Page last updated: 2024-08-25

oxazolidin-2-one and Dyslipidemias

oxazolidin-2-one has been researched along with Dyslipidemias in 29 studies

Research

Studies (29)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (13.79)29.6817
2010's25 (86.21)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Avorn, J; Franklin, JM; Hey, SP; Kesselheim, AS1
Chen, D; Gao, P; Wang, Y; Zhang, Q; Zhou, J1
Ballantyne, CM; Catapano, AL; Norata, GD1
Akinsanya, KO; Castro-Perez, J; Chen, Y; Daniels, E; Johns, DG; Previs, SF; Roddy, TP; Wang, SP; Zhou, H1
Kikuchi, M; McCrary Sisk, C; Nakagomi, M; Numaguchi, H; Shirakawa, M; Surks, HK; Tamura, S; Teramoto, T1
Cai, J; Chen, C; Hu, Z; Li, C; Li, Y; Liu, L; Luo, H; Pei, F; Zeng, C; Zhang, W; Zhou, F; Zhou, L1
Dong, B; Fung, C; Kan, K; Liu, J; Singh, AB1
Briand, F; Burr, N; Johns, DG; Muzotte, E; Sulpice, T; Thieblemont, Q; Urbain, I1
Berbée, JF; Havekes, LM; Jukema, JW; Kühnast, S; Pieterman, EJ; Princen, HM; Rensen, PC; van der Hoorn, JW; van der Tuin, SJ; Verschuren, L; Wang, Y; Willems van Dijk, K1
Burnett, JR; Hooper, AJ; Page, MM1
Asztalos, B; Baer, AL; Coromilas, E; deGoma, EM; Donovan, DS; Dunbar, RL; Ginsberg, HN; Gutstein, DE; Holleran, S; Johnson-Levonas, AO; Jumes, P; Karmally, W; Lassman, ME; Liu, Y; Millar, JS; Ngai, C; Rader, DJ; Rafeek, H; Ramakrishnan, R; Reyes-Soffer, G; Thomas, T; Wagner, JA1
Borghi, C; Cicero, AF1
Ashraf, TB; Ballantyne, CM; Cressman, MD; Gill, GG; Hunter, JA; Johnson-Levonas, AO; Kher, U; Mitchel, YB; Shah, S1
Crucet, M; Doycheva, P; Giral, H; Jukema, JW; Kratzer, A; Kühnast, S; Landmesser, U; Lüscher, TF; Mocharla, P; Osto, E; Princen, HM; Simic, B; Speer, T; Staels, B; Stivala, S; Tailleux, A; van der Hoorn, JW1
Bloomfield, D; Carlson, GL; Littlejohn, TW; McKenney, JM; Mitchel, Y; Pasternak, RC; Sapre, A; Sisk, CM; Tribble, D1
Al-Huniti, N; Archer, L; Bergman, AJ; Chavez-Eng, C; Chen, J; Cote, J; Dykstra, K; Garg, A; Gottesdiener, K; Hilliard, D; Jin, B; Krishna, R; Laethem, T; Lasseter, KC; Lutz, R; Panebianco, D; Snyder, K; Van Bortel, L; Van Dyck, K; Van Hoydonck, P; Wagner, JA1
Fisher, T; Hubbard, B; Kling, J; Li, H; Pagler, T; Sparrow, CP; Taggart, AK; Tall, AR; Yvan-Charvet, L1
Miyares, MA1
Athyros, VG; Katsiki, N; Mikhailidis, DP1
Devaraj, S; Jialal, I1
Briand, F; Castro-Perez, J; Chen, Y; Gagen, K; Hankemeier, T; Hubbard, BK; Johns, DG; McLaren, DG; Roddy, TP; Shah, V; Sulpice, T; Vreeken, RJ; Wang, SP1
Alivanis, P; Aperis, G; Paliouras, C; Papakonstantinou, N; Tsampikaki, E1
Shinkai, H1
Davis, K; Miyares, MA1
Goldberg, AS; Hegele, RA1
Anderson, MS; Bergman, AJ; Bieberdorf, F; Bloomfield, DM; Chavez-Eng, C; Chodakewitz, J; Cote, J; Doherty, J; Fallon, M; Gottesdiener, KM; Gutierrez, M; Jin, B; Krishna, R; Lutz, R; Rosko, K; Wagner, JA1
Duriez, P1

Reviews

11 review(s) available for oxazolidin-2-one and Dyslipidemias

ArticleYear
Success, Failure, and Transparency in Biomarker-Based Drug Development: A Case Study of Cholesteryl Ester Transfer Protein Inhibitors.
    Circulation. Cardiovascular quality and outcomes, 2017, Volume: 10, Issue:6

    Topics: Amides; Anticholesteremic Agents; Benzodiazepines; Biomarkers, Pharmacological; Cholesterol Ester Transfer Proteins; Drug Approval; Drug Discovery; Dyslipidemias; Endpoint Determination; Esters; Humans; Lipids; Oxazolidinones; Predictive Value of Tests; Quinolines; Reproducibility of Results; Sulfhydryl Compounds; Time Factors; Treatment Outcome

2017
The effect and safety of anacetrapib in the treatment of dyslipidemia: a systematic review and meta-analysis.
    Postgraduate medicine, 2018, Volume: 130, Issue:1

    Topics: Anticholesteremic Agents; Dyslipidemias; Humans; Oxazolidinones

2018
New therapeutic principles in dyslipidaemia: focus on LDL and Lp(a) lowering drugs.
    European heart journal, 2013, Volume: 34, Issue:24

    Topics: Azetidines; Benzimidazoles; Benzodiazepines; Carrier Proteins; Cholesterol, LDL; Dicarboxylic Acids; Dyslipidemias; Ezetimibe; Fatty Acids; Humans; Hypolipidemic Agents; Lipoprotein(a); Oligonucleotides; Oxazolidinones; Proprotein Convertase 9; Proprotein Convertases; Serine Endopeptidases

2013
Cholesteryl ester transfer protein inhibitors in the treatment of dyslipidemia: a systematic review and meta-analysis.
    PloS one, 2013, Volume: 8, Issue:10

    Topics: Adult; Amides; Anticholesteremic Agents; Benzodiazepines; Blood Pressure; Cholesterol; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Drug Therapy, Combination; Dyslipidemias; Esters; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Oxazolidinones; Quinolines; Randomized Controlled Trials as Topic; Sulfhydryl Compounds; Treatment Outcome; Triglycerides

2013
Anacetrapib for the treatment of dyslipidaemia: the last bastion of the cholesteryl ester transfer protein inhibitors?
    Expert opinion on pharmacotherapy, 2016, Volume: 17, Issue:2

    Topics: Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Clinical Trials, Phase II as Topic; Clinical Trials, Phase III as Topic; Drug Therapy, Combination; Dyslipidemias; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypolipidemic Agents; Molecular Targeted Therapy; Oxazolidinones; Risk Factors

2016
Pharmacokinetic drug evaluation of anacetrapib for the treatment of dyslipidemia.
    Expert opinion on drug metabolism & toxicology, 2017, Volume: 13, Issue:2

    Topics: Animals; Anticholesteremic Agents; Area Under Curve; Cytochrome P-450 CYP3A Inhibitors; Drug Interactions; Dyslipidemias; Half-Life; Humans; Liver Diseases; Oxazolidinones

2017
Anacetrapib and dalcetrapib: two novel cholesteryl ester transfer protein inhibitors.
    The Annals of pharmacotherapy, 2011, Volume: 45, Issue:1

    Topics: Amides; Animals; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Drug Interactions; Dyslipidemias; Esters; Humans; Lipid Regulating Agents; Oxazolidinones; Sulfhydryl Compounds

2011
Anacetrapib: a new weapon against dyslipidemia.
    Current clinical pharmacology, 2011, Volume: 6, Issue:4

    Topics: Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Clinical Trials as Topic; Drug Therapy, Combination; Dyslipidemias; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypercholesterolemia; Metabolic Syndrome; Oxazolidinones

2011
Cholesteryl ester transfer-protein modulator and inhibitors and their potential for the treatment of cardiovascular diseases.
    Vascular health and risk management, 2012, Volume: 8

    Topics: Amides; Animals; Biomarkers; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Dyslipidemias; Esters; Humans; Hypolipidemic Agents; Oxazolidinones; Quinolines; Sulfhydryl Compounds; Treatment Outcome

2012
Patient considerations and clinical impact of cholesteryl ester transfer protein inhibitors in the management of dyslipidemia: focus on anacetrapib.
    Vascular health and risk management, 2012, Volume: 8

    Topics: Biomarkers; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Drug Therapy, Combination; Dyslipidemias; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypolipidemic Agents; Lipids; Oxazolidinones; Patient Selection; Risk Assessment; Risk Factors; Treatment Outcome

2012
Cholesteryl ester transfer protein inhibitors for dyslipidemia: focus on dalcetrapib.
    Drug design, development and therapy, 2012, Volume: 6

    Topics: Amides; Anticholesteremic Agents; Benzodiazepines; Cholesterol Ester Transfer Proteins; Dyslipidemias; Esters; Humans; Lipoproteins, HDL; Oxazolidinones; Sulfhydryl Compounds

2012

Trials

6 trial(s) available for oxazolidin-2-one and Dyslipidemias

ArticleYear
Efficacy and safety of the cholesteryl ester transfer protein inhibitor anacetrapib in Japanese patients with dyslipidemia.
    Atherosclerosis, 2013, Volume: 230, Issue:1

    Topics: Adult; Aged; Anticholesteremic Agents; Atorvastatin; Cholesterol Ester Transfer Proteins; Dose-Response Relationship, Drug; Double-Blind Method; Dyslipidemias; Female; Gene Expression Regulation; Heptanoic Acids; Humans; Japan; Male; Middle Aged; Oxazolidinones; Patient Safety; Pyrroles; Time Factors; Treatment Outcome; Young Adult

2013
Cholesteryl Ester Transfer Protein Inhibition With Anacetrapib Decreases Fractional Clearance Rates of High-Density Lipoprotein Apolipoprotein A-I and Plasma Cholesteryl Ester Transfer Protein.
    Arteriosclerosis, thrombosis, and vascular biology, 2016, Volume: 36, Issue:5

    Topics: Adult; Aged; Anticholesteremic Agents; Apolipoprotein A-I; Apolipoprotein A-II; Biomarkers; Cholesterol Ester Transfer Proteins; Double-Blind Method; Dyslipidemias; Female; Humans; Lipoproteins, HDL; Male; Middle Aged; Oxazolidinones; Time Factors; Treatment Outcome

2016
Lipid-Modifying Efficacy and Tolerability of Anacetrapib Added to Ongoing Statin Therapy in Patients with Hypercholesterolemia or Low High-Density Lipoprotein Cholesterol.
    The American journal of cardiology, 2017, Feb-01, Volume: 119, Issue:3

    Topics: Aged; Anticholesteremic Agents; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Double-Blind Method; Drug Therapy, Combination; Dyslipidemias; Ezetimibe; Female; Fibric Acids; Humans; Hydroxymethylglutaryl-CoA Reductase Inhibitors; Hypercholesterolemia; Male; Middle Aged; Niacin; Oxazolidinones; Treatment Outcome

2017
Efficacy and safety of the cholesteryl ester transfer protein inhibitor anacetrapib as monotherapy and coadministered with atorvastatin in dyslipidemic patients.
    American heart journal, 2009, Volume: 157, Issue:2

    Topics: Aged; Anticholesteremic Agents; Atorvastatin; Cholesterol Ester Transfer Proteins; Dose-Response Relationship, Drug; Double-Blind Method; Drug Therapy, Combination; Dyslipidemias; Female; Heptanoic Acids; Humans; Male; Middle Aged; Oxazolidinones; Pyrroles; Treatment Outcome

2009
Single-dose pharmacokinetics and pharmacodynamics of anacetrapib, a potent cholesteryl ester transfer protein (CETP) inhibitor, in healthy subjects.
    British journal of clinical pharmacology, 2009, Volume: 68, Issue:4

    Topics: Adolescent; Adult; Age Factors; Aged; Aged, 80 and over; Cholesterol Ester Transfer Proteins; Cross-Over Studies; Double-Blind Method; Dyslipidemias; Fasting; Female; Humans; Male; Middle Aged; Obesity; Oxazolidinones; Sex Factors; Treatment Outcome; Young Adult

2009
Effect of the cholesteryl ester transfer protein inhibitor, anacetrapib, on lipoproteins in patients with dyslipidaemia and on 24-h ambulatory blood pressure in healthy individuals: two double-blind, randomised placebo-controlled phase I studies.
    Lancet (London, England), 2007, Dec-08, Volume: 370, Issue:9603

    Topics: Adolescent; Adult; Aged; Blood Pressure; Cholesterol Ester Transfer Proteins; Dose-Response Relationship, Drug; Double-Blind Method; Dyslipidemias; Electrocardiography; Female; Humans; Male; Middle Aged; Oxazolidinones

2007

Other Studies

12 other study(ies) available for oxazolidin-2-one and Dyslipidemias

ArticleYear
In vivo effects of anacetrapib on preβ HDL: improvement in HDL remodeling without effects on cholesterol absorption.
    Journal of lipid research, 2013, Volume: 54, Issue:10

    Topics: Amides; Animals; Anticholesteremic Agents; Area Under Curve; Azetidines; Cholesterol; Cholesterol Ester Transfer Proteins; Cricetinae; Diet, High-Fat; Drug Evaluation, Preclinical; Dyslipidemias; Esters; Ezetimibe; High-Density Lipoproteins, Pre-beta; Humans; Intestinal Absorption; Male; Mesocricetus; Oxazolidinones; Sulfhydryl Compounds

2013
CETP inhibitors downregulate hepatic LDL receptor and PCSK9 expression in vitro and in vivo through a SREBP2 dependent mechanism.
    Atherosclerosis, 2014, Volume: 235, Issue:2

    Topics: Amides; Animals; Anticholesteremic Agents; Cholesterol; Cholesterol Ester Transfer Proteins; Down-Regulation; Dyslipidemias; Esters; Hep G2 Cells; Hepatocytes; Humans; Lipids; Male; Oxazolidinones; Proprotein Convertase 9; Proprotein Convertases; Receptors, LDL; Serine Endopeptidases; Sterol Regulatory Element Binding Protein 2; Sulfhydryl Compounds

2014
Anacetrapib and dalcetrapib differentially alters HDL metabolism and macrophage-to-feces reverse cholesterol transport at similar levels of CETP inhibition in hamsters.
    European journal of pharmacology, 2014, Oct-05, Volume: 740

    Topics: Amides; Animals; Anticholesteremic Agents; Biological Transport; Cholesterol; Cholesterol Ester Transfer Proteins; Cricetinae; Dyslipidemias; Esters; Feces; Macrophages; Male; Oxazolidinones; Sulfhydryl Compounds; Triglycerides

2014
Anacetrapib reduces (V)LDL cholesterol by inhibition of CETP activity and reduction of plasma PCSK9.
    Journal of lipid research, 2015, Volume: 56, Issue:11

    Topics: Animals; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Cholesterol, VLDL; Down-Regulation; Drug Evaluation, Preclinical; Dyslipidemias; Female; Gene Expression; Gene Regulatory Networks; Hypolipidemic Agents; Lipid Metabolism; Metabolic Networks and Pathways; Mice, Transgenic; Oxazolidinones; Proprotein Convertase 9; Proprotein Convertases; Serine Endopeptidases

2015
Anacetrapib, but not evacetrapib, impairs endothelial function in CETP-transgenic mice in spite of marked HDL-C increase.
    Atherosclerosis, 2017, Volume: 257

    Topics: Animals; Anticholesteremic Agents; Apolipoprotein E3; Aryldialkylphosphatase; Benzodiazepines; Biomarkers; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Diet, High-Fat; Disease Models, Animal; Dyslipidemias; Endothelium, Vascular; Female; Genetic Predisposition to Disease; Humans; Mice, Transgenic; Oxazolidinones; Phenotype; Reactive Oxygen Species; Triglycerides; Up-Regulation; Vasodilation

2017
Cholesterol efflux potential and antiinflammatory properties of high-density lipoprotein after treatment with niacin or anacetrapib.
    Arteriosclerosis, thrombosis, and vascular biology, 2010, Volume: 30, Issue:7

    Topics: Animals; Anti-Inflammatory Agents; ATP Binding Cassette Transporter 1; ATP Binding Cassette Transporter, Subfamily G, Member 1; ATP-Binding Cassette Transporters; Cells, Cultured; Cholesterol; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Clinical Trials as Topic; Dyslipidemias; Foam Cells; Humans; Hypolipidemic Agents; Inflammation; Inflammation Mediators; Lipoproteins; Macrophages; Mice; Mice, Knockout; Niacin; Oxazolidinones; Time Factors; Toll-Like Receptor 4; Treatment Outcome

2010
Anacetrapib.
    American journal of cardiovascular drugs : drugs, devices, and other interventions, 2010, Volume: 10, Issue:4

    Topics: Atherosclerosis; Cholesterol Ester Transfer Proteins; Clinical Trials as Topic; Coronary Disease; Dyslipidemias; Humans; Hypercholesterolemia; Oxazolidinones

2010
Trial watch: hope renewed for strategy to raise HDL cholesterol.
    Nature reviews. Drug discovery, 2011, Volume: 10, Issue:1

    Topics: Anticholesteremic Agents; Cardiovascular Diseases; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Clinical Trials, Phase II as Topic; Dyslipidemias; Humans; Oxazolidinones; Quinolines; Risk Factors

2011
The DEFINE study: a bright future for CETP inhibitors?
    Expert opinion on investigational drugs, 2011, Volume: 20, Issue:3

    Topics: Animals; Anticholesteremic Agents; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Dyslipidemias; Humans; Oxazolidinones; Quinolines

2011
Novel cholesteryl ester transfer protein inhibitors: promising therapy for dyslipidemia?
    Metabolic syndrome and related disorders, 2011, Volume: 9, Issue:3

    Topics: Cholesterol Ester Transfer Proteins; Drugs, Investigational; Dyslipidemias; Humans; Hypolipidemic Agents; Molecular Targeted Therapy; Oxazolidinones; Quinolines

2011
Anacetrapib promotes reverse cholesterol transport and bulk cholesterol excretion in Syrian golden hamsters.
    Journal of lipid research, 2011, Volume: 52, Issue:11

    Topics: Animals; Biological Transport; Cell Line; Cholesterol; Cholesterol Ester Transfer Proteins; Cricetinae; Dyslipidemias; Feces; Lipoproteins, HDL; Macrophages; Male; Mice; Oxazolidinones

2011
Treating high-density lipoprotein cholesterol: a return to inhibition of cholesteryl ester transfer protein?
    Current atherosclerosis reports, 2008, Volume: 10, Issue:3

    Topics: Anticholesteremic Agents; Atherosclerosis; Cholesterol Ester Transfer Proteins; Cholesterol, HDL; Cholesterol, LDL; Dyslipidemias; Heart Diseases; Humans; Oxazolidinones; Quinolines; Risk Factors

2008