Page last updated: 2024-08-17

quinoline and Malaria, Falciparum

quinoline has been researched along with Malaria, Falciparum in 12 studies

Research

Studies (12)

TimeframeStudies, this research(%)All Research%
pre-19901 (8.33)18.7374
1990's0 (0.00)18.2507
2000's2 (16.67)29.6817
2010's7 (58.33)24.3611
2020's2 (16.67)2.80

Authors

AuthorsStudies
Fidock, DA; Mok, S; Wicht, KJ1
Hoda, N; Kalamuddin, M; Malhotra, P; Maqbool, M; Mohmmed, A; Singh, A1
de Dios, A; Gorka, AP; Roepe, PD1
D'hooghe, M; Vandekerckhove, S1
JOSEPH, AA; LOUGHLIN, EH; RAPPAPORT, I; RICE, JB; WELLS, HS1
Edaye, S; Georges, E; Leimanis, ML; Reiling, SJ; Rohrbach, P; Wunderlich, J1
Au, A; Egan, TJ; Guzgay, H; Hendricks, DT; Land, KM; Shokar, A; Smith, GS; Smith, PJ; Stringer, T; Taylor, D1
Agomo, CO; Hallet, R; Oguike, M; Oyibo, WA; Sutherland, C1
Chookajorn, T; Fidock, DA; Gabryszewski, SJ; Modchang, C; Musset, L1
Roepe, PD1
Burrows, JN; Chibale, K; Wells, TN1
Ginsburg, H; Macreadie, I; Sirawaraporn, W; Tilley, L1

Reviews

5 review(s) available for quinoline and Malaria, Falciparum

ArticleYear
Molecular Mechanisms of Drug Resistance in
    Annual review of microbiology, 2020, 09-08, Volume: 74

    Topics: Antimalarials; Artemisinins; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Membrane Transport Proteins; Mutation; Plasmodium falciparum; Protozoan Proteins; Quinolines

2020
Quinoline drug-heme interactions and implications for antimalarial cytostatic versus cytocidal activities.
    Journal of medicinal chemistry, 2013, Jul-11, Volume: 56, Issue:13

    Topics: Antimalarials; Crystallization; Drug Resistance; Heme; Hemeproteins; Humans; Malaria, Falciparum; Molecular Structure; Plasmodium falciparum; Quinolines

2013
Molecular and physiologic basis of quinoline drug resistance in Plasmodium falciparum malaria.
    Future microbiology, 2009, Volume: 4, Issue:4

    Topics: Animals; Antimalarials; Drug Resistance; Humans; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines

2009
The state of the art in anti-malarial drug discovery and development.
    Current topics in medicinal chemistry, 2011, Volume: 11, Issue:10

    Topics: Antimalarials; Clinical Trials as Topic; Drug Combinations; Drug Design; Drug Discovery; Drug Therapy, Combination; Humans; Malaria; Malaria, Falciparum; Plasmodium falciparum; Quinolines

2011
Antimalarial drug development and new targets.
    Parasitology today (Personal ed.), 2000, Volume: 16, Issue:10

    Topics: Animals; Antimalarials; Drug Design; Drug Resistance; Folic Acid Antagonists; Humans; Malaria, Falciparum; Plasmodium falciparum; Quinolines

2000

Other Studies

7 other study(ies) available for quinoline and Malaria, Falciparum

ArticleYear
Quinoline carboxamide core moiety-based compounds inhibit P. falciparumfalcipain-2: Design, synthesis and antimalarial efficacy studies.
    Bioorganic chemistry, 2021, Volume: 108

    Topics: Antimalarials; Cysteine Endopeptidases; Dose-Response Relationship, Drug; Drug Design; Malaria, Falciparum; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Quinolines; Structure-Activity Relationship

2021
Exploration of aziridine- and β-lactam-based hybrids as both bioactive substances and synthetic intermediates in medicinal chemistry.
    Bioorganic & medicinal chemistry, 2013, Jul-01, Volume: 21, Issue:13

    Topics: Animals; Antimalarials; Antiviral Agents; Aziridines; beta-Lactams; Chemistry, Pharmaceutical; Drug Discovery; Humans; Malaria, Falciparum; Plasmodium falciparum; Purines; Quinolines

2013
The treatment of Plasmodium falciparum malaria with a single dose antimalarial; a preliminary report of the use of hydroxychloroquine, 7-chloro-4(4-(N-ethyl-N-B-hydroxyethylamino)-1-methylbutylamino)-quinoline diphosphate.
    Antibiotics & chemotherapy (Northfield, Ill.), 1952, Volume: 2, Issue:4

    Topics: Antimalarials; Chloroquine; Humans; Hydroxychloroquine; Malaria; Malaria, Falciparum; Quinolines

1952
A 2-amino quinoline, 5-(3-(2-(7-chloroquinolin-2-yl)ethenyl)phenyl)-8-dimethylcarbamyl-4,6-dithiaoctanoic acid, interacts with PfMDR1 and inhibits its drug transport in Plasmodium falciparum.
    Molecular and biochemical parasitology, 2014, Volume: 195, Issue:1

    Topics: Antimalarials; Biological Transport; Chloroquine; Drug Resistance; Humans; Malaria, Falciparum; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Plasmodium falciparum; Protozoan Proteins; Quinolines

2014
Polyamine quinoline rhodium complexes: synthesis and pharmacological evaluation as antiparasitic agents against Plasmodium falciparum and Trichomonas vaginalis.
    Dalton transactions (Cambridge, England : 2003), 2015, Sep-07, Volume: 44, Issue:33

    Topics: Antiparasitic Agents; Coordination Complexes; Female; Humans; Malaria, Falciparum; Plasmodium falciparum; Polyamines; Quinolines; Rhodium; Structure-Activity Relationship; Trichomonas vaginalis; Trichomonas Vaginitis

2015
Assessment of Markers of Antimalarial Drug Resistance in Plasmodium falciparum Isolates from Pregnant Women in Lagos, Nigeria.
    PloS one, 2016, Volume: 11, Issue:1

    Topics: Adult; Antimalarials; Drug Resistance; Female; Humans; Malaria, Falciparum; Membrane Transport Proteins; Nigeria; Plasmodium falciparum; Pregnancy; Pregnancy Complications; Pregnant Women; Protozoan Proteins; Quinolines; Young Adult

2016
Combinatorial Genetic Modeling of pfcrt-Mediated Drug Resistance Evolution in Plasmodium falciparum.
    Molecular biology and evolution, 2016, Volume: 33, Issue:6

    Topics: Alleles; Antimalarials; Chloroquine; Drug Resistance; Haplotypes; Humans; Malaria, Falciparum; Membrane Transport Proteins; Models, Genetic; Mutation; Plasmodium falciparum; Polymorphism, Single Nucleotide; Protozoan Proteins; Quinolines

2016