Page last updated: 2024-08-21

podophyllotoxin and Malaria, Falciparum

podophyllotoxin has been researched along with Malaria, Falciparum in 7 studies

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's0 (0.00)29.6817
2010's6 (85.71)24.3611
2020's1 (14.29)2.80

Authors

AuthorsStudies
Brun, R; Carballeira, NM; Herman, R; Kappe, SH; Lauinger, IL; Perozzo, R; Sanabria, D; Tarun, A; Tasdemir, D; Zloh, M1
Brun, R; Huang, TL; Kaiser, M; Mayence, A; Vanden Eynde, JJ; Yarlett, N1
Amewu, RK; Burrell-Saward, H; Chadwick, J; Hussain, A; Janneh, O; Miguel, C; O'Neill, PM; Panda, S; Rinki, R; Vivas, L; Ward, SA1
Brun, R; Göker, H; Kaiser, M; Karaaslan, C1
Aponte, RA; Bonnert, R; Chaiyen, P; Charman, SA; Chitnumsub, P; Diederich, F; Freiberg, GM; Ittarat, W; Jaruwat, A; Kundu, A; Leartsakulpanich, U; Lloyd, M; Rottmann, M; Sadhukhan, S; Schäfer, A; Schwertz, G; Siggel, M; Srikumaran, M; White, KL; Witschel, MC; Zwyssig, A1
Brun, R; Calvet, CM; Costi, R; De Leo, A; De Vita, D; Di Santo, R; Jennings, GK; Kaiser, M; Madia, VN; Mäser, P; Messore, A; Pescatori, L; Podust, LM; Saccoliti, F; Scipione, L; Tudino, V1
Horiuchi, M; Ihara, M; Ikegami-Kawai, M; Itoh, I; Kaiser, M; Kojima, M; Miyagi, S; Mizukawa, Y; Nanga Chick, C; Sakanoue, S; Togashi, H; Tsubuki, M; Usuki, T1

Reviews

1 review(s) available for podophyllotoxin and Malaria, Falciparum

ArticleYear
Quest for a potent antimalarial drug lead: Synthesis and evaluation of 6,7-dimethoxyquinazoline-2,4-diamines.
    Bioorganic & medicinal chemistry, 2021, 03-01, Volume: 33

    Topics: Animals; Antimalarials; Dose-Response Relationship, Drug; Drug Discovery; Female; Malaria, Falciparum; Mice; Mice, Inbred ICR; Molecular Structure; Parasitic Sensitivity Tests; Plasmodium falciparum; Structure-Activity Relationship

2021

Other Studies

6 other study(ies) available for podophyllotoxin and Malaria, Falciparum

ArticleYear
2-Hexadecynoic acid inhibits plasmodial FAS-II enzymes and arrests erythrocytic and liver stage Plasmodium infections.
    Bioorganic & medicinal chemistry, 2010, Nov-01, Volume: 18, Issue:21

    Topics: Alkynes; Antimalarials; Binding Sites; Cell Line, Tumor; Computer Simulation; Erythrocytes; Fatty Acid Synthase, Type II; Fatty Acids, Unsaturated; Humans; Kinetics; Liver; Malaria, Falciparum; Plasmodium falciparum; Protozoan Proteins

2010
Bis(oxyphenylene)benzimidazoles: a novel class of anti-Plasmodium falciparum agents.
    Bioorganic & medicinal chemistry, 2011, Dec-15, Volume: 19, Issue:24

    Topics: Animals; Antimalarials; Benzimidazoles; Cell Line; Humans; Inhibitory Concentration 50; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats

2011
Synthesis and evaluation of the antimalarial, anticancer, and caspase 3 activities of tetraoxane dimers.
    Bioorganic & medicinal chemistry, 2013, Dec-01, Volume: 21, Issue:23

    Topics: Antimalarials; Antineoplastic Agents; Caspase 3; Cell Line, Tumor; Dimerization; Humans; Malaria, Falciparum; Neoplasms; Plasmodium falciparum; Tetraoxanes

2013
Synthesis and potent antiprotozoal activity of mono/di amidino 2-anilinobenzimidazoles versus Plasmodium falciparum and Trypanosoma brucei rhodesiense.
    Bioorganic & medicinal chemistry, 2016, 09-15, Volume: 24, Issue:18

    Topics: Aniline Compounds; Animals; Antiprotozoal Agents; Benzimidazoles; Cell Line; Humans; Malaria, Falciparum; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosomiasis, African

2016
Antimalarial Inhibitors Targeting Serine Hydroxymethyltransferase (SHMT) with in Vivo Efficacy and Analysis of their Binding Mode Based on X-ray Cocrystal Structures.
    Journal of medicinal chemistry, 2017, 06-22, Volume: 60, Issue:12

    Topics: Animals; Antimalarials; Arabidopsis Proteins; Chemistry Techniques, Synthetic; Crystallography, X-Ray; Cysteine; Drug Stability; Enzyme Inhibitors; Glycine Hydroxymethyltransferase; Half-Life; Ligands; Malaria, Falciparum; Mice, SCID; Plasmodium falciparum; Plasmodium vivax; Protein Conformation; Rats; Structure-Activity Relationship; Thiophenes

2017
Biological evaluation and structure-activity relationships of imidazole-based compounds as antiprotozoal agents.
    European journal of medicinal chemistry, 2018, Aug-05, Volume: 156

    Topics: Animals; Antiprotozoal Agents; Cell Line; Chagas Disease; Female; Humans; Imidazoles; Inhibitory Concentration 50; Leishmania donovani; Leishmaniasis, Visceral; Malaria, Falciparum; Mice; Mice, Inbred BALB C; Parasitic Sensitivity Tests; Plasmodium falciparum; Rats; Structure-Activity Relationship; Trypanosoma brucei rhodesiense; Trypanosoma cruzi; Trypanosomiasis, African

2018