quinazolines has been researched along with Adjuvant Arthritis in 22 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 5 (22.73) | 18.7374 |
1990's | 4 (18.18) | 18.2507 |
2000's | 6 (27.27) | 29.6817 |
2010's | 6 (27.27) | 24.3611 |
2020's | 1 (4.55) | 2.80 |
Authors | Studies |
---|---|
Gao, WL; Li, YT; Lu, M; Wang, J; Yin, L; Yin, ZS; Zhang, H | 1 |
Abuelizz, HA; Al-Salahi, R; Ali, AA; Ezzeldin, E; Hassane, AE; Marzouk, M | 1 |
Bai, X; Cai, D; Huang, B; Jiang, W; Jiang, Y; Li, K; Li, M; Liu, A; Shen, J; Song, Q; Xu, S; Zhang, Y | 1 |
Dagli, AF; Erman, F; Gundogdu, B; Isik, A; Karatas, A; Koca, SS; Ozgen, M; Sahin, K | 1 |
Cao, D; Chen, L; Li, D; Pei, H; Pu, Y; Tang, M; Xie, C | 1 |
Ishikawa, M; Miyaki, S; Nakasa, T; Ochi, M; Takada, T | 1 |
Akama-Garren, EH; Edalati, A; Lindstrom, TM; Petralia, JD; Robinson, WH; Ruiz, PJ; Stein, EA; Swanson, CD | 1 |
Hayashi, H; Isobe, Y; Nagasaki, T; Obara, F; Tobe, M; Tomizawa, H | 1 |
Achira, M; Kume, T; Totsuka, R | 1 |
Beaton, HG; Boughton-Smith, N; Cook, TR; Cooper, SL; Fraser-Rae, L; Hallam, K; Hamley, P; McInally, T; Nicholls, DJ; Pimm, AD; Tinker, AC; Wallace, AV | 1 |
Bennett, BL; Desai, S; Erdman, PE; Manning, A; Ow, A; Palanki, MS; Ransone, L; Ren, M; Spooner, C; Suto, M; Toriumi, W; Totsuka, R; Tsao, P | 1 |
Baharav, E; Bar-Yehuda, S; Fishman, P; Halpren, M; Madi, L; Ochaion, A; Rath-Wolfson, L; Silberman, D; Weinberger, A | 1 |
Diacovo, TG; Puri, KD; Randis, TM; Zhou, H | 1 |
Houlihan, WJ; Perrine, JW; Takesue, EI | 1 |
Ghia, M; Mattioli, F; Minganti, V; Novelli, F | 1 |
Bateman-Fite, R; Brackeen, MF; Clark, RL; Connolly, KM; Menius, JA; Noel, LS; Sekut, L; Stimpson, SA; Yarnall, D | 1 |
Baba, A; Kawamura, N; Makino, H; Ohta, Y; Sohda, T; Taketomi, S | 1 |
Diamantis, W; Ludwig, BJ; Sofia, RD | 1 |
Baggiolini, M; Gubler, HU | 1 |
Awata, H; Inukai, T; Koga, Y; Kurokawa, H; Yanagi, Y | 1 |
Chand, D; Kaul, A; Khajuria, A; Sharma, ML | 1 |
Fujii, T; Fujitsu, T; Hiroi, J; Kobayashi, K; Mori, J; Motoyama, Y; Ohara, K; Shibayama, F | 1 |
22 other study(ies) available for quinazolines and Adjuvant Arthritis
Article | Year |
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Evodiamine attenuates adjuvant-induced arthritis in rats by inhibiting synovial inflammation and restoring the Th17/Treg balance.
Topics: Animals; Arthritis, Experimental; Interleukin-10; Interleukin-6; Joints; Male; Quinazolines; Rats; Rats, Inbred Lew; STAT3 Transcription Factor; STAT5 Transcription Factor; Synovial Membrane; Synovitis; T-Lymphocytes, Regulatory; Th17 Cells; Tumor Necrosis Factor-alpha | 2020 |
Molecular modeling, enzyme activity, anti-inflammatory and antiarthritic activities of newly synthesized quinazoline derivatives.
Topics: Animals; Antirheumatic Agents; Arthritis, Experimental; Carrageenan; Cyclooxygenase 1; Cyclooxygenase 2; Cyclooxygenase Inhibitors; Dose-Response Relationship, Drug; Edema; Membrane Proteins; Molecular Docking Simulation; Molecular Structure; Quinazolines; Rats; Structure-Activity Relationship | 2017 |
Tyrosine kinase Fyn promotes osteoarthritis by activating the β-catenin pathway.
Topics: Aging; Animals; Arthritis, Experimental; Benzodioxoles; beta Catenin; Cartilage, Articular; Cells, Cultured; Chondrocytes; Enzyme Inhibitors; Gene Knockout Techniques; Humans; Mice, Knockout; Molecular Targeted Therapy; Osteoarthritis; Proto-Oncogene Proteins c-fyn; Pyrazoles; Pyrimidines; Quinazolines; Signal Transduction | 2018 |
Lapatinib ameliorates experimental arthritis in rats.
Topics: Animals; Arthritis, Experimental; Female; Inflammation Mediators; Lapatinib; Quinazolines; Random Allocation; Rats; Rats, Wistar | 2015 |
Anti-arthritis effect of a novel quinazoline derivative through inhibiting production of TNF-α mediated by TNF-α converting enzyme in murine collagen-induced arthritis model.
Topics: ADAM Proteins; ADAM17 Protein; Animals; Arthritis, Experimental; Cell Line; Collagen; Disease Models, Animal; Enzyme-Linked Immunosorbent Assay; Male; Mice; Mice, Inbred DBA; Quinazolines; RNA, Messenger; Tumor Necrosis Factor-alpha | 2015 |
Attenuation of cartilage degeneration by calcitonin gene-related paptide receptor antagonist via inhibition of subchondral bone sclerosis in osteoarthritis mice.
Topics: Animals; Arthritis, Experimental; Bone Remodeling; Calcitonin Gene-Related Peptide Receptor Antagonists; Cartilage; Cells, Cultured; Dipeptides; Drug Evaluation, Preclinical; Humans; Male; Mice, Inbred C57BL; Osteoarthritis; Osteogenesis; Piperazines; Quinazolines | 2016 |
Inhibition of epidermal growth factor receptor tyrosine kinase ameliorates collagen-induced arthritis.
Topics: Animals; Arthritis, Experimental; Arthritis, Rheumatoid; Becaplermin; Cell Division; Cyclooxygenase 2; Cytokines; Drug Evaluation, Preclinical; Endothelial Cells; ErbB Receptors; Erlotinib Hydrochloride; Fibroblasts; Gene Expression Regulation; Human Umbilical Vein Endothelial Cells; Humans; Male; Mice; Mice, Inbred DBA; Neovascularization, Pathologic; Osteoclasts; Protein Kinase Inhibitors; Proto-Oncogene Proteins c-sis; Quinazolines; Synovial Membrane | 2012 |
Structure-activity relationships of 6-fluoroquinazolines: dual-acting compounds with inhibitory activities toward both TNF-alpha production and T cell proliferation.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Area Under Curve; Arthritis, Experimental; B-Lymphocytes; Cell Division; Concanavalin A; Depression, Chemical; Drug Design; Edema; Humans; In Vitro Techniques; Lipopolysaccharides; Magnetic Resonance Spectroscopy; Male; Mice; Neutrophils; Quinazolines; Rats; Rats, Sprague-Dawley; Spleen; Structure-Activity Relationship; T-Lymphocytes; Tumor Necrosis Factor-alpha | 2003 |
Differences in pharmacokinetics and hepatobiliary transport of a novel anti-inflammatory agent between normal and adjuvant arthritis rats.
Topics: Administration, Oral; Animals; Anti-Inflammatory Agents; Area Under Curve; Arthritis, Experimental; Biological Transport; Caco-2 Cells; Chromatography, High Pressure Liquid; Dose-Response Relationship, Drug; Female; Humans; Hydrazines; Injections, Intravenous; Liver; Models, Chemical; Quinazolines; Quinidine; Rats; Rats, Inbred Lew; Time Factors | 2002 |
1,2-Dihydro-4-quinazolinamines: potent, highly selective inhibitors of inducible nitric oxide synthase which show antiinflammatory activity in vivo.
Topics: Acute Disease; Administration, Oral; Amines; Animals; Arthritis, Experimental; Cell Line; Chronic Disease; Enzyme Inhibitors; Injections, Intravenous; Isoenzymes; Nitric Oxide Synthase; Nitric Oxide Synthase Type II; Quinazolines; Rats; Spiro Compounds; Structure-Activity Relationship | 2003 |
The design and synthesis of novel orally active inhibitors of AP-1 and NF-kappaB mediated transcriptional activation. SAR of in vitro and in vivo studies.
Topics: Administration, Oral; Animals; Arthritis, Experimental; Disease Models, Animal; Drug Design; Humans; Jurkat Cells; NF-kappa B; Quinazolines; Rats; Structure-Activity Relationship; Transcription Factor AP-1; Transcriptional Activation | 2003 |
Antiinflammatory effect of A3 adenosine receptor agonists in murine autoimmune arthritis models.
Topics: Adenosine; Adenosine A3 Receptor Agonists; Adenosine A3 Receptor Antagonists; Animals; Anti-Inflammatory Agents; Arthritis, Experimental; Collagen; Dose-Response Relationship, Drug; Female; Joints; Lymph Nodes; Male; Mice; Mice, Inbred DBA; Quinazolines; Rats; Receptor, Adenosine A3; Spleen; Triazoles; Tumor Necrosis Factor-alpha | 2005 |
Role of PI3Kdelta and PI3Kgamma in inflammatory arthritis and tissue localization of neutrophils.
Topics: Adenine; Animals; Arthritis, Experimental; Chemotaxis, Leukocyte; Class I Phosphatidylinositol 3-Kinases; Class Ib Phosphatidylinositol 3-Kinase; Edema; Enzyme Inhibitors; Hindlimb; Isoenzymes; Leukotriene B4; Mice; Mice, Inbred NOD; Mice, Inbred Strains; Mice, Knockout; Mice, Transgenic; N-Formylmethionine Leucyl-Phenylalanine; Neutrophil Infiltration; Neutrophils; Phosphatidylinositol 3-Kinases; Phosphoinositide-3 Kinase Inhibitors; Quinazolines | 2008 |
Anti-inflammatory and other pharmacodynamic properties of five members of the 4-aryl-1-isopropyl-2(1H)-quinazolinone series.
Topics: Animals; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Blood Glucose; Bronchodilator Agents; Central Nervous System; Chemical Phenomena; Chemistry; Chickens; Fever; Guinea Pigs; Hemodynamics; Hypoglycemic Agents; Male; Mice; Quinazolines; Rabbits; Rats; Rats, Inbred Strains; Stomach Ulcer; Time Factors | 1984 |
Inhibitory properties of triethylphosphine goldlupinylsulfide in adjuvant-induced arthritis in rats.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Antirheumatic Agents; Arthritis, Experimental; Gold; Male; Organogold Compounds; Organometallic Compounds; Quinazolines; Rats; Rats, Sprague-Dawley | 1995 |
Anti-inflammatory activity of phosphodiesterase (PDE)-IV inhibitors in acute and chronic models of inflammation.
Topics: Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Carrageenan; Female; Galactosamine; Inflammation; Lipopolysaccharides; Macrophages; Male; Mice; Mice, Inbred C3H; Mice, Inbred C57BL; Phosphodiesterase Inhibitors; Purinones; Pyridazines; Pyrrolidinones; Quinazolines; Rats; Rats, Inbred Lew; Rolipram; Shock, Septic; Tumor Necrosis Factor-alpha | 1995 |
Studies on disease-modifying antirheumatic drugs: synthesis of novel quinoline and quinazoline derivatives and their anti-inflammatory effect.
Topics: Animals; Antirheumatic Agents; Arthritis, Experimental; Bone Resorption; Dinoprostone; Disease Models, Animal; Female; Magnetic Resonance Spectroscopy; Male; Pregnancy; Quinazolines; Quinolines; Rats; Rats, Inbred Lew; Rats, Sprague-Dawley; Structure-Activity Relationship | 1996 |
Pharmacological properties of 2,3-dihydro-9H-isoxazolo [3,2-b] quinazolin-9-one (W-2429. Part 1: Analgesic, antipyretic and antiedema activity.
Topics: Administration, Oral; Analgesics, Opioid; Animals; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Aspirin; Body Temperature; Dextropropoxyphene; Drug Interactions; Drug Tolerance; Edema; Fever; Humans; Injections, Intravenous; Isoxazoles; Lethal Dose 50; Male; Mice; Narcotic Antagonists; Oxazoles; Quinazolines; Rats; Substance-Related Disorders; Time Factors | 1977 |
Pharmacological properties of proquazone.
Topics: Animals; Anti-Inflammatory Agents; Anti-Inflammatory Agents, Non-Steroidal; Arthritis, Experimental; Drug Evaluation, Preclinical; Gastrointestinal Hemorrhage; Indomethacin; Inflammation; Quinazolines; Rats | 1978 |
[Anti-inflammatory activity of SL-573 (author's transl)].
Topics: Adrenalectomy; Animals; Anti-Inflammatory Agents; Arthritis, Experimental; Capillary Permeability; Depression, Chemical; Edema; Granuloma; Intestinal Perforation; Male; Mice; Quinazolines; Quinazolinones; Rats; Wound Healing | 1978 |
Immunopharmacological properties of azepino [2, 1-b] quinazolin-12(6H)-one-7, 8, 9, 10-tetrahydro (RLX).
Topics: Animals; Antibody Formation; Arthritis, Experimental; Bronchodilator Agents; Hypersensitivity, Delayed; Immunosuppressive Agents; In Vitro Techniques; Lymphocyte Activation; Male; Mice; Neutrophils; Pleurisy; Quinazolines; Rabbits; Rats | 1992 |
Effects of FR50948, a new orally active antiallergic agent, in experimental allergic models.
Topics: Animals; Arthritis, Experimental; Arthus Reaction; Bronchi; Forssman Antigen; Guinea Pigs; Histamine Release; Hypersensitivity; Male; Mast Cells; Mice; Mice, Inbred ICR; Neutrophils; Passive Cutaneous Anaphylaxis; Quinazolines; Rats; Rats, Inbred Strains | 1988 |