Page last updated: 2024-08-21

pyrazines and Androgen-Independent Prostatic Cancer

pyrazines has been researched along with Androgen-Independent Prostatic Cancer in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's4 (100.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Butler, LM; Castillo, L; Centenera, MM; Daly, RJ; Grogan, J; Haynes, AM; Horvath, LG; Kench, JG; Lee, BY; Lin, HM; Shreeve, SM; Spielman, C; Stricker, PD; Yeung, NK1
Barata, P; Cooney, M; Dreicer, R; Garcia, JA; Tyler, A; Wright, J1
Kuna, M; Mikecin, AM; Raucher, D; Walker, LR1
Franco, OE; Hayward, SW; Jin, R; Matusik, RJ; Wang, J; Wang, Y; Yamashita, H; Yu, X1

Trials

1 trial(s) available for pyrazines and Androgen-Independent Prostatic Cancer

ArticleYear
A phase 2 study of OSI-906 (linsitinib, an insulin-like growth factor receptor-1 inhibitor) in patients with asymptomatic or mildly symptomatic (non-opioid requiring) metastatic castrate resistant prostate cancer (CRPC).
    Investigational new drugs, 2018, Volume: 36, Issue:3

    Topics: Aged; Endothelial Cells; Humans; Imidazoles; Male; Middle Aged; Neoplasm Metastasis; Neoplastic Cells, Circulating; Prostate-Specific Antigen; Prostatic Neoplasms, Castration-Resistant; Pyrazines; Receptor, IGF Type 1; Receptors, Somatomedin

2018

Other Studies

3 other study(ies) available for pyrazines and Androgen-Independent Prostatic Cancer

ArticleYear
Effect of FAK inhibitor VS-6063 (defactinib) on docetaxel efficacy in prostate cancer.
    The Prostate, 2018, Volume: 78, Issue:4

    Topics: Animals; Antineoplastic Agents; Apoptosis; Benzamides; Cell Count; Cell Line, Tumor; Cell Proliferation; Cell Survival; Docetaxel; Drug Resistance, Neoplasm; Focal Adhesion Kinase 1; Humans; Immunoblotting; Immunohistochemistry; Male; Mice; Prostate; Prostatic Neoplasms, Castration-Resistant; Pyrazines; Sulfonamides; Xenograft Model Antitumor Assays

2018
Thermally targeted p21 peptide enhances bortezomib cytotoxicity in androgen-independent prostate cancer cell lines.
    Anti-cancer drugs, 2014, Volume: 25, Issue:2

    Topics: Androgens; Antineoplastic Agents; Apoptosis; Boronic Acids; Bortezomib; Cell Cycle Checkpoints; Cell Proliferation; Cyclin-Dependent Kinase Inhibitor p21; Drug Synergism; Hot Temperature; Humans; Male; Molecular Mimicry; Peptides; Prostatic Neoplasms, Castration-Resistant; Protein Engineering; Pyrazines; Recombinant Fusion Proteins; Tumor Cells, Cultured

2014
Inhibition of NF-kappa B signaling restores responsiveness of castrate-resistant prostate cancer cells to anti-androgen treatment by decreasing androgen receptor-variant expression.
    Oncogene, 2015, Volume: 34, Issue:28

    Topics: Androgen Antagonists; Anilides; Antineoplastic Agents; Antineoplastic Combined Chemotherapy Protocols; Boronic Acids; Bortezomib; Cell Line, Tumor; Humans; Male; NF-kappa B; Nitriles; Prostatic Neoplasms, Castration-Resistant; Pyrazines; Receptors, Androgen; Signal Transduction; Tosyl Compounds; Xenograft Model Antitumor Assays

2015