Compounds > piperidine
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piperidine and Pain

piperidine has been researched along with Pain in 5 studies

Research

Studies (5)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's2 (40.00)29.6817
2010's3 (60.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Journigan, VB; Khroyan, TV; Polgar, WE; Zaveri, NT1
Albrecht, C; Bartolozzi, A; Berry, AK; Ceci, A; Cirillo, PF; Gemkow, MJ; Hickey, ER; Nagaraja, NV; Riether, D; Romig, H; Sauer, A; Thomson, DS; Wu, L; Zindell, R1
Diaz, JL; Holenz, J; Oberdorf, C; Schepmann, D; Vela, JM; Wünsch, B1
Ahn, K; Beidler, D; Bhattacharya, K; Cravatt, BF; Johnson, DS; Kamtekar, S; Lazerwith, S; Liimatta, M; Long, JZ; McKinney, MK; Mileni, M; Sadagopan, N; Smith, SE; Stevens, RC; Stiff, C; Swaney, S; Van Becelaere, K; Weerapana, E; Zhang, Y1
Bennett, C; Bridal, T; Burnett, DA; Correll, CC; Czarniecki, M; Dong, Z; Greenlee, WJ; Jia, YP; Kieselgof, J; Kim, HM; Knutson, C; McKittrick, BA; Mullins, D; Nechuta, TL; Priestley, T; Rindgen, D; Smith, EM; Sorota, S; Tan, Z; Tulshian, D; Zhang, X; Zhou, X1

Other Studies

5 other study(ies) available for piperidine and Pain

ArticleYear
Designing bifunctional NOP receptor-mu opioid receptor ligands from NOP-receptor selective scaffolds. Part II.
    Bioorganic & medicinal chemistry, 2014, Apr-15, Volume: 22, Issue:8

    Topics: Analgesics; Animals; Ligands; Mice; Models, Animal; Nociceptin Receptor; Pain; Piperidines; Protein Binding; Receptors, Opioid; Receptors, Opioid, mu; Structure-Activity Relationship

2014
Selective CB2 receptor agonists. Part 3: the optimization of a piperidine-based series that demonstrated efficacy in an in vivo neuropathic pain model.
    Bioorganic & medicinal chemistry letters, 2015, Feb-01, Volume: 25, Issue:3

    Topics: Animals; Diabetic Neuropathies; Half-Life; Humans; Ligands; Male; Microsomes, Liver; Pain; Pipecolic Acids; Piperidines; Protein Binding; Rats; Rats, Wistar; Receptor, Cannabinoid, CB1; Receptor, Cannabinoid, CB2; Solubility; Structure-Activity Relationship; Thiazines

2015
Thiophene bioisosteres of spirocyclic sigma receptor ligands. 1. N-substituted spiro[piperidine-4,4'-thieno[3,2-c]pyrans].
    Journal of medicinal chemistry, 2008, Oct-23, Volume: 51, Issue:20

    Topics: Alkylation; Animals; Cyclization; Ligands; Mice; Models, Molecular; Molecular Structure; Oxidation-Reduction; Pain; Piperidines; Protein Binding; Pyrans; Rats; Receptors, sigma; Spiro Compounds; Structure-Activity Relationship; Thiophenes

2008
Discovery and characterization of a highly selective FAAH inhibitor that reduces inflammatory pain.
    Chemistry & biology, 2009, Apr-24, Volume: 16, Issue:4

    Topics: Amidohydrolases; Animals; Arachidonic Acids; Brain; Crystallography, X-Ray; Endocannabinoids; Enzyme Inhibitors; Humans; Male; Pain; Piperazine; Piperazines; Piperidines; Polyunsaturated Alkamides; Rats; Rats, Sprague-Dawley; Receptors, Cannabinoid; Structure-Activity Relationship; Urea

2009
T-type calcium channel blockers: spiro-piperidine azetidines and azetidinones-optimization, design and synthesis.
    Bioorganic & medicinal chemistry letters, 2010, Aug-01, Volume: 20, Issue:15

    Topics: Animals; Azetidines; Calcium Channel Blockers; Calcium Channels, T-Type; Drug Design; Humans; Pain; Piperidines; Protein Binding; Rats; Spiro Compounds; Structure-Activity Relationship

2010