Page last updated: 2024-10-21

pk 11195 and Allergic Encephalomyelitis

pk 11195 has been researched along with Allergic Encephalomyelitis in 4 studies

PK-11195 : A monocarboxylic acid amide obtained by formal condensation of the carboxy group of 1-(2-chlorophenyl)isoquinoline-3-carboxylic acid with the amino group of sec-butylmethylamine

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (25.00)18.2507
2000's2 (50.00)29.6817
2010's1 (25.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Abourbeh, G1
Thézé, B1
Maroy, R1
Dubois, A1
Brulon, V1
Fontyn, Y1
Dollé, F1
Tavitian, B1
Boisgard, R1
Vowinckel, E1
Reutens, D1
Becher, B1
Verge, G1
Evans, A1
Owens, T1
Antel, JP1
Agnello, D1
Carvelli, L1
Muzio, V1
Villa, P1
Bottazzi, B1
Polentarutti, N1
Mennini, T1
Mantovani, A1
Ghezzi, P1
Banati, RB1
Newcombe, J1
Gunn, RN1
Cagnin, A1
Turkheimer, F1
Heppner, F1
Price, G1
Wegner, F1
Giovannoni, G1
Miller, DH1
Perkin, GD1
Smith, T1
Hewson, AK1
Bydder, G1
Kreutzberg, GW1
Jones, T1
Cuzner, ML1
Myers, R1

Clinical Trials (5)

Trial Overview

TrialPhaseEnrollmentStudy TypeStart DateStatus
Brain Inflammation In Major Depressive Disorder[NCT01851356]61 participants (Actual)Observational2013-05-08Completed
Assessment of [11C]ER-176 to Image Translocator Protein in Brain and Whole-Body of Healthy Subjects[NCT02147392]Early Phase 116 participants (Actual)Interventional2014-05-14Completed
Assessment of [11C]DPA-713 in Temporal Lobe Epilepsy[NCT01793532]38 participants (Actual)Observational2013-01-31Completed
Molecular Imaging Modality by Positron Emission Tomography Using 18F-X : Study of Microglial Activation in Amyotrophic Lateral Sclerosis[NCT00563537]Phase 130 participants (Anticipated)Interventional2007-01-31Recruiting
PET Imaging of Peripheral Benzodiazepine Receptors Using [11C](R)-PK 11195 and [11C]PBR28[NCT00696371]15 participants (Actual)Observational2008-06-06Completed
[information is prepared from clinicaltrials.gov, extracted Sep-2024]

Other Studies

4 other studies available for pk 11195 and Allergic Encephalomyelitis

ArticleYear
Imaging microglial/macrophage activation in spinal cords of experimental autoimmune encephalomyelitis rats by positron emission tomography using the mitochondrial 18 kDa translocator protein radioligand [¹⁸F]DPA-714.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2012, Apr-25, Volume: 32, Issue:17

    Topics: Animals; Antigens, CD; Carrier Proteins; Disease Models, Animal; Encephalomyelitis, Autoimmune, Expe

2012
PK11195 binding to the peripheral benzodiazepine receptor as a marker of microglia activation in multiple sclerosis and experimental autoimmune encephalomyelitis.
    Journal of neuroscience research, 1997, Oct-15, Volume: 50, Issue:2

    Topics: Animals; Biomarkers; Brain; Encephalomyelitis, Autoimmune, Experimental; Humans; Isoquinolines; Magn

1997
Increased peripheral benzodiazepine binding sites and pentraxin 3 expression in the spinal cord during EAE: relation to inflammatory cytokines and modulation by dexamethasone and rolipram.
    Journal of neuroimmunology, 2000, Sep-22, Volume: 109, Issue:2

    Topics: Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; C-Reactive Protein; Dexamethasone; E

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000
The peripheral benzodiazepine binding site in the brain in multiple sclerosis: quantitative in vivo imaging of microglia as a measure of disease activity.
    Brain : a journal of neurology, 2000, Volume: 123 ( Pt 11)

    Topics: Adult; Animals; Antineoplastic Agents; Benzodiazepines; Binding Sites; Brain; Carbon Radioisotopes;

2000