Page last updated: 2024-08-21

quinazolines and Cardiovascular Diseases

quinazolines has been researched along with Cardiovascular Diseases in 42 studies

Research

Studies (42)

TimeframeStudies, this research(%)All Research%
pre-19902 (4.76)18.7374
1990's4 (9.52)18.2507
2000's7 (16.67)29.6817
2010's28 (66.67)24.3611
2020's1 (2.38)2.80

Authors

AuthorsStudies
Li, WQ; Li, YJ; Ma, WJ; Yin, YC; Zhang, BK1
Calosing, C; Gilham, D; Halliday, C; Jahagirdar, R; Johansson, J; Kulikowski, E; Sweeney, M; Tsujikawa, LM; Wasiak, S; Wong, NC1
Aglietta, M; Bonzano, A; Cagnazzo, C; Depetris, I; Filippi, R; Leone, F; Marino, D1
Dziadziuszko, R; Palczewski, P; Płatek, AE; Szymański, FM; Łęgosz, P1
Braconi, C; Chau, I; Cunningham, D; Forster, M; Gerlinger, M; Kalaitzaki, E; Khan, K; Rane, JK; Rao, S; Starling, N; Valeri, N; Watkins, D1
Li, JJ; Tian, KM; Xu, SW1
Emser, A; Gong, Y; von Eynatten, M; Woerle, HJ1
Grunberger, G1
Capdevila, J; Filetti, S; Grande, E; Kreissl, MC; Newbold, K; Reinisch, W; Robert, C; Schlumberger, M; Tolstrup, LK; Zamorano, JL1
Gu, JA; Huang, SH; Huang, ST; Lee, CM; Lin, CM; Lin, FY; Rau, TG; Yang, CH; Yang, WC1
Anastassiadis, E; Diessel, S; Forst, T; Löffler, A; Pfützner, A1
Abdel-Rahman, O; Fouad, M1
Hasegawa, Y; Katayama, T; Kim-Mitsuyama, S; Koibuchi, N; Kusaka, H; Lin, B; Ma, M; Nakagawa, T; Sueta, D; Toyama, K; Uekawa, K1
Chinetti-Gbaguidi, G; Colin, S; Kuivenhoven, JA; Staels, B1
Birtolo, C; Codeluppi, K; Cortelazzo, S; Fama, A; Gastl, G; Gugliotta, G; Gugliotta, L; Marcheselli, L; Piccin, A; Santoro, U; Steurer, M; Tieghi, A; Tortorella, G1
Davis, J; Gadkar, K; Lu, J; Mazer, NA; Ramanujan, S; Sahasranaman, S1
Gilham, D; Gordon, A; Halliday, C; Johansson, J; Kulikowski, E; McLure, K; Norek, K; Patel, RG; Sweeney, M; Tsujikawa, LM; Wasiak, S; Wong, NC; Young, P1
Chen, L; Fang, Q; Li, W; Li, X; Liang, G; Wang, J; Wang, L; Wang, Y; Zhang, Y; Zhong, P1
Birgegård, G1
Castaldo, V; Ferrara, ML; Gridelli, C; Maione, P; Mazzeo, N; Palazzolo, G; Rossi, A1
McNeill, E1
Vannucchi, AM1
Awada, A; Azim, HA; Metzger Filho, O; Saini, KS1
Catalano, O; De Giuli, L; Della Porta, MG; Eleuteri, E; Riccardi, A; Tondini, C; Zambelli, A1
Cacciola, E; Cacciola, R; Candoni, A; Ciancia, R; Codeluppi, K; Crugnola, M; Grossi, A; Gugliotta, L; Iurlo, A; Liberati, AM; Lunghi, M; Martinelli, V; Mazzucconi, MG; Palmieri, F; Pierri, I; Scalzulli, PR; Specchia, G; Tieghi, A; Tortorella, G; Usala, E; Vannucchi, AM; Vianelli, N1
Besses, C; Martínez-Sellés, M1
Johansen, OE; Neubacher, D; Patel, S; von Eynatten, M; Woerle, HJ1
Joy, TR1
Abbineni, C; Balaji, G; Balasubrahmanyam, D; Cheera, S; Elster, L; Frimurer, TM; Harinder Reddy, K; Högberg, T; Jadhav, VP; Kanna Reddy, HR; Khanna, I; Rist, Ø; Sasmal, PK; Sasmal, S; Sebastian, VJ; Shashikumar, D; Sihorkar, V; Singh, MP; Srinivas, G; Suresh, J; Talwar, R1
Imaizumi, S; Miura, S; Saku, K; Uehara, Y; Yahiro, E1
Goto, K1
Frantz, S1
Alcaraz, A; Elhilali, M; Emberton, M; Hartung, R; Harving, N; Matzkin, H; Vallancien, G; van Moorselaar, J1
O'Leary, MP1
Brogden, RN; Kellerman, D; Romankiewicz, JA; Stanaszek, WF1
Kather, H1
Buzelin, JM; Delauche-Cavallier, MC; Geffriaud-Ricouard, C; Roth, S; Santoni, JP1
Hara, Y; Harano, Y; Kanazawa, A; Nishioheda, Y; Ryomoto, K; Shinozaki, K; Suzuki, M; Tsushima, M1
Mesa, RA; Petitt, RM; Silverstein, MN; Solberg, LA; Tefferi, A1
Green, AR1
De la Rosette, JJ; Farmer, RD; Herings, RM; Leufkens, HG; Man in 't Veld, AJ; Souverein, PC1
Ijzerman, AP; Timmerman, H; van Muijlwijk-Koezen, JE1

Reviews

23 review(s) available for quinazolines and Cardiovascular Diseases

ArticleYear
Calcitonin gene‑related peptide‑mediated pharmacological effects in cardiovascular and gastrointestinal diseases (Review).
    Molecular medicine reports, 2021, Volume: 23, Issue:1

    Topics: Calcitonin Gene-Related Peptide; Cardiovascular Diseases; Gastrointestinal Diseases; Gene Expression Regulation; Humans; Indole Alkaloids; Molecular Targeted Therapy; Nitroglycerin; Quinazolines; Up-Regulation

2021
Fluoropyrimidine-induced cardiotoxicity.
    Critical reviews in oncology/hematology, 2018, Volume: 124

    Topics: Acetates; Capecitabine; Cardiotoxicity; Cardiovascular Diseases; Drug Combinations; Fluorouracil; Humans; Neoplasms; Pyrimidines; Pyrrolidines; Quinazolines; Thiophenes; Thymine; Trifluridine; Uracil; Uridine

2018
Rutaecarpine: A promising cardiovascular protective alkaloid from Evodia rutaecarpa (Wu Zhu Yu).
    Pharmacological research, 2019, Volume: 141

    Topics: Alkaloids; Animals; Anti-Inflammatory Agents; Antioxidants; Cardiotonic Agents; Cardiovascular Diseases; Evodia; Humans; Hypolipidemic Agents; Indole Alkaloids; Platelet Aggregation Inhibitors; Quinazolines; Vasodilator Agents

2019
Efficacy and safety of linagliptin in type 2 diabetes subjects at high risk for renal and cardiovascular disease: a pooled analysis of six phase III clinical trials.
    Cardiovascular diabetology, 2013, Apr-09, Volume: 12

    Topics: Cardiovascular Diseases; Clinical Trials, Phase III as Topic; Diabetes Mellitus, Type 2; Humans; Hypoglycemic Agents; Kidney Diseases; Linagliptin; Purines; Quinazolines; Randomized Controlled Trials as Topic; Risk Factors; Treatment Outcome

2013
Clinical utility of the dipeptidyl peptidase-4 inhibitor linagliptin.
    Postgraduate medicine, 2013, Volume: 125, Issue:3

    Topics: Cardiovascular Diseases; Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Humans; Hyperglycemia; Hypoglycemic Agents; Linagliptin; Purines; Quinazolines

2013
Vandetanib in advanced medullary thyroid cancer: review of adverse event management strategies.
    Advances in therapy, 2013, Volume: 30, Issue:11

    Topics: Carcinoma, Neuroendocrine; Cardiovascular Diseases; Dose-Response Relationship, Drug; Drug Administration Schedule; Drug Eruptions; Drug-Related Side Effects and Adverse Reactions; Female; Gastrointestinal Diseases; Humans; Male; Neoplasm Invasiveness; Neoplasm Staging; Patient Selection; Piperidines; Prognosis; Quinazolines; Risk Assessment; Thyroid Neoplasms; Treatment Outcome

2013
Risk of cardiovascular toxicities in patients with solid tumors treated with sunitinib, axitinib, cediranib or regorafenib: an updated systematic review and comparative meta-analysis.
    Critical reviews in oncology/hematology, 2014, Volume: 92, Issue:3

    Topics: Angiogenesis Inhibitors; Antineoplastic Agents; Axitinib; Cardiovascular Diseases; Humans; Imidazoles; Incidence; Indazoles; Indoles; Neoplasms; Phenylurea Compounds; Protein Kinase Inhibitors; Pyridines; Pyrroles; Quinazolines; Risk; Sunitinib

2014
Emerging small molecule drugs.
    Handbook of experimental pharmacology, 2015, Volume: 224

    Topics: Animals; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Drug Design; Dyslipidemias; Humans; Hypolipidemic Agents; Liver X Receptors; Molecular Targeted Therapy; Orphan Nuclear Receptors; Peroxisome Proliferator-Activated Receptors; Quinazolines; Quinazolinones; Signal Transduction

2015
The Use of Anagrelide in Myeloproliferative Neoplasms, with Focus on Essential Thrombocythemia.
    Current hematologic malignancy reports, 2016, Volume: 11, Issue:5

    Topics: Age Factors; Bone Marrow; Cardiovascular Diseases; Humans; Interferon-alpha; Myeloproliferative Disorders; Platelet Aggregation Inhibitors; Quinazolines; Tachycardia; Thrombocythemia, Essential

2016
Treatment of advanced non-small-cell lung cancer in the elderly.
    Lung cancer (Amsterdam, Netherlands), 2009, Volume: 66, Issue:3

    Topics: Age Factors; Aged; Aged, 80 and over; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Bevacizumab; Carcinoma, Non-Small-Cell Lung; Cardiovascular Diseases; Cisplatin; Clinical Trials as Topic; Comorbidity; Contraindications; ErbB Receptors; Erlotinib Hydrochloride; Gefitinib; Humans; Lung Neoplasms; Quinazolines; Radiation-Sensitizing Agents; Vascular Endothelial Growth Factor A

2009
RVX-208, a stimulator of apolipoprotein AI gene expression for the treatment of cardiovascular diseases.
    Current opinion in investigational drugs (London, England : 2000), 2010, Volume: 11, Issue:3

    Topics: Animals; Apolipoprotein A-I; Cardiovascular Diseases; Clinical Trials as Topic; Gene Expression; Humans; Quinazolines; Quinazolinones

2010
JAK2 mutation and thrombosis in the myeloproliferative neoplasms.
    Current hematologic malignancy reports, 2010, Volume: 5, Issue:1

    Topics: Amino Acid Substitution; Aspirin; Cardiovascular Diseases; Clinical Trials as Topic; Fibrinolytic Agents; Humans; Incidence; Interferon-alpha; Janus Kinase 2; Multicenter Studies as Topic; Mutation, Missense; Myeloproliferative Disorders; Phenotype; Point Mutation; Quinazolines; Thrombophilia; Thrombosis

2010
Prevention and management of major side effects of targeted agents in breast cancer.
    Critical reviews in oncology/hematology, 2012, Volume: 84 Suppl 1

    Topics: Animals; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Bevacizumab; Breast; Breast Neoplasms; Cardiovascular Diseases; Female; Gastrointestinal Diseases; Humans; Lapatinib; Molecular Targeted Therapy; Quinazolines; Skin Diseases; Trastuzumab

2012
Predicting and preventing cardiotoxicity in the era of breast cancer targeted therapies. Novel molecular tools for clinical issues.
    Breast (Edinburgh, Scotland), 2011, Volume: 20, Issue:2

    Topics: Angiogenesis Inhibitors; Antibodies, Monoclonal; Antibodies, Monoclonal, Humanized; Antineoplastic Agents; Benzenesulfonates; Bevacizumab; Biomarkers; Breast Neoplasms; Cardiotoxins; Cardiovascular Diseases; Female; Heart Failure; Humans; Indoles; Lapatinib; Molecular Targeted Therapy; Niacinamide; Phenylurea Compounds; Protein Kinase Inhibitors; Pyridines; Pyrroles; Quinazolines; Risk Assessment; Sorafenib; Sunitinib; Trastuzumab

2011
Cardiovascular safety with linagliptin in patients with type 2 diabetes mellitus: a pre-specified, prospective, and adjudicated meta-analysis of a phase 3 programme.
    Cardiovascular diabetology, 2012, Jan-10, Volume: 11

    Topics: Aged; Angina, Unstable; Biomarkers; Blood Glucose; Cardiovascular Diseases; Clinical Trials, Phase III as Topic; Diabetes Complications; Diabetes Mellitus, Type 2; Dipeptidyl-Peptidase IV Inhibitors; Evidence-Based Medicine; Female; Glycated Hemoglobin; Hospitalization; Humans; Linagliptin; Male; Middle Aged; Myocardial Infarction; Patient Safety; Proportional Hazards Models; Prospective Studies; Purines; Quinazolines; Randomized Controlled Trials as Topic; Risk Assessment; Risk Factors; Stroke; Treatment Outcome

2012
Novel HDL-based therapeutic agents.
    Pharmacology & therapeutics, 2012, Volume: 135, Issue:1

    Topics: Animals; Apolipoprotein A-I; Biomarkers; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Dyslipidemias; Humans; Hypolipidemic Agents; Molecular Mimicry; Quinazolines; Quinazolinones; Treatment Outcome

2012
Chymase inhibitors.
    Current pharmaceutical design, 2013, Volume: 19, Issue:17

    Topics: Acetamides; Animals; Atrial Fibrillation; Azetidines; Benzoates; Cardiovascular Diseases; Chymases; Heart Failure; Humans; Hypertension; Mast Cells; Oxazoles; Pyrimidines; Quinazolines; Sulfonamides

2013
[Prospects for endothelin-related drugs].
    Nihon rinsho. Japanese journal of clinical medicine, 2004, Volume: 62 Suppl 9

    Topics: Animals; Aspartic Acid Endopeptidases; Bosentan; Cardiovascular Diseases; Drug Design; Endothelin Receptor Antagonists; Endothelin-1; Endothelin-Converting Enzymes; Hemodynamics; Humans; Metalloendopeptidases; Organophosphonates; Peptides, Cyclic; Quinazolines; Receptors, Endothelin; Sulfonamides; Sulfonylurea Compounds; Tetracyclines; Tetrazoles

2004
Treatment and pharmacologic management of BPH in the context of common comorbidities.
    The American journal of managed care, 2006, Volume: 12, Issue:5 Suppl

    Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Azasteroids; Cardiovascular Diseases; Comorbidity; Doxazosin; Drug Therapy, Combination; Dutasteride; Enzyme Inhibitors; Erectile Dysfunction; Finasteride; Global Health; Humans; Male; Prazosin; Prostatic Hyperplasia; Quinazolines; Sulfonamides; Tamsulosin; Transurethral Resection of Prostate; Treatment Outcome

2006
Prazosin update. A review of its pharmacological properties and therapeutic use in hypertension and congestive heart failure.
    Drugs, 1983, Volume: 25, Issue:4

    Topics: Adrenergic alpha-Antagonists; Blood Pressure; Cardiovascular Diseases; Clinical Trials as Topic; Heart Failure; Heart Rate; Hemodynamics; Humans; Hypertension; Kidney; Lipid Metabolism; Prazosin; Quinazolines; Regional Blood Flow; Renin-Angiotensin System

1983
Anagrelide as a new platelet-lowering agent in essential thrombocythemia: mechanism of actin, efficacy, toxicity, current indications.
    Seminars in thrombosis and hemostasis, 1997, Volume: 23, Issue:4

    Topics: Animals; Bone Marrow; Cardiovascular Diseases; Clinical Trials as Topic; Cohort Studies; Hematopoiesis; Hemodynamics; Humans; Megakaryocytes; Middle Aged; Myeloproliferative Disorders; Platelet Aggregation Inhibitors; Quinazolines; Thrombocythemia, Essential; Thrombosis

1997
The pathogenesis and management of essential thrombocythaemia.
    Haematologica, 1999, Volume: 84 Suppl EHA-4

    Topics: Acute Disease; Alkylating Agents; Aspirin; Cardiovascular Diseases; Clone Cells; Gene Expression; Hemorrhage; Humans; Hydroxyurea; Leukemia, Myeloid; Megakaryocytes; Platelet Aggregation Inhibitors; Quinazolines; Risk; Thrombocythemia, Essential; Thrombophilia

1999
The adenosine A3 receptor and its ligands.
    Progress in medicinal chemistry, 2001, Volume: 38

    Topics: Adenosine; Amino Acid Sequence; Animals; Cardiovascular Diseases; Cloning, Molecular; Flavonoids; Humans; Immune System Diseases; Lung Diseases; Models, Animal; Molecular Sequence Data; Protein Binding; Pyrans; Pyridines; Quinazolines; Receptors, Purinergic; Sequence Alignment; Species Specificity; Triazoles; Xanthines

2001

Trials

4 trial(s) available for quinazolines and Cardiovascular Diseases

ArticleYear
Effect of linagliptin compared with glimepiride on postprandial glucose metabolism, islet cell function and vascular function parameters in patients with type 2 diabetes mellitus receiving ongoing metformin treatment.
    Diabetes/metabolism research and reviews, 2014, Volume: 30, Issue:7

    Topics: Aged; Biomarkers; Blood Glucose; Cardiovascular Diseases; Diabetes Mellitus, Type 2; Drug Therapy, Combination; Female; Glucagon; Glucagon-Like Peptide 1; Humans; Hypoglycemic Agents; Insulin; Islets of Langerhans; Linagliptin; Male; Metformin; Middle Aged; Plasminogen Activator Inhibitor 1; Postprandial Period; Proinsulin; Purines; Quinazolines; Risk Factors; Sulfonylurea Compounds

2014
Anagrelide treatment and cardiovascular monitoring in essential thrombocythemia. A prospective observational study.
    Leukemia research, 2015, Volume: 39, Issue:6

    Topics: Adult; Aged; Cardiovascular Diseases; Electrocardiography; Female; Follow-Up Studies; Humans; Male; Middle Aged; Monitoring, Physiologic; Natriuretic Peptide, Brain; Peptide Fragments; Platelet Aggregation Inhibitors; Prospective Studies; Quinazolines; Thrombocythemia, Essential; Troponin I

2015
Prazosin update. A review of its pharmacological properties and therapeutic use in hypertension and congestive heart failure.
    Drugs, 1983, Volume: 25, Issue:4

    Topics: Adrenergic alpha-Antagonists; Blood Pressure; Cardiovascular Diseases; Clinical Trials as Topic; Heart Failure; Heart Rate; Hemodynamics; Humans; Hypertension; Kidney; Lipid Metabolism; Prazosin; Quinazolines; Regional Blood Flow; Renin-Angiotensin System

1983
Clinical uroselectivity: evidence from patients treated with slow-release alfuzosin for symptomatic benign prostatic obstruction.
    British journal of urology, 1997, Volume: 79, Issue:6

    Topics: Adrenergic alpha-Antagonists; Aged; Antihypertensive Agents; Blood Pressure; Cardiovascular Diseases; Delayed-Action Preparations; Double-Blind Method; Humans; Hypertension; Male; Prostatic Hyperplasia; Quinazolines; Treatment Outcome; Urinary Retention; Urination

1997

Other Studies

16 other study(ies) available for quinazolines and Cardiovascular Diseases

ArticleYear
Downregulation of the Complement Cascade In Vitro, in Mice and in Patients with Cardiovascular Disease by the BET Protein Inhibitor Apabetalone (RVX-208).
    Journal of cardiovascular translational research, 2017, Volume: 10, Issue:4

    Topics: Animals; Cardiovascular Diseases; Cells, Cultured; Complement Activation; Complement Inactivating Agents; Complement System Proteins; Cytokines; Gene Expression Profiling; Hepatocytes; Humans; Immunity, Innate; Mice, SCID; Primary Cell Culture; Proteins; Proteomics; Quinazolines; Quinazolinones; Signal Transduction

2017
Cardiovascular safety of novel non-small cell lung cancer oncotherapy in a patient treated with novel generations of tyrosine kinase inhibitors.
    Kardiologia polska, 2018, Volume: 76, Issue:3

    Topics: Acrylamides; Afatinib; Aniline Compounds; Antineoplastic Agents; Carcinoma, Non-Small-Cell Lung; Cardiotonic Agents; Cardiovascular Diseases; Gefitinib; Humans; Lung Neoplasms; Middle Aged; Nebivolol; Piperazines; Protein Kinase Inhibitors; Quinazolines; Ramipril

2018
Efficacy and Cardiotoxic Safety Profile of Raltitrexed in Fluoropyrimidines-Pretreated or High-Risk Cardiac Patients With GI Malignancies: Large Single-Center Experience.
    Clinical colorectal cancer, 2019, Volume: 18, Issue:1

    Topics: Adult; Aged; Aged, 80 and over; Antineoplastic Combined Chemotherapy Protocols; Capecitabine; Cardiotoxicity; Cardiovascular Diseases; Female; Fluorouracil; Follow-Up Studies; Gastrointestinal Neoplasms; Humans; Male; Middle Aged; Prognosis; Quinazolines; Retrospective Studies; Safety; Survival Rate; Thiophenes

2019
Low-cytotoxic synthetic bromorutaecarpine exhibits anti-inflammation and activation of transient receptor potential vanilloid type 1 activities.
    BioMed research international, 2013, Volume: 2013

    Topics: Anti-Inflammatory Agents; Cardiovascular Diseases; Drugs, Chinese Herbal; Evodia; Gene Expression Regulation; Humans; Indole Alkaloids; Inflammation; Macrophages; Nitric Oxide Synthase Type II; Quinazolines; TRPV Cation Channels

2013
DPP-4 inhibitor linagliptin ameliorates cardiovascular injury in salt-sensitive hypertensive rats independently of blood glucose and blood pressure.
    Cardiovascular diabetology, 2014, Nov-29, Volume: 13

    Topics: Animals; Blood Glucose; Blood Pressure; Blood Pressure Determination; Cardiovascular Diseases; Dipeptidyl-Peptidase IV Inhibitors; Disease Models, Animal; Heart; Hypertension; Linagliptin; Male; Purines; Quinazolines; Rats; Rats, Inbred Dahl; Sodium Chloride, Dietary

2014
Evaluation of HDL-modulating interventions for cardiovascular risk reduction using a systems pharmacology approach.
    Journal of lipid research, 2016, Volume: 57, Issue:1

    Topics: Apolipoprotein A-I; Biological Transport; Biomarkers; Cardiovascular Diseases; Cholesterol; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Humans; Hypolipidemic Agents; Lipoproteins, HDL; Models, Biological; Quinazolines; Quinazolinones; Risk Factors; Up-Regulation

2016
RVX-208, a BET-inhibitor for treating atherosclerotic cardiovascular disease, raises ApoA-I/HDL and represses pathways that contribute to cardiovascular disease.
    Atherosclerosis, 2016, Volume: 247

    Topics: Apolipoprotein A-I; Atherosclerosis; Cardiovascular Diseases; Cells, Cultured; Cholesterol, HDL; Clinical Trials, Phase II as Topic; Dose-Response Relationship, Drug; Gene Expression Profiling; Hepatocytes; Humans; Hypolipidemic Agents; Liver; Male; Oligonucleotide Array Sequence Analysis; Quinazolines; Quinazolinones; Randomized Controlled Trials as Topic; Retrospective Studies; Signal Transduction; Time Factors; Up-Regulation

2016
EGFR Inhibition Blocks Palmitic Acid-induced inflammation in cardiomyocytes and Prevents Hyperlipidemia-induced Cardiac Injury in Mice.
    Scientific reports, 2016, Apr-18, Volume: 6

    Topics: Animals; Apolipoproteins E; Apoptosis; Cardiovascular Diseases; Cell Line; Diet, High-Fat; ErbB Receptors; Hyperlipidemias; Male; Mice; Mice, Inbred C57BL; Myocytes, Cardiac; Palmitic Acid; Protein Kinase Inhibitors; Quinazolines; Rats; src-Family Kinases; Toll-Like Receptor 4; Tyrphostins

2016
Low impact of cardiovascular adverse events on anagrelide treatment discontinuation in a cohort of 232 patients with essential thrombocythemia.
    Leukemia research, 2011, Volume: 35, Issue:12

    Topics: Adolescent; Adult; Aged; Aged, 80 and over; Cardiovascular Diseases; Child; Cohort Studies; Drug-Related Side Effects and Adverse Reactions; Female; Follow-Up Studies; Humans; Male; Middle Aged; Platelet Aggregation Inhibitors; Quinazolines; Retrospective Studies; Thrombocythemia, Essential; Withholding Treatment; Young Adult

2011
Anagrelide and cardiovascular events. Much ado about nothing?
    Leukemia research, 2011, Volume: 35, Issue:12

    Topics: Cardiovascular Diseases; Female; Humans; Male; Quinazolines; Thrombocythemia, Essential; Withholding Treatment

2011
Design and optimization of quinazoline derivatives as melanin concentrating hormone receptor 1 (MCHR1) antagonists: part 2.
    Bioorganic & medicinal chemistry letters, 2012, May-01, Volume: 22, Issue:9

    Topics: Cardiovascular Diseases; Drug Design; Humans; Quinazolines; Receptors, Pituitary Hormone; Receptors, Somatostatin; Structure-Activity Relationship

2012
Drug discovery: playing dirty.
    Nature, 2005, Oct-13, Volume: 437, Issue:7061

    Topics: Animals; Benzamides; Cardiovascular Diseases; Clinical Trials as Topic; Clozapine; Depression; Drug Approval; Drug Design; Drug Evaluation, Preclinical; Drug Industry; Gefitinib; Humans; Imatinib Mesylate; Neoplasms; Piperazines; Pyrimidines; Quinazolines; Sensitivity and Specificity; Substrate Specificity; Therapeutics; United States; United States Food and Drug Administration

2005
Age, comorbidity and hypertensive co-medication do not affect cardiovascular tolerability of 10 mg alfuzosin once daily.
    The Journal of urology, 2006, Volume: 175, Issue:2

    Topics: Adrenergic alpha-Antagonists; Age Factors; Aged; Antihypertensive Agents; Cardiovascular Diseases; Diabetes Complications; Drug Administration Schedule; Humans; Hypertension; Male; Middle Aged; Myocardial Ischemia; Quinazolines; Urination Disorders

2006
[Hypertensive therapy with prazosin. Concomitant cardiovascular, metabolic and respiratory diseases. Proven facts and potential aspects].
    Fortschritte der Medizin, 1984, Apr-26, Volume: 102, Issue:16

    Topics: Adolescent; Adult; Arrhythmias, Cardiac; Cardiovascular Diseases; Diabetes Complications; Humans; Hypertension; Kidney; Lipids; Myocardial Infarction; Prazosin; Quinazolines; Respiratory Tract Diseases

1984
Clinical impact of insulin resistance syndrome in cardiovascular diseases and its therapeutic approach.
    Hypertension research : official journal of the Japanese Society of Hypertension, 1996, Volume: 19 Suppl 1

    Topics: Adrenergic alpha-Antagonists; Adult; Aged; Amlodipine; Angiotensin-Converting Enzyme Inhibitors; Blood Pressure; Calcium Channel Blockers; Cardiovascular Diseases; Cilazapril; Humans; Insulin Resistance; Middle Aged; Quinazolines

1996
Evaluating adverse cardiovascular effects of drug treatment for benign prostatic hyperplasia (BPH): methodological considerations.
    Journal of clinical epidemiology, 2001, Volume: 54, Issue:5

    Topics: 5-alpha Reductase Inhibitors; Adrenergic alpha-Antagonists; Adult; Aged; Bias; Cardiovascular Diseases; Case-Control Studies; Finasteride; Humans; Male; Middle Aged; Morbidity; Netherlands; Prazosin; Prognosis; Prostatic Hyperplasia; Quinazolines; Research Design; Risk Factors; Sulfonamides; Tamsulosin

2001