Page last updated: 2024-08-21

quinazolines and Uterine Neoplasms

quinazolines has been researched along with Uterine Neoplasms in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's5 (38.46)29.6817
2010's8 (61.54)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Carson, DD; Engel, BJ1
Bedard, PL; Castonguay, V; Chen, EX; Chen, H; Chen, Z; Clarke, B; Cohen, B; Hirte, HW; Hotte, SJ; Ivy, SP; Kamel-Reid, S; Liu, G; McGarrity, A; Oza, AM; Razak, AR; Reedijk, M; Sahebjam, S; Siu, LL; Wang, L; Zhang, T; Zhang, WJ1
Muggia, F; Teplinsky, E1
Azodi, M; Bellone, S; Bonazzoli, E; Bortolomai, I; Cocco, E; English, DP; Lopez, S; Nicoletti, R; Ratner, E; Roque, DM; Rutherford, TJ; Santin, AD; Schwab, CL; Schwartz, PE; Silasi, DA1
Borger, DR; Byron, VF; DiGloria, CM; Foster, R; Groeneweg, JW; Growdon, WB; Hernandez, SF; Kim, M; Lopez, H; Rueda, BR; Scialabba, V; Tambouret, R; Zhang, L1
Borger, D; Chisholm, S; Foster, R; Growdon, WB; Hernandez, SF; Rueda, BR1
Bai, Y; Black, J; Carvajal-Hausdorf, DE; Rimm, DL; Santin, AD; Schalper, KA1
Bolshakov, S; Dicker, A; Korchin, B; Lahat, G; Lazar, A; Lev, D; Merritt, W; Nguyen, T; Pollock, RE; Ren, W; Sood, A; Wei, C1
Golabi, N; Jean-Claude, BJ; Larroque-Lombard, AL; Todorova, M; Williams, C1
Al-Hendy, A; Copland, JA; Young, SL1
Ben-Bassat, H; Hartzstark, Z; Klein, BY; Laufer, N; Levitzki, R; Rojansky, N; Shlomai, Z; Shushan, A1
Ben-Bassat, H; Klein, BY; Laufer, N; Mishani, E; Rojansky, N; Shushan, A1
Nowak, RA1

Reviews

2 review(s) available for quinazolines and Uterine Neoplasms

ArticleYear
Targeting HER2 in ovarian and uterine cancers: challenges and future directions.
    Gynecologic oncology, 2014, Volume: 135, Issue:2

    Topics: Adenocarcinoma, Mucinous; Ado-Trastuzumab Emtansine; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Carcinoma; Endometrial Neoplasms; Female; Genes, erbB-2; Humans; Lapatinib; Maytansine; Molecular Targeted Therapy; Ovarian Neoplasms; Quinazolines; Trastuzumab; Uterine Neoplasms

2014
Potential nonhormonal therapeutics for medical treatment of leiomyomas.
    Seminars in reproductive medicine, 2004, Volume: 22, Issue:2

    Topics: Bexarotene; Female; Heparin; Humans; Interferon-alpha; Leiomyoma; ortho-Aminobenzoates; Piperidines; Pyridones; Quinazolines; Quinazolinones; Reproduction; Tetrahydronaphthalenes; Thiazolidinediones; Tocopherols; Uterine Neoplasms

2004

Trials

1 trial(s) available for quinazolines and Uterine Neoplasms

ArticleYear
A phase I study of the combination of ro4929097 and cediranib in patients with advanced solid tumours (PJC-004/NCI 8503).
    British journal of cancer, 2013, Aug-20, Volume: 109, Issue:4

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Benzazepines; Breast Neoplasms; Carcinoma, Neuroendocrine; Carcinoma, Renal Cell; Colorectal Neoplasms; Female; Humans; Kidney Neoplasms; Leiomyosarcoma; Male; Middle Aged; Neoplasms; Quinazolines; Sarcoma, Endometrial Stromal; Thyroid Neoplasms; Treatment Outcome; Uterine Neoplasms; Young Adult

2013

Other Studies

10 other study(ies) available for quinazolines and Uterine Neoplasms

ArticleYear
Activated EGFR stimulates MUC1 expression in human uterine and pancreatic cancer cell lines.
    Journal of cellular biochemistry, 2013, Volume: 114, Issue:10

    Topics: Blotting, Western; Cell Line, Tumor; Epidermal Growth Factor; ErbB Receptors; Female; Gene Expression; Humans; Mucin-1; Pancreatic Neoplasms; Quinazolines; Rosiglitazone; Thiazolidinediones; Tyrphostins; Uterine Neoplasms

2013
Afatinib demonstrates remarkable activity against HER2-amplified uterine serous endometrial cancer in vitro and in vivo.
    British journal of cancer, 2014, Oct-28, Volume: 111, Issue:9

    Topics: Adult; Afatinib; Aged; Aged, 80 and over; Animals; Apoptosis; Cell Cycle; Cell Proliferation; Cystadenocarcinoma, Serous; Endometrial Neoplasms; Female; Humans; Immunoenzyme Techniques; In Situ Hybridization, Fluorescence; In Vitro Techniques; Mice; Mice, SCID; Middle Aged; Phosphorylation; Quinazolines; Receptor, ErbB-2; Signal Transduction; Tumor Cells, Cultured; Uterine Neoplasms; Xenograft Model Antitumor Assays

2014
Dual HER2 targeting impedes growth of HER2 gene-amplified uterine serous carcinoma xenografts.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2014, Dec-15, Volume: 20, Issue:24

    Topics: Animals; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Apoptosis; Cell Line, Tumor; Cell Proliferation; Cystadenocarcinoma, Serous; Disease Models, Animal; Female; Gene Amplification; Gene Expression; Humans; Lapatinib; Mice; Protein Kinase Inhibitors; Quinazolines; Receptor, ErbB-2; Signal Transduction; Trastuzumab; Tumor Burden; Uterine Neoplasms; Xenograft Model Antitumor Assays

2014
Ridaforolimus improves the anti-tumor activity of dual HER2 blockade in uterine serous carcinoma in vivo models with HER2 gene amplification and PIK3CA mutation.
    Gynecologic oncology, 2016, Volume: 141, Issue:3

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; Apoptosis; Benzoxazoles; Cell Cycle; Cell Proliferation; Class I Phosphatidylinositol 3-Kinases; Cystadenoma, Serous; Drug Synergism; Female; Gene Amplification; Humans; Lapatinib; Mice; Mice, Inbred NOD; Mice, SCID; Phosphatidylinositol 3-Kinases; Pyrimidines; Quinazolines; Receptor, ErbB-2; Sirolimus; TOR Serine-Threonine Kinases; Trastuzumab; Uterine Neoplasms; Xenograft Model Antitumor Assays

2016
Objective, domain-specific HER2 measurement in uterine and ovarian serous carcinomas and its clinical significance.
    Gynecologic oncology, 2017, Volume: 145, Issue:1

    Topics: Ado-Trastuzumab Emtansine; Afatinib; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Cohort Studies; Extracellular Space; Female; Fluorescent Antibody Technique; Humans; Intracellular Space; Lapatinib; Maytansine; Middle Aged; Neoplasms, Cystic, Mucinous, and Serous; Ovarian Neoplasms; Protein Domains; Quinazolines; Receptor, ErbB-2; Retrospective Studies; Tissue Array Analysis; Trastuzumab; Uterine Neoplasms

2017
Combined vascular endothelial growth factor receptor/epidermal growth factor receptor blockade with chemotherapy for treatment of local, uterine, and metastatic soft tissue sarcoma.
    Clinical cancer research : an official journal of the American Association for Cancer Research, 2008, Sep-01, Volume: 14, Issue:17

    Topics: Animals; Antineoplastic Combined Chemotherapy Protocols; ErbB Receptors; Female; Humans; Lung Neoplasms; Mice; Mice, Nude; Muscle Neoplasms; Piperidines; Quinazolines; Receptors, Vascular Endothelial Growth Factor; Sarcoma; Tumor Cells, Cultured; Uterine Neoplasms; Xenograft Model Antitumor Assays

2008
Synthesis and uptake of fluorescence-labeled Combi-molecules by P-glycoprotein-proficient and -deficient uterine sarcoma cells MES-SA and MES-SA/DX5.
    Journal of medicinal chemistry, 2010, Mar-11, Volume: 53, Issue:5

    Topics: Antineoplastic Agents; ATP Binding Cassette Transporter, Subfamily B, Member 1; Cell Line, Tumor; Cell Proliferation; Comet Assay; Dansyl Compounds; DNA; DNA Damage; ErbB Receptors; Female; Flow Cytometry; Half-Life; Humans; Magnetic Resonance Spectroscopy; Microscopy, Fluorescence; Quinazolines; Sarcoma; Spectrometry, Mass, Electrospray Ionization; Structure-Activity Relationship; Uterine Neoplasms

2010
The AG1478 tyrosine kinase inhibitor is an effective suppressor of leiomyoma cell growth.
    Human reproduction (Oxford, England), 2004, Volume: 19, Issue:9

    Topics: Adult; Apoptosis; Cell Cycle; Cell Division; Cells, Cultured; Enzyme Inhibitors; ErbB Receptors; Estradiol; Female; Humans; Leiomyoma; Myometrium; Phosphorylation; Progesterone; Protein-Tyrosine Kinases; Quinazolines; Tyrphostins; Uterine Neoplasms

2004
Inhibition of leiomyoma cell proliferation in vitro by genistein and the protein tyrosine kinase inhibitor TKS050.
    Fertility and sterility, 2007, Volume: 87, Issue:1

    Topics: Antineoplastic Agents; Cell Proliferation; Dose-Response Relationship, Drug; Female; Genistein; Humans; Leiomyoma; Protein-Tyrosine Kinases; Quinazolines; Tumor Cells, Cultured; Uterine Neoplasms

2007
Novel therapeutic strategies for leiomyomas: targeting growth factors and their receptors.
    Environmental health perspectives, 2000, Volume: 108 Suppl 5

    Topics: Antineoplastic Agents; Blotting, Western; Chromatography, Liquid; Female; Growth Inhibitors; Growth Substances; Humans; Hysterectomy; Hysteroscopy; Immunohistochemistry; Interferon-alpha; Leiomyoma; Phenoxyacetates; Piperidines; Polymers; Protein Synthesis Inhibitors; Pyridones; Quinazolines; Quinazolinones; Receptors, Growth Factor; Uterine Neoplasms

2000