quinazolines has been researched along with Muscle Relaxation in 38 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 7 (18.42) | 18.7374 |
1990's | 15 (39.47) | 18.2507 |
2000's | 13 (34.21) | 29.6817 |
2010's | 2 (5.26) | 24.3611 |
2020's | 1 (2.63) | 2.80 |
Authors | Studies |
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Ahn, JH; Bae, EJ; Cho, S; Jo, H; Kim, SJ; Kwon, JW; Lee, N; Park, CS | 1 |
Agrawal, KC; Chandra, S; Gur, S; Hellstrom, WJ; Kadowitz, PJ; Koka, PS; Sikka, SC | 1 |
Alexandre, L; Behr-Roussel, D; Denoux, Y; Giuliano, F; Gorny, D; Lebret, T; Oger, S | 1 |
Abdulkadir, NA; Cetinkaya, M; Demirturk, K; Gur, S; Hellstrom, WJ; Karabakan, M; Ozgur-Akdemir, A; Volkan-Oztekin, C | 1 |
Barras, M; Palea, S | 1 |
Baur, F; Fozard, JR; Wolber, C | 1 |
Azegami, Y; Kaneda, T; Nakajyo, S; Shimizu, K; Urakawa, N; Yamamoto, H | 1 |
Akaishi, T; Hara, H; Ishida, N; Kashiwagi, K; Matsugi, T; Takagi, Y | 1 |
Chen, CF; Chen, CM; Chen, KT; Ko, HC; Su, JP; Wang, GJ | 1 |
Alexandre, L; Behr-Roussel, D; Charles Tremeaux, J; Combes, M; Giuliano, F; Gorny, D; Oger, S | 1 |
Ishihara, Y; Kitamura, S; Kosaka, K; Yotsumoto, H | 1 |
Ruskoaho, H | 1 |
Miyazaki, M; Nakajima, M; Okamura, T; Toda, N | 1 |
Bernabé, J; Burvenich, C; Peeters, G; Vandeputte-Van Messom, G | 1 |
Forssmann, WG; Jonas, U; Meyer, M; Schulz-Knappe, P; Stief, CG; Taher, A; Truss, M | 1 |
Chen, CF; Chiou, WF; Chou, CJ; Liao, JF; Sham, AY | 1 |
Fujimoto, M; Saeki, T; Saito, I; Takase, Y | 1 |
Isaka, N; Ito, M; Itoh, H; Konishi, T; Miyahara, M; Nakano, T; Shiraishi, T | 1 |
Lee, YM; Peng, IH; Sheu, JR; Yen, MH | 1 |
Chen, CF; Chiou, WF; Liao, JF; Shum, AY | 1 |
Aktan, Y; Erol, K; Ertan, M; Saraç, S; Yarim, M | 1 |
Boydağ, S; Erol, K; Ertan, M; Saraç, S; Yarim, M | 1 |
Adachi, H; Ishihara, H; Kabasawa, Y; Kodama, K; Matsukura, M; Miyazaki, K; Takase, Y; Watanabe, N | 1 |
Chiu, JH; Jiang, JK; Lin, JK; Yu, IT | 1 |
Adachi, H; Ishibashi, K; Ishihara, H; Kabasawa, Y; Kakiki, M; Kodama, K; Matsukura, M; Miyazaki, K; Nishino, M; Ozaki, H; Takase, Y; Watanabe, N | 1 |
Andersson, K; Fujiwara, M; Persson, K | 1 |
Bumann, K; Kaumann, AJ; Verheggen, R | 1 |
Ahlawat, S; Bhatti, RS; Gupta, R; Jindal, DP | 1 |
Chen, CF; Chiou, WF | 1 |
Bolzano, K | 1 |
Andersson, KE; Mikkelsen, E; Pedersen, OL | 1 |
Chen, CF; Chiou, WF; Chou, CJ; Shum, AY | 1 |
Buyuktimkin, N; Buyuktimkin, S; Ekinci, AC; Otuk, G | 1 |
Hayashi, Y; Ikeda, K; Ohnishi, H; Watanabe, K | 1 |
Ebisawa, H; Eguchi, Y; Ishikawa, M; Sasaki, F; Sugimoto, A | 1 |
Bertaux, L; Crouzette, J; Dussaucy, E; Fournier, PE; Girre, C; Palombo, S | 1 |
Brown, GL; Douglas, FL; Kotake, AN; Mustafa, SJ; Sabouni, MH | 1 |
Hamrick, ME; Millen, J; Riley, TN; Waters, IW | 1 |
1 trial(s) available for quinazolines and Muscle Relaxation
Article | Year |
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Comparative effects on psychomotor performance of the muscle relaxant afloqualone, alone and with ethanol.
Topics: Administration, Oral; Adolescent; Adult; Diazepam; Double-Blind Method; Drug Interactions; Ethanol; Humans; Male; Muscle Relaxants, Central; Muscle Relaxation; Psychomotor Performance; Quinazolines | 1991 |
37 other study(ies) available for quinazolines and Muscle Relaxation
Article | Year |
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Discovery and characterization of a potent activator of the BK
Topics: Animals; Membrane Potentials; Muscle Relaxation; Myocytes, Smooth Muscle; Quinazolines; Rats; Urinary Bladder, Overactive | 2022 |
Alfuzosin attenuates erectile dysfunction in rats with partial bladder outlet obstruction.
Topics: Adrenergic alpha-Antagonists; Animals; Blotting, Western; Erectile Dysfunction; Immunohistochemistry; Male; Muscle Contraction; Muscle Relaxation; Nitric Oxide Synthase; Penile Erection; Penis; Quinazolines; Rats; Rats, Sprague-Dawley; Urinary Bladder Neck Obstruction | 2008 |
Combination of alfuzosin and tadalafil exerts an additive relaxant effect on human detrusor and prostatic tissues in vitro.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Agonists; Aged; Carbachol; Carbolines; Cholinergic Agonists; Dose-Response Relationship, Drug; Drug Therapy, Combination; Electric Stimulation; Humans; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth; Norepinephrine; Phosphodiesterase 5 Inhibitors; Prostate; Quinazolines; Tadalafil; Urinary Bladder | 2010 |
Imatinib mesylate (Gleevec) as protein-tyrosine kinase inhibitor elicits smooth muscle relaxation in isolated human prostatic tissue.
Topics: Adrenergic alpha-Antagonists; Aged; Benzamides; Humans; Hyperplasia; Imatinib Mesylate; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Piperazines; Prostate; Prostatic Diseases; Protein Kinase Inhibitors; Protein-Tyrosine Kinases; Pyrimidines; Quinazolines | 2011 |
Comparison of the relaxant effects of alfuzosin, phentolamine and sildenafil on rabbit isolated corpus cavernosum.
Topics: Adrenergic alpha-Antagonists; Animals; Erectile Dysfunction; Male; Muscle Relaxation; Penile Erection; Phentolamine; Phosphodiesterase Inhibitors; Piperazines; Prostatic Hyperplasia; Purines; Quinazolines; Rabbits; Sildenafil Citrate; Sulfones | 2003 |
Antagonist pharmacology of adenosine A2B receptors from rat, guinea pig and dog.
Topics: Adenosine A2 Receptor Antagonists; Adenosine-5'-(N-ethylcarboxamide); Animals; Dogs; Dose-Response Relationship, Drug; Female; Guinea Pigs; In Vitro Techniques; Male; Muscle Relaxation; Quinazolines; Rats; Receptor, Adenosine A2B; Species Specificity; Triazoles | 2003 |
Lack of cyclic nucleotide regulation of MBCQ-induced relaxation of rat ileal smooth muscle.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Animals; Carbachol; Cholinergic Agonists; Cyclic AMP; Cyclic GMP; Cyclic Nucleotide Phosphodiesterases, Type 5; Dipyridamole; Ileum; Male; Muscle Relaxation; Muscle, Smooth; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Potassium; Purinones; Quinazolines; Rats; Rats, Wistar | 2003 |
Effects of bunazosin hydrochloride on ciliary muscle constriction and matrix metalloproteinase activities.
Topics: Adrenergic alpha-Antagonists; Animals; Antihypertensive Agents; Aqueous Humor; Cattle; Cells, Cultured; Ciliary Body; Drug Combinations; Intraocular Pressure; Isometric Contraction; Latanoprost; Macaca fascicularis; Male; Matrix Metalloproteinases; Muscle Relaxation; Muscle, Smooth; Phenylephrine; Prostaglandins F, Synthetic; Quinazolines; Trabecular Meshwork | 2004 |
Chemical and biological comparisons on Evodia with two related species of different locations and conditions.
Topics: Alkaloids; Animals; Aorta; China; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Evodia; Female; Fruit; In Vitro Techniques; Indole Alkaloids; Male; Methanol; Molecular Structure; Muscle Relaxation; Muscle, Smooth; Muscle, Smooth, Vascular; Myometrium; Plant Extracts; Quinazolines; Rats; Rats, Sprague-Dawley; Species Specificity; Synephrine; Taiwan | 2006 |
Combination of alfuzosin and tadalafil exerts in vitro an additive relaxant effect on human corpus cavernosum.
Topics: Adrenergic alpha-Antagonists; Carbolines; Dose-Response Relationship, Drug; Drug Therapy, Combination; Erectile Dysfunction; Humans; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Penile Erection; Phosphodiesterase Inhibitors; Quinazolines; Tadalafil | 2008 |
The potentiating effect of an alpha-adrenergic blocking agent (E-643) on the action of bronchodilators.
Topics: Adrenergic alpha-Antagonists; Animals; Bronchodilator Agents; Cyclic AMP; Cyclic GMP; Drug Synergism; Epinephrine; Guinea Pigs; Isoproterenol; Male; Muscle Relaxation; Muscle, Smooth; Prostaglandins E; Quinazolines; Trachea | 1980 |
Prevention of cardiac hypertrophy by long-term treatment with isosorbide dinitrate and prazosin but not by minoxidil in spontaneously hypertensive rats.
Topics: Animals; Blood Pressure; Cardiomegaly; Female; Hypertension; Isosorbide Dinitrate; Male; Minoxidil; Muscle Relaxation; Nitroglycerin; Prazosin; Pyrimidines; Quinazolines; Rats; Rats, Inbred Strains | 1984 |
Modification by yohimbine and prazosin of the mechanical response of isolated dog mesenteric, renal and coronary arteries to transmural stimulation and norepinephrine.
Topics: Animals; Coronary Vessels; Dogs; Electric Stimulation; Female; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Norepinephrine; Prazosin; Quinazolines; Renal Artery; Yohimbine | 1984 |
Effect of prazosin on the function of the teat sphincter in lactating cows.
Topics: Animals; Cattle; Female; Injections, Intra-Arterial; Injections, Intravenous; Lactation; Mammary Glands, Animal; Milk Ejection; Muscle Relaxation; Muscle, Smooth; Oxytocin; Plethysmography; Prazosin; Pregnancy; Quinazolines | 1984 |
Characterization of cyclic nucleotide phosphodiesterase isoenzymes in the human ureter and their functional role in vitro.
Topics: 3',5'-Cyclic-AMP Phosphodiesterases; Calmodulin; Chromatography, DEAE-Cellulose; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Humans; Hydrolysis; In Vitro Techniques; Muscle Relaxation; Muscle Tonus; Muscle, Smooth; Papaverine; Phosphodiesterase Inhibitors; Purinones; Pyrrolidinones; Quinazolines; Rolipram; Ureter | 1994 |
The mechanism of the vasodilator effect of rutaecarpine, an alkaloid isolated from Evodia rutaecarpa.
Topics: Acetylcholine; Alkaloids; Animals; Arginine; Atropine; Calcium; Dose-Response Relationship, Drug; Endothelium, Vascular; In Vitro Techniques; Indole Alkaloids; Male; Mesenteric Arteries; Methylene Blue; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroarginine; Phenylephrine; Quinazolines; Rats; Rats, Sprague-Dawley; Triprolidine; Vasodilation; Yohimbine | 1994 |
Cyclic GMP phosphodiesterase inhibitors. 1. The discovery of a novel potent inhibitor, 4-((3,4-(methylenedioxy)benzyl)amino)-6,7,8-trimethoxyquinazoline.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Animals; Aorta; Chromones; Coronary Vessels; Cyclic GMP; Dinoprost; Isoenzymes; Molecular Structure; Muscle Relaxation; Purinones; Quinazolines; Structure-Activity Relationship; Swine | 1993 |
Isoenzymes of cyclic nucleotide phosphodiesterase in the human aorta: characterization and the effects of E4021.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Aorta; Calcium-Calmodulin-Dependent Protein Kinases; Cytosol; Dinoprost; Humans; In Vitro Techniques; Isoenzymes; Kidney; Kinetics; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Piperidines; Quinazolines; Subcellular Fractions; Vasodilator Agents | 1995 |
Effects of DC-015, a novel potent and selective alpha 1-adrenoceptor antagonist on plasma lipid and vascular reactivity in hyperlipidaemic rats.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-Antagonists; Animals; Aorta; Blood Pressure; Dose-Response Relationship, Drug; Hyperlipidemias; In Vitro Techniques; Lipids; Lipoproteins; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Prazosin; Quinazolines; Rats; Rats, Inbred SHR; Rats, Inbred WKY | 1996 |
Studies of the cellular mechanisms underlying the vasorelaxant effects of rutaecarpine, a bioactive component extracted from an herbal drug.
Topics: Acetylcholine; Alkaloids; Animals; Aorta, Thoracic; Calcimycin; Calcium; Calcium Channel Blockers; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Estrenes; Gallic Acid; Guanylate Cyclase; Histamine; Indole Alkaloids; Ionophores; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Nitric Oxide; Pertussis Toxin; Phenylephrine; Pyrrolidinones; Quinazolines; Rats; Rats, Sprague-Dawley; Type C Phospholipases; Vasodilator Agents; Virulence Factors, Bordetella | 1997 |
4-aryl-5-oxo-1,2,3,4,5,6,7,8-octahydroquinazoline-2-thione derivatives: synthesis, enantiomeric separation and in vitro screening as calcium antagonists.
Topics: Animals; Calcium Channel Blockers; Drug Evaluation, Preclinical; Female; Ileum; In Vitro Techniques; Male; Muscle Relaxation; Quinazolines; Rats | 1997 |
Synthesis, chemical and pharmacological properties of some 4-aryl-1,2,3,4,5,6,7,8-octahydroquinazoline-2,5-diones.
Topics: Animals; Calcium Channel Blockers; Female; Guinea Pigs; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Muscle Relaxation; Quinazolines; Rats; Spectrophotometry, Infrared; Spectrophotometry, Ultraviolet | 1998 |
4-Benzylamino-1-chloro-6-substituted phthalazines: synthesis and inhibitory activity toward phosphodiesterase 5.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Animals; Blood Platelets; Coronary Vessels; Cyclic Nucleotide Phosphodiesterases, Type 5; Dinoprost; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Phthalazines; Piperidines; Quinazolines; Swine; Vasodilator Agents | 1998 |
In vitro relaxation of rabbit and human internal anal sphincter by rutaecarpine, an alkaloid isolated from Evodia rutaecarpa.
Topics: Acetylcholine; Alkaloids; Anal Canal; Animals; Calcium; Dose-Response Relationship, Drug; Drugs, Chinese Herbal; Edetic Acid; Enzyme Inhibitors; Ethylmaleimide; Humans; In Vitro Techniques; Indole Alkaloids; Male; Methylene Blue; Muscle Relaxation; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nifedipine; Quinazolines; Rabbits; Species Specificity; Vasodilator Agents | 2000 |
4-(3-Chloro-4-methoxybenzyl)aminophthalazines: synthesis and inhibitory activity toward phosphodiesterase 5.
Topics: 3',5'-Cyclic-GMP Phosphodiesterases; Animals; Antihypertensive Agents; Biological Availability; Blood Pressure; Coronary Vessels; Cyclic Nucleotide Phosphodiesterases, Type 5; Dinoprost; Hypertension, Pulmonary; In Vitro Techniques; Male; Muscle Relaxation; Muscle, Smooth, Vascular; Phosphodiesterase Inhibitors; Phosphoric Diester Hydrolases; Phthalazines; Piperidines; Quinazolines; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Swine; Vasodilator Agents | 2000 |
Nitric oxide-induced cGMP accumulation in the mouse bladder is not related to smooth muscle relaxation.
Topics: Animals; Arginine; Carbachol; Cyclic AMP; Cyclic GMP; Dose-Response Relationship, Drug; Electric Stimulation; Enzyme Inhibitors; Female; In Vitro Techniques; Mice; Mice, Inbred BALB C; Molsidomine; Muscle Relaxation; Muscle, Smooth; Nitric Oxide Donors; Nitric Oxide Synthase; Nitroarginine; Nitroprusside; Phosphodiesterase Inhibitors; Piperazines; Piperidines; Purines; Quinazolines; Sildenafil Citrate; Sulfones; Urethra; Urinary Bladder | 2000 |
BIBN4096BS is a potent competitive antagonist of the relaxant effects of alpha-CGRP on human temporal artery: comparison with CGRP(8-37).
Topics: Adolescent; Adult; Aged; Calcitonin Gene-Related Peptide; Female; Humans; In Vitro Techniques; Male; Middle Aged; Muscle Relaxation; Muscle, Smooth, Vascular; Nitroprusside; Papaverine; Peptide Fragments; Piperazines; Quinazolines; Receptors, Calcitonin Gene-Related Peptide; Temporal Arteries; Vasodilator Agents | 2002 |
Synthesis and bronchodilatory activity of some nitrogen bridgehead compounds.
Topics: Acetylcholine; Animals; Bridged-Ring Compounds; Bronchodilator Agents; Guinea Pigs; In Vitro Techniques; Muscle Relaxation; Muscle, Smooth; Nitrogen; Quinazolines; Trachea | 2002 |
Pharmacological profile of evodiamine in isolated rabbit corpus cavernosum.
Topics: Aging; Animals; Colforsin; Electric Stimulation; In Vitro Techniques; Isometric Contraction; Male; Muscle Contraction; Muscle Relaxation; Nitric Oxide Donors; Nitroprusside; Nucleotides, Cyclic; Penis; Plant Extracts; Potassium; Potassium Channel Blockers; Quinazolines; Rabbits | 2002 |
[A clinical study with prazosin].
Topics: Adrenergic alpha-Antagonists; Adult; Aged; Benzothiadiazines; Depression; Diuretics; Drug Therapy, Combination; Female; Humans; Hypertension; Male; Middle Aged; Muscle Contraction; Muscle Relaxation; Prazosin; Quinazolines; Sexual Behavior; Sodium Chloride Symporter Inhibitors; Urination Disorders | 1978 |
Comparison of the in vitro effects of prazosin, nifedipine, and dihydralazine in isolated human mesenteric and crural vessels.
Topics: Adolescent; Adult; Aged; Calcium; Dihydralazine; Humans; Hydralazine; In Vitro Techniques; Leg; Mesenteric Arteries; Mesenteric Veins; Middle Aged; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Nifedipine; Norepinephrine; Potassium; Prazosin; Pyridines; Quinazolines | 1979 |
The vasorelaxant effect of evodiamine in rat isolated mesenteric arteries: mode of action.
Topics: Animals; Calcium; Calcium Channels; Calcium Chloride; Endothelium, Vascular; In Vitro Techniques; Male; Mesenteric Arteries; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Phenylephrine; Plant Extracts; Potassium Channels; Quinazolines; Rats; Rats, Sprague-Dawley; Tetraethylammonium Compounds; Vasodilator Agents | 1992 |
Pharmacological studies on quaternized 4(3H)-quinazolinones.
Topics: Animals; Anti-Infective Agents; Anticonvulsants; Hypnotics and Sedatives; Mice; Muscle Relaxation; Quinazolines | 1992 |
[Effect of moxisylyte on the lower urinary tracts (2). Effect on the urethra in anesthetized dogs].
Topics: Adrenergic alpha-Antagonists; Animals; Blood Pressure; Dogs; Dose-Response Relationship, Drug; Female; Heart Rate; Moxisylyte; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Phentolamine; Phenylephrine; Prazosin; Quinazolines; Urethra; Yohimbine | 1991 |
Studies on hypotensive agents. Synthesis of 1-substituted 3-(2-chlorophenyl)-6-ethoxycarbonyl-5,7-dimethyl-2,4(1H,3H)-quinazoline diones.
Topics: Animals; Antihypertensive Agents; In Vitro Techniques; Muscle Contraction; Muscle Relaxation; Muscle, Smooth, Vascular; Quinazolines; Rabbits | 1991 |
Effects of CGS-15943A on the relaxations produced by adenosine analogs in human blood vessels.
Topics: Adenosine; Adult; Coronary Vessels; Humans; In Vitro Techniques; Mammary Arteries; Middle Aged; Muscle Relaxation; Muscle, Smooth, Vascular; Potassium Chloride; Quinazolines; Saphenous Vein; Theophylline; Triazoles | 1990 |
2-(beta-Arylethylamino)- and 4-(beta-arylethylamino)quinazolines as phosphodiesterase inhibitors.
Topics: Animals; Cattle; Ethylamines; Female; Guinea Pigs; Muscle Relaxation; Muscle, Smooth; Myocardium; Phosphodiesterase Inhibitors; Quinazolines; Theophylline | 1985 |