Page last updated: 2024-08-18

piperidine and Disease Models, Animal

piperidine has been researched along with Disease Models, Animal in 11 studies

Research

Studies (11)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's1 (9.09)18.2507
2000's2 (18.18)29.6817
2010's7 (63.64)24.3611
2020's1 (9.09)2.80

Authors

AuthorsStudies
Chen, Y; Gao, L; Hao, C; Jin, J; Liu, BF; Liu, X; Xiong, J; Zhang, G1
Ahmad Bhat, M; Al-Omar, MA; Naglah, AM1
Barnes, KD; Blaner, WS; Chen, P; Cioffi, CL; Conlon, MP; Freeman, EE; Johnson, G; Kitchen, DB; Martin, WH; Pearson, PG; Petrukhin, K; Racz, B; Varadi, A; Zhu, L1
Chiba, K; Fujimoto, T; Inoue, S; Miyazaki, S; Mochizuki, A; Mori, Y; Nagai, Y; Nagayama, T; Nakamura, Y; Nishi, T; Ogawa, Y; Sugita, C; Tamaki, K1
Bhosale, VM; Chaudhari, SS; Gudi, GS; Kadam, AB; Karnik, PV; Khairatkar-Joshi, N; Mukhopadhyay, I; Raghuram, A; Rao, SS; Sangana, RR; Thomas, A; Vaiyapuri, TS; Wale, DP1
Gogineni, A; Hanson, JE; Herrington, J; Meilandt, WJ; Reynen, P; Scearce-Levie, K; Weimer, RM; Zhou, Q1
Beretta, EE; Cameron, KO; Chen, Y; Chu-Moyer, M; Fernando, D; Gao, H; Gautreau, D; Guzman-Perez, A; Hadcock, JR; Hoth, C; Jardine, Pda S; Kohrt, J; Lavergne, S; Makowski, M; Perez, S; Perry, DA; Polivkova, J; Rogers, L; Scott, DO; Swick, AG; Thiede, L; Trebino, CE; Trilles, RV; Wilmowski, J; Zhang, Y1
Chen, Y; Liu, BF; Liu, X; Xu, X; Zhang, G1
Ahmad, FJ; Ali, MM; Aqil, M; Chowdhary, I; Sultana, Y; Talegaonkar, S1
Aritake, K; Hayashi, K; Hayashi, M; Hirotsu, I; Hizue, M; Kimura, Y; Matsushita, N; Mitsui, K; Nakajima, H; Takada, A; Tani, T1
Hasegawa, S; Hirota, TK; Komoto, T; Kotake, J; Koya, H; Otsuka, M; Sakamoto, T; Sato, S1

Other Studies

11 other study(ies) available for piperidine and Disease Models, Animal

ArticleYear
Piperidine propionamide as a scaffold for potent sigma-1 receptor antagonists and mu opioid receptor agonists for treating neuropathic pain.
    European journal of medicinal chemistry, 2020, Apr-01, Volume: 191

    Topics: Amides; Animals; Disease Models, Animal; Dose-Response Relationship, Drug; Formaldehyde; Guinea Pigs; Injections, Subcutaneous; Mice; Mice, Inbred ICR; Molecular Structure; Neuralgia; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Opioid, mu; Receptors, sigma; Sciatic Nerve; Sigma-1 Receptor; Structure-Activity Relationship

2020
Synthesis and in vivo anti-ulcer evaluation of some novel piperidine linked dihydropyrimidinone derivatives.
    Journal of enzyme inhibition and medicinal chemistry, 2018, Volume: 33, Issue:1

    Topics: Animals; Anti-Ulcer Agents; Crystallography, X-Ray; Disease Models, Animal; Dose-Response Relationship, Drug; Ethanol; Models, Molecular; Molecular Structure; Piperidines; Pyrimidinones; Rats; Rats, Wistar; Stomach Ulcer; Structure-Activity Relationship

2018
Design, Synthesis, and Preclinical Efficacy of Novel Nonretinoid Antagonists of Retinol-Binding Protein 4 in the Mouse Model of Hepatic Steatosis.
    Journal of medicinal chemistry, 2019, 06-13, Volume: 62, Issue:11

    Topics: Animals; Chemistry Techniques, Synthetic; Disease Models, Animal; Drug Design; Fatty Liver; Male; Mice; Piperidines; Rats; Retinol-Binding Proteins, Plasma; Tissue Distribution

2019
Synthesis and optimization of novel (3S,5R)-5-(2,2-dimethyl-5-oxo-4-phenylpiperazin-1-yl)piperidine-3-carboxamides as orally active renin inhibitors.
    Bioorganic & medicinal chemistry, 2013, Sep-15, Volume: 21, Issue:18

    Topics: Administration, Oral; Amides; Animals; Blood Pressure; Disease Models, Animal; Furosemide; Half-Life; Hypertension; Macaca fascicularis; Piperazines; Piperidines; Protease Inhibitors; Rats; Rats, Transgenic; Renin; Structure-Activity Relationship

2013
Synthesis and pharmacological evaluation of novel N-aryl-3,4-dihydro-1'H-spiro[chromene-2,4'-piperidine]-1'-carboxamides as TRPM8 antagonists.
    Bioorganic & medicinal chemistry, 2013, Nov-01, Volume: 21, Issue:21

    Topics: Administration, Oral; Amides; Analgesics; Animals; Disease Models, Animal; Half-Life; Male; Mice; Mice, Inbred C57BL; Neuralgia; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Spiro Compounds; Stereoisomerism; Structure-Activity Relationship; TRPM Cation Channels

2013
Chronic GluN2B antagonism disrupts behavior in wild-type mice without protecting against synapse loss or memory impairment in Alzheimer's disease mouse models.
    The Journal of neuroscience : the official journal of the Society for Neuroscience, 2014, Jun-11, Volume: 34, Issue:24

    Topics: Alzheimer Disease; Amyloid beta-Peptides; Amyloid beta-Protein Precursor; Animals; Attention Deficit and Disruptive Behavior Disorders; Behavior, Animal; Disease Models, Animal; Female; HEK293 Cells; Humans; In Vitro Techniques; Male; Maze Learning; Membrane Potentials; Memory Disorders; Mice; Mice, Inbred C57BL; Mice, Transgenic; Mutation; Piperidines; Synapses

2014
Discovery of new piperidine amide triazolobenzodiazepinones as intestinal-selective CCK1 receptor agonists.
    Bioorganic & medicinal chemistry letters, 2012, Apr-15, Volume: 22, Issue:8

    Topics: Amides; Animals; Cells, Cultured; Disease Models, Animal; Drug Discovery; Humans; Inhibitory Concentration 50; Male; Mice; Mice, Obese; Piperidines; Protein Binding; Rats; Rats, Sprague-Dawley; Receptor, Cholecystokinin A; Structure-Activity Relationship; Weight Loss

2012
Synthesis and evaluation of a series of piperidine-2,6-dione-piperazine (piperidine) derivatives as multireceptor atypical antipsychotics.
    Archiv der Pharmazie, 2012, Volume: 345, Issue:11

    Topics: Animals; Antipsychotic Agents; Apomorphine; Behavior, Animal; Clozapine; Disease Models, Animal; Dizocilpine Maleate; Mice; Piperidines; Rats; Rats, Sprague-Dawley; Receptors, Dopamine; Receptors, Histamine H1; Receptors, Serotonin; Structure-Activity Relationship

2012
Transdermal therapeutic system of enalapril maleate using piperidine as penetration enhancer.
    Current drug delivery, 2008, Volume: 5, Issue:2

    Topics: Acrylates; Administration, Cutaneous; Animals; Antihypertensive Agents; Biological Availability; Blood Pressure; Disease Models, Animal; Drug Stability; Drug Storage; Enalapril; Excipients; Female; Hypertension; Male; Permeability; Piperidines; Polymers; Povidone; Rats; Skin Absorption

2008
Pharmacological studies on the novel antiallergic drug HQL-79: I. Antiallergic and antiasthmatic effects in various experimental models.
    Japanese journal of pharmacology, 1998, Volume: 78, Issue:1

    Topics: Animals; Anti-Allergic Agents; Anti-Asthmatic Agents; Antigens; Bronchoconstriction; Capillary Permeability; Dibenzazepines; Disease Models, Animal; Dose-Response Relationship, Drug; Guinea Pigs; Histamine H1 Antagonists; Hypersensitivity, Delayed; Imidazoles; Ketotifen; Leukocytes; Male; Mice; Mice, Inbred ICR; Nasal Mucosa; Passive Cutaneous Anaphylaxis; Piperidines; Rats; Rats, Wistar; Respiratory Hypersensitivity

1998
New strong fibrates with piperidine moiety.
    Chemical & pharmaceutical bulletin, 2000, Volume: 48, Issue:12

    Topics: Animals; Disease Models, Animal; Hypercholesterolemia; Hypertriglyceridemia; Hypoglycemic Agents; Hypolipidemic Agents; Male; Mice; Mice, Inbred ICR; Piperazine; Piperazines; Piperidines; Propionates; Rats; Rats, Sprague-Dawley

2000