Page last updated: 2024-08-21

oxazoles and Seizures

oxazoles has been researched along with Seizures in 66 studies

Research

Studies (66)

TimeframeStudies, this research(%)All Research%
pre-199055 (83.33)18.7374
1990's2 (3.03)18.2507
2000's2 (3.03)29.6817
2010's4 (6.06)24.3611
2020's3 (4.55)2.80

Authors

AuthorsStudies
Biggerstaff, A; Cerne, R; Cook, JM; Jin, X; Kivell, BM; Knutson, DE; Lippa, A; Mian, MY; Pandey, KP; Ping, X; Sharmin, D; Smith, JL; Witkin, JM1
Arnold, LA; Cerne, R; Cook, JM; Divović, B; Golani, LK; Jin, X; Lippa, A; Meyer, MJ; Mondal, P; Pandey, KP; Ping, X; Revanian, S; Savić, MM; Sharmin, D; Smith, JL; Witkin, JM; Zahn, NM1
Chen, S; Deng, X; Wang, S; Xiao, F; Yan, R; Zhang, Y; Zhou, N1
Brodney, MA; Davoren, JE; Edgerton, JR; Fortin, JP; Garnsey, M; Grimwood, S; Harris, AR; Jenkinson, S; Kenakin, T; Lazzaro, JT; Lee, CW; Lotarski, SM; Nottebaum, L; O'Neil, SV; Pettersen, B; Popiolek, M; Ramsey, S; Steyn, SJ; Thorn, CA; Webb, D; Zhang, L1
Cho, HP; Conn, PJ; Hanson, RM; Lindsley, CW; Maksymetz, J; Moran, SP; Niswender, CM; Remke, DH; Rook, JM1
Babaei, J; Gavzan, H; Hashemi, F; Sayyah, M1
Aghaei, HN; Dehpour, AR; Ebrahimi, A; Gholizadeh, R; Gooshe, M; Mousavizadeh, K; Payandemehr, B; Rahimian, R; Varastehmoradi, B1
BROWN, WC; GOODMAN, LS; SWINYARD, EA1
LAWRENCE, DE1
BALDWIN, RW1
FRIEDEL, B; LEMPP, R1
Fishback, JA; Green, AM; Kaushal, N; Matsumoto, RR; McCurdy, CR; Mésangeau, C; Narayanan, S; Poupaert, JH; Shaikh, J; Viard, E; Xu, YT1
Minchin, MC; Nutt, DJ1
DeFeudis, FV1
Engel, J; Liljequist, S1
Aldinio, C; French, ED; Schwarcz, R1
Breese, GR; Frye, GD; McCown, TJ1
Dewhurst, IC; Ekuwem, CE; Griffiths, R; O'Neill, C; Sinclair, CD; Williams, DC1
Gonzalez, LP; Hettinger, MK1
Sarhan, S; Seiler, N1
Albala, BJ; Moshé, SL1
Horton, R; Meldrum, B1
Johnson, DD; Krogsgaard-Larsen, P; Schousboe, A; Wood, JD1
Guldin, WO; Markowitsch, HJ1
Back, KC; George, ME; Pinkerton, MK1
Collins, RC1
Kamei, C; Masuda, Y; Oka, M; Shimizu, M; Yoshida, K1
Menon, MK; Vivonia, CA1
Pizzi, WJ; Unnerstall, JR1
Hori, M; Karasawa, T; Masuda, Y; Shimizu, M; Shiraishi, Y; Yoshida, K1
Cacciaguerra, S; Delarge, J; Depovere, P; Isa, M; Masereel, B; Poupaert, JH; Spampinato, S; Stables, JP; Ucar, H; Van derpoorten, K1
Hanson, GR; Jensen, M; Johnson, M; White, HS1
Harindran, J; Naik, SR; Varde, AB1
Hasegawa, K; Ishibashi, C1
Horton, RW; Meldrum, BS; Pedley, TA1
Karasawa, T; Masuda, Y; Shimizu, M; Shiraishi, Y; Utsui, Y; Yoshida, K1
Mayevsky, A1
Matthews, WD; McCafferty, GP1
Anhut, H; Hertting, G; Steinhauer, HB1
Gorecki, DK; Peesker, SJ; Wood, JD1
Chiu, P; Colasanti, BK; Craig, CR1
Ito, T; Shimizu, M; Yoshida, K1
Lee, CM; Plotnikoff, NP1
Gonsalves, SF; Harbaugh, RE; Krogsgaard-Larsen, P; Schousboe, A; Twitchell, B1
Kaijima, M; Tanaka, S; Tanaka, T; Yonemasu, Y1
Kunimoto, M; Tanaka, T; Yonemasu, Y1
Bagri, A; Di Scala, G; Sandner, G1
Hjeds, H; Krogsgaard-Larsen, P; Sarhan, S; Schousboe, A; Seiler, N1
Chweh, AY; Swinyard, EA; Ulloque, RA1
Tanaka, T; Watanabe, K; Yonemasu, Y1
Hubauer, H; Nitsch, C1
Calcet, J; Corriol, J; Dimov, S; Joanny, P1
Brink, JJ; Freeman, EA1
Millichap, JG1
Hooshmand, H; Suter, CG1
Greenblatt, EN; Osterberg, AC1
Tettenborn, D1
Böszörményi, M1
Kamioka, T; Kobayashi, S; Suzuki, Y; Takagi, H1
Borrelli, F; Caprino, L; Falchetti, R2
Karasawa, T; Masuda, M; Oka, M; Shimizu, M; Yoshida, K1
Kamioka, T; Kobayashi, S; Suzuki, Y; Tachikawa, R; Takagi, H1
Frey, HH; Kretschmer, BH1
Clark, DG; McElligott, TF1
Southgate, PJ1

Reviews

2 review(s) available for oxazoles and Seizures

ArticleYear
The imidazodiazepine, KRM-II-81: An example of a newly emerging generation of GABAkines for neurological and psychiatric disorders.
    Pharmacology, biochemistry, and behavior, 2022, Volume: 213

    Topics: Animals; Anti-Anxiety Agents; Anticonvulsants; Antidepressive Agents; Anxiety; Epilepsy; GABA Agents; GABA-A Receptor Agonists; Humans; Mental Disorders; Nervous System Diseases; Neuralgia; Oxazoles; Receptors, GABA; Receptors, GABA-A; Seizures

2022
Physiological and behavioral studies with muscimol.
    Neurochemical research, 1980, Volume: 5, Issue:10

    Topics: Animals; Behavior; Behavior, Animal; Blood-Brain Barrier; Dopamine; Feeding Behavior; gamma-Aminobutyric Acid; Humans; Learning; Memory; Muscimol; Oxazoles; Receptors, Cell Surface; Receptors, GABA-A; Seizures

1980

Trials

1 trial(s) available for oxazoles and Seizures

ArticleYear
[Triple placebo test for comparison of side effects of terizidone (terivalidin) and cycloserine].
    International journal of clinical pharmacology, therapy and toxicology, 1973, Volume: 8, Issue:1

    Topics: Clinical Trials as Topic; Cycloserine; Female; Humans; Imines; Male; Mental Disorders; Oxazoles; Seizures; Sleep Initiation and Maintenance Disorders; Tremor; Tuberculosis, Pulmonary; Vertigo

1973

Other Studies

63 other study(ies) available for oxazoles and Seizures

ArticleYear
Comparative anticonvulsant activity of the GABAkine KRM-II-81 and a deuterated analog.
    Drug development research, 2023, Volume: 84, Issue:3

    Topics: Animals; Anticonvulsants; Diazepam; Mice; Oxazoles; Seizures

2023
Synthesis and antiseizure effect evaluation of nonimidazole histamine H
    Archiv der Pharmazie, 2021, Volume: 354, Issue:4

    Topics: Animals; Anticonvulsants; Dose-Response Relationship, Drug; Histamine Antagonists; Imidazoles; Mice; Mice, Inbred Strains; Molecular Docking Simulation; Molecular Structure; N-Methylaspartate; Oxazoles; Receptors, Histamine H3; Seizures; Structure-Activity Relationship

2021
Design and Synthesis of γ- and δ-Lactam M
    Journal of medicinal chemistry, 2017, 08-10, Volume: 60, Issue:15

    Topics: Allosteric Regulation; Amphetamine; Animals; Ataxia; Diarrhea; Dogs; Donepezil; Drug Design; Female; Humans; Indans; Isoindoles; Lactams; Male; Mice, Inbred C57BL; Microsomes, Liver; Oxazoles; Piperidines; Rats, Wistar; Receptor, Muscarinic M1; Scopolamine; Seizures; Structure-Activity Relationship; Sulfonamides; Thiadiazoles; Vomiting

2017
PF-06827443 Displays Robust Allosteric Agonist and Positive Allosteric Modulator Activity in High Receptor Reserve and Native Systems.
    ACS chemical neuroscience, 2018, 09-19, Volume: 9, Issue:9

    Topics: Allosteric Regulation; Animals; Calcium; CHO Cells; Cricetulus; Dogs; Humans; Isoindoles; Mice; Oxazoles; Patch-Clamp Techniques; Prefrontal Cortex; Rats; Receptor, Muscarinic M1; Seizures

2018
A role for peroxisome proliferator-activated receptor α in anticonvulsant activity of docosahexaenoic acid against seizures induced by pentylenetetrazole.
    Neuroscience letters, 2018, 08-10, Volume: 681

    Topics: Animals; Anticonvulsants; Docosahexaenoic Acids; Injections, Intraventricular; Male; Mice; Oxazoles; Pentylenetetrazole; PPAR alpha; Seizures; Tyrosine

2018
Involvement of PPAR receptors in the anticonvulsant effects of a cannabinoid agonist, WIN 55,212-2.
    Progress in neuro-psychopharmacology & biological psychiatry, 2015, Mar-03, Volume: 57

    Topics: Anilides; Animals; Anticonvulsants; Benzoxazines; Cannabinoid Receptor Antagonists; Disease Models, Animal; Dose-Response Relationship, Drug; Drug Interactions; Male; Mice; Morpholines; Naphthalenes; Oxazoles; Pentylenetetrazole; Peroxisome Proliferator-Activated Receptors; Pioglitazone; Piperidines; Pyrazoles; Receptor, Cannabinoid, CB1; Seizures; Thiazolidinediones; Tyrosine

2015
Comparative assays of antiepileptic drugs in mice and rats.
    The Journal of pharmacology and experimental therapeutics, 1952, Volume: 106, Issue:3

    Topics: Animals; Anticonvulsants; Barbiturates; Biological Assay; Hydantoins; Mice; Oxazoles; Rats; Seizures; Urea

1952
Near fatal hemolytic anemia during anti-epileptiform convulsion therapy with tridione.
    Journal of the American Veterinary Medical Association, 1952, Volume: 121, Issue:907

    Topics: Anemia, Hemolytic; Animals; Dog Diseases; Dogs; Epilepsy; Oxazoles; Seizures; Trimethadione

1952
The dione drugs in petit mal seizures.
    Maryland state medical journal, 1953, Volume: 2, Issue:11

    Topics: Epilepsy; Epilepsy, Absence; Humans; Oxazoles; Seizures

1953
[Grand mal provocation in the treatment of petit mal in children with oxazolidines or succinimides and its therapeutic consequences].
    Zeitschrift fur Kinderheilkunde, 1962, Volume: 87

    Topics: Anticonvulsants; Child; Epilepsy; Epilepsy, Absence; Epilepsy, Tonic-Clonic; Humans; Infant; Oxazoles; Pyrrolidinones; Seizures; Succinimides

1962
Conversion of a highly selective sigma-1 receptor-ligand to sigma-2 receptor preferring ligands with anticocaine activity.
    Journal of medicinal chemistry, 2008, Mar-13, Volume: 51, Issue:5

    Topics: Animals; Anticonvulsants; Brain; Cocaine; Cocaine-Related Disorders; In Vitro Techniques; Ligands; Mice; Oxazoles; Piperazines; Radioligand Assay; Rats; Receptors, sigma; Seizures; Sigma-1 Receptor; Structure-Activity Relationship; Thiazoles

2008
The effect of repeated electroconvulsive shock on the function of THIP, a GABA agonist.
    Pharmacology, biochemistry, and behavior, 1984, Volume: 21, Issue:4

    Topics: Animals; Anticonvulsants; Blood-Brain Barrier; Dose-Response Relationship, Drug; Electroshock; Isoxazoles; Male; Oxazoles; Pentylenetetrazole; Rats; Rats, Inbred Strains; Receptors, GABA-A; Seizures; Sensory Thresholds

1984
Effects of GABAergic agonists and antagonists on various ethanol-induced behavioral changes.
    Psychopharmacology, 1982, Volume: 78, Issue:1

    Topics: Animals; Behavior, Animal; Bicuculline; Body Temperature Regulation; Dose-Response Relationship, Drug; Ethanol; Female; Motor Activity; Muridae; Muscimol; Oxazoles; Pentylenetetrazole; Picrotoxin; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Sleep Stages; Strychnine

1982
The effects of intrahippocampal ibotenic acid and their blockade by (-) 2-amino-7-phosphonoheptanoic acid: morphological and electroencephalographical analysis.
    Experimental brain research, 1983, Volume: 51, Issue:1

    Topics: 2-Amino-5-phosphonovalerate; Amino Acids; Animals; Behavior, Animal; Dose-Response Relationship, Drug; Electroencephalography; Evoked Potentials; Hippocampus; Ibotenic Acid; Male; Neurons; Oxazoles; Rats; Rats, Inbred Strains; Seizures; Synaptic Transmission

1983
Characterization of susceptibility to audiogenic seizures in ethanol-dependent rats after microinjection of gamma-aminobutyric acid (GABA) agonists into the inferior colliculus, substantia nigra or medial septum.
    The Journal of pharmacology and experimental therapeutics, 1983, Volume: 227, Issue:3

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Bicuculline; Ethanol; GABA Antagonists; Humans; Inferior Colliculi; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Receptors, Neurotransmitter; Seizures; Septum Pellucidum; Substance Withdrawal Syndrome; Substantia Nigra

1983
Synergistic inhibition of [3H]muscimol binding to calf-brain synaptic membranes in the presence of L-homocysteine and pyridoxal 5'-phosphate. A possible mechanism for homocysteine-induced seizures.
    European journal of biochemistry, 1983, Dec-15, Volume: 137, Issue:3

    Topics: Animals; Binding, Competitive; Brain; Cattle; Drug Synergism; Homocysteine; In Vitro Techniques; Kinetics; Models, Chemical; Muscimol; Oxazoles; Pyridoxal Phosphate; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Synaptic Membranes

1983
Intranigral muscimol suppresses ethanol withdrawal seizures.
    Brain research, 1984, Apr-23, Volume: 298, Issue:1

    Topics: Acoustic Stimulation; Alcoholism; Animals; gamma-Aminobutyric Acid; Humans; Male; Muscimol; Oxazoles; Rats; Rats, Inbred Strains; Receptors, Cell Surface; Receptors, GABA-A; Seizures; Substance Withdrawal Syndrome; Substantia Nigra

1984
Synergistic anticonvulsant effects of a GABA agonist and glycine.
    General pharmacology, 1984, Volume: 15, Issue:4

    Topics: 3-Mercaptopropionic Acid; Animals; Anticonvulsants; Drug Synergism; gamma-Aminobutyric Acid; Glycine; Male; Mice; Muscimol; Oxazoles; Seizures

1984
Nigral muscimol infusions facilitate the development of seizures in immature rats.
    Brain research, 1984, Volume: 315, Issue:2

    Topics: Age Factors; Animals; Flurothyl; gamma-Aminobutyric Acid; Muscimol; Oxazoles; Rats; Seizures; Substantia Nigra

1984
Effects of the bicyclic GABA agonist, THIP, on myoclonic and seizure responses in mice and baboons with reflex epilepsy.
    European journal of pharmacology, 1980, Feb-08, Volume: 61, Issue:3

    Topics: Animals; Anticonvulsants; Electroencephalography; gamma-Aminobutyric Acid; Haplorhini; Isoxazoles; Mice; Mice, Inbred DBA; Myoclonus; Oxazoles; Papio; Photic Stimulation; Seizures; Time Factors

1980
Anticonvulsant activity of the glial-selective GABA uptake inhibitor, THPO.
    Neuropharmacology, 1983, Volume: 22, Issue:1

    Topics: 4-Aminobutyrate Transaminase; Animals; Animals, Newborn; Anticonvulsants; Chickens; Cyclohexanecarboxylic Acids; Isoniazid; Isoxazoles; Male; Mice; Oxazoles; Seizures; Transaminases

1983
Epidural kainate, but not ibotenate, produces lesions in local and distant regions of the brain. A comparison of the intracerebral actions of kainic acid and ibotenic acid.
    Journal of neuroscience methods, 1982, Volume: 5, Issue:1-2

    Topics: Animals; Brain; Brain Mapping; Cerebral Cortex; Dose-Response Relationship, Drug; Hippocampus; Ibotenic Acid; Kainic Acid; Neurons; Oxazoles; Pyrrolidines; Rats; Seizures

1982
Therapeutics of monomethylhydrazine intoxication.
    Toxicology and applied pharmacology, 1982, Volume: 63, Issue:2

    Topics: Animals; Diazepam; Dose-Response Relationship, Drug; Drug Therapy, Combination; Male; Methylhydrazines; Mice; Mice, Inbred ICR; Monomethylhydrazine; Muscimol; Oxazoles; Pyridoxine; Seizures

1982
Anticonvulsant effects of muscimol.
    Neurology, 1980, Volume: 30, Issue:6

    Topics: Animals; Bicuculline; GABA Antagonists; Muscimol; Neurons; Oxazoles; Penicillins; Picrotoxin; Rats; Receptors, Drug; Seizures; Strychnine

1980
Effects of 3-sulfamoylmethyl-1,2-benzisoxazole (AD-810) and some antiepileptics on the kindled seizures in the neocortex, hippocampus and amygdala in rats.
    Archives internationales de pharmacodynamie et de therapie, 1981, Volume: 249, Issue:1

    Topics: Amygdala; Animals; Anticonvulsants; Cerebral Cortex; Electric Stimulation; Electroencephalography; Hippocampus; Isoxazoles; Male; Oxazoles; Rats; Seizures; Zonisamide

1981
Muscimol-induced myoclonic jerks in mice.
    Neuropharmacology, 1981, Volume: 20, Issue:5

    Topics: Animals; Drug Interactions; Kinetics; Male; Mice; Muscimol; Oxazoles; Picrotoxin; Seizures

1981
Muscimol and gamma-hydroxybutyrate: similar interactions with convulsant agents.
    Life sciences, 1981, Jul-27, Volume: 29, Issue:4

    Topics: 3-Mercaptopropionic Acid; Animals; Anticonvulsants; Bicuculline; Dose-Response Relationship, Drug; Drug Synergism; Hydroxybutyrates; Male; Mice; Muscimol; Oxazoles; Pentylenetetrazole; Seizures; Sodium Oxybate; Strychnine; Sulfhydryl Compounds

1981
3-Sulfamoylmethyl-1,2-benzisoxazole, a new type of anticonvulsant drug. Pharmacological profile.
    Arzneimittel-Forschung, 1980, Volume: 30, Issue:3

    Topics: Animals; Anticonvulsants; Barbiturates; Carbonic Anhydrase Inhibitors; Dogs; Electroshock; Isoxazoles; Motor Activity; Oxazoles; Rabbits; Rats; Seizures; Sleep; Species Specificity; Time Factors; Zonisamide

1980
Synthesis and anticonvulsant activity of 2(3H)-benzoxazolone and 2(3H)-benzothiazolone derivatives.
    Journal of medicinal chemistry, 1998, Mar-26, Volume: 41, Issue:7

    Topics: Animals; Anticonvulsants; Electric Stimulation; Injections, Intraperitoneal; Male; Mice; Oxazoles; Rats; Seizures; Thiazoles

1998
Distinct features of seizures induced by cocaine and amphetamine analogs.
    European journal of pharmacology, 1999, Jul-21, Volume: 377, Issue:2-3

    Topics: Animals; Central Nervous System Agents; Central Nervous System Stimulants; Diazepam; Dose-Response Relationship, Drug; Flunarizine; Hallucinogens; Male; Methamphetamine; Mice; N-Methyl-3,4-methylenedioxyamphetamine; Oxazoles; Rats; Rats, Sprague-Dawley; Seizures; Time Factors; Valproic Acid

1999
Pimprinine, an extracellular alkaloid produced by Streptomyces CDRIL-312: fermentation, isolation and pharmacological activity.
    Journal of biotechnology, 2001, Jun-01, Volume: 88, Issue:1

    Topics: Animals; Anticonvulsants; Biotechnology; Chromatography, Thin Layer; Dose-Response Relationship, Drug; Fermentation; Lethal Dose 50; Mice; Mice, Inbred Strains; Microbial Sensitivity Tests; Oxazoles; Phenytoin; Respiratory Insufficiency; Seizures; Streptomyces; Toxicity Tests; Tremor; Tremorine

2001
[Effects of a new minor tranquilizer, 10-chloro-3-methyl-1 1b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo [6,7]-1,4-diazepino [5,4-b]-oxazol-6-one (CS-386), on the after-discharge and behavior induced by electrical stimulation of the amygdala in freely-
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1977, Volume: 73, Issue:3

    Topics: Administration, Oral; Amygdala; Animals; Anti-Anxiety Agents; Benzodiazepines; Cats; Electric Stimulation; Electroencephalography; Female; Male; Muscle Contraction; Oxazoles; Salivation; Seizures; Time Factors

1977
Electroencephalographic and behavioral effects of a GABA agonist (muscimol) on photosensitive epilepsy in the baboon, papio papio.
    Epilepsia, 1979, Volume: 20, Issue:4

    Topics: Animals; Anticonvulsants; Drug Evaluation, Preclinical; Electroencephalography; Haplorhini; Muscimol; Oxazoles; Papio; Photic Stimulation; Seizures

1979
Relationships between plasma concentrations of diphenylhydantoin, phenobarbital, carbamazepine, and 3-sulfamoylmethyl-1,2-benzisoxazole (AD-810), a new anticonvulsant agent, and their anticonvulsant or neurotoxic effects in experimental animals.
    Epilepsia, 1979, Volume: 20, Issue:6

    Topics: Animals; Anticonvulsants; Brain; Carbamazepine; Dogs; Dose-Response Relationship, Drug; Haplorhini; Isoxazoles; Male; Mice; Motor Skills; Oxazoles; Phenobarbital; Phenytoin; Rabbits; Rats; Seizures; Species Specificity

1979
The effect of trimethadione on brain energy metabolism and EEG activity of the conscious rat exposed to HPO.
    Journal of neuroscience research, 1975, Volume: 1, Issue:2

    Topics: Animals; Brain; Electroencephalography; Energy Metabolism; Hyperbaric Oxygenation; Male; NAD; Oxazoles; Rats; Seizures; Trimethadione

1975
Anticonvulsant activity of muscimol against seizures induced by impairment of GABA-mediated neurotransmission.
    Neuropharmacology, 1979, Volume: 18, Issue:11

    Topics: Animals; Anticonvulsants; Bicuculline; gamma-Aminobutyric Acid; Isoniazid; Male; Muscimol; Oxazoles; Pentylenetetrazole; Picrotoxin; Rats; Seizures; Strychnine; Synaptic Transmission

1979
The synthesis of prostaglandins and thromboxane in the mouse brain in vivo. Influence of drug induced convulsions, hypoxia and the anticonvulsants trimethadione and diazepam.
    Naunyn-Schmiedeberg's archives of pharmacology, 1979, Volume: 310, Issue:1

    Topics: Animals; Brain; Diazepam; In Vitro Techniques; Male; Mice; Oxazoles; Oxygen; Pentylenetetrazole; Picrotoxin; Prostaglandins; Seizures; Thromboxanes; Time Factors; Trimethadione

1979
3-Isoxazolidone--an inhibitor of GABA metabolism.
    Biochemical pharmacology, 1976, Jul-15, Volume: 25, Issue:14

    Topics: Aminobutyrates; Animals; Brain; Chickens; Depression, Chemical; GABA Antagonists; gamma-Aminobutyric Acid; Glutamate Decarboxylase; In Vitro Techniques; Isoniazid; Isoxazoles; Male; Mice; Oxazoles; Oxazolidinones; Rats; Seizures; Time Factors

1976
Effects of diphenylhydantoin and trimethadione on seizure activity during cobalt experimental epilepsy in the rat.
    Neuropharmacology, 1976, Volume: 15, Issue:8

    Topics: Animals; Cobalt; Female; Oxazoles; Phenytoin; Rats; Seizures; Time Factors; Trimethadione

1976
Effect of 1,2-benzisoxazole-3-acetamidoxime on caudato-thalamo-cortical system in cats.
    Chemical & pharmaceutical bulletin, 1976, Volume: 24, Issue:12

    Topics: Animals; Cats; Caudate Nucleus; Cerebral Cortex; Electroencephalography; Female; Isoxazoles; Male; Oxazoles; Oximes; Seizures; Thalamus

1976
Antidepressant and anticonvulsant activity of 1-(5-phenyl-4-oxazolin-2-yl)-4-substituted piperazines.
    Journal of medicinal chemistry, 1976, Volume: 19, Issue:5

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Antidepressive Agents; Behavior, Animal; Dihydroxyphenylalanine; Mice; Oxazoles; Pemoline; Piperazines; Seizures

1976
Anticonvulsant activity of the glial GABA uptake inhibitor, THAO, in chemical seizures.
    European journal of pharmacology, 1989, Sep-13, Volume: 168, Issue:2

    Topics: Animals; Anticonvulsants; gamma-Aminobutyric Acid; Isoniazid; Isoxazoles; Male; Nervous System; Neuroglia; Neurotransmitter Uptake Inhibitors; Oxazoles; Pentylenetetrazole; Rats; Rats, Inbred Strains; Seizures

1989
Ibotenic acid-induced nigral lesion and limbic seizure in cats.
    Brain research, 1989, Oct-02, Volume: 498, Issue:2

    Topics: Animals; Brain Diseases; Cats; Electroencephalography; Female; Ibotenic Acid; Kainic Acid; Limbic System; Male; Oxazoles; Seizures; Substantia Nigra

1989
[Limbic seizure and ibotenic acid-induced lesions of substantia innominata in cats].
    No to shinkei = Brain and nerve, 1989, Volume: 41, Issue:7

    Topics: Amygdala; Animals; Basal Ganglia; Cats; Cholinergic Fibers; Ibotenic Acid; Kainic Acid; Limbic System; Oxazoles; Seizures; Substantia Innominata

1989
Effects of unilateral microinjections of GABAergic drugs into the inferior colliculus on auditory evoked potentials and on audiogenic seizure susceptibility.
    Experimental neurology, 1989, Volume: 104, Issue:1

    Topics: Acoustic Stimulation; Animals; Anticonvulsants; Bicuculline; Evoked Potentials, Auditory; Functional Laterality; gamma-Aminobutyric Acid; Inferior Colliculi; Isoxazoles; Male; Microinjections; Oxazoles; Rats; Rats, Inbred Strains; Reference Values; Seizures

1989
Amplification by glycine of the anticonvulsant effect of THPO, a GABA uptake inhibitor.
    General pharmacology, 1985, Volume: 16, Issue:5

    Topics: 3-Mercaptopropionic Acid; Animals; Anticonvulsants; Brain Chemistry; Drug Synergism; gamma-Aminobutyric Acid; Glycine; Isoxazoles; Male; Mice; Neurotransmitter Uptake Inhibitors; Oxazoles; Pentylenetetrazole; Seizures

1985
Effects of gamma-aminobutyric acid (GABA) receptor agonists on the neurotoxicity and anticonvulsant activity of barbiturates in mice.
    The Journal of pharmacology and experimental therapeutics, 1986, Volume: 237, Issue:2

    Topics: Animals; Anticonvulsants; Baclofen; Barbiturates; Dose-Response Relationship, Drug; Drug Synergism; Electroshock; gamma-Aminobutyric Acid; Isoxazoles; Male; Mice; Nervous System; Oxazoles; Receptors, GABA-A; Seizures

1986
[Ibotenic acid-induced limbic seizures and neuronal degeneration].
    No to shinkei = Brain and nerve, 1987, Volume: 39, Issue:6

    Topics: Amygdala; Animals; Cats; Electroencephalography; Hippocampus; Ibotenic Acid; Injections; Limbic System; Nerve Degeneration; Oxazoles; Seizures

1987
Distant blood-brain barrier opening in subfields of the rat hippocampus after intrastriatal injections of kainic acid but not ibotenic acid.
    Neuroscience letters, 1986, Feb-14, Volume: 64, Issue:1

    Topics: Animals; Blood-Brain Barrier; Corpus Striatum; Hippocampus; Ibotenic Acid; Kainic Acid; Male; Oxazoles; Pinocytosis; Rats; Rats, Inbred Strains; Seizures

1986
The protection against the cerebral and pulmonary effects of hyperbaric oxygen by pharmacological agents and lithium salts in mice.
    Resuscitation, 1973, Volume: 2, Issue:1

    Topics: Acetates; Aminobutyrates; Animals; Anticonvulsants; Antipsychotic Agents; Brain; Chlorpromazine; Female; Hydroxybutyrates; Hyperbaric Oxygenation; Lithium; Lung; Mice; Oxazoles; Phenobarbital; Phenytoin; Prochlorperazine; Promazine; Pulmonary Edema; Seizures; Water

1973
Effects of 5-phenyloxazolidinedione on sodium-potassium-magnesium-activated adenosine triphosphatase activity in mouse brain.
    Journal of neurochemistry, 1972, Volume: 19, Issue:7

    Topics: Adenosine Triphosphatases; Animals; Anticonvulsants; Brain; Carbon Isotopes; Chemical Phenomena; Chemistry; Enzyme Activation; Female; Imines; Ketones; Lethal Dose 50; Magnesium; Mice; Ouabain; Oxazoles; Potassium; Seizures; Sodium; Trimethadione

1972
Drug treatment of convulsive disorders.
    The New England journal of medicine, 1972, Mar-02, Volume: 286, Issue:9

    Topics: Acetazolamide; Adrenocorticotropic Hormone; Adult; Anticonvulsants; Barbiturates; Child; Diazepam; Epilepsy; Epilepsy, Absence; Epilepsy, Tonic-Clonic; Ethosuximide; Humans; Infant; Myoclonus; Oxazoles; Phenobarbital; Phenytoin; Primidone; Pyrrolidinones; Seizures; Trimethadione

1972
Classification and treatment of seizure disorders in children.
    Virginia medical monthly, 1970, Volume: 97, Issue:2

    Topics: Acetazolamide; Adolescent; Adrenocorticotropic Hormone; Anticonvulsants; Barbiturates; Child; Child, Preschool; Diazepam; Electroencephalography; Epilepsy, Absence; Epilepsy, Temporal Lobe; Epilepsy, Tonic-Clonic; Ethosuximide; Humans; Infant; Infant, Newborn; Male; Nitrazepam; Oxazoles; Phenytoin; Seizures; Succinimides; Trimethadione

1970
Some pharmacologic properties of thozalinone, a new excitant.
    Toxicology and applied pharmacology, 1965, Volume: 7, Issue:4

    Topics: Amphetamine; Animals; Appetite; Central Nervous System Stimulants; Liver; Mice; Monoamine Oxidase; Movement; Oxazoles; Rats; Reserpine; Seizures; Tetrabenazine

1965
[The toxicology of glisoxepide, a new oral antidiabetic. Results of animal studies].
    Arzneimittel-Forschung, 1974, Volume: 24, Issue:0

    Topics: Abnormalities, Drug-Induced; Administration, Oral; Animals; Azepines; Blood Glucose; Body Weight; Cats; Depression, Chemical; Dogs; Drug Evaluation, Preclinical; Female; Fertility; Glucose Tolerance Test; Hypoglycemia; Hypoglycemic Agents; Injections, Intravenous; Lethal Dose 50; Mice; Neoplasms; Oxazoles; Pregnancy; Rabbits; Rats; Seizures; Sulfonylurea Compounds; Time Factors

1974
Pharmacological studies on 10-chloro-11b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo-(6,7)-1,4-diazepino(5,4-b)-oxazol-6-one (CS-370), a new psychosedative agent.
    Arzneimittel-Forschung, 1972, Volume: 22, Issue:5

    Topics: Aggression; Animals; Anxiety; Avoidance Learning; Behavior, Animal; Benzazepines; Cats; Conditioning, Psychological; Cricetinae; Diazepam; Dogs; Female; Haplorhini; Humans; Ketones; Male; Mice; Motor Activity; Oxazoles; Rats; Seizures; Tranquilizing Agents

1972
Pharmacological research on 4,5-diphenyl-2-bis(2-hydroxyethyl)-aminoxazol (Ditazol), a new synthetic oxazole derivative as an anti-inflammatory agent.
    Arzneimittel-Forschung, 1973, Volume: 23, Issue:9

    Topics: Administration, Oral; Administration, Topical; Adrenalectomy; Analgesics; Animals; Anti-Inflammatory Agents; Arthritis, Rheumatoid; Body Temperature; Capillary Permeability; Edema; Ethanolamines; Female; Granuloma; Guanethidine; Hot Temperature; Male; Mice; Oxazoles; Phenylbutazone; Rats; Reserpine; Seizures

1973
General pharmacological properties of 4,5-diphenyl-2-bis-(2-hydroxyethyl)-aminoxazol (ditazol).
    Arzneimittel-Forschung, 1973, Volume: 23, Issue:9

    Topics: Amphetamine; Animals; Anti-Inflammatory Agents; Atropine; Blood Pressure; Cats; Chlorpromazine; Ethanolamines; Female; Gastrointestinal Motility; Guinea Pigs; Heart Rate; In Vitro Techniques; Indomethacin; Lethal Dose 50; Male; Meprobamate; Mice; Motor Activity; Muscle Contraction; Oxazoles; Peptic Ulcer; Phenylbutazone; Rabbits; Rats; Reserpine; Seizures; Sleep

1973
1,2-Benzisoxazole-3-acetamidoxime hydrochloride, a new psychotropic agent.
    Experientia, 1974, Apr-15, Volume: 30, Issue:4

    Topics: Acetamides; Aggression; Animals; Antidepressive Agents; Behavior, Animal; Brain; Brain Chemistry; Dopamine; Dose-Response Relationship, Drug; Electroencephalography; Female; Humans; Ileum; In Vitro Techniques; Isoxazoles; Norepinephrine; Oxazoles; Oximes; Reserpine; Seizures; Sleep; Tranquilizing Agents

1974
[Pharmacological studies of oxazolazepam, a new psychotropic agent. I. Actions on the central nervous system, especially on the behavioral aspect].
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1970, Volume: 66, Issue:1

    Topics: Adaptation, Biological; Analgesics; Anesthesia; Animals; Anticonvulsants; Apomorphine; Avoidance Learning; Azepines; Behavior, Animal; Central Nervous System; Chlordiazepoxide; Chlorpromazine; Cricetinae; Diazepam; Dogs; Drug Synergism; Drug Tolerance; Electric Stimulation; Female; Guinea Pigs; Haplorhini; Male; Mice; Morphine; Oxazoles; Rats; Seizures; Thiopental; Tranquilizing Agents; Tremorine

1970
Anticonvulsant effect of trimethadione in mice during continued treatment via the drinking water.
    Archives internationales de pharmacodynamie et de therapie, 1971, Volume: 193, Issue:1

    Topics: Animals; Anticonvulsants; Female; Male; Mice; Osmolar Concentration; Oxazoles; Pentylenetetrazole; Seizures; Trimethadione; Water

1971
Acute and short-term toxicity of drazoxolon (4-(2-chlorophenylhydrazone)-3-methyl-5-isoxazolone).
    Food and cosmetics toxicology, 1969, Volume: 7, Issue:5

    Topics: Animals; Antifungal Agents; Blood Pressure; Body Weight; Cats; Columbidae; Dogs; Eye; Female; Guinea Pigs; Heart Block; Male; Mice; Oxazoles; Poultry; Rabbits; Rats; Reflex; Seizures; Skin; Spermatozoa

1969
A comparison of the anticonvulsant properties of 2-diethylaminopento-4-ynoyl-2',6'-xylidide (WY 21745) with lignocaine, phenytoin, phenobarbitone and trimethadione.
    Archives internationales de pharmacodynamie et de therapie, 1971, Volume: 191, Issue:2

    Topics: Anesthetics, Local; Animals; Anticonvulsants; Drug Antagonism; Electroshock; Lethal Dose 50; Lidocaine; Mice; Oxazoles; Pentylenetetrazole; Phenobarbital; Phenytoin; Seizures; Trimethadione

1971