Page last updated: 2024-09-03

pd 142893 and Muscle Contraction

pd 142893 has been researched along with Muscle Contraction in 10 studies

*Muscle Contraction: A process leading to shortening and/or development of tension in muscle tissue. Muscle contraction occurs by a sliding filament mechanism whereby actin filaments slide inward among the myosin filaments. [MeSH]

Research

Studies (10)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's9 (90.00)18.2507
2000's1 (10.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Cody, WL; DePue, PL; Doherty, AM; Dudley, DT; He, JX; Hingorani, GP; Leitz, NL; Leonard, DM; Rapundalo, ST; Waite, LA1
Cheng, XM; Cody, WL; Davis, LS; DePue, PL; Doherty, AM; Flynn, MA; He, JX; LaDouceur, DM; Reynolds, EE; Welch, KM1
Cody, WL; DePue, PL; Flynn, MA; Haleen, SJ; He, JX; Kaltenbronn, JS; Leonard, DM; Sefler, AM; Waite, LA; Walker, DM1
Allcock, GH; Corder, R; Vane, JR; Warner, TD1
Allcock, GH; Mickley, EJ; Vane, JR; Warner, TD1
de Wit, D; Kimura, S; Masaki, T; Masuda, Y; Mizuguchi, T; Moroi, K; Nishiyama, M; Saito, T; Tanaka, H; Yanagisawa, M1
Cody, WL; Doherty, AM; Haleen, SJ; He, JX; Reily, MD; Reyner, EL; Stewart, BH; Walker, DM1
Alvarez, BV; CamiliĆ³n de Hurtado, MC; Cingolani, HE; Ennis, IL1
Bodelsson, G; Laursen, M; Stjernquist, M1
Curtis, LA; Holm, AS; Holmes, EP; Koch, CE; Moore, RM; Venugopal, CS1

Other Studies

10 other study(ies) available for pd 142893 and Muscle Contraction

ArticleYear
Structure-activity relationships of C-terminal endothelin hexapeptide antagonists.
    Journal of medicinal chemistry, 1993, Sep-03, Volume: 36, Issue:18

    Topics: Amino Acid Sequence; Animals; Arachidonic Acid; Cerebellum; Endothelin Receptor Antagonists; Endothelins; Heart Ventricles; Inositol Phosphates; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Rabbits; Rats; Receptors, Endothelin; Structure-Activity Relationship

1993
In vitro and in vivo studies with a series of hexapeptide endothelin antagonists.
    Journal of cardiovascular pharmacology, 1993, Volume: 22 Suppl 8

    Topics: Amino Acid Sequence; Animals; Arachidonic Acid; Azepines; Endothelin Receptor Antagonists; Endothelins; Ganglionic Blockers; Hemodynamics; In Vitro Techniques; Indoles; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Rabbits; Rats; Receptors, Endothelin; Structure-Activity Relationship; Vasoconstriction

1993
Structure-activity relationships of the potent combined endothelin-A/endothelin-B receptor antagonist Ac-DDip16-Leu-Asp-Ile-Ile-Trp21: development of endothelin-B receptor selective antagonists.
    Journal of medicinal chemistry, 1995, Jul-21, Volume: 38, Issue:15

    Topics: Amino Acid Sequence; Animals; Endothelin Receptor Antagonists; Endothelins; Humans; In Vitro Techniques; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Peptides; Rabbits; Rats; Receptor, Endothelin A; Receptor, Endothelin B; Sensitivity and Specificity; Structure-Activity Relationship

1995
Use of the endothelin antagonists BQ-123 and PD 142893 to reveal three endothelin receptors mediating smooth muscle contraction and the release of EDRF.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Amino Acid Sequence; Animals; Aorta, Thoracic; Endothelin Receptor Antagonists; Endothelins; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Nitric Oxide; Oligopeptides; Peptides, Cyclic; Pulmonary Artery; Rabbits; Rats; Rats, Wistar; Receptors, Endothelin; Stomach; Vasoconstrictor Agents; Vasodilation; Viper Venoms

1993
Characterization of endothelin receptors mediating the effects of the endothelin/sarafotoxin peptides on autonomic neurotransmission in the rat vas deferens and guinea-pig ileum.
    British journal of pharmacology, 1993, Volume: 110, Issue:2

    Topics: Amino Acid Sequence; Animals; Autonomic Nervous System; Electric Stimulation; Endothelin Receptor Antagonists; Endothelins; Guinea Pigs; Ileum; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; Oligopeptides; Peptides, Cyclic; Rats; Rats, Wistar; Receptors, Endothelin; Synaptic Transmission; Vas Deferens; Vasoconstrictor Agents; Viper Venoms

1993
Analysis of two pharmacologically predicted endothelin B receptor subtypes by using the endothelin B receptor gene knockout mouse.
    British journal of pharmacology, 1997, Volume: 120, Issue:8

    Topics: Animals; Aorta; Endothelin-1; Gastric Fundus; In Vitro Techniques; Mice; Mice, Knockout; Muscle Contraction; Muscle Relaxation; Oligopeptides; Peptides, Cyclic; Phenylephrine; Receptor, Endothelin B; Receptors, Endothelin

1997
Design of a potent combined pseudopeptide endothelin-A/endothelin-B receptor antagonist, Ac-DBhg16-Leu-Asp-Ile-[NMe]Ile-Trp21 (PD 156252): examination of its pharmacokinetic and spectral properties.
    Journal of medicinal chemistry, 1997, Jul-04, Volume: 40, Issue:14

    Topics: Amino Acid Sequence; Animals; Drug Design; Endothelin Receptor Antagonists; Endothelin-1; Femoral Artery; Humans; In Vitro Techniques; Kinetics; Magnetic Resonance Spectroscopy; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Protein Conformation; Pulmonary Artery; Rabbits; Rats; Receptor, Endothelin A; Receptor, Endothelin B; Renal Circulation; Structure-Activity Relationship; Tumor Cells, Cultured

1997
Stretch-induced alkalinization of feline papillary muscle: an autocrine-paracrine system.
    Circulation research, 1998, Oct-19, Volume: 83, Issue:8

    Topics: Alkalies; Alkaloids; Amiloride; Angiotensin II; Animals; Anti-Arrhythmia Agents; Autocrine Communication; Benzophenanthridines; Cats; Endothelin Receptor Antagonists; Endothelins; Enzyme Inhibitors; Heart; Hydrogen-Ion Concentration; Losartan; Muscle Contraction; Muscle Fibers, Skeletal; Oligopeptides; Papillary Muscles; Paracrine Communication; Peptides, Cyclic; Phenanthridines; Protein Kinase C; Sodium-Hydrogen Exchangers

1998
Atypical receptors mediate the response to endothelin-1 and sarafotoxin S6b in the human umbilical artery.
    European journal of pharmacology, 1998, Dec-04, Volume: 362, Issue:2-3

    Topics: Endothelin Receptor Antagonists; Endothelin-1; Endothelium, Vascular; Humans; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Piperidines; Receptor, Endothelin B; Umbilical Arteries; Vasoconstriction; Vasoconstrictor Agents; Viper Venoms

1998
In vitro pharmacologic effect of two endothelin-1 antagonists on equine colonic arteries and veins.
    American journal of veterinary research, 2001, Volume: 62, Issue:2

    Topics: Animals; Arteries; Colon; Dose-Response Relationship, Drug; Drug Synergism; Endothelin-1; Horses; In Vitro Techniques; Muscle Contraction; Muscle, Smooth, Vascular; Oligopeptides; Vasoconstriction; Veins

2001