalines; Urologic Neoplasms

2020
Identifying fibroblast growth factor receptor genetic alterations using RNA-based assays in patients with metastatic or locally advanced, surgically unresectable, urothelial carcinoma who may benefit from erdafitinib treatment.
    The journal of pathology. Clinical research, 2020, Volume: 6, Issue:3

    Topics: Aged; Carcinoma, Transitional Cell; Female; Humans; Male; Middle Aged; Pyrazoles; Quinoxalines; Real-Time Polymerase Chain Reaction; Receptor, Fibroblast Growth Factor, Type 2; Receptor, Fibroblast Growth Factor, Type 3; Urologic Neoplasms

2020
Biomolecular interactions and binding dynamics of tyrosine kinase inhibitor erdafitinib, with human serum albumin.
    Journal of biomolecular structure & dynamics, 2021, Volume: 39, Issue:11

    Topics: Binding Sites; Carcinoma, Transitional Cell; Circular Dichroism; Humans; Molecular Docking Simulation; Protein Binding; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Serum Albumin, Human; Spectrometry, Fluorescence; Thermodynamics; Tumor Microenvironment; Urinary Bladder Neoplasms

2021
FGFR alterations in urothelial carcinoma: Picking the right target.
    Bulletin du cancer, 2021, Volume: 108, Issue:6

    Topics: Carcinoma, Transitional Cell; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Gene Fusion; Humans; Molecular Targeted Therapy; Morpholines; Mutation; Phenylurea Compounds; Piperazines; Protein Kinase Inhibitors; Pyrazoles; Pyrimidines; Pyrroles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 2; Receptor, Fibroblast Growth Factor, Type 3; Thiophenes; Urinary Bladder Neoplasms

2021
Erdafitinib: First Global Approval.
    Drugs, 2019, Volume: 79, Issue:9

    Topics: Antineoplastic Agents; Carcinoma, Transitional Cell; Drug Approval; Humans; Protein Kinase Inhibitors; Pyrazoles; Quinoxalines; Receptor, Fibroblast Growth Factor, Type 2; Receptor, Fibroblast Growth Factor, Type 3; Treatment Outcome; United States; United States Food and Drug Administration; Urologic Neoplasms

2019
Synergistic inhibition of GP130 and ERK signaling blocks chemoresistant bladder cancer cell growth.
    Cellular signalling, 2019, Volume: 63

    Topics: Butadienes; Carcinoma, Transitional Cell; Cell Line, Tumor; Cell Movement; Cell Survival; Drug Resistance, Neoplasm; Drug Synergism; Enzyme Inhibitors; Gene Expression Regulation, Neoplastic; Glycoproteins; Humans; Hydrazines; MAP Kinase Signaling System; Mitogen-Activated Protein Kinase 1; Nitriles; Quinoxalines; Urinary Bladder Neoplasms

2019
Carcinogenicity of the N-hydroxy derivative of 2-amino-1-methyl-6-phenylimidazo[4,5-b]pyridine, 2-amino-3, 8-dimethyl-imidazo[4,5-f]quinoxaline and 3, 2'-dimethyl-4-aminobiphenyl in the rat.
    Cancer letters, 2000, Jul-03, Volume: 155, Issue:1

    Topics: Aminobiphenyl Compounds; Animals; Animals, Newborn; Body Weight; Carcinogens; Carcinoma, Transitional Cell; Colonic Neoplasms; Hyperplasia; Imidazoles; Male; Mutagens; Prostatic Neoplasms; Pyridines; Quinoxalines; Rats; Rats, Inbred ACI; Urinary Bladder Neoplasms

2000