Page last updated: 2024-08-18

pyrroles and Plasmodium falciparum Malaria

pyrroles has been researched along with Plasmodium falciparum Malaria in 9 studies

Research

Studies (9)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's3 (33.33)29.6817
2010's5 (55.56)24.3611
2020's1 (11.11)2.80

Authors

AuthorsStudies
Andrew, AK; Cooper, CA; Moore, JM; Morffy Smith, CD; Russ, BN1
Angulo-Barturen, I; Barker, H; Burrows, JN; Charman, SA; Chen, G; Chittimalla, R; Chiu, FCK; Crighton, E; Deng, X; El Mazouni, F; Ferrer, S; Huertas-Valentin, L; Jimenez-Diaz, MB; Katneni, K; Kokkonda, S; Lafuente-Monasterio, MJ; Martinez-Martinez, MS; Matthews, D; McLaren, J; Palmer, MJ; Phillips, MA; Rathod, PK; Shackleford, DM; Shahi, SP; Tomchick, D; Waterson, D; White, J; White, KL; Wittlin, S1
Abdullahi, M; Arang, N; Austin, LS; Billman, ZP; Douglass, AN; Hume, JCC; Kain, HS; Kappe, SHI; Kaushansky, A; Mikolajczak, SA; Murphy, SC1
Bienvenu, AL; Picot, S1
Amalvict, R; Baret, E; Briolant, S; Dormoi, J; Gil, M; Henry, M; Parquet, V; Pradines, B; Rogier, C; Wurtz, N1
Cassera, MB; Hazleton, KZ; Schramm, VL; Zhang, Y1
Büchhold, C; Ehlers, M; Gelhaus, C; Langolf, S; Machon, U; Rosenthal, PJ; Schirmeister, T; Schmuck, C; Sicking, W1
Davis, TM; Hamzah, J; Skinner-Adams, TS1
Baret, E; Briolant, S; Fontaine, A; Fusai, T; Henry, M; Mosnier, J; Pradines, B; Rogier, C; Torrentino-Madamet, M1

Reviews

1 review(s) available for pyrroles and Plasmodium falciparum Malaria

ArticleYear
Purine and pyrimidine pathways as targets in Plasmodium falciparum.
    Current topics in medicinal chemistry, 2011, Volume: 11, Issue:16

    Topics: Antimalarials; Binding Sites; Drug Design; Enzyme Inhibitors; Humans; Malaria, Falciparum; Models, Molecular; Plasmodium falciparum; Protein Binding; Protozoan Proteins; Purine Nucleosides; Purines; Pyrimidines; Pyrimidinones; Pyrroles; Substrate Specificity

2011

Other Studies

8 other study(ies) available for pyrroles and Plasmodium falciparum Malaria

ArticleYear
A novel murine model for assessing fetal and birth outcomes following transgestational maternal malaria infection.
    Scientific reports, 2019, 12-20, Volume: 9, Issue:1

    Topics: Animals; Cell Survival; Chromosome Pairing; Disease Models, Animal; Female; Finite Element Analysis; Malaria; Malaria, Falciparum; Mice; Nerve Regeneration; Polymers; Pregnancy; Pregnancy Complications, Parasitic; Pyrroles; Tissue Scaffolds

2019
Lead Optimization of a Pyrrole-Based Dihydroorotate Dehydrogenase Inhibitor Series for the Treatment of Malaria.
    Journal of medicinal chemistry, 2020, 05-14, Volume: 63, Issue:9

    Topics: Animals; Antimalarials; Cell Line, Tumor; Crystallography, X-Ray; Dihydroorotate Dehydrogenase; Dogs; Enzyme Inhibitors; Female; Humans; Malaria, Falciparum; Male; Mice, SCID; Microsomes, Liver; Molecular Structure; Oxidoreductases Acting on CH-CH Group Donors; Parasitic Sensitivity Tests; Plasmodium falciparum; Plasmodium vivax; Protein Binding; Pyrroles; Rats; Structure-Activity Relationship

2020
Host-based Prophylaxis Successfully Targets Liver Stage Malaria Parasites.
    Molecular therapy : the journal of the American Society of Gene Therapy, 2015, Volume: 23, Issue:5

    Topics: Animals; Antimalarials; Cell Line; Disease Models, Animal; Female; Imidazoles; Indoles; Life Cycle Stages; Liver; Malaria; Malaria, Falciparum; Mice; Mice, Transgenic; Parasite Load; Piperazines; Plasmodium; Plasmodium falciparum; Post-Exposure Prophylaxis; Proto-Oncogene Proteins c-bcl-2; Pyrroles; Tumor Suppressor Protein p53

2015
Statins alone are ineffective in cerebral malaria but potentiate artesunate.
    Antimicrobial agents and chemotherapy, 2008, Volume: 52, Issue:11

    Topics: Animals; Antimalarials; Artemisinins; Artesunate; Atorvastatin; Disease Models, Animal; Drug Synergism; Fatty Acids, Monounsaturated; Fluvastatin; Heptanoic Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Indoles; Malaria, Cerebral; Malaria, Falciparum; Mice; Neuroprotective Agents; Pravastatin; Pyrroles; Simvastatin

2008
Atorvastatin as a potential anti-malarial drug: in vitro synergy in combinational therapy with quinine against Plasmodium falciparum.
    Malaria journal, 2010, May-25, Volume: 9

    Topics: Antimalarials; Atorvastatin; ATP-Binding Cassette Transporters; Drug Resistance; Drug Synergism; Gene Dosage; Genetic Variation; Genotype; Heptanoic Acids; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Inhibitory Concentration 50; Malaria, Falciparum; Membrane Transport Proteins; Multidrug Resistance-Associated Proteins; Mutation; Parasitic Sensitivity Tests; Plasmodium falciparum; Protozoan Proteins; Pyrroles; Quinine

2010
Development of antitrypanosomal and antiplasmodial nonpeptidic cysteine protease inhibitors based on N-protected-guanidino-furan and -pyrrole building blocks.
    ChemMedChem, 2011, Sep-05, Volume: 6, Issue:9

    Topics: Animals; Antimalarials; Cysteine Proteinase Inhibitors; Furans; Guanidines; Humans; Malaria, Falciparum; Plasmodium falciparum; Pyrroles; Structure-Activity Relationship; Trypanocidal Agents; Trypanosoma brucei brucei; Trypanosomiasis

2011
In vitro antimalarial activity of retinoids and the influence of selective retinoic acid receptor antagonists.
    Acta tropica, 2003, Volume: 87, Issue:3

    Topics: Animals; Anthracenes; Antimalarials; Benzoates; Chromans; Drug Interactions; Hypoxanthine; Inhibitory Concentration 50; Malaria, Falciparum; Plasmodium falciparum; Pyrroles; Receptors, Retinoic Acid; Retinoids; Tretinoin; Vitamin A

2003
Atorvastatin is 10-fold more active in vitro than other statins against Plasmodium falciparum.
    Antimicrobial agents and chemotherapy, 2007, Volume: 51, Issue:7

    Topics: Animals; Antimalarials; Atorvastatin; Dose-Response Relationship, Drug; Heptanoic Acids; Hydroxymethylglutaryl-CoA Reductase Inhibitors; In Vitro Techniques; Inhibitory Concentration 50; Malaria, Falciparum; Microbial Sensitivity Tests; Plasmodium falciparum; Pyrroles; Structure-Activity Relationship

2007