Page last updated: 2024-08-21

pyrazines and Malaria

pyrazines has been researched along with Malaria in 14 studies

Research

Studies (14)

TimeframeStudies, this research(%)All Research%
pre-199011 (78.57)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's2 (14.29)24.3611
2020's1 (7.14)2.80

Authors

AuthorsStudies
Ospina-Villa, JD; Soto-Sánchez, J1
Borboa, R; Campo, B; Chatterjee, AK; Chen, Z; Diagana, TT; Gagaring, K; Glynne, RJ; Klooster, EJ; Kocken, CH; Kuhen, K; Leroy, D; Luty, A; McNamara, CW; Nagle, A; Plouffe, DM; Remarque, EJ; Roland, J; Sauerwein, R; Thomas, AW; van Amsterdam, SM; van den Berg, A; van Gemert, GJ; Voorberg-van der Wel, A; Winzeler, EA; Yeung, BK; Zeeman, AM1
Angulo-Barturen, I; Antonova-Koch, Y; Bashyam, S; Birkholtz, LM; Botha, ME; Charman, SA; Chibale, K; Ferrer, S; Gonzàlez Cabrera, D; Han, Z; Jiménez-Díaz, MB; Lawrence, N; Le Manach, C; Martínez, MS; Meister, S; Nchinda, AT; Nondaba, SH; Paquet, T; Reader, J; Street, LJ; Taylor, D; Waterson, D; White, KL; Winzeler, EA; Wittlin, S; Witty, MJ; Younis, Y; Zabiulla, M1
Carson, PE; Frischer, H; Rieckmann, KH; Trenholme, GM; Williams, RL1
Bowman, JE; Carson, PE; Frischer, H; Kass, L; Richard, L; Rieckmann, KH; Willerson, D1
Colwell, EJ1
Clyde, DF; McCarthy, VC1
Brogger, S; Duby, C; Gramiccia, G; Lietaert, P; Mandel, SP; Matsushima, T; Rossi-Espagnet, A; Storey, J; Thomas, D1
Clyde, DF1
Clyde, DF; DuPont, HL; Hornick, RB; Miller, RM1
Canfield, CJ; Hall, WH; MacDonald, BS; Whiting, EG1
Clyde, DF; Levine, MM; Miller, RM; Schwartz, AR1
Jacobus, DP; Rothe, WE; Walter, WG1
Peters, W1

Reviews

2 review(s) available for pyrazines and Malaria

ArticleYear
Current status of quinoxaline and quinoxaline 1,4-di-N-oxides derivatives as potential antiparasitic agents.
    Chemical biology & drug design, 2021, Volume: 98, Issue:4

    Topics: Animals; Antiparasitic Agents; Benzene; Chagas Disease; Humans; Leishmaniasis; Malaria; Oxidation-Reduction; Oxides; Pyrazines; Quinoxalines; Structure-Activity Relationship

2021
A review of the drug sensitivity of Plasmodium falciparum in Thailand.
    The Southeast Asian journal of tropical medicine and public health, 1972, Volume: 3, Issue:2

    Topics: Chloroquine; Drug Resistance; Geography; Humans; Malaria; Methylamines; Naphthacenes; Plasmodium falciparum; Pyrazines; Pyrimethamine; Pyrimidines; Quinine; Sulfamethoxazole; Sulfonamides; Tetracycline; Thailand; Trimethoprim

1972

Trials

1 trial(s) available for pyrazines and Malaria

ArticleYear
Sulfalene with pyrimethamine and chloroquine with pyrimethamine in single-dose treatment of Plasmodium falciparum infections. A trial in a rural population in northern Nigeria.
    Bulletin of the World Health Organization, 1973, Volume: 49, Issue:3

    Topics: Adult; Antimalarials; Child; Child, Preschool; Chloroquine; Drug Combinations; Humans; Infant; Malaria; Nigeria; Plasmodium falciparum; Pyrazines; Pyrimethamine; Rural Health; Sulfanilamides

1973

Other Studies

11 other study(ies) available for pyrazines and Malaria

ArticleYear
KAI407, a potent non-8-aminoquinoline compound that kills Plasmodium cynomolgi early dormant liver stage parasites in vitro.
    Antimicrobial agents and chemotherapy, 2014, Volume: 58, Issue:3

    Topics: Animals; Antimalarials; Drug Evaluation, Preclinical; Female; Hepatocytes; Imidazoles; In Vitro Techniques; Liver; Macaca mulatta; Malaria; Mice; Mice, Inbred ICR; Plasmodium cynomolgi; Pyrazines; Sporozoites

2014
Identification of a Potential Antimalarial Drug Candidate from a Series of 2-Aminopyrazines by Optimization of Aqueous Solubility and Potency across the Parasite Life Cycle.
    Journal of medicinal chemistry, 2016, 11-10, Volume: 59, Issue:21

    Topics: Animals; Antimalarials; Disease Models, Animal; Dose-Response Relationship, Drug; Ether-A-Go-Go Potassium Channels; Hep G2 Cells; Humans; Life Cycle Stages; Malaria; Mice; Mice, SCID; Microsomes, Liver; Molecular Structure; Parasitic Diseases, Animal; Parasitic Sensitivity Tests; Plasmodium berghei; Plasmodium falciparum; Pyrazines; Solubility; Structure-Activity Relationship; Water

2016
Host failure in treatment of malaria with sulfalene and pyrimethamine.
    Annals of internal medicine, 1975, Volume: 82, Issue:2

    Topics: Adult; Amodiaquine; Drug Resistance; Drug Therapy, Combination; Erythrocytes; Humans; Malaria; Male; Phenotype; Plasmodium falciparum; Pyrazines; Pyrimethamine; Sulfanilamides; Sulfonamides; Tetracycline

1975
Chemotherapeutic results in a multi-drug resistant strain of Plasmodium falciparum malaria from Vietnam.
    Military medicine, 1974, Volume: 139, Issue:3

    Topics: Adult; Alanine Transaminase; Anopheles; Antimalarials; Aspartate Aminotransferases; Dapsone; Drug Resistance, Microbial; Drug Therapy, Combination; Humans; Malaria; Male; Methylamines; Military Medicine; Phenanthrenes; Plasmodium falciparum; Pyrazines; Pyrimethamine; Quinine; Sulfanilamides; Trimethoprim; Vietnam

1974
Influence of sulfalene upon gametocytogenesis of Plasmodium falciparum and subsequent infection patterns in Anopheles stephensi.
    Experimental parasitology, 1973, Volume: 33, Issue:1

    Topics: Anopheles; Antimalarials; Drug Resistance, Microbial; Humans; Malaria; Male; Plasmodium falciparum; Pyrazines; Quinine; Sulfonamides

1973
Sulfalene and trimethoprim in acute falciparum malaria.
    JAMA, 1969, Jul-28, Volume: 209, Issue:4

    Topics: Aniline Compounds; Folic Acid Antagonists; Humans; Malaria; Plasmodium falciparum; Pyrazines; Pyrimidines; Quinine

1969
Treatment of falciparum malaria caused by strain resistant to quinine.
    JAMA, 1970, Sep-21, Volume: 213, Issue:12

    Topics: Adult; Aniline Compounds; Drug Resistance, Microbial; Humans; Malaria; Male; Plasmodium falciparum; Pyrazines; Quinine; United States; Vietnam

1970
Treatment of acute falciparum malaria from Vietnam with trimethoprim and sulfalene.
    The American journal of tropical medicine and hygiene, 1971, Volume: 20, Issue:4

    Topics: Acute Disease; Administration, Oral; Antimalarials; Folic Acid Antagonists; Humans; Malaria; Military Medicine; Plasmodium falciparum; Pyrazines; Pyrimidines; Sulfonamides; United States; Vietnam

1971
Treatment of falciparum malaria with sulfalene and trimethoprim.
    The American journal of tropical medicine and hygiene, 1971, Volume: 20, Issue:6

    Topics: Adult; Anti-Infective Agents; Antimalarials; Drug Combinations; Drug Resistance, Microbial; Folic Acid Antagonists; Humans; Malaria; Male; Plasmodium falciparum; Pyrazines; Pyrimidines; Sulfonamides; Time Factors; Trimethoprim

1971
Treatment of trophozoite-induced Plasmodium knowlesi infection in the rhesus monkey with Trimethoprim and sulfalene.
    The American journal of tropical medicine and hygiene, 1969, Volume: 18, Issue:4

    Topics: Aniline Compounds; Animals; Antimalarials; Drug Synergism; Folic Acid Antagonists; Haplorhini; Malaria; Plasmodium; Pyrazines; Pyrimidines

1969
Potentiating action of sulfalene-pyrimethamine mixtures against drug-resistant strains of Plasmodium berghei.
    Chemotherapy, 1971, Volume: 16, Issue:6

    Topics: Animals; Drug Combinations; Drug Resistance, Microbial; Drug Synergism; Injections, Intraperitoneal; Malaria; Male; Mice; Mice, Inbred Strains; Plasmodium; Pyrazines; Pyrimethamine; Sulfamethoxypyridazine; Sulfonamides; Time Factors

1971