Page last updated: 2024-08-17

quinoline and Malaria

quinoline has been researched along with Malaria in 48 studies

Research

Studies (48)

TimeframeStudies, this research(%)All Research%
pre-199031 (64.58)18.7374
1990's0 (0.00)18.2507
2000's2 (4.17)29.6817
2010's9 (18.75)24.3611
2020's6 (12.50)2.80

Authors

AuthorsStudies
Bharate, SB; Mudududdla, R; Nuthakki, VK1
Gao, F; Kong, F; Sun, Z; Xiao, J1
Chang, L; Ding, C; Feng, LS; Gao, C; Li, C; Shi, F; Wu, X; Xu, Z; Yan, XF; Zhao, F1
Chibale, K; Combrinck, J; D'hooghe, M; Minić, A; Smith, PJ; Van de Walle, T; Van Hecke, K1
Cheong, SL; Ng, CH; Tibon, NS1
Egan, TJ; Joshi, MC1
Avery, SV; Vallières, C1
Faist, J; Hochegger, P; Kaiser, M; Mäser, P; Saf, R; Seebacher, W; Weis, R1
Gorka, AP; Jacobs, LM; Roepe, PD1
Bohn, K; Chmielewski, J; Ferdig, M; Fidock, DA; Henrich, PP; Hrycyna, CA; Kirk, K; Kuriakose, J; Lehane, AM; Martin, RE; Namanja, H; Pires, MM; Summers, RL1
JOSEPH, AA; LOUGHLIN, EH; RAPPAPORT, I; RICE, JB; WELLS, HS1
Gryzło, B; Kulig, K1
D'hooghe, M; Vandekerckhove, S1
Boechat, N; Ferreira, Mde L; Jesus, AM; Júnior, CC; Krettli, AU; Leite, MM; Pinheiro, LC; Souza, NB1
CRAIGE, B; JONES, R1
BERLINER, RW; EARLE, DP1
ARCHIBALD, RM; WEISIGER, JR1
TOLMAN, LL1
SARGENT, H1
RAPPORT, MM; SENEAR, AE1
SARGENT, H; SENEAR, AE1
BROWN, RF; JACOBS, TL1
KOEPFLI, JB; MEAD, JF; SENEAR, AE1
BUCHMAN, ER; SARGENT, H1
JACOBS, TL; WINSTEIN, S1
NORTON, TR; SEIBERT, RA1
CREECH, HJ; DRAKE, NL2
BLOOM, MS; BRESLOW, DS1
FUSON, RC; PARHAM, WE; REED, LJ1
ASHBURN, G; LUTZ, RE; ROWLETT, RJ1
DEINET, AJ; LUTZ, RE1
CAMPBELL, KN; SOMMERS, AH1
Burrows, JN; Chibale, K; Wells, TN1
Breytenbach, JC; Denti, P; Kolesnikova, NI; Lombard, MC; N'Da, DD; Norman, J; Tran Van Ba, C; Vial, H; Wein, S; Wiesner, L1
COVELL, G1
HERRERO, MT1
de LUCENA, DT1
DE, NN; RAMA RAO, R; SIRSI, M1
BERTAGNA, P1
HOEKENGA, MT1
COOPER, WC; RUHE, DS1
DRAKE, NL; HAYES, RA1
COPE, AC; NACE, HR1
GRAY, A; HILL, J1
BOLDT, TH; GOODWINE, CH1
Dali Ali, F; Delarue, S; Girault, S; Grellier, P; Maes, L; Sergheraert, C1
Garg, SK; Gupta, A; Tekwani, BL; Tripathi, AK1

Reviews

8 review(s) available for quinoline and Malaria

ArticleYear
Role of basic aminoalkyl chains in the lead optimization of Indoloquinoline alkaloids.
    European journal of medicinal chemistry, 2022, Jan-05, Volume: 227

    Topics: Alkaloids; Antimalarials; Antineoplastic Agents; Cell Proliferation; Indoles; Malaria; Molecular Structure; Neoplasms; Quinolines

2022
Current scenario of ferrocene-containing hybrids for antimalarial activity.
    European journal of medicinal chemistry, 2020, Jan-01, Volume: 185

    Topics: Antimalarials; Artemisinins; Ferrous Compounds; Humans; Malaria; Metallocenes; Molecular Structure; Parasitic Sensitivity Tests; Peroxides; Plasmodium falciparum; Quinolines

2020
Hybrid molecules with potential in vitro antiplasmodial and in vivo antimalarial activity against drug-resistant Plasmodium falciparum.
    Medicinal research reviews, 2020, Volume: 40, Issue:3

    Topics: Animals; Antimalarials; CHO Cells; Cricetulus; Drug Design; Drug Resistance; Humans; In Vitro Techniques; Inhibitory Concentration 50; Malaria; Molecular Structure; Pharmaceutical Preparations; Plasmodium falciparum; Quinolines; Quinolones

2020
Current progress in antimalarial pharmacotherapy and multi-target drug discovery.
    European journal of medicinal chemistry, 2020, Feb-15, Volume: 188

    Topics: Animals; Antimalarials; Artemisinins; Drug Discovery; Drug Resistance; Humans; Malaria; Molecular Structure; Paclitaxel; Quinolines

2020
Quinoline Containing Side-chain Antimalarial Analogs: Recent Advances and Therapeutic Application.
    Current topics in medicinal chemistry, 2020, Volume: 20, Issue:8

    Topics: Animals; Antimalarials; Humans; Malaria; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines

2020
Quinoline--a promising fragment in the search for new antimalarials.
    Mini reviews in medicinal chemistry, 2014, Volume: 14, Issue:4

    Topics: Antimalarials; Drug Design; Humans; Malaria; Plasmodium falciparum; Quinolines

2014
Quinoline-based antimalarial hybrid compounds.
    Bioorganic & medicinal chemistry, 2015, Aug-15, Volume: 23, Issue:16

    Topics: Animals; Antimalarials; Drug Discovery; Humans; Malaria; Plasmodium; Quinolines

2015
The state of the art in anti-malarial drug discovery and development.
    Current topics in medicinal chemistry, 2011, Volume: 11, Issue:10

    Topics: Antimalarials; Clinical Trials as Topic; Drug Combinations; Drug Design; Drug Discovery; Drug Therapy, Combination; Humans; Malaria; Malaria, Falciparum; Plasmodium falciparum; Quinolines

2011

Other Studies

40 other study(ies) available for quinoline and Malaria

ArticleYear
Design and synthesis of novel ferrocene-quinoline conjugates and evaluation of their electrochemical and antiplasmodium properties.
    European journal of medicinal chemistry, 2020, Feb-01, Volume: 187

    Topics: Antimalarials; Dose-Response Relationship, Drug; Drug Design; Electrochemical Techniques; Ferrous Compounds; Humans; Malaria; Metallocenes; Models, Molecular; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2020
The Candidate Antimalarial Drug MMV665909 Causes Oxygen-Dependent mRNA Mistranslation and Synergizes with Quinoline-Derived Antimalarials.
    Antimicrobial agents and chemotherapy, 2017, Volume: 61, Issue:9

    Topics: Amodiaquine; Antimalarials; Artemisinins; Chloroquine; Malaria; Oxygen; Primaquine; Protein Biosynthesis; Quinolines; Reactive Oxygen Species; RNA, Messenger; Saccharomyces cerevisiae

2017
Synthesis and structure-activity relationships for new 6-fluoroquinoline derivatives with antiplasmodial activity.
    Bioorganic & medicinal chemistry, 2019, 05-15, Volume: 27, Issue:10

    Topics: Animals; Antimalarials; Cell Line; Cell Survival; Disease Models, Animal; Drug Resistance; Malaria; Mice; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2019
Cytostatic versus cytocidal profiling of quinoline drug combinations via modified fixed-ratio isobologram analysis.
    Malaria journal, 2013, Sep-18, Volume: 12

    Topics: Animals; Antimalarials; Cell Division; Cell Survival; Drug Combinations; Drug Synergism; Drug Therapy, Combination; Humans; Inhibitory Concentration 50; Malaria; Plasmodium falciparum; Quinolines

2013
Quinine dimers are potent inhibitors of the Plasmodium falciparum chloroquine resistance transporter and are active against quinoline-resistant P. falciparum.
    ACS chemical biology, 2014, Mar-21, Volume: 9, Issue:3

    Topics: Animals; Antimalarials; Dimerization; Dose-Response Relationship, Drug; Drug Resistance; Drug Stability; Malaria; Membrane Transport Proteins; Mice; Molecular Structure; Oocytes; Plasmodium berghei; Plasmodium falciparum; Protozoan Proteins; Quinine; Quinolines; Transfection; Xenopus laevis

2014
The treatment of Plasmodium falciparum malaria with a single dose antimalarial; a preliminary report of the use of hydroxychloroquine, 7-chloro-4(4-(N-ethyl-N-B-hydroxyethylamino)-1-methylbutylamino)-quinoline diphosphate.
    Antibiotics & chemotherapy (Northfield, Ill.), 1952, Volume: 2, Issue:4

    Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Malaria; Malaria, Falciparum; Quinolines

1952
Anti-Plasmodium falciparum activity of quinoline-sulfonamide hybrids.
    Bioorganic & medicinal chemistry, 2015, Sep-01, Volume: 23, Issue:17

    Topics: Animals; Humans; Malaria; Mice; Molecular Structure; Plasmodium falciparum; Quinolines; Sulfonamides

2015
A study of the prophylactic effectiveness of several 8-aminoquinolines in sporozoite-induced vivax malaria, Chesson strain.
    The Journal of clinical investigation, 1948, Volume: 27, Issue:3 Pt1

    Topics: Aminoquinolines; Animals; Humans; Malaria; Malaria, Vivax; Quinolines; Sporozoites

1948
Studies on the chemotherapy of the human malarias; of the human malarias the physiological disposition, antimalarial activity, and toxicity of several derivatives of 4-aminoquinoline.
    The Journal of clinical investigation, 1948, Volume: 27, Issue:3 Pt1

    Topics: Aminoquinolines; Antimalarials; Humans; Malaria; Quinolines

1948
A study of the mechanism of degradation of antimalarial drugs reactions of 8-aminoquinoline derivatives and other secondary aromatic amines with aldehydes.
    Proceedings. American Federation for Clinical Research, 1947, Volume: 3

    Topics: Aldehydes; Amines; Aminoquinolines; Antimalarials; Humans; Malaria; Pharmaceutical Preparations; Quinolines

1947
Fluorine and sulfur quinoline derivatives as anti-malarial agents.
    Iowa State College journal of science, 1946, Volume: 21, Issue:1

    Topics: Antimalarials; Drug Therapy; Fluorides; Fluorine; Humans; Hydroxychloroquine; Malaria; Quinolines; Sulfur

1946
Potential antimalarials; (6-methoxyquinolyl-4)-alpha-piperidylcarbinols.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Antimalarials; Humans; Malaria; Methanol; Quinolines

1946
The synthesis of potential antimalarials; 2-phenyl-alpha-(2-piperidyl)-4-quinolinemethanols.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Antimalarials; Malaria; Methanol; Quinolines

1946
The synthesis of potential antimalarials; 7-chloro-alpha-(2-piperidyl)-4-quinolinemethanol.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Antimalarials; Humans; Malaria; Methanol; Quinolines

1946
alpha-(2-Piperidyl)-2-aryl-4-quinolinemethanols.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Malaria; Methanol; Quinolines

1946
The synthesis of potential antimalarials; 2-alkyl-alpha-(2-piperidyl)-4-quinolinemethanols.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Antimalarials; Malaria; Methanol; Quinolines

1946
Potential antimalarials (chloro-2-phenylquinolyl-4)-alpha-piperidylcarbinols.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Antimalarials; Humans; Malaria; Methanol; Quinolines

1946
alpha-Piperidyl-4-quinolinemethanols substituted in the 2-position.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Humans; Malaria; Methanol; Quinolines

1946
The synthesis of some alpha-(piperidyl)-quinolinemethanols.
    Journal of the American Chemical Society, 1946, Volume: 68, Issue:12

    Topics: Humans; Malaria; Methanol; Quinolines

1946
Synthetic antimalarials; the preparation of certain 4-aminoquinolines.
    Journal of the American Chemical Society, 1946, Volume: 68

    Topics: Aminoquinolines; Antimalarials; Malaria; Quinolines

1946
Synthetic antimalarials; the preparation and properties of 7-chloro-4-(4-diethylamino-l-methylbutylamino)-quinoline (SN-7618).
    Journal of the American Chemical Society, 1946, Volume: 68

    Topics: Antimalarials; Malaria; Quinolines

1946
Synthesis of antimalarials; the synthesis of certain 4-aminoquinoline derivatives.
    Journal of the American Chemical Society, 1946, Volume: 68

    Topics: Aminoquinolines; Antimalarials; Malaria; Quinolines

1946
The synthesis of 7-chloro-4-(l-ethyl-4-piperidylamino)-quinoline (SN-13,425).
    Journal of the American Chemical Society, 1946, Volume: 68

    Topics: Chromans; Malaria; Quinolines; Thiosemicarbazones

1946
Antimalarials; dl-7-chloro-2-(4-diethylamino-l-methylbutylamino)-quinoline.
    Journal of the American Chemical Society, 1946, Volume: 68

    Topics: Antimalarials; Malaria; Quinolines

1946
Antimalarials; 2-chloro-5-(3-diethylaminopropylamino)-quinoline; useful preparations of 2-chloro-5- and 8-nitroquinolines.
    Journal of the American Chemical Society, 1946, Volume: 68

    Topics: Antimalarials; Malaria; Nitroquinolines; Quinolines

1946
Studies in the quinoline series; the preparation of some 8-(omega-alkylaminoalkylamino)-quinolines.
    Journal of the American Chemical Society, 1946, Volume: 68

    Topics: Malaria; Quinolines

1946
Antimalarial and anticancer activities of artemisinin-quinoline hybrid-dimers and pharmacokinetic properties in mice.
    European journal of pharmaceutical sciences : official journal of the European Federation for Pharmaceutical Sciences, 2012, Dec-18, Volume: 47, Issue:5

    Topics: Animals; Antimalarials; Antineoplastic Agents; Artemisinins; Cell Line, Tumor; Humans; Malaria; Male; Mice; Mice, Inbred C57BL; Parasitemia; Plasmodium falciparum; Quinolines

2012
MALARIA STRAINS RESISTANT TO 4-AMINO-QUINOLINE DRUGS.
    British medical journal, 1965, Aug-21, Volume: 2, Issue:5459

    Topics: Antimalarials; Drug Resistance; Drug Resistance, Microbial; Humans; Malaria; Plasmodium falciparum; Quinolines

1965
[Synthetic antimalarials; camoquin].
    La Medicina colonial, 1950, Volume: 16, Issue:3

    Topics: Amodiaquine; Antimalarials; Malaria; Quinolines

1950
[Treatment of malaria with camoquin].
    Revista brasileira de medicina, 1950, Volume: 7, Issue:9

    Topics: Amodiaquine; Humans; Malaria; Quinolines

1950
Antibacterial properties of some quinoline substituted guanides with special reference to the acute toxicity and the bacteriostatic activity of N'-(p-chlorophenyl)-N5-(8'chloro-5'quinolyl) biguanide acetate.
    Current science, 1950, Volume: 19, Issue:10

    Topics: Acetates; Anti-Bacterial Agents; Biguanides; DDT; Malaria; Quinolines

1950
[General sketch on documentation relative to amodiaquine].
    Bulletin of the World Health Organization, 1951, Volume: 4, Issue:2

    Topics: Amodiaquine; Documentation; Humans; Malaria; Quinolines

1951
Camoquin treatment of malaria a preliminary report.
    The American journal of tropical medicine and hygiene, 1950, Volume: 30, Issue:1

    Topics: Amodiaquine; Humans; Malaria; Quinolines

1950
Studies in human malaria; the protective and therapeutic action of SN 6911 against St. Elizabeth strain vivax malaria.
    American journal of hygiene, 1949, Volume: 49, Issue:1

    Topics: Hydroxychloroquine; Malaria; Malaria, Vivax; Quinolines

1949
Synthetic antimalarials; some derivatives of 8-aminoquinoline.
    Journal of the American Chemical Society, 1949, Volume: 71, Issue:2

    Topics: Aminoquinolines; Antimalarials; Malaria; Quinolines

1949
Synthesis of 6-methoxy-8-aminoquinoline derivatives; ethyleneimine rearrangements in attachment of monoalkylaminoalkyl side chains.
    Journal of the American Chemical Society, 1949, Volume: 71, Issue:2

    Topics: Amino Acids; Aminoquinolines; Aziridines; Malaria; Quinolines

1949
Antimalarial studies in the quinoline series.
    Annals of tropical medicine and parasitology, 1949, Volume: 43, Issue:1

    Topics: Antimalarials; Humans; Malaria; Quinolines

1949
A second year's field trial with chloroquine suppression of high endemic malaria in a Panamanian village.
    Journal. National Malaria Society (U.S.), 1949, Volume: 8, Issue:3

    Topics: Chloroquine; Humans; Malaria; Quinolines

1949
"One-pot" synthesis and antimalarial activity of formamidine derivatives of 4-anilinoquinoline.
    Chemical & pharmaceutical bulletin, 2001, Volume: 49, Issue:8

    Topics: Amidines; Amodiaquine; Animals; Antimalarials; Cell Line; Humans; Inhibitory Concentration 50; Macrophages; Malaria; Mice; Plasmodium berghei; Quinolines

2001
In vitro beta-hematin formation assays with plasma of mice infected with Plasmodium yoelii and other parasite preparations: comparative inhibition with quinoline and endoperoxide antimalarials.
    Life sciences, 2001, Oct-26, Volume: 69, Issue:23

    Topics: Animals; Antimalarials; Artemisinins; Biological Assay; Dose-Response Relationship, Drug; Erythrocytes; Hemeproteins; Hemin; In Vitro Techniques; Malaria; Male; Mice; Parasitemia; Peroxides; Plasmodium yoelii; Quinolines; Sesquiterpenes

2001