Page last updated: 2024-08-21

pyrimidine and Angiogenesis, Pathologic

pyrimidine has been researched along with Angiogenesis, Pathologic in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (25.00)29.6817
2010's1 (25.00)24.3611
2020's2 (50.00)2.80

Authors

AuthorsStudies
Bhandari, S; Bhargava, SK; Reddy, TS; Reddy, VG; Sakla, AP; Sana, S; Shankaraiah, N; Tokala, R1
Cui, DB; Guan, HY; Li, YJ; Liao, SG; Liu, T; Wang, S; Wang, YC; Xu, GB; Yan, GY; Yang, D; Zhang, H; Zhang, RH; Zhao, YL; Zhou, M; Zhou, YH1
Kim, D; Kwon, A; Lee, BY; Min, KH; Nguyen, HK; Song, J; Suh, W; Yoo, J1
Buttar, D; Edge, M; Emery, SC; Fitzek, M; Forder, C; Griffen, A; Hayter, B; Hayward, CF; Hopcroft, PJ; Luke, RW; Page, K; Stawpert, J; Wright, A1

Other Studies

4 other study(ies) available for pyrimidine and Angiogenesis, Pathologic

ArticleYear
Exploration of carbamide derived pyrimidine-thioindole conjugates as potential VEGFR-2 inhibitors with anti-angiogenesis effect.
    European journal of medicinal chemistry, 2020, Aug-15, Volume: 200

    Topics: Angiogenesis Inhibitors; Antineoplastic Agents; Cell Proliferation; Cell Survival; Dose-Response Relationship, Drug; Drug Screening Assays, Antitumor; Humans; Indoles; Molecular Structure; Neovascularization, Pathologic; Protein Kinase Inhibitors; Pyrimidines; Structure-Activity Relationship; Tumor Cells, Cultured; Urea; Vascular Endothelial Growth Factor Receptor-2

2020
Design, synthesis, and biological evaluation of 2,4-diamino pyrimidine derivatives as potent FAK inhibitors with anti-cancer and anti-angiogenesis activities.
    European journal of medicinal chemistry, 2021, Oct-15, Volume: 222

    Topics: Angiogenesis Inhibitors; Antineoplastic Agents; Cell Proliferation; Cells, Cultured; Dose-Response Relationship, Drug; Drug Design; Drug Screening Assays, Antitumor; Focal Adhesion Kinase 1; Humans; Molecular Structure; Neovascularization, Pathologic; Protein Kinase Inhibitors; Pyrimidines; Structure-Activity Relationship

2021
Structure-Activity Relationship of Indole-Tethered Pyrimidine Derivatives that Concurrently Inhibit Epidermal Growth Factor Receptor and Other Angiokinases.
    PloS one, 2015, Volume: 10, Issue:9

    Topics: Angiogenesis Inhibitors; Carcinoma, Non-Small-Cell Lung; Cell Proliferation; ErbB Receptors; Human Umbilical Vein Endothelial Cells; Humans; Indazoles; Indoles; Inhibitory Concentration 50; Lung Neoplasms; Molecular Docking Simulation; Neovascularization, Pathologic; Protein Kinase Inhibitors; Protein Kinases; Pyrimidines; Structure-Activity Relationship; Sulfonamides; Vascular Endothelial Growth Factor A

2015
Discovery of imidazole vinyl pyrimidines as a novel class of kinase inhibitors which inhibit Tie-2 and are orally bioavailable.
    Bioorganic & medicinal chemistry letters, 2008, Aug-15, Volume: 18, Issue:16

    Topics: Administration, Oral; Biological Availability; Chemistry, Pharmaceutical; Drug Design; Humans; Imidazoles; Inhibitory Concentration 50; Models, Chemical; Molecular Conformation; Neovascularization, Pathologic; Protein Kinase Inhibitors; Pyrimidines; Receptor, TIE-2; Structure-Activity Relationship

2008