Page last updated: 2024-08-17

quinoline and Trypanosomiasis, African

quinoline has been researched along with Trypanosomiasis, African in 2 studies

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's1 (50.00)24.3611
2020's1 (50.00)2.80

Authors

AuthorsStudies
Basta, A; Biancofiore, I; Ciammaichella, A; D'Amico, M; Ferrigno, F; Fini, I; Gennari, N; Graziani, R; Harper, S; Nardi, V; Ontoria, JM; Paonessa, G; Ponzi, S; Summa, V; Vittoria Orsale, M1
Bland, ND; Campbell, RK; Ochiana, SO; Pollastri, MP; Settimo, L1

Other Studies

2 other study(ies) available for quinoline and Trypanosomiasis, African

ArticleYear
Optimization of 2-(1H-imidazo-2-yl)piperazines series of Trypanosoma brucei growth inhibitors as potential treatment for the second stage of HAT.
    Bioorganic & medicinal chemistry letters, 2020, 06-15, Volume: 30, Issue:12

    Topics: Cell Survival; Drug Evaluation, Preclinical; Growth Inhibitors; Human Umbilical Vein Endothelial Cells; Humans; Isomerism; Morpholines; Piperazines; Quinolines; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis, African

2020
Repurposing human PDE4 inhibitors for neglected tropical diseases. Evaluation of analogs of the human PDE4 inhibitor GSK-256066 as inhibitors of PDEB1 of Trypanosoma brucei.
    Chemical biology & drug design, 2015, Volume: 85, Issue:5

    Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Aminoquinolines; Binding Sites; Cyclic Nucleotide Phosphodiesterases, Type 4; Drug Repositioning; Humans; Molecular Docking Simulation; Neglected Diseases; Phosphodiesterase 4 Inhibitors; Protein Structure, Tertiary; Protozoan Proteins; Quinolines; Structure-Activity Relationship; Sulfones; Trypanosoma brucei brucei; Trypanosomiasis, African

2015