Page last updated: 2024-09-03

pd 128042 and Elevated Cholesterol

pd 128042 has been researched along with Elevated Cholesterol in 4 studies

Research

Studies (4)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's4 (100.00)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Burnett, DA; Burrier, RE; Caplen, MA; Clader, JW; Davis, HR1
Anderson, M; Bocan, T; Bousley, R; Hamelehle, KL; Homan, R; Krause, BR; Lee, HT; Lee, P; Mueller, SB; O'Brien, PM; Picard, JA; Purchase, CF; Reindel, JF; Roth, BD; Sliskovic, DR; Stanfield, RL; Turluck, D; White, AD1
Auerbach, B; Bisgaier, CL; Homan, R; Kieft, K; Krause, BR; Newton, RS; Pape, ME1
Hagihara, H; Ito, Y; Mutoh, S; Nagayoshi, A; Notsu, Y; Ohne, K; Okuhara, M; Sakuma, Y1

Other Studies

4 other study(ies) available for pd 128042 and Elevated Cholesterol

ArticleYear
2-Azetidinones as inhibitors of cholesterol absorption.
    Journal of medicinal chemistry, 1994, Jun-10, Volume: 37, Issue:12

    Topics: Absorption; Animals; Anticholesteremic Agents; Azetidines; Cholesterol; Cricetinae; Disease Models, Animal; Hypercholesterolemia; Male; Mesocricetus; Microsomes; Rats; Sterol O-Acyltransferase; Structure-Activity Relationship

1994
Inhibitors of acyl-CoA:cholesterol O-acyltransferase. synthesis and pharmacological activity of (+/-)-2-dodecyl-alpha-phenyl-N-(2,4,6-trimethoxyphenyl)-2H-tetrazole-5- acetamide and structurally related tetrazole amide derivatives.
    Journal of medicinal chemistry, 1996, Jun-07, Volume: 39, Issue:12

    Topics: Animals; Anticholesteremic Agents; Arteriosclerosis; Cholesterol; Cholesterol, Dietary; Drug Design; Drug Evaluation, Preclinical; Enzyme Inhibitors; Guinea Pigs; Hypercholesterolemia; Macrophages; Male; Microsomes, Liver; Molecular Structure; Rabbits; Rats; Sterol O-Acyltransferase; Structure-Activity Relationship; Tetrazoles

1996
ACAT inhibition decreases LDL cholesterol in rabbits fed a cholesterol-free diet. Marked changes in LDL cholesterol without changes in LDL receptor mRNA abundance.
    Arteriosclerosis and thrombosis : a journal of vascular biology, 1994, Volume: 14, Issue:4

    Topics: Anilides; Animals; Aryl Hydrocarbon Hydroxylases; Cholesterol; Cholesterol, LDL; Cytochrome P-450 Enzyme System; Dietary Fats; Hydroxymethylglutaryl CoA Reductases; Hypercholesterolemia; Male; Rabbits; Receptors, LDL; RNA, Messenger; Steroid Hydroxylases; Sterol O-Acyltransferase

1994
Plasma cholesterol reducing effect of FR129169, a novel acyl-CoA:cholesterol acyltransferase inhibitor, in the rat.
    Japanese journal of pharmacology, 1996, Volume: 70, Issue:1

    Topics: Acetamides; Administration, Oral; Anilides; Animals; Anticholesteremic Agents; Cholesterol; Enzyme Inhibitors; Hypercholesterolemia; Liver; Male; Rabbits; Rats; Rats, Sprague-Dawley; Sterol O-Acyltransferase

1996