oxazoles has been researched along with Muscle Contraction in 82 studies
Timeframe | Studies, this research(%) | All Research% |
---|---|---|
pre-1990 | 28 (34.15) | 18.7374 |
1990's | 22 (26.83) | 18.2507 |
2000's | 21 (25.61) | 29.6817 |
2010's | 11 (13.41) | 24.3611 |
2020's | 0 (0.00) | 2.80 |
Authors | Studies |
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Chiba, Y; Ikebe, M; Kai, Y; Sakai, H; Sato, K | 1 |
Hozaki, M; Matsumoto, T; Mizutani, E; Nakamura, M; Sugita, S | 1 |
Liu, QH; Savoia, CP; Wang, YX; Wu, LG; Yadav, V; Zhang, Z; Zheng, YM | 1 |
Koh, SD; O'Driscoll, K; Sanders, KM; Sung, TS; Zhu, MH | 1 |
Aimbire, F; Albertini, R; Bjordal, JM; Correa, JC; Costa, MS; de Lima, FM; Iversen, VV | 1 |
das Graças Fernandes Sales, M; do Carmo, PL; Sudo, RT; Trachez, MM; Zapata-Sudo, G | 1 |
Hagood, JS; Lu, B; Merryman, WD; Murphy-Ullrich, JE; Zhou, Y | 1 |
Azuma, YT; Morioka, A; Nakajima, H; Nishiyama, K; Takeuchi, T | 1 |
Albinsson, S; Ekman, M; Rippe, C; Sadegh, MK; Swärd, K; Uvelius, B | 1 |
Ajima, K; Kaidoh, M; Kawai, Y; Kimizuka, K; Maejima, D; Ohhashi, T | 1 |
Dahan, D; Ducret, T; Estève, E; Marthan, R; Quignard, JF; Savineau, JP | 1 |
Joseph, L; Mei, L; Song, T; Wang, YX; Yadav, VR; Zheng, YM | 1 |
Ahn, DS; Hori, M; Karaki, H; Kim, YS; Kobayashi, M; Kwon, SC; Nakazawa, H; Ozaki, H | 1 |
Barrish, JC; Bird, E; Chen, P; Chong, S; Gu, Z; Hermsmeier, M; Humphreys, WG; Koplowitz, B; Leith, L; Liu, EC; Marino, A; Mathur, A; Moreland, S; Morrison, RA; Murugesan, N; Spergel, S; Trippodo, N; Waldron, T; Webb, ML; Young, M; Zhang, R | 1 |
Artigues-Varin, C; Mulder, P; Richard, V; Thuillez, C; Varin, R | 1 |
Bosc, JJ; Girodet, PO; Jarry, C; Molimard, M; Pourageaud, F | 1 |
Breemen, Cv; Dai, J; Kuo, KH; Lee, CH; Leo, JM; Seow, CY | 1 |
Liu, L; Xu, J | 1 |
Imaizumi, Y; Morimura, K; Muraki, K; Ohi, Y; Ohya, S; Yamamura, H | 1 |
Honjo, H; Ito, S; Kamiya, K; Kodama, I; Kume, H; Oguma, T; Shimokata, K; Takeda, N | 1 |
Austin, C; Jones, CJ; O'Neill, SC; Shaw, L; Sweeney, MA; Taggart, MJ | 1 |
Al-Chalabi, M; Ferraro, P; Govindaraju, V; Martin, JG; Michoud, MC; Powell, WS | 1 |
Cornell, CL; Fliri, HG; Garst, ME; Kharlamb, AB; Landsverk, KJ; Martos, JL; Pettit, SN; Stamer, WD; Struble, CS; Wan, Z; Wang, JW; Wheeler, LA; Woodward, DF | 1 |
Carmo, PL; Sudo, RT; Trachez, MM; Zapata-Sudo, G | 1 |
Bakker, RA; Celanire, S; Christophe, B; Collart, PP; de Esch, IJ; Gelens, E; Gillard, MR; Hulscher, S; Lallemand, BI; Lebon, F; Leurs, R; Snip, E; Talaga, PE; Timmerman, H; van der Goot, H; Venhuis, BJ; Wijtmans, M | 1 |
Antonetti, F; Caprino, L; Martelli, F; McCraw, AP; Morelli, L; Sim, AK | 1 |
Canonico, PL; Di Chiara, G; Imperato, A; Nicoletti, F; Piacente, B; Raffaele, R; Scapagnini, U | 1 |
Caroon, JM; Clark, RD; Kluge, AF; Lee, CH; Strosberg, AM | 1 |
Sone, H; Takayanagi, I | 1 |
Kadokawa, T; Kawashima, K; Sohji, Y; Sone, H; Takayanagi, I | 1 |
File, SE | 1 |
Jones, RL; Qian, YM; Wise, H | 1 |
Gallant, EM; Lentz, LR; Taylor, SR | 1 |
Dannhardt, G; Lambrecht, G; Laufer, S; Mutschler, E; Schweiger, J | 1 |
Mills, I; Murata, K; Packer, CS; Sumpio, BE | 1 |
Itoh, T; Suzuki, A | 1 |
Harris, DN; Misra, RN; Ogletree, ML; Schumacher, WA; Webb, ML | 1 |
Fusetani, N; Hori, M; Karaki, H; Ozaki, H; Saito, S; Shin, YZ | 1 |
Amano, M; Chihara, K; Feng, J; Fukata, Y; Ito, M; Iwamatsu, A; Kaibuchi, K; Kimura, K; Nakafuku, M; Nakano, T; Okawa, K; Yamamori, B | 1 |
Boulanger, CM; Illiano, S; Marsault, R; Taddei, S; Vanhoutte, PM | 1 |
Avellar, MC; Markus, RP | 1 |
Barrett, VJ; Buckingham, J; Giles, H; Honey, AC; MacLennan, SJ; Martin, GR; Moncada, S; Prentice, DJ; Robertson, AD | 1 |
Cario-Toumaniantz, C; Loirand, G; Pacaud, P | 1 |
Ali, A; Cheng, HY; Ting, KN; Wilson, VG | 1 |
Hori, M; Karaki, H; Kim, BK; Ozaki, H; Takahashi, K | 1 |
Dobashi, K; Harada, T; Horie, T; Iizuka, K; Mori, M; Nakazawa, T; Yoshii, A | 1 |
Blue, DR; Dillon, MP; Eglen, RM; Jasper, JR; Lesnick, JD; MacLennan, SJ; Zhu, QM | 1 |
Broten, TP; Chan, TB; Chang, RS; Forray, C; Freidinger, RO; Gluchowski, C; Jeon, Y; Kassahun, K; Lagu, B; Li, C; Nagarathnam, D; O'Malley, SS; Pettibone, DJ; Ransom, RW; Rodrigues, AD; Schorn, TW; Shen, Q; Tian, D; Wetzel, JM | 1 |
Barrish, JC; Bird, E; Gu, Z; Leith, L; Liu, EC; Marino, A; Mathur, A; Moreland, S; Morrison, RA; Murugesan, N; Spergel, S; Stein, PD; Waldron, T; Webb, ML; Zhang, R | 1 |
Fridén, J; Lieber, RL | 1 |
Grover, GJ; Rosenfeld, L; Stier, CT | 1 |
Dyker, H; Lösel, P; Plant, A; Scherkenbeck, J; Stieber, F | 1 |
Boissard, C; Chung, NN; Keller, M; Lemieux, C; Mutter, M; Patiny, L; Schiller, PW | 1 |
Fukuta, H; Hashitani, H; Keller, S; Lang, RJ; Mulholland, EL; Suzuki, H; Takano, H | 1 |
Hasegawa, K; Ishibashi, C | 1 |
Diamantis, W; Edelson, J; Gordon, R; Ludwig, BJ; Sofia, RD | 1 |
Fregnan, GB; Vidali, M | 1 |
Amlacher, R; Güttner, J; Härtl, A; Hillesheim, HG; Hoffmann, H; Horn, U; Kirchner, E; Knappe, H; Ulbricht, H | 1 |
Allen, DG; Westerblad, H | 1 |
Han, YG; Hartshorne, DJ; Hori, M; Karaki, H; Magae, J | 1 |
Higuchi, H; Hiraoka, N; Ito, M; Itoh, H; Konishi, T; Lederis, K; Nakano, T | 1 |
Denborough, MA; Foster, PS; Hopkinson, KC; Payne, N | 1 |
Karaki, H; Obara, K; Ozaki, H; Someya, T; Usuki, T; Yabu, H; Yoshino, M | 1 |
Fusetani, N; Hashimoto, K; Hori, M; Ishihara, H; Karaki, H; Kato, Y; Ozaki, H; Sato, K; Uemura, D; Watabe, S | 1 |
Ohara, K; Someya, T; Usuki, T; Yabu, H | 1 |
Karaki, H; Ohara, K; Ozaki, H; Someya, T; Usuki, T; Yabu, H | 1 |
Carenzi, A; Chiarino, D; Napoletano, M; Reggiani, A; Sala, A; Sala, R | 1 |
Leslie, GC; Part, NJ | 1 |
Bourreau, JP; Tricoche, R | 1 |
Kadokawa, T; Kawashima, K; Mizuta, H; Naruto, S; Ueda, S; Yoshida, T | 1 |
Hikino, H; Kasahara, Y; Konno, C; Ogata, K | 1 |
Dikstein, S; Himelstein, R; Maran, M | 1 |
Schümann, HJ; Starke, K; Werner, U | 1 |
Arrigoni, E; Benzi, G; Bermudez, E; Berte, F | 1 |
Mittag, TW; Tormay, A | 1 |
Lea, TJ; Usherwood, PN | 1 |
Borrelli, F; Caprino, L; Falchetti, R | 1 |
Bottari, F; Nannipieri, E; Saettone, MF; Serafini, MF; Tellini, N | 1 |
Hudgins, PM; Putney, JW | 1 |
Madenli, M | 1 |
Weiss, GB | 1 |
Büch, O; Heimann, H; Krupp, P; Kunz, HA; Stenger, EG; Theobald, W | 1 |
1 review(s) available for oxazoles and Muscle Contraction
Article | Year |
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Ifetroban sodium: an effective TxA2/PGH2 receptor antagonist.
Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hypertension; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Ischemia; Oxazoles; Platelet Aggregation Inhibitors; Prostaglandin H2; Prostaglandins H; Randomized Controlled Trials as Topic; Receptors, Prostaglandin; Receptors, Thromboxane; Stroke; Thrombosis; Thromboxane A2 | 2001 |
81 other study(ies) available for oxazoles and Muscle Contraction
Article | Year |
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Rac1 modulates G-protein-coupled receptor-induced bronchial smooth muscle contraction.
Topics: Animals; Bronchi; Carbachol; Endothelin-1; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Oxazoles; Phorbol 12,13-Dibutyrate; Phosphorylation; Potassium; Protein Phosphatase 1; rac1 GTP-Binding Protein; Rats; Rats, Wistar; Receptors, G-Protein-Coupled | 2018 |
Photoelasticity-based evaluation of cellular contractile force for phenotypic discrimination of vascular smooth muscle cells.
Topics: Actin Cytoskeleton; Amides; Animals; Cells, Cultured; Elasticity; Fluorescence; Marine Toxins; Microscopy, Fluorescence; Muscle Contraction; Muscle, Smooth, Vascular; Oxazoles; Phenotype; Pyridines; Swine | 2019 |
Calcineurin upregulates local Ca(2+) signaling through ryanodine receptor-1 in airway smooth muscle cells.
Topics: Animals; Calcineurin; Calcineurin Inhibitors; Calcium Signaling; Cell Line; Female; Macrocyclic Compounds; Male; Mice; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Oxazoles; Peptides; Protein Phosphatase 2; Ryanodine; Ryanodine Receptor Calcium Release Channel; Trachea; Up-Regulation | 2014 |
Intracellular Ca(2+) release from endoplasmic reticulum regulates slow wave currents and pacemaker activity of interstitial cells of Cajal.
Topics: Animals; Anoctamin-1; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cells, Cultured; Chloride Channels; Endoplasmic Reticulum; Enzyme Activation; Enzyme Inhibitors; HEK293 Cells; Humans; Indoles; Inositol 1,4,5-Trisphosphate; Interstitial Cells of Cajal; Intestine, Small; Macrocyclic Compounds; Membrane Potentials; Mice; Muscle Contraction; Myocytes, Smooth Muscle; Oxazoles; Patch-Clamp Techniques; Ryanodine; Ryanodine Receptor Calcium Release Channel; Thapsigargin | 2015 |
Effect of low level laser therapy on bronchial hyper-responsiveness.
Topics: Animals; Base Sequence; Bronchial Hyperreactivity; Calcium; Carbachol; DNA Primers; Gene Expression; In Vitro Techniques; Inositol 1,4,5-Trisphosphate Receptors; Inositol Phosphates; Low-Level Light Therapy; Macrocyclic Compounds; Male; Muscle Contraction; Myocytes, Smooth Muscle; Oxazoles; Rats; Rats, Wistar; RNA, Messenger; Tumor Necrosis Factor-alpha | 2009 |
Toxicological evaluation of azumolene after repeated intraperitoneal administration in rats.
Topics: Animals; Caffeine; Dose-Response Relationship, Drug; Imidazoles; Injections, Intraperitoneal; Kidney; Liver; Male; Muscle Contraction; Muscle, Skeletal; Neuromuscular Agents; Oxazoles; Rats; Rats, Wistar; Solubility; Toxicity Tests, Chronic | 2010 |
Thy-1-integrin alphav beta5 interactions inhibit lung fibroblast contraction-induced latent transforming growth factor-beta1 activation and myofibroblast differentiation.
Topics: Amino Acid Motifs; Animals; Cell Differentiation; Cell Membrane; Cell-Free System; Endothelin-1; Fibroblasts; Humans; Immobilized Proteins; Lung; Mice; Muscle Contraction; Myoblasts; Oxazoles; Protein Binding; Rats; Receptors, Vitronectin; Solubility; Thy-1 Antigens; Transforming Growth Factor beta1 | 2010 |
Clofibrate relaxes the longitudinal smooth muscle of the mouse distal colon through calcium-mediated desensitisation of contractile machinery.
Topics: Anilides; Animals; Anticholesteremic Agents; Benzamides; Calcium; Clofibrate; Colon; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Drug Evaluation, Preclinical; Guanylate Cyclase; Male; Marine Toxins; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Nitric Oxide Synthase; Oxazoles; Potassium Channel Blockers; PPAR alpha; Pyridines; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Sodium Channel Blockers; Soluble Guanylyl Cyclase | 2011 |
Deletion of Dicer in smooth muscle affects voiding pattern and reduces detrusor contractility and neuroeffector transmission.
Topics: Adenosine Triphosphate; Animals; Calcium Channels, L-Type; Calcium-Binding Proteins; Calponins; DEAD-box RNA Helicases; Desmin; Electric Stimulation; Gene Expression; Male; Marine Toxins; Mice; Microfilament Proteins; MicroRNAs; Muscle Contraction; Muscle, Smooth; Neuroeffector Junction; Oxazoles; Real-Time Polymerase Chain Reaction; Ribonuclease III; Synaptic Transmission; Tissue Culture Techniques; Urinary Bladder; Urination | 2012 |
Sphingosine 1-phosphate (S1P) induces S1P2 receptor-dependent tonic contraction in murine iliac lymph vessels.
Topics: Animals; Aspirin; Biomechanical Phenomena; Calcium Signaling; Endothelium, Lymphatic; Estrenes; Lymphatic Vessels; Lysophospholipids; Macrocyclic Compounds; Male; Mice; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide; Oxazoles; Pressure; Pyrazoles; Pyridines; Pyrrolidinones; Receptors, Lysosphingolipid; Signal Transduction; Sphingosine | 2013 |
Implication of the ryanodine receptor in TRPV4-induced calcium response in pulmonary arterial smooth muscle cells from normoxic and chronically hypoxic rats.
Topics: Animals; Caffeine; Calcium Channel Agonists; Calcium Signaling; Cell Hypoxia; Cells, Cultured; Dantrolene; Hypertension, Pulmonary; Hypoxia; In Vitro Techniques; Macrocyclic Compounds; Male; Morpholines; Muscle Contraction; Muscle Relaxants, Central; Myocytes, Smooth Muscle; Oxazoles; Patch-Clamp Techniques; Phorbols; Pulmonary Artery; Pyrroles; Rats; Rats, Wistar; Ryanodine; Ryanodine Receptor Calcium Release Channel; TRPV Cation Channels | 2012 |
Important role of PLC-γ1 in hypoxic increase in intracellular calcium in pulmonary arterial smooth muscle cells.
Topics: Animals; Boron Compounds; Calcium; Electron Transport Complex III; Estrenes; Gene Expression; Hypoxia; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Lentivirus; Macrocyclic Compounds; Methacrylates; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Oxazoles; Phospholipase C gamma; Pulmonary Artery; Pyrrolidinones; Reactive Oxygen Species; RNA, Small Interfering; Thiazoles; Vasoconstriction | 2013 |
Inhibitory mechanism of xestospongin-C on contraction and ion channels in the intestinal smooth muscle.
Topics: Animals; Calcium Channels; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Inositol 1,4,5-Trisphosphate Receptors; Ion Channels; Macrocyclic Compounds; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Receptors, Cytoplasmic and Nuclear | 2002 |
Biphenylsulfonamide endothelin receptor antagonists. 4. Discovery of N-[[2'-[[(4,5-dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1'-biphenyl]- 2-yl]methyl]-N,3,3-trimethylbutanamide (BMS-207940), a highly potent and orally active ET(A) selective
Topics: Administration, Oral; Animals; Blood Pressure; Caco-2 Cells; Carotid Arteries; CHO Cells; Cricetinae; Endothelin Receptor Antagonists; Humans; In Vitro Techniques; Isoxazoles; Macaca fascicularis; Male; Muscle Contraction; Oxazoles; Rabbits; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptor, Endothelin B; Structure-Activity Relationship; Sulfonamides | 2003 |
Alpha2-adrenoceptor ligands inhibit alpha1-adrenoceptor-mediated contraction of isolated rat arteries.
Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Azepines; Brimonidine Tartrate; Clonidine; Idazoxan; In Vitro Techniques; Ligands; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Oxazoles; Prostaglandins; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Rilmenidine; Yohimbine | 2002 |
Synthesis and anti-histaminic evaluation of N-phenyl-(alkyl)-5-(dialkylamino)methyl-2-amino-2-oxazolines.
Topics: Acetylcholine; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Male; Molecular Structure; Muscle Contraction; Muscle, Smooth; Oxazoles; Phenylephrine; Rats; Structure-Activity Relationship; Trachea | 2003 |
Calyculin-A disrupts subplasmalemmal junction and recurring Ca2+ waves in vascular smooth muscle.
Topics: Action Potentials; Animals; Calcium; Calcium Signaling; Calcium-Transporting ATPases; Cell Membrane; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Marine Toxins; Microscopy, Electron, Transmission; Muscle Contraction; Muscle, Smooth, Vascular; Organ Culture Techniques; Oxazoles; Phenylephrine; Rabbits; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Vasoconstrictor Agents; Vena Cava, Inferior | 2005 |
The role of calcium desensitization in vascular hyporeactivity and its regulation after hemorrhagic shock in the rat.
Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Blood Vessels; Calcium; Carbazoles; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Indoles; Insulin; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Oxazoles; Perfusion; Protein Kinase Inhibitors; Rats; Rats, Wistar; Shock, Hemorrhagic; Staurosporine; Tetradecanoylphorbol Acetate | 2005 |
Two-step Ca2+ intracellular release underlies excitation-contraction coupling in mouse urinary bladder myocytes.
Topics: Action Potentials; Animals; Calcium; Calcium Channels; Calcium Signaling; Cells, Cultured; Enzyme Inhibitors; Female; Indoles; Macrocyclic Compounds; Male; Mice; Mice, Inbred C57BL; Microscopy, Confocal; Muscle Contraction; Myocytes, Smooth Muscle; Oxazoles; Patch-Clamp Techniques; Ryanodine; Urinary Bladder | 2006 |
Involvement of reduced sensitivity to Ca in beta-adrenergic action on airway smooth muscle.
Topics: Adrenergic beta-Agonists; Amides; Animals; Asthma; Bucladesine; Calcium; Calcium Channel Blockers; Colforsin; Cyclic AMP Receptor Protein; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Fura-2; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Isoproterenol; Male; Maleimides; Marine Toxins; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Oxazoles; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Trachea | 2006 |
Caveolae and sarcoplasmic reticular coupling in smooth muscle cells of pressurised arteries: the relevance for Ca2+ oscillations and tone.
Topics: Animals; Anticholesteremic Agents; beta-Cyclodextrins; Calcium; Caveolae; In Vitro Techniques; Marine Toxins; Mesenteric Arteries; Microscopy, Electron; Muscle Contraction; Myocytes, Smooth Muscle; Myography; Oxazoles; Phosphoric Monoester Hydrolases; Rats; Sarcoplasmic Reticulum | 2006 |
Interleukin-8: novel roles in human airway smooth muscle cell contraction and migration.
Topics: Antibodies; Calcium; Cell Movement; Cells, Cultured; Estrenes; Flow Cytometry; Gene Expression Regulation; Humans; Inositol 1,4,5-Trisphosphate Receptors; Interleukin-8; Macrocyclic Compounds; Muscle Contraction; Myocytes, Smooth Muscle; Neutralization Tests; Oxazoles; Pyrrolidinones; Receptors, Interleukin-8A; Receptors, Interleukin-8B; Respiratory System; RNA, Messenger; Type C Phospholipases | 2006 |
Bimatoprost, prostamide activity, and conventional drainage.
Topics: Aged; Aged, 80 and over; Amides; Animals; Antihypertensive Agents; Aqueous Humor; Bimatoprost; Calcium; Calcium Signaling; Cats; Cell Culture Techniques; Cloprostenol; Dinoprost; Dinoprostone; Female; Humans; Intraocular Pressure; Iris; Lipids; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Oxazoles; Receptors, Thromboxane; Recombinant Proteins; Trabecular Meshwork | 2007 |
Effects of azumolene on normal and malignant hyperthermia-susceptible skeletal muscle.
Topics: Animals; Dantrolene; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Imidazoles; In Vitro Techniques; Inhibitory Concentration 50; Male; Malignant Hyperthermia; Mice; Muscle Contraction; Muscle Relaxants, Central; Muscle, Skeletal; Oxazoles; Solubility | 2008 |
4-benzyl-1H-imidazoles with oxazoline termini as histamine H3 receptor agonists.
Topics: Animals; CHO Cells; Combinatorial Chemistry Techniques; Cricetinae; Cricetulus; Cytochrome P-450 Enzyme System; Drug Design; Guinea Pigs; Histamine Agonists; Humans; Imidazoles; In Vitro Techniques; Intestines; Models, Molecular; Muscle Contraction; Muscle, Smooth; Oxazoles; Protein Binding; Radioligand Assay; Receptors, Histamine H3; Structure-Activity Relationship | 2008 |
The vascular protection of ditazole and its effect on arachidonic acid metabolism.
Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Coagulation; Cheek; Cricetinae; Epoprostenol; Fibrinolytic Agents; Male; Mesocricetus; Microcirculation; Muscle Contraction; Muscle, Smooth, Vascular; Oxazoles; Rabbits; Thromboxane A2 | 1983 |
Motor and postural effects of kainic acid or GABA agonist and antagonist injection into the cerebellar nucleus fastigii.
Topics: Animals; Cerebellar Nuclei; Kainic Acid; Motor Skills; Muscimol; Muscle Contraction; Oxazoles; Picrotoxin; Posture; Pyrrolidines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission | 1983 |
Synthesis and antihypertensive activity of a series of spiro[1,3,4,6,7,11b-hexahydro-2H-benzo[a]quinolizine-2,5'-oxazolidin-2'-one]s.
Topics: 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; Animals; Antihypertensive Agents; Aorta; Drug Evaluation, Preclinical; In Vitro Techniques; Magnetic Resonance Spectroscopy; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship | 1983 |
Inhibitory action of 2-(1-,2-benzisoxazol-3-yl)-3-[2-(2-piperidinoethoxy) phenyl]acrylonitrile (SX-284) on acetylcholine release from vagus nerve in guinea pig ileum.
Topics: Acetylcholine; Animals; Choline; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Isoxazoles; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Tetrodotoxin; Vagus Nerve; Vas Deferens | 1983 |
A possible mechanism of a new antispasmodic drug, 2-(1,2-benzisoxazol-3-yl)-3-[2-(2-piperidinoethoxy) phenyl]acrylonitrile (SX-284).
Topics: Animals; Cecum; Gastric Fundus; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Isoxazoles; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Parasympatholytics; Phrenic Nerve; Trachea; Urinary Bladder | 1982 |
Chlordiazepoxide-induced ataxia, muscle relaxation and sedation in the rat: effects of muscimol, picrotoxin and naloxone.
Topics: Animals; Arousal; Chlordiazepoxide; Exploratory Behavior; Male; Motor Activity; Motor Skills; Muridae; Muscimol; Muscle Contraction; Muscle Relaxation; Naloxone; Oxazoles; Picrotoxin; Rats; Reaction Time | 1982 |
A study of prostacyclin mimetics distinguishes neuronal from neutrophil IP receptors.
Topics: Acetates; Amino Acid Sequence; Animals; Bridged Bicyclo Compounds; Cell Aggregation; Colon; Cyclohexanols; Drug Interactions; Epoprostenol; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; N-Formylmethionine Leucyl-Phenylalanine; Neurons; Neutrophils; Oxazoles; Phenoxyacetates; Platelet Aggregation Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Epoprostenol; Receptors, Prostaglandin; Stimulation, Chemical | 1995 |
Modulation of caffeine contractures in mammalian skeletal muscles by variation of extracellular potassium.
Topics: Animals; Caffeine; Dantrolene; Drug Synergism; Extracellular Space; Imidazoles; Mice; Muscle Contraction; Muscle Relaxants, Central; Muscle, Skeletal; Oxazoles; Perchlorates; Potassium; Sodium Compounds; Swine | 1995 |
Regioisomeric 5(3)-aminomethyl-3(5)-phenylisoxazoles: synthesis, spectroscopic discrimination, and muscarinic activity.
Topics: Animals; Cholinergic Agents; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Oxazoles; Rabbits; Vas Deferens | 1995 |
Cyclic strain stimulates dephosphorylation of the 20kDa regulatory myosin light chain in vascular smooth muscle cells.
Topics: Animals; Cattle; Cell Adhesion; Cells, Cultured; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Phosphatase 1; Stress, Mechanical | 1994 |
Effects of calyculin A on tension and myosin phosphorylation in skinned smooth muscle of the rabbit mesenteric artery.
Topics: Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cyclic AMP; In Vitro Techniques; Inosine Triphosphate; Isometric Contraction; Male; Marine Toxins; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Myosins; Oxazoles; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Rabbits; Vasoconstrictor Agents | 1993 |
Pharmacological profile of BMS 180,291: a potent, long-acting, orally active thromboxane A2/prostaglandin endoperoxide receptor antagonist.
Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Administration, Oral; Animals; Aorta; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Coronary Vessels; Dinoprostone; Fatty Acids, Unsaturated; Guinea Pigs; Humans; Hydrazines; In Vitro Techniques; Male; Mice; Muscle Contraction; Oxazoles; Platelet Aggregation; Propionates; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin; Receptors, Thromboxane; Swine; Thromboxane B2; Trachea | 1993 |
Mycalolide-B, a novel and specific inhibitor of actomyosin ATPase isolated from marine sponge.
Topics: Actins; Animals; Chickens; In Vitro Techniques; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Myosins; Oxazoles; Porifera; Rabbits; Rats; Rats, Wistar | 1993 |
Regulation of myosin phosphatase by Rho and Rho-associated kinase (Rho-kinase)
Topics: 3T3 Cells; Actins; Amino Acid Sequence; Animals; Cattle; GTP Phosphohydrolases; GTP-Binding Proteins; Intracellular Signaling Peptides and Proteins; Isopropyl Thiogalactoside; Marine Toxins; Mice; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Myosin-Light-Chain Phosphatase; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Serine-Threonine Kinases; rho-Associated Kinases; rhoA GTP-Binding Protein | 1996 |
Rilmenidine activates postjunctional alpha 1- and alpha 2-adrenoceptors in the canine saphenous vein.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dogs; Female; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isotope Labeling; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Osmolar Concentration; Oxazoles; Phenoxybenzamine; Prazosin; Protein Binding; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Tritium; Yohimbine | 1996 |
Are imidazoline receptors involved in sympathetic neurotransmission in rat vas deferens?
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Idazoxan; Imidazoline Receptors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxazoles; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens; Yohimbine | 1996 |
Receptor specificity and trigemino-vascular inhibitory actions of a novel 5-HT1B/1D receptor partial agonist, 311C90 (zolmitriptan).
Topics: Animals; Coronary Vessels; Dose-Response Relationship, Drug; Guinea Pigs; Heart; Humans; Male; Muscle Contraction; Oxazoles; Oxazolidinones; Rabbits; Serotonin Receptor Agonists; Trigeminal Ganglion; Tryptamines | 1997 |
Antagonism of alpha1-adrenoceptor agonist-induced responses by rilmenidine in vascular smooth muscle.
Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Calcium; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Phenylephrine; Portal Vein; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Rilmenidine | 1998 |
Rilmenidine reveals differences in the pharmacological characteristics of prejunctional alpha2-adrenoceptors in the guinea-pig, rat and pig.
Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Arteries; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Ileum; Male; Muscle Contraction; Oxazoles; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Rilmenidine; Species Specificity; Swine; Vas Deferens | 1998 |
Increased contractility of rat uterine smooth muscle at the end of pregnancy.
Topics: Actins; Animals; Calcium; Enzyme Inhibitors; Female; Marine Toxins; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Oxazoles; Oxytocin; Phosphoprotein Phosphatases; Phosphorylation; Potassium; Pregnancy; Pregnancy, Animal; Protein Kinases; Rats; Rats, Wistar; Type C Phospholipases; Uterus | 1998 |
Relaxation of contracted rabbit tracheal and human bronchial smooth muscle by Y-27632 through inhibition of Ca2+ sensitization.
Topics: 1-Methyl-3-isobutylxanthine; Amides; Animals; Bronchi; Calcium; Carbachol; Cholinergic Agents; Detergents; Dose-Response Relationship, Drug; Endothelin-1; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Intracellular Signaling Peptides and Proteins; Marine Toxins; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Kinase; Octoxynol; Oxazoles; Phosphodiesterase Inhibitors; Protein Serine-Threonine Kinases; Pyridines; Rabbits; rho-Associated Kinases; Signal Transduction; Trachea; Type C Phospholipases | 1999 |
alpha 2A-adrenoceptors, not I1-imidazoline receptors, mediate the hypotensive effects of rilmenidine and moxonidine in conscious mice. In vivo and in vitro studies.
Topics: Animals; Antihypertensive Agents; Blood Pressure; Cell Line; Dogs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypotension; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Transfection | 1999 |
De novo design of a novel oxazolidinone analogue as a potent and selective alpha1A adrenergic receptor antagonist with high oral bioavailability.
Topics: Administration, Oral; Adrenergic alpha-Antagonists; Animals; Aorta; Binding, Competitive; Biological Availability; Blood Pressure; Dogs; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Pressure; Prostate; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Urethra | 2000 |
Biphenylsulfonamide endothelin receptor antagonists. 2. Discovery of 4'-oxazolyl biphenylsulfonamides as a new class of potent, highly selective ET(A) antagonists.
Topics: Administration, Oral; Animals; Biological Availability; Blood Pressure; Carotid Arteries; Drug Evaluation, Preclinical; Endothelin Receptor Antagonists; Hypertension; In Vitro Techniques; Injections, Intravenous; Macaca fascicularis; Muscle Contraction; Muscle, Smooth, Vascular; Oxazoles; Rabbits; Radioligand Assay; Rats; Receptor, Endothelin A; Structure-Activity Relationship; Sulfonamides | 2000 |
Serum creatine kinase level is a poor predictor of muscle function after injury.
Topics: Animals; Biomarkers; Creatine Kinase; Isoenzymes; Models, Animal; Muscle Contraction; Muscle, Skeletal; Oxazoles; Rabbits | 2001 |
Syntheses of analogues of the insect neuropeptide proctolin containing an oxazole ring as an amide bond replacement.
Topics: Amides; Animals; Digestive System; Grasshoppers; In Vitro Techniques; Indicators and Reagents; Muscle Contraction; Neuropeptides; Oligopeptides; Oxazoles; Oxidation-Reduction | 2001 |
Pseudoproline-containing analogues of morphiceptin and endomorphin-2: evidence for a cis Tyr-Pro amide bond in the bioactive conformation.
Topics: Animals; Brain; Endorphins; Guinea Pigs; Ileum; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Mice; Muscle Contraction; Muscle, Smooth; Oligopeptides; Oxazoles; Proline; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Thiazoles; Vas Deferens | 2001 |
Modulators of internal Ca2+ stores and the spontaneous electrical and contractile activity of the guinea-pig renal pelvis.
Topics: Animals; Boron Compounds; Caffeine; Calcium; Electric Conductivity; Electrophysiology; Estrenes; Guinea Pigs; Indoles; Kidney Pelvis; Macrocyclic Compounds; Muscle Contraction; Muscle, Smooth; Neomycin; Oxazoles; Pyrrolidinones; Ryanodine | 2002 |
[Effects of a new minor tranquilizer, 10-chloro-3-methyl-1 1b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo [6,7]-1,4-diazepino [5,4-b]-oxazol-6-one (CS-386), on the after-discharge and behavior induced by electrical stimulation of the amygdala in freely-
Topics: Administration, Oral; Amygdala; Animals; Anti-Anxiety Agents; Benzodiazepines; Cats; Electric Stimulation; Electroencephalography; Female; Male; Muscle Contraction; Oxazoles; Salivation; Seizures; Time Factors | 1977 |
Pharmacological properties of 2,3-dihydro-9H-isoxazolo[3,2-b]-quinazolin-9-one (W-2429. Part 2: General pharmacological investigation.
Topics: Anesthetics, Local; Animals; Anti-Inflammatory Agents, Non-Steroidal; Anticonvulsants; Antidepressive Agents, Tricyclic; Antitussive Agents; Cats; Diuresis; Dogs; Enzyme Induction; Female; Gastrointestinal Hemorrhage; Gastrointestinal Motility; Guinea Pigs; Hemodynamics; Isoxazoles; Male; Mice; Motor Activity; Muscle Contraction; Muscle, Smooth; Oxazoles; Postural Balance; Prostaglandin-Endoperoxide Synthases; Quinazolines; Rabbits; Rats; Respiration; Sleep; Stomach Ulcer; Time Factors | 1977 |
Pharmacological profile of a new psychotherapeutic agent: 4-p-fluorophenyl-5-N(N'-o-methoxyphenyl)piperazinoethyl-4-oxazolin-2-one (LR 511).
Topics: Aggression; Analgesics; Animals; Anticonvulsants; Antidepressive Agents; Autonomic Nervous System; Behavior, Animal; Catalepsy; Conditioning, Psychological; Dogs; Drug Synergism; Exploratory Behavior; Female; Humans; Hypnotics and Sedatives; Lethal Dose 50; Male; Mice; Motor Activity; Muscle Contraction; Oxazoles; Piperazines; Psychotropic Drugs; Rabbits; Rats; Tranquilizing Agents | 1977 |
[2-Amino-oxazoles as potential H-bonding agents in virostatic research. 4. Pharmacokinetics and pharmacologic-toxicologic profile of 2-guanidino-4,5-dipropyloxazole hydrochloride].
Topics: Administration, Oral; Animals; Antiviral Agents; Digestive System; Dogs; Female; Guinea Pigs; Half-Life; Heart Rate; Hydrogen Bonding; In Vitro Techniques; Injections, Subcutaneous; Male; Mice; Muscle Contraction; Myocardial Contraction; Oxazoles; Rabbits; Rats; Rats, Wistar; Swine | 1992 |
Myoplasmic free Mg2+ concentration during repetitive stimulation of single fibres from mouse skeletal muscle.
Topics: Adenosine Triphosphate; Animals; Benzofurans; Fura-2; Hydrogen-Ion Concentration; Magnesium; Male; Mice; Muscle Contraction; Muscles; Oxazoles; Sodium | 1992 |
A novel protein phosphatase inhibitor, tautomycin. Effect on smooth muscle.
Topics: Animals; Antifungal Agents; Aorta; Calcium; Enzyme Inhibitors; Ethers, Cyclic; Guinea Pigs; Kinetics; Macromolecular Substances; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Myosins; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Pyrans; Rabbits; Rats; Spiro Compounds; Verapamil | 1991 |
Contraction of rat thoracic aorta strips by endothelin-1 in the absence of extracellular Ca2+.
Topics: Animals; Aorta, Thoracic; Caffeine; Calcium; Endothelins; In Vitro Techniques; Indicators and Reagents; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Phorbol 12,13-Dibutyrate; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Urotensins; Vasoconstrictor Agents | 1991 |
The effect of azumolene on hypercontractility and sarcoplasmic reticulum Ca(2+)-dependent ATPase activity of malignant hyperpyrexia-susceptible porcine skeletal muscle.
Topics: Animals; Caffeine; Calcium-Transporting ATPases; Dantrolene; Halothane; Imidazoles; Malignant Hyperthermia; Muscle Contraction; Muscle Relaxants, Central; Muscles; Oxazoles; Potassium Chloride; Sarcoplasmic Reticulum | 1991 |
Modification by calyculin A of inward Ca currents in smooth muscle cells isolated from guinea pig taenia coli.
Topics: Animals; Benzofurans; Calcium; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Guinea Pigs; In Vitro Techniques; Intestine, Large; Marine Toxins; Muscle Contraction; Muscle, Smooth; Oxazoles | 1990 |
Calcium-independent activation of contractile apparatus in smooth muscle by calyculin-A.
Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Actomyosin; Animals; Aorta, Thoracic; Ca(2+) Mg(2+)-ATPase; Calcium; Calcium-Transporting ATPases; Cecum; Egtazic Acid; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Oxazoles; Phosphorylation; Porifera; Rats; Rats, Inbred Strains; Verapamil | 1989 |
[Action of cytochalasin B on the contraction of smooth muscle of guinea pig taenia coli].
Topics: Animals; Calcium Channels; Colon; Cytochalasin B; Guinea Pigs; In Vitro Techniques; Marine Toxins; Muscle Contraction; Muscle, Smooth; Oxazoles; Potassium | 1989 |
[Effect of calyculin A on the contraction of colonic smooth muscle of guinea pigs].
Topics: Animals; Calcium; Calcium Channels; Colon; Guinea Pigs; In Vitro Techniques; Marine Toxins; Muscle Contraction; Muscle, Smooth; Oxazoles | 1989 |
New isoxazole derivatives provided with antihypertensive activity.
Topics: Animals; Antihypertensive Agents; Aorta, Thoracic; Binding, Competitive; Chemical Phenomena; Chemistry; Clonidine; In Vitro Techniques; Isoxazoles; Magnetic Resonance Spectroscopy; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Vas Deferens; Yohimbine | 1989 |
The effect of EU4093 (azumolene sodium) on the contraction of intrafusal muscle in the soleus muscle of the anaesthetized rat.
Topics: Anesthesia; Animals; Electric Stimulation; Female; Imidazoles; In Vitro Techniques; Muscle Contraction; Muscle Relaxants, Central; Muscles; Neurons; Oxazoles; Rats; Rats, Inbred Strains | 1989 |
Prejunctional alpha 2-adrenergic properties of S-3341 (dicyclopropylmethyl)amino-2-delta-2-oxazoline: a comparison with clonidine.
Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Oxazoles; Prazosin; Rats; Rats, Inbred WKY; Rilmenidine; Vas Deferens; Yohimbine | 1987 |
Synthesis and spasmolytic activity of aminoalkyl 2-substituted-2-(1,2-benzisoxazol-3-yl)acetates.
Topics: Animals; Chemical Phenomena; Chemistry; Guinea Pigs; In Vitro Techniques; Isoxazoles; Male; Muscle Contraction; Oxazoles; Parasympatholytics | 1987 |
Pharmacology of ephedroxanes.
Topics: Analgesics; Anesthesia; Animals; Anticonvulsants; Anura; Blepharoptosis; Blood Pressure; Body Temperature; Chickens; Drug Synergism; Electroshock; Guinea Pigs; Heart Rate; Hexobarbital; In Vitro Techniques; Male; Mice; Motor Activity; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxazoles; Pentylenetetrazole; Postural Balance; Rats; Rats, Inbred Strains; Strychnine | 1985 |
Vorticella--a model for chemopharmacodynamic action on smooth muscle.
Topics: Adenosine; Amides; Anesthetics, Local; Animals; Ciliophora; Culture Media; Cyanides; Ferricyanides; Lanthanum; Lead; Models, Biological; Muscle Contraction; Muscle, Smooth; Nicotine; Oxazoles; Papaverine; Phenazines; Potassium Chloride; Tetrazolium Salts; Time Factors; Vitamin K | 1972 |
Actions of clonidine and 2-(2-methyl-6-ethyl-cyclohexylamino)-2-oxazoline on postganglionic autonomic nerves.
Topics: Acetylcholine; Animals; Antihypertensive Agents; Autonomic Fibers, Postganglionic; Clonidine; Cyclohexylamines; Depression, Chemical; Electric Stimulation; Guinea Pigs; Heart; Heart Rate; Hexamethonium Compounds; Ileum; Imidazoles; In Vitro Techniques; Muscle Contraction; Neurosecretion; Norepinephrine; Oxazoles; Rabbits; Synaptic Transmission | 1972 |
Action of antibiotics on respiratory tract. II. Dicloxacillin.
Topics: Acetylcholine; Ampicillin; Animals; Barium; Bronchi; Chlorides; Dicloxacillin; Dogs; Ephedrine; Female; Histamine H1 Antagonists; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Penicillins; Respiration; Respiratory System | 1970 |
Effects of isoxazolium cations on some isolated muscle preparations.
Topics: Acetylcholine; Angiotensin II; Animals; Aorta; Cholinesterase Inhibitors; Diaphragm; Diphenhydramine; Electric Stimulation; Guinea Pigs; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Muscles; Norepinephrine; Oxazoles; Parasympathomimetics; Perchlorates; Pilocarpine; Piperazines; Rabbits; Rats; Serotonin Antagonists | 1971 |
The site of action of ibotenic acid and the identification of two populations of glutamate receptors on insect muscle-fibres.
Topics: Aminobutyrates; Animals; Basidiomycota; Binding, Competitive; Dose-Response Relationship, Drug; Glutamates; Grasshoppers; In Vitro Techniques; Iontophoresis; Membrane Potentials; Membranes; Muscle Contraction; Muscles; Neural Conduction; Neurons; Oxazoles; Perfusion; Picrotoxin; Quaternary Ammonium Compounds; Receptors, Drug; Serotonin; Time Factors; Tryptamines | 1973 |
General pharmacological properties of 4,5-diphenyl-2-bis-(2-hydroxyethyl)-aminoxazol (ditazol).
Topics: Amphetamine; Animals; Anti-Inflammatory Agents; Atropine; Blood Pressure; Cats; Chlorpromazine; Ethanolamines; Female; Gastrointestinal Motility; Guinea Pigs; Heart Rate; In Vitro Techniques; Indomethacin; Lethal Dose 50; Male; Meprobamate; Mice; Motor Activity; Muscle Contraction; Oxazoles; Peptic Ulcer; Phenylbutazone; Rabbits; Rats; Reserpine; Seizures; Sleep | 1973 |
Synthesis and biological activity of some 4-aryl-substituted 4-oxazolin-2-ones.
Topics: Animals; Barbiturates; Central Nervous System; Cyclization; Guinea Pigs; Ileum; Injections, Intraperitoneal; Ketones; Lethal Dose 50; Mice; Muscle Contraction; Muscles; Oxazoles; Oxidation-Reduction; Structure-Activity Relationship | 1972 |
Distribution of local anesthetics and the intracellular pH in vascular smooth muscle.
Topics: Anesthetics, Local; Animals; Aorta; Binding Sites; Calcium; Carbon Isotopes; Cocaine; Extracellular Space; Hydrogen-Ion Concentration; In Vitro Techniques; Ketones; Kinetics; Lidocaine; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxazoles; Potassium; Procaine; Rabbits; Structure-Activity Relationship; Tetracaine | 1972 |
[Study of a new myorelaxant combined with an analgesic: Dorsilon].
Topics: Acetaminophen; Adult; Analgesics; Catechols; Drug Synergism; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle Relaxants, Central; Oxazoles | 1970 |
Actions of procaine on nicotine-induced effects in frog sartorius muscle.
Topics: Animals; Anura; Biological Transport; Calcium; Calcium Isotopes; Carbon Isotopes; Depression, Chemical; Hydrogen-Ion Concentration; In Vitro Techniques; Iodoacetates; Muscle Contraction; Muscles; Nialamide; Nicotine; Oxazoles; Procaine; Stimulation, Chemical; Thigh | 1968 |
[Pharmacological and experimental psychological studies with 2 components of fly agaric (Amanita muscaria)].
Topics: Animals; Autonomic Nervous System; Basidiomycota; Behavior, Animal; Blood Pressure; Body Temperature; Conditioning, Classical; Electroencephalography; Guinea Pigs; Humans; Mice; Motor Activity; Muscle Contraction; Oxazoles; Psychological Tests; Psychoses, Substance-Induced; Rabbits; Rats; Reflex, Monosynaptic; Respiration | 1968 |