Page last updated: 2024-09-05

piboserod and Muscle Contraction

piboserod has been researched along with Muscle Contraction in 7 studies

*Muscle Contraction: A process leading to shortening and/or development of tension in muscle tissue. Muscle contraction occurs by a sliding filament mechanism whereby actin filaments slide inward among the myosin filaments. [MeSH]

Research

Studies (7)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's2 (28.57)18.2507
2000's5 (71.43)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Bingham, S; Ellis, ES; Gaster, LM; Joiner, GF; King, FD; Sanger, GJ; Sutton, JM; Wardle, KA; Wyman, PA1
Armstrong, SR; Beattie, DT; Humphrey, PP; Mai, N; Marquess, D; McCullough, JL; Pulido-Rios, T; Richardson, C; Sandlund, C; Smith, JA; Vickery, RG1
De Maeyer, JH; Lefebvre, RA; Schuurkes, JA1
Eda, H; Kimura, N; Komada, T; Mikami, T; Naganeo, R; Nakata, E; Nakatani, K; Ohmi, T; Sakakibara, M; Sugimoto, H; Suzuki, K; Toga, T1
Karaki, S; Kuwahara, A; Mitsui, R; Ono, S1
Becker, DP; Flynn, DL; Gullikson, GW; Loeffler, R; Moormann, AE; Moummi, C; Nosal, R; Villamil, CI; Yang, DC1
Bingham, S; Ellis, ES; Gaster, LM; Rushant, B; Sanger, GJ; Smith, MI; Wardle, KA1

Other Studies

7 other study(ies) available for piboserod and Muscle Contraction

ArticleYear
N-[(1-butyl-4-piperidinyl)methyl]-3,4dihydro-2H-[1,3]oxazino[3,2- a]indole10-carboxamide hydrochloride: the first potent and selective 5-HT4 receptor antagonist amide with oral activity.
    Journal of medicinal chemistry, 1995, Nov-24, Volume: 38, Issue:24

    Topics: Administration, Oral; Animals; Dioxanes; Dogs; Guinea Pigs; Indoles; Muscle Contraction; Piperidines; Receptors, Serotonin; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Structure-Activity Relationship; Sulfonamides

1995
The 5-HT4 receptor agonist, tegaserod, is a potent 5-HT2B receptor antagonist in vitro and in vivo.
    British journal of pharmacology, 2004, Volume: 143, Issue:5

    Topics: Animals; Cell Membrane; Cells, Cultured; Colon; Cyclic AMP; Esophagus; Gastric Fundus; Gastrointestinal Transit; Guinea Pigs; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Pressure; Protein Binding; Radioligand Assay; Rats; Rats, Sprague-Dawley; Receptor, Serotonin, 5-HT2B; Receptors, Serotonin, 5-HT4; Serotonin Antagonists; Serotonin Receptor Agonists

2004
Selective desensitization of the 5-HT4 receptor-mediated response in pig atrium but not in stomach.
    British journal of pharmacology, 2009, Volume: 156, Issue:2

    Topics: Animals; Atrial Function, Left; Benzofurans; Female; In Vitro Techniques; Models, Biological; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Organ Specificity; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Stomach; Swine; Synaptic Transmission; Tachyphylaxis

2009
In vitro and in vivo pharmacological characterization of PF-01354082, a novel partial agonist selective for the 5-HT(4) receptor.
    European journal of pharmacology, 2009, May-01, Volume: 609, Issue:1-3

    Topics: Administration, Oral; Animals; Benzimidazoles; Carbachol; Cell Line; CHO Cells; Cholinergic Agonists; Cricetinae; Cricetulus; Cyclic AMP; Dogs; Dose-Response Relationship, Drug; Esophagus; Gastrointestinal Motility; Humans; Indoles; Kidney; Male; Muscle Contraction; Muscle, Smooth; Piperidines; Rats; Rats, Inbred Strains; Sensitivity and Specificity; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Serotonin Receptor Agonists; Time Factors

2009
Muscarinic and 5-HT4 receptors participate in the regulation of the frequency of spontaneous contractions of the longitudinal muscle in rat distal colon.
    Biomedical research (Tokyo, Japan), 2005, Volume: 26, Issue:4

    Topics: Animals; Atropine; Colon; Dioxanes; Gastrointestinal Motility; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Piperidines; Rats; Rats, Wistar; Receptors, Muscarinic; Receptors, Serotonin, 5-HT4; Serotonin 5-HT4 Receptor Antagonists; Serotonin Antagonists

2005
Pyrrolizidine esters and amides as 5-HT4 receptor agonists and antagonists.
    Journal of medicinal chemistry, 2006, Feb-09, Volume: 49, Issue:3

    Topics: Amides; Animals; Benzamides; Bradycardia; Brain; Dogs; Esophagus; Esters; Female; Gastric Emptying; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Male; Mice; Muscle Contraction; Muscle, Smooth; Pyloric Antrum; Pyrroles; Pyrrolizidine Alkaloids; Radioligand Assay; Rats; Rats, Wistar; Serotonin 5-HT4 Receptor Agonists; Serotonin 5-HT4 Receptor Antagonists; Structure-Activity Relationship

2006
Selective and functional 5-hydroxytryptamine4 receptor antagonism by SB 207266.
    British journal of pharmacology, 1996, Volume: 118, Issue:3

    Topics: Animals; Benzimidazoles; Bridged Bicyclo Compounds, Heterocyclic; Colon; Dogs; Dose-Response Relationship, Drug; Guinea Pigs; Indoles; Male; Muscle Contraction; Piperidines; Serotonin; Serotonin Antagonists; Time Factors

1996