Page last updated: 2024-08-21

oxazoles and Muscle Contraction

oxazoles has been researched along with Muscle Contraction in 82 studies

Research

Studies (82)

TimeframeStudies, this research(%)All Research%
pre-199028 (34.15)18.7374
1990's22 (26.83)18.2507
2000's21 (25.61)29.6817
2010's11 (13.41)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Chiba, Y; Ikebe, M; Kai, Y; Sakai, H; Sato, K1
Hozaki, M; Matsumoto, T; Mizutani, E; Nakamura, M; Sugita, S1
Liu, QH; Savoia, CP; Wang, YX; Wu, LG; Yadav, V; Zhang, Z; Zheng, YM1
Koh, SD; O'Driscoll, K; Sanders, KM; Sung, TS; Zhu, MH1
Aimbire, F; Albertini, R; Bjordal, JM; Correa, JC; Costa, MS; de Lima, FM; Iversen, VV1
das Graças Fernandes Sales, M; do Carmo, PL; Sudo, RT; Trachez, MM; Zapata-Sudo, G1
Hagood, JS; Lu, B; Merryman, WD; Murphy-Ullrich, JE; Zhou, Y1
Azuma, YT; Morioka, A; Nakajima, H; Nishiyama, K; Takeuchi, T1
Albinsson, S; Ekman, M; Rippe, C; Sadegh, MK; Swärd, K; Uvelius, B1
Ajima, K; Kaidoh, M; Kawai, Y; Kimizuka, K; Maejima, D; Ohhashi, T1
Dahan, D; Ducret, T; Estève, E; Marthan, R; Quignard, JF; Savineau, JP1
Joseph, L; Mei, L; Song, T; Wang, YX; Yadav, VR; Zheng, YM1
Ahn, DS; Hori, M; Karaki, H; Kim, YS; Kobayashi, M; Kwon, SC; Nakazawa, H; Ozaki, H1
Barrish, JC; Bird, E; Chen, P; Chong, S; Gu, Z; Hermsmeier, M; Humphreys, WG; Koplowitz, B; Leith, L; Liu, EC; Marino, A; Mathur, A; Moreland, S; Morrison, RA; Murugesan, N; Spergel, S; Trippodo, N; Waldron, T; Webb, ML; Young, M; Zhang, R1
Artigues-Varin, C; Mulder, P; Richard, V; Thuillez, C; Varin, R1
Bosc, JJ; Girodet, PO; Jarry, C; Molimard, M; Pourageaud, F1
Breemen, Cv; Dai, J; Kuo, KH; Lee, CH; Leo, JM; Seow, CY1
Liu, L; Xu, J1
Imaizumi, Y; Morimura, K; Muraki, K; Ohi, Y; Ohya, S; Yamamura, H1
Honjo, H; Ito, S; Kamiya, K; Kodama, I; Kume, H; Oguma, T; Shimokata, K; Takeda, N1
Austin, C; Jones, CJ; O'Neill, SC; Shaw, L; Sweeney, MA; Taggart, MJ1
Al-Chalabi, M; Ferraro, P; Govindaraju, V; Martin, JG; Michoud, MC; Powell, WS1
Cornell, CL; Fliri, HG; Garst, ME; Kharlamb, AB; Landsverk, KJ; Martos, JL; Pettit, SN; Stamer, WD; Struble, CS; Wan, Z; Wang, JW; Wheeler, LA; Woodward, DF1
Carmo, PL; Sudo, RT; Trachez, MM; Zapata-Sudo, G1
Bakker, RA; Celanire, S; Christophe, B; Collart, PP; de Esch, IJ; Gelens, E; Gillard, MR; Hulscher, S; Lallemand, BI; Lebon, F; Leurs, R; Snip, E; Talaga, PE; Timmerman, H; van der Goot, H; Venhuis, BJ; Wijtmans, M1
Antonetti, F; Caprino, L; Martelli, F; McCraw, AP; Morelli, L; Sim, AK1
Canonico, PL; Di Chiara, G; Imperato, A; Nicoletti, F; Piacente, B; Raffaele, R; Scapagnini, U1
Caroon, JM; Clark, RD; Kluge, AF; Lee, CH; Strosberg, AM1
Sone, H; Takayanagi, I1
Kadokawa, T; Kawashima, K; Sohji, Y; Sone, H; Takayanagi, I1
File, SE1
Jones, RL; Qian, YM; Wise, H1
Gallant, EM; Lentz, LR; Taylor, SR1
Dannhardt, G; Lambrecht, G; Laufer, S; Mutschler, E; Schweiger, J1
Mills, I; Murata, K; Packer, CS; Sumpio, BE1
Itoh, T; Suzuki, A1
Harris, DN; Misra, RN; Ogletree, ML; Schumacher, WA; Webb, ML1
Fusetani, N; Hori, M; Karaki, H; Ozaki, H; Saito, S; Shin, YZ1
Amano, M; Chihara, K; Feng, J; Fukata, Y; Ito, M; Iwamatsu, A; Kaibuchi, K; Kimura, K; Nakafuku, M; Nakano, T; Okawa, K; Yamamori, B1
Boulanger, CM; Illiano, S; Marsault, R; Taddei, S; Vanhoutte, PM1
Avellar, MC; Markus, RP1
Barrett, VJ; Buckingham, J; Giles, H; Honey, AC; MacLennan, SJ; Martin, GR; Moncada, S; Prentice, DJ; Robertson, AD1
Cario-Toumaniantz, C; Loirand, G; Pacaud, P1
Ali, A; Cheng, HY; Ting, KN; Wilson, VG1
Hori, M; Karaki, H; Kim, BK; Ozaki, H; Takahashi, K1
Dobashi, K; Harada, T; Horie, T; Iizuka, K; Mori, M; Nakazawa, T; Yoshii, A1
Blue, DR; Dillon, MP; Eglen, RM; Jasper, JR; Lesnick, JD; MacLennan, SJ; Zhu, QM1
Broten, TP; Chan, TB; Chang, RS; Forray, C; Freidinger, RO; Gluchowski, C; Jeon, Y; Kassahun, K; Lagu, B; Li, C; Nagarathnam, D; O'Malley, SS; Pettibone, DJ; Ransom, RW; Rodrigues, AD; Schorn, TW; Shen, Q; Tian, D; Wetzel, JM1
Barrish, JC; Bird, E; Gu, Z; Leith, L; Liu, EC; Marino, A; Mathur, A; Moreland, S; Morrison, RA; Murugesan, N; Spergel, S; Stein, PD; Waldron, T; Webb, ML; Zhang, R1
Fridén, J; Lieber, RL1
Grover, GJ; Rosenfeld, L; Stier, CT1
Dyker, H; Lösel, P; Plant, A; Scherkenbeck, J; Stieber, F1
Boissard, C; Chung, NN; Keller, M; Lemieux, C; Mutter, M; Patiny, L; Schiller, PW1
Fukuta, H; Hashitani, H; Keller, S; Lang, RJ; Mulholland, EL; Suzuki, H; Takano, H1
Hasegawa, K; Ishibashi, C1
Diamantis, W; Edelson, J; Gordon, R; Ludwig, BJ; Sofia, RD1
Fregnan, GB; Vidali, M1
Amlacher, R; Güttner, J; Härtl, A; Hillesheim, HG; Hoffmann, H; Horn, U; Kirchner, E; Knappe, H; Ulbricht, H1
Allen, DG; Westerblad, H1
Han, YG; Hartshorne, DJ; Hori, M; Karaki, H; Magae, J1
Higuchi, H; Hiraoka, N; Ito, M; Itoh, H; Konishi, T; Lederis, K; Nakano, T1
Denborough, MA; Foster, PS; Hopkinson, KC; Payne, N1
Karaki, H; Obara, K; Ozaki, H; Someya, T; Usuki, T; Yabu, H; Yoshino, M1
Fusetani, N; Hashimoto, K; Hori, M; Ishihara, H; Karaki, H; Kato, Y; Ozaki, H; Sato, K; Uemura, D; Watabe, S1
Ohara, K; Someya, T; Usuki, T; Yabu, H1
Karaki, H; Ohara, K; Ozaki, H; Someya, T; Usuki, T; Yabu, H1
Carenzi, A; Chiarino, D; Napoletano, M; Reggiani, A; Sala, A; Sala, R1
Leslie, GC; Part, NJ1
Bourreau, JP; Tricoche, R1
Kadokawa, T; Kawashima, K; Mizuta, H; Naruto, S; Ueda, S; Yoshida, T1
Hikino, H; Kasahara, Y; Konno, C; Ogata, K1
Dikstein, S; Himelstein, R; Maran, M1
Schümann, HJ; Starke, K; Werner, U1
Arrigoni, E; Benzi, G; Bermudez, E; Berte, F1
Mittag, TW; Tormay, A1
Lea, TJ; Usherwood, PN1
Borrelli, F; Caprino, L; Falchetti, R1
Bottari, F; Nannipieri, E; Saettone, MF; Serafini, MF; Tellini, N1
Hudgins, PM; Putney, JW1
Madenli, M1
Weiss, GB1
Büch, O; Heimann, H; Krupp, P; Kunz, HA; Stenger, EG; Theobald, W1

Reviews

1 review(s) available for oxazoles and Muscle Contraction

ArticleYear
Ifetroban sodium: an effective TxA2/PGH2 receptor antagonist.
    Cardiovascular drug reviews, 2001,Summer, Volume: 19, Issue:2

    Topics: Animals; Bridged Bicyclo Compounds, Heterocyclic; Humans; Hypertension; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Ischemia; Oxazoles; Platelet Aggregation Inhibitors; Prostaglandin H2; Prostaglandins H; Randomized Controlled Trials as Topic; Receptors, Prostaglandin; Receptors, Thromboxane; Stroke; Thrombosis; Thromboxane A2

2001

Other Studies

81 other study(ies) available for oxazoles and Muscle Contraction

ArticleYear
Rac1 modulates G-protein-coupled receptor-induced bronchial smooth muscle contraction.
    European journal of pharmacology, 2018, Jan-05, Volume: 818

    Topics: Animals; Bronchi; Carbachol; Endothelin-1; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Oxazoles; Phorbol 12,13-Dibutyrate; Phosphorylation; Potassium; Protein Phosphatase 1; rac1 GTP-Binding Protein; Rats; Rats, Wistar; Receptors, G-Protein-Coupled

2018
Photoelasticity-based evaluation of cellular contractile force for phenotypic discrimination of vascular smooth muscle cells.
    Scientific reports, 2019, 03-08, Volume: 9, Issue:1

    Topics: Actin Cytoskeleton; Amides; Animals; Cells, Cultured; Elasticity; Fluorescence; Marine Toxins; Microscopy, Fluorescence; Muscle Contraction; Muscle, Smooth, Vascular; Oxazoles; Phenotype; Pyridines; Swine

2019
Calcineurin upregulates local Ca(2+) signaling through ryanodine receptor-1 in airway smooth muscle cells.
    American journal of physiology. Lung cellular and molecular physiology, 2014, Nov-15, Volume: 307, Issue:10

    Topics: Animals; Calcineurin; Calcineurin Inhibitors; Calcium Signaling; Cell Line; Female; Macrocyclic Compounds; Male; Mice; Mice, Knockout; Muscle Contraction; Muscle, Smooth; Oxazoles; Peptides; Protein Phosphatase 2; Ryanodine; Ryanodine Receptor Calcium Release Channel; Trachea; Up-Regulation

2014
Intracellular Ca(2+) release from endoplasmic reticulum regulates slow wave currents and pacemaker activity of interstitial cells of Cajal.
    American journal of physiology. Cell physiology, 2015, Apr-15, Volume: 308, Issue:8

    Topics: Animals; Anoctamin-1; Calcium; Calcium Channel Blockers; Calcium-Transporting ATPases; Cells, Cultured; Chloride Channels; Endoplasmic Reticulum; Enzyme Activation; Enzyme Inhibitors; HEK293 Cells; Humans; Indoles; Inositol 1,4,5-Trisphosphate; Interstitial Cells of Cajal; Intestine, Small; Macrocyclic Compounds; Membrane Potentials; Mice; Muscle Contraction; Myocytes, Smooth Muscle; Oxazoles; Patch-Clamp Techniques; Ryanodine; Ryanodine Receptor Calcium Release Channel; Thapsigargin

2015
Effect of low level laser therapy on bronchial hyper-responsiveness.
    Lasers in medical science, 2009, Volume: 24, Issue:4

    Topics: Animals; Base Sequence; Bronchial Hyperreactivity; Calcium; Carbachol; DNA Primers; Gene Expression; In Vitro Techniques; Inositol 1,4,5-Trisphosphate Receptors; Inositol Phosphates; Low-Level Light Therapy; Macrocyclic Compounds; Male; Muscle Contraction; Myocytes, Smooth Muscle; Oxazoles; Rats; Rats, Wistar; RNA, Messenger; Tumor Necrosis Factor-alpha

2009
Toxicological evaluation of azumolene after repeated intraperitoneal administration in rats.
    Fundamental & clinical pharmacology, 2010, Volume: 24, Issue:4

    Topics: Animals; Caffeine; Dose-Response Relationship, Drug; Imidazoles; Injections, Intraperitoneal; Kidney; Liver; Male; Muscle Contraction; Muscle, Skeletal; Neuromuscular Agents; Oxazoles; Rats; Rats, Wistar; Solubility; Toxicity Tests, Chronic

2010
Thy-1-integrin alphav beta5 interactions inhibit lung fibroblast contraction-induced latent transforming growth factor-beta1 activation and myofibroblast differentiation.
    The Journal of biological chemistry, 2010, Jul-16, Volume: 285, Issue:29

    Topics: Amino Acid Motifs; Animals; Cell Differentiation; Cell Membrane; Cell-Free System; Endothelin-1; Fibroblasts; Humans; Immobilized Proteins; Lung; Mice; Muscle Contraction; Myoblasts; Oxazoles; Protein Binding; Rats; Receptors, Vitronectin; Solubility; Thy-1 Antigens; Transforming Growth Factor beta1

2010
Clofibrate relaxes the longitudinal smooth muscle of the mouse distal colon through calcium-mediated desensitisation of contractile machinery.
    Pharmacology, 2011, Volume: 88, Issue:1-2

    Topics: Anilides; Animals; Anticholesteremic Agents; Benzamides; Calcium; Clofibrate; Colon; Cyclic AMP-Dependent Protein Kinases; Disease Models, Animal; Drug Evaluation, Preclinical; Guanylate Cyclase; Male; Marine Toxins; Mice; Mice, Inbred C57BL; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Nitric Oxide Synthase; Oxazoles; Potassium Channel Blockers; PPAR alpha; Pyridines; Pyrimidines; Receptors, Cytoplasmic and Nuclear; Sodium Channel Blockers; Soluble Guanylyl Cyclase

2011
Deletion of Dicer in smooth muscle affects voiding pattern and reduces detrusor contractility and neuroeffector transmission.
    PloS one, 2012, Volume: 7, Issue:4

    Topics: Adenosine Triphosphate; Animals; Calcium Channels, L-Type; Calcium-Binding Proteins; Calponins; DEAD-box RNA Helicases; Desmin; Electric Stimulation; Gene Expression; Male; Marine Toxins; Mice; Microfilament Proteins; MicroRNAs; Muscle Contraction; Muscle, Smooth; Neuroeffector Junction; Oxazoles; Real-Time Polymerase Chain Reaction; Ribonuclease III; Synaptic Transmission; Tissue Culture Techniques; Urinary Bladder; Urination

2012
Sphingosine 1-phosphate (S1P) induces S1P2 receptor-dependent tonic contraction in murine iliac lymph vessels.
    Microcirculation (New York, N.Y. : 1994), 2013, Volume: 20, Issue:1

    Topics: Animals; Aspirin; Biomechanical Phenomena; Calcium Signaling; Endothelium, Lymphatic; Estrenes; Lymphatic Vessels; Lysophospholipids; Macrocyclic Compounds; Male; Mice; Muscle Contraction; Muscle, Smooth; NG-Nitroarginine Methyl Ester; Nifedipine; Nitric Oxide; Oxazoles; Pressure; Pyrazoles; Pyridines; Pyrrolidinones; Receptors, Lysosphingolipid; Signal Transduction; Sphingosine

2013
Implication of the ryanodine receptor in TRPV4-induced calcium response in pulmonary arterial smooth muscle cells from normoxic and chronically hypoxic rats.
    American journal of physiology. Lung cellular and molecular physiology, 2012, Nov-01, Volume: 303, Issue:9

    Topics: Animals; Caffeine; Calcium Channel Agonists; Calcium Signaling; Cell Hypoxia; Cells, Cultured; Dantrolene; Hypertension, Pulmonary; Hypoxia; In Vitro Techniques; Macrocyclic Compounds; Male; Morpholines; Muscle Contraction; Muscle Relaxants, Central; Myocytes, Smooth Muscle; Oxazoles; Patch-Clamp Techniques; Phorbols; Pulmonary Artery; Pyrroles; Rats; Rats, Wistar; Ryanodine; Ryanodine Receptor Calcium Release Channel; TRPV Cation Channels

2012
Important role of PLC-γ1 in hypoxic increase in intracellular calcium in pulmonary arterial smooth muscle cells.
    American journal of physiology. Lung cellular and molecular physiology, 2013, Feb-01, Volume: 304, Issue:3

    Topics: Animals; Boron Compounds; Calcium; Electron Transport Complex III; Estrenes; Gene Expression; Hypoxia; Inositol 1,4,5-Trisphosphate; Inositol 1,4,5-Trisphosphate Receptors; Lentivirus; Macrocyclic Compounds; Methacrylates; Mice; Muscle Contraction; Muscle, Smooth, Vascular; Myocytes, Smooth Muscle; Oxazoles; Phospholipase C gamma; Pulmonary Artery; Pyrrolidinones; Reactive Oxygen Species; RNA, Small Interfering; Thiazoles; Vasoconstriction

2013
Inhibitory mechanism of xestospongin-C on contraction and ion channels in the intestinal smooth muscle.
    British journal of pharmacology, 2002, Volume: 137, Issue:8

    Topics: Animals; Calcium Channels; Dose-Response Relationship, Drug; Guinea Pigs; Ileum; Inositol 1,4,5-Trisphosphate Receptors; Ion Channels; Macrocyclic Compounds; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Receptors, Cytoplasmic and Nuclear

2002
Biphenylsulfonamide endothelin receptor antagonists. 4. Discovery of N-[[2'-[[(4,5-dimethyl-3-isoxazolyl)amino]sulfonyl]-4-(2-oxazolyl)[1,1'-biphenyl]- 2-yl]methyl]-N,3,3-trimethylbutanamide (BMS-207940), a highly potent and orally active ET(A) selective
    Journal of medicinal chemistry, 2003, Jan-02, Volume: 46, Issue:1

    Topics: Administration, Oral; Animals; Blood Pressure; Caco-2 Cells; Carotid Arteries; CHO Cells; Cricetinae; Endothelin Receptor Antagonists; Humans; In Vitro Techniques; Isoxazoles; Macaca fascicularis; Male; Muscle Contraction; Oxazoles; Rabbits; Rats; Rats, Sprague-Dawley; Receptor, Endothelin A; Receptor, Endothelin B; Structure-Activity Relationship; Sulfonamides

2003
Alpha2-adrenoceptor ligands inhibit alpha1-adrenoceptor-mediated contraction of isolated rat arteries.
    Fundamental & clinical pharmacology, 2002, Volume: 16, Issue:4

    Topics: Adrenergic alpha-1 Receptor Antagonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Aorta, Thoracic; Arteries; Azepines; Brimonidine Tartrate; Clonidine; Idazoxan; In Vitro Techniques; Ligands; Male; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Nitric Oxide; Oxazoles; Prostaglandins; Quinoxalines; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Rilmenidine; Yohimbine

2002
Synthesis and anti-histaminic evaluation of N-phenyl-(alkyl)-5-(dialkylamino)methyl-2-amino-2-oxazolines.
    Journal of enzyme inhibition and medicinal chemistry, 2003, Volume: 18, Issue:2

    Topics: Acetylcholine; Animals; Aorta, Thoracic; Dose-Response Relationship, Drug; Guinea Pigs; Histamine; Histamine H1 Antagonists; In Vitro Techniques; Male; Molecular Structure; Muscle Contraction; Muscle, Smooth; Oxazoles; Phenylephrine; Rats; Structure-Activity Relationship; Trachea

2003
Calyculin-A disrupts subplasmalemmal junction and recurring Ca2+ waves in vascular smooth muscle.
    Cell calcium, 2005, Volume: 37, Issue:1

    Topics: Action Potentials; Animals; Calcium; Calcium Signaling; Calcium-Transporting ATPases; Cell Membrane; Dose-Response Relationship, Drug; Enzyme Inhibitors; Male; Marine Toxins; Microscopy, Electron, Transmission; Muscle Contraction; Muscle, Smooth, Vascular; Organ Culture Techniques; Oxazoles; Phenylephrine; Rabbits; Sarcoplasmic Reticulum; Sarcoplasmic Reticulum Calcium-Transporting ATPases; Vasoconstrictor Agents; Vena Cava, Inferior

2005
The role of calcium desensitization in vascular hyporeactivity and its regulation after hemorrhagic shock in the rat.
    Shock (Augusta, Ga.), 2005, Volume: 23, Issue:6

    Topics: 8-Bromo Cyclic Adenosine Monophosphate; Animals; Blood Vessels; Calcium; Carbazoles; Cyclic GMP-Dependent Protein Kinases; Dose-Response Relationship, Drug; Enzyme Inhibitors; Female; Indoles; Insulin; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Phosphatase; Oxazoles; Perfusion; Protein Kinase Inhibitors; Rats; Rats, Wistar; Shock, Hemorrhagic; Staurosporine; Tetradecanoylphorbol Acetate

2005
Two-step Ca2+ intracellular release underlies excitation-contraction coupling in mouse urinary bladder myocytes.
    American journal of physiology. Cell physiology, 2006, Volume: 290, Issue:2

    Topics: Action Potentials; Animals; Calcium; Calcium Channels; Calcium Signaling; Cells, Cultured; Enzyme Inhibitors; Female; Indoles; Macrocyclic Compounds; Male; Mice; Mice, Inbred C57BL; Microscopy, Confocal; Muscle Contraction; Myocytes, Smooth Muscle; Oxazoles; Patch-Clamp Techniques; Ryanodine; Urinary Bladder

2006
Involvement of reduced sensitivity to Ca in beta-adrenergic action on airway smooth muscle.
    Clinical and experimental allergy : journal of the British Society for Allergy and Clinical Immunology, 2006, Volume: 36, Issue:2

    Topics: Adrenergic beta-Agonists; Amides; Animals; Asthma; Bucladesine; Calcium; Calcium Channel Blockers; Colforsin; Cyclic AMP Receptor Protein; Cyclic AMP-Dependent Protein Kinases; Depression, Chemical; Fura-2; Guinea Pigs; Imidazoles; In Vitro Techniques; Indoles; Intracellular Signaling Peptides and Proteins; Isoproterenol; Male; Maleimides; Marine Toxins; Methacholine Chloride; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Phosphatase; Oxazoles; Protein Kinase C; Protein Serine-Threonine Kinases; Pyridines; rho-Associated Kinases; Trachea

2006
Caveolae and sarcoplasmic reticular coupling in smooth muscle cells of pressurised arteries: the relevance for Ca2+ oscillations and tone.
    Cardiovascular research, 2006, Mar-01, Volume: 69, Issue:4

    Topics: Animals; Anticholesteremic Agents; beta-Cyclodextrins; Calcium; Caveolae; In Vitro Techniques; Marine Toxins; Mesenteric Arteries; Microscopy, Electron; Muscle Contraction; Myocytes, Smooth Muscle; Myography; Oxazoles; Phosphoric Monoester Hydrolases; Rats; Sarcoplasmic Reticulum

2006
Interleukin-8: novel roles in human airway smooth muscle cell contraction and migration.
    American journal of physiology. Cell physiology, 2006, Volume: 291, Issue:5

    Topics: Antibodies; Calcium; Cell Movement; Cells, Cultured; Estrenes; Flow Cytometry; Gene Expression Regulation; Humans; Inositol 1,4,5-Trisphosphate Receptors; Interleukin-8; Macrocyclic Compounds; Muscle Contraction; Myocytes, Smooth Muscle; Neutralization Tests; Oxazoles; Pyrrolidinones; Receptors, Interleukin-8A; Receptors, Interleukin-8B; Respiratory System; RNA, Messenger; Type C Phospholipases

2006
Bimatoprost, prostamide activity, and conventional drainage.
    Investigative ophthalmology & visual science, 2007, Volume: 48, Issue:9

    Topics: Aged; Aged, 80 and over; Amides; Animals; Antihypertensive Agents; Aqueous Humor; Bimatoprost; Calcium; Calcium Signaling; Cats; Cell Culture Techniques; Cloprostenol; Dinoprost; Dinoprostone; Female; Humans; Intraocular Pressure; Iris; Lipids; Male; Middle Aged; Muscle Contraction; Muscle, Smooth; Organ Culture Techniques; Oxazoles; Receptors, Thromboxane; Recombinant Proteins; Trabecular Meshwork

2007
Effects of azumolene on normal and malignant hyperthermia-susceptible skeletal muscle.
    Basic & clinical pharmacology & toxicology, 2008, Volume: 102, Issue:3

    Topics: Animals; Dantrolene; Dose-Response Relationship, Drug; Guinea Pigs; Humans; Imidazoles; In Vitro Techniques; Inhibitory Concentration 50; Male; Malignant Hyperthermia; Mice; Muscle Contraction; Muscle Relaxants, Central; Muscle, Skeletal; Oxazoles; Solubility

2008
4-benzyl-1H-imidazoles with oxazoline termini as histamine H3 receptor agonists.
    Journal of medicinal chemistry, 2008, May-22, Volume: 51, Issue:10

    Topics: Animals; CHO Cells; Combinatorial Chemistry Techniques; Cricetinae; Cricetulus; Cytochrome P-450 Enzyme System; Drug Design; Guinea Pigs; Histamine Agonists; Humans; Imidazoles; In Vitro Techniques; Intestines; Models, Molecular; Muscle Contraction; Muscle, Smooth; Oxazoles; Protein Binding; Radioligand Assay; Receptors, Histamine H3; Structure-Activity Relationship

2008
The vascular protection of ditazole and its effect on arachidonic acid metabolism.
    Thrombosis research, 1983, Dec-01, Volume: 32, Issue:5

    Topics: Animals; Arachidonic Acid; Arachidonic Acids; Blood Coagulation; Cheek; Cricetinae; Epoprostenol; Fibrinolytic Agents; Male; Mesocricetus; Microcirculation; Muscle Contraction; Muscle, Smooth, Vascular; Oxazoles; Rabbits; Thromboxane A2

1983
Motor and postural effects of kainic acid or GABA agonist and antagonist injection into the cerebellar nucleus fastigii.
    Birth defects original article series, 1983, Volume: 19, Issue:4

    Topics: Animals; Cerebellar Nuclei; Kainic Acid; Motor Skills; Muscimol; Muscle Contraction; Oxazoles; Picrotoxin; Posture; Pyrrolidines; Rats; Receptors, Cell Surface; Receptors, GABA-A; Synaptic Transmission

1983
Synthesis and antihypertensive activity of a series of spiro[1,3,4,6,7,11b-hexahydro-2H-benzo[a]quinolizine-2,5'-oxazolidin-2'-one]s.
    Journal of medicinal chemistry, 1983, Volume: 26, Issue:10

    Topics: 2H-Benzo(a)quinolizin-2-ol, 2-Ethyl-1,3,4,6,7,11b-hexahydro-3-isobutyl-9,10-dimethoxy-; Animals; Antihypertensive Agents; Aorta; Drug Evaluation, Preclinical; In Vitro Techniques; Magnetic Resonance Spectroscopy; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Rats; Receptors, Adrenergic, alpha; Structure-Activity Relationship

1983
Inhibitory action of 2-(1-,2-benzisoxazol-3-yl)-3-[2-(2-piperidinoethoxy) phenyl]acrylonitrile (SX-284) on acetylcholine release from vagus nerve in guinea pig ileum.
    Journal of pharmacobio-dynamics, 1983, Volume: 6, Issue:4

    Topics: Acetylcholine; Animals; Choline; Electric Stimulation; Guinea Pigs; Ileum; In Vitro Techniques; Isoxazoles; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Tetrodotoxin; Vagus Nerve; Vas Deferens

1983
A possible mechanism of a new antispasmodic drug, 2-(1,2-benzisoxazol-3-yl)-3-[2-(2-piperidinoethoxy) phenyl]acrylonitrile (SX-284).
    Japanese journal of pharmacology, 1982, Volume: 32, Issue:6

    Topics: Animals; Cecum; Gastric Fundus; Gastrointestinal Motility; Guinea Pigs; Ileum; In Vitro Techniques; Isoxazoles; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Parasympatholytics; Phrenic Nerve; Trachea; Urinary Bladder

1982
Chlordiazepoxide-induced ataxia, muscle relaxation and sedation in the rat: effects of muscimol, picrotoxin and naloxone.
    Pharmacology, biochemistry, and behavior, 1982, Volume: 17, Issue:6

    Topics: Animals; Arousal; Chlordiazepoxide; Exploratory Behavior; Male; Motor Activity; Motor Skills; Muridae; Muscimol; Muscle Contraction; Muscle Relaxation; Naloxone; Oxazoles; Picrotoxin; Rats; Reaction Time

1982
A study of prostacyclin mimetics distinguishes neuronal from neutrophil IP receptors.
    European journal of pharmacology, 1995, May-24, Volume: 278, Issue:3

    Topics: Acetates; Amino Acid Sequence; Animals; Bridged Bicyclo Compounds; Cell Aggregation; Colon; Cyclohexanols; Drug Interactions; Epoprostenol; In Vitro Techniques; Male; Molecular Sequence Data; Muscle Contraction; N-Formylmethionine Leucyl-Phenylalanine; Neurons; Neutrophils; Oxazoles; Phenoxyacetates; Platelet Aggregation Inhibitors; Rats; Rats, Sprague-Dawley; Receptors, Epoprostenol; Receptors, Prostaglandin; Stimulation, Chemical

1995
Modulation of caffeine contractures in mammalian skeletal muscles by variation of extracellular potassium.
    Journal of cellular physiology, 1995, Volume: 165, Issue:2

    Topics: Animals; Caffeine; Dantrolene; Drug Synergism; Extracellular Space; Imidazoles; Mice; Muscle Contraction; Muscle Relaxants, Central; Muscle, Skeletal; Oxazoles; Perchlorates; Potassium; Sodium Compounds; Swine

1995
Regioisomeric 5(3)-aminomethyl-3(5)-phenylisoxazoles: synthesis, spectroscopic discrimination, and muscarinic activity.
    Archiv der Pharmazie, 1995, Volume: 328, Issue:5

    Topics: Animals; Cholinergic Agents; Guinea Pigs; Ileum; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Myocardial Contraction; Oxazoles; Rabbits; Vas Deferens

1995
Cyclic strain stimulates dephosphorylation of the 20kDa regulatory myosin light chain in vascular smooth muscle cells.
    Biochemical and biophysical research communications, 1994, Nov-30, Volume: 205, Issue:1

    Topics: Animals; Cattle; Cell Adhesion; Cells, Cultured; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosins; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Phosphatase 1; Stress, Mechanical

1994
Effects of calyculin A on tension and myosin phosphorylation in skinned smooth muscle of the rabbit mesenteric artery.
    British journal of pharmacology, 1993, Volume: 109, Issue:3

    Topics: Animals; Calcium; Calcium-Calmodulin-Dependent Protein Kinases; Cyclic AMP; In Vitro Techniques; Inosine Triphosphate; Isometric Contraction; Male; Marine Toxins; Mesenteric Arteries; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Myosins; Oxazoles; Phosphorylation; Protein Kinase C; Protein Kinase Inhibitors; Protein Kinases; Rabbits; Vasoconstrictor Agents

1993
Pharmacological profile of BMS 180,291: a potent, long-acting, orally active thromboxane A2/prostaglandin endoperoxide receptor antagonist.
    The Journal of pharmacology and experimental therapeutics, 1993, Volume: 264, Issue:2

    Topics: 15-Hydroxy-11 alpha,9 alpha-(epoxymethano)prosta-5,13-dienoic Acid; Administration, Oral; Animals; Aorta; Bridged Bicyclo Compounds, Heterocyclic; Cattle; Coronary Vessels; Dinoprostone; Fatty Acids, Unsaturated; Guinea Pigs; Humans; Hydrazines; In Vitro Techniques; Male; Mice; Muscle Contraction; Oxazoles; Platelet Aggregation; Propionates; Prostaglandin Endoperoxides, Synthetic; Rats; Rats, Sprague-Dawley; Receptors, Prostaglandin; Receptors, Thromboxane; Swine; Thromboxane B2; Trachea

1993
Mycalolide-B, a novel and specific inhibitor of actomyosin ATPase isolated from marine sponge.
    FEBS letters, 1993, May-10, Volume: 322, Issue:2

    Topics: Actins; Animals; Chickens; In Vitro Techniques; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myocardial Contraction; Myosins; Oxazoles; Porifera; Rabbits; Rats; Rats, Wistar

1993
Regulation of myosin phosphatase by Rho and Rho-associated kinase (Rho-kinase)
    Science (New York, N.Y.), 1996, Jul-12, Volume: 273, Issue:5272

    Topics: 3T3 Cells; Actins; Amino Acid Sequence; Animals; Cattle; GTP Phosphohydrolases; GTP-Binding Proteins; Intracellular Signaling Peptides and Proteins; Isopropyl Thiogalactoside; Marine Toxins; Mice; Molecular Sequence Data; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Myosin-Light-Chain Phosphatase; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Protein Serine-Threonine Kinases; rho-Associated Kinases; rhoA GTP-Binding Protein

1996
Rilmenidine activates postjunctional alpha 1- and alpha 2-adrenoceptors in the canine saphenous vein.
    Fundamental & clinical pharmacology, 1996, Volume: 10, Issue:4

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Brimonidine Tartrate; Calcium Channel Blockers; Clonidine; Dihydropyridines; Dogs; Female; Idazoxan; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Isotope Labeling; Male; Medetomidine; Muscle Contraction; Muscle, Smooth; Osmolar Concentration; Oxazoles; Phenoxybenzamine; Prazosin; Protein Binding; Quinoxalines; Radioligand Assay; Receptors, Adrenergic, alpha-1; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Tritium; Yohimbine

1996
Are imidazoline receptors involved in sympathetic neurotransmission in rat vas deferens?
    General pharmacology, 1996, Volume: 27, Issue:7

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Adrenergic alpha-Antagonists; Animals; Electric Stimulation; Idazoxan; Imidazoline Receptors; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxazoles; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Sympathetic Nervous System; Synaptic Transmission; Vas Deferens; Yohimbine

1996
Receptor specificity and trigemino-vascular inhibitory actions of a novel 5-HT1B/1D receptor partial agonist, 311C90 (zolmitriptan).
    British journal of pharmacology, 1997, Volume: 121, Issue:2

    Topics: Animals; Coronary Vessels; Dose-Response Relationship, Drug; Guinea Pigs; Heart; Humans; Male; Muscle Contraction; Oxazoles; Oxazolidinones; Rabbits; Serotonin Receptor Agonists; Trigeminal Ganglion; Tryptamines

1997
Antagonism of alpha1-adrenoceptor agonist-induced responses by rilmenidine in vascular smooth muscle.
    European journal of pharmacology, 1998, Jan-12, Volume: 341, Issue:2-3

    Topics: Adrenergic alpha-1 Receptor Agonists; Adrenergic alpha-Agonists; Animals; Calcium; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Phenylephrine; Portal Vein; Rats; Rats, Wistar; Receptors, Adrenergic, alpha-1; Rilmenidine

1998
Rilmenidine reveals differences in the pharmacological characteristics of prejunctional alpha2-adrenoceptors in the guinea-pig, rat and pig.
    British journal of pharmacology, 1998, Volume: 125, Issue:1

    Topics: Adrenergic alpha-2 Receptor Agonists; Adrenergic alpha-2 Receptor Antagonists; Adrenergic alpha-Agonists; Animals; Arteries; Brimonidine Tartrate; Clonidine; Dose-Response Relationship, Drug; Electric Stimulation; Guinea Pigs; Ileum; Male; Muscle Contraction; Oxazoles; Quinoxalines; Rats; Receptors, Adrenergic, alpha-2; Rilmenidine; Species Specificity; Swine; Vas Deferens

1998
Increased contractility of rat uterine smooth muscle at the end of pregnancy.
    Comparative biochemistry and physiology. Part A, Molecular & integrative physiology, 1998, Volume: 121, Issue:2

    Topics: Actins; Animals; Calcium; Enzyme Inhibitors; Female; Marine Toxins; Muscle Contraction; Muscle, Smooth; Myosin Light Chains; Oxazoles; Oxytocin; Phosphoprotein Phosphatases; Phosphorylation; Potassium; Pregnancy; Pregnancy, Animal; Protein Kinases; Rats; Rats, Wistar; Type C Phospholipases; Uterus

1998
Relaxation of contracted rabbit tracheal and human bronchial smooth muscle by Y-27632 through inhibition of Ca2+ sensitization.
    American journal of respiratory cell and molecular biology, 1999, Volume: 20, Issue:6

    Topics: 1-Methyl-3-isobutylxanthine; Amides; Animals; Bronchi; Calcium; Carbachol; Cholinergic Agents; Detergents; Dose-Response Relationship, Drug; Endothelin-1; GTP-Binding Proteins; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Intracellular Signaling Peptides and Proteins; Marine Toxins; Muscle Contraction; Muscle, Smooth; Myosin-Light-Chain Kinase; Octoxynol; Oxazoles; Phosphodiesterase Inhibitors; Protein Serine-Threonine Kinases; Pyridines; Rabbits; rho-Associated Kinases; Signal Transduction; Trachea; Type C Phospholipases

1999
alpha 2A-adrenoceptors, not I1-imidazoline receptors, mediate the hypotensive effects of rilmenidine and moxonidine in conscious mice. In vivo and in vitro studies.
    Annals of the New York Academy of Sciences, 1999, Jun-21, Volume: 881

    Topics: Animals; Antihypertensive Agents; Blood Pressure; Cell Line; Dogs; Guanosine 5'-O-(3-Thiotriphosphate); Humans; Hypotension; Imidazoles; Imidazoline Receptors; In Vitro Techniques; Male; Mice; Mice, Inbred Strains; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Quinolizines; Receptors, Adrenergic, alpha-2; Receptors, Drug; Rilmenidine; Saphenous Vein; Transfection

1999
De novo design of a novel oxazolidinone analogue as a potent and selective alpha1A adrenergic receptor antagonist with high oral bioavailability.
    Journal of medicinal chemistry, 2000, Jul-27, Volume: 43, Issue:15

    Topics: Administration, Oral; Adrenergic alpha-Antagonists; Animals; Aorta; Binding, Competitive; Biological Availability; Blood Pressure; Dogs; Humans; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Pressure; Prostate; Radioligand Assay; Rats; Receptors, Adrenergic, alpha-1; Recombinant Proteins; Urethra

2000
Biphenylsulfonamide endothelin receptor antagonists. 2. Discovery of 4'-oxazolyl biphenylsulfonamides as a new class of potent, highly selective ET(A) antagonists.
    Journal of medicinal chemistry, 2000, Aug-10, Volume: 43, Issue:16

    Topics: Administration, Oral; Animals; Biological Availability; Blood Pressure; Carotid Arteries; Drug Evaluation, Preclinical; Endothelin Receptor Antagonists; Hypertension; In Vitro Techniques; Injections, Intravenous; Macaca fascicularis; Muscle Contraction; Muscle, Smooth, Vascular; Oxazoles; Rabbits; Radioligand Assay; Rats; Receptor, Endothelin A; Structure-Activity Relationship; Sulfonamides

2000
Serum creatine kinase level is a poor predictor of muscle function after injury.
    Scandinavian journal of medicine & science in sports, 2001, Volume: 11, Issue:2

    Topics: Animals; Biomarkers; Creatine Kinase; Isoenzymes; Models, Animal; Muscle Contraction; Muscle, Skeletal; Oxazoles; Rabbits

2001
Syntheses of analogues of the insect neuropeptide proctolin containing an oxazole ring as an amide bond replacement.
    Organic letters, 2001, Nov-01, Volume: 3, Issue:22

    Topics: Amides; Animals; Digestive System; Grasshoppers; In Vitro Techniques; Indicators and Reagents; Muscle Contraction; Neuropeptides; Oligopeptides; Oxazoles; Oxidation-Reduction

2001
Pseudoproline-containing analogues of morphiceptin and endomorphin-2: evidence for a cis Tyr-Pro amide bond in the bioactive conformation.
    Journal of medicinal chemistry, 2001, Nov-08, Volume: 44, Issue:23

    Topics: Animals; Brain; Endorphins; Guinea Pigs; Ileum; In Vitro Techniques; Magnetic Resonance Spectroscopy; Male; Mice; Muscle Contraction; Muscle, Smooth; Oligopeptides; Oxazoles; Proline; Protein Conformation; Radioligand Assay; Rats; Receptors, Opioid; Receptors, Opioid, delta; Receptors, Opioid, mu; Thiazoles; Vas Deferens

2001
Modulators of internal Ca2+ stores and the spontaneous electrical and contractile activity of the guinea-pig renal pelvis.
    British journal of pharmacology, 2002, Volume: 135, Issue:6

    Topics: Animals; Boron Compounds; Caffeine; Calcium; Electric Conductivity; Electrophysiology; Estrenes; Guinea Pigs; Indoles; Kidney Pelvis; Macrocyclic Compounds; Muscle Contraction; Muscle, Smooth; Neomycin; Oxazoles; Pyrrolidinones; Ryanodine

2002
[Effects of a new minor tranquilizer, 10-chloro-3-methyl-1 1b-(2-chlorophenyl)-2,3,5,6,7,11b-hexahydrobenzo [6,7]-1,4-diazepino [5,4-b]-oxazol-6-one (CS-386), on the after-discharge and behavior induced by electrical stimulation of the amygdala in freely-
    Nihon yakurigaku zasshi. Folia pharmacologica Japonica, 1977, Volume: 73, Issue:3

    Topics: Administration, Oral; Amygdala; Animals; Anti-Anxiety Agents; Benzodiazepines; Cats; Electric Stimulation; Electroencephalography; Female; Male; Muscle Contraction; Oxazoles; Salivation; Seizures; Time Factors

1977
Pharmacological properties of 2,3-dihydro-9H-isoxazolo[3,2-b]-quinazolin-9-one (W-2429. Part 2: General pharmacological investigation.
    Arzneimittel-Forschung, 1977, Volume: 27, Issue:4

    Topics: Anesthetics, Local; Animals; Anti-Inflammatory Agents, Non-Steroidal; Anticonvulsants; Antidepressive Agents, Tricyclic; Antitussive Agents; Cats; Diuresis; Dogs; Enzyme Induction; Female; Gastrointestinal Hemorrhage; Gastrointestinal Motility; Guinea Pigs; Hemodynamics; Isoxazoles; Male; Mice; Motor Activity; Muscle Contraction; Muscle, Smooth; Oxazoles; Postural Balance; Prostaglandin-Endoperoxide Synthases; Quinazolines; Rabbits; Rats; Respiration; Sleep; Stomach Ulcer; Time Factors

1977
Pharmacological profile of a new psychotherapeutic agent: 4-p-fluorophenyl-5-N(N'-o-methoxyphenyl)piperazinoethyl-4-oxazolin-2-one (LR 511).
    Pharmacology, 1977, Volume: 15, Issue:6

    Topics: Aggression; Analgesics; Animals; Anticonvulsants; Antidepressive Agents; Autonomic Nervous System; Behavior, Animal; Catalepsy; Conditioning, Psychological; Dogs; Drug Synergism; Exploratory Behavior; Female; Humans; Hypnotics and Sedatives; Lethal Dose 50; Male; Mice; Motor Activity; Muscle Contraction; Oxazoles; Piperazines; Psychotropic Drugs; Rabbits; Rats; Tranquilizing Agents

1977
[2-Amino-oxazoles as potential H-bonding agents in virostatic research. 4. Pharmacokinetics and pharmacologic-toxicologic profile of 2-guanidino-4,5-dipropyloxazole hydrochloride].
    Die Pharmazie, 1992, Volume: 47, Issue:5

    Topics: Administration, Oral; Animals; Antiviral Agents; Digestive System; Dogs; Female; Guinea Pigs; Half-Life; Heart Rate; Hydrogen Bonding; In Vitro Techniques; Injections, Subcutaneous; Male; Mice; Muscle Contraction; Myocardial Contraction; Oxazoles; Rabbits; Rats; Rats, Wistar; Swine

1992
Myoplasmic free Mg2+ concentration during repetitive stimulation of single fibres from mouse skeletal muscle.
    The Journal of physiology, 1992, Volume: 453

    Topics: Adenosine Triphosphate; Animals; Benzofurans; Fura-2; Hydrogen-Ion Concentration; Magnesium; Male; Mice; Muscle Contraction; Muscles; Oxazoles; Sodium

1992
A novel protein phosphatase inhibitor, tautomycin. Effect on smooth muscle.
    FEBS letters, 1991, Jul-08, Volume: 285, Issue:1

    Topics: Animals; Antifungal Agents; Aorta; Calcium; Enzyme Inhibitors; Ethers, Cyclic; Guinea Pigs; Kinetics; Macromolecular Substances; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Myosins; Okadaic Acid; Oxazoles; Phosphoprotein Phosphatases; Phosphorylation; Pyrans; Rabbits; Rats; Spiro Compounds; Verapamil

1991
Contraction of rat thoracic aorta strips by endothelin-1 in the absence of extracellular Ca2+.
    British journal of pharmacology, 1991, Volume: 104, Issue:4

    Topics: Animals; Aorta, Thoracic; Caffeine; Calcium; Endothelins; In Vitro Techniques; Indicators and Reagents; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Phorbol 12,13-Dibutyrate; Rats; Rats, Inbred Strains; Tetradecanoylphorbol Acetate; Urotensins; Vasoconstrictor Agents

1991
The effect of azumolene on hypercontractility and sarcoplasmic reticulum Ca(2+)-dependent ATPase activity of malignant hyperpyrexia-susceptible porcine skeletal muscle.
    Clinical and experimental pharmacology & physiology, 1991, Volume: 18, Issue:7

    Topics: Animals; Caffeine; Calcium-Transporting ATPases; Dantrolene; Halothane; Imidazoles; Malignant Hyperthermia; Muscle Contraction; Muscle Relaxants, Central; Muscles; Oxazoles; Potassium Chloride; Sarcoplasmic Reticulum

1991
Modification by calyculin A of inward Ca currents in smooth muscle cells isolated from guinea pig taenia coli.
    Progress in clinical and biological research, 1990, Volume: 327

    Topics: Animals; Benzofurans; Calcium; Enzyme Inhibitors; Fluorescent Dyes; Fura-2; Guinea Pigs; In Vitro Techniques; Intestine, Large; Marine Toxins; Muscle Contraction; Muscle, Smooth; Oxazoles

1990
Calcium-independent activation of contractile apparatus in smooth muscle by calyculin-A.
    The Journal of pharmacology and experimental therapeutics, 1989, Volume: 250, Issue:1

    Topics: 2',3'-Cyclic-Nucleotide Phosphodiesterases; Actomyosin; Animals; Aorta, Thoracic; Ca(2+) Mg(2+)-ATPase; Calcium; Calcium-Transporting ATPases; Cecum; Egtazic Acid; Guinea Pigs; In Vitro Techniques; Kinetics; Male; Marine Toxins; Muscle Contraction; Muscle, Smooth; Muscle, Smooth, Vascular; Myosin-Light-Chain Kinase; Oxazoles; Phosphorylation; Porifera; Rats; Rats, Inbred Strains; Verapamil

1989
[Action of cytochalasin B on the contraction of smooth muscle of guinea pig taenia coli].
    Nihon Heikatsukin Gakkai zasshi, 1989, Volume: 25, Issue:6

    Topics: Animals; Calcium Channels; Colon; Cytochalasin B; Guinea Pigs; In Vitro Techniques; Marine Toxins; Muscle Contraction; Muscle, Smooth; Oxazoles; Potassium

1989
[Effect of calyculin A on the contraction of colonic smooth muscle of guinea pigs].
    Nihon Heikatsukin Gakkai zasshi, 1989, Volume: 25, Issue:6

    Topics: Animals; Calcium; Calcium Channels; Colon; Guinea Pigs; In Vitro Techniques; Marine Toxins; Muscle Contraction; Muscle, Smooth; Oxazoles

1989
New isoxazole derivatives provided with antihypertensive activity.
    Arzneimittel-Forschung, 1989, Volume: 39, Issue:6

    Topics: Animals; Antihypertensive Agents; Aorta, Thoracic; Binding, Competitive; Chemical Phenomena; Chemistry; Clonidine; In Vitro Techniques; Isoxazoles; Magnetic Resonance Spectroscopy; Male; Muscle Contraction; Muscle, Smooth, Vascular; Norepinephrine; Oxazoles; Prazosin; Rats; Rats, Inbred SHR; Rats, Inbred Strains; Rats, Inbred WKY; Vas Deferens; Yohimbine

1989
The effect of EU4093 (azumolene sodium) on the contraction of intrafusal muscle in the soleus muscle of the anaesthetized rat.
    British journal of pharmacology, 1989, Volume: 97, Issue:4

    Topics: Anesthesia; Animals; Electric Stimulation; Female; Imidazoles; In Vitro Techniques; Muscle Contraction; Muscle Relaxants, Central; Muscles; Neurons; Oxazoles; Rats; Rats, Inbred Strains

1989
Prejunctional alpha 2-adrenergic properties of S-3341 (dicyclopropylmethyl)amino-2-delta-2-oxazoline: a comparison with clonidine.
    Canadian journal of physiology and pharmacology, 1987, Volume: 65, Issue:12

    Topics: Adrenergic alpha-Agonists; Animals; Clonidine; Electric Stimulation; In Vitro Techniques; Male; Muscle Contraction; Muscle, Smooth; Neuromuscular Junction; Oxazoles; Prazosin; Rats; Rats, Inbred WKY; Rilmenidine; Vas Deferens; Yohimbine

1987
Synthesis and spasmolytic activity of aminoalkyl 2-substituted-2-(1,2-benzisoxazol-3-yl)acetates.
    Chemical & pharmaceutical bulletin, 1987, Volume: 35, Issue:5

    Topics: Animals; Chemical Phenomena; Chemistry; Guinea Pigs; In Vitro Techniques; Isoxazoles; Male; Muscle Contraction; Oxazoles; Parasympatholytics

1987
Pharmacology of ephedroxanes.
    Journal of ethnopharmacology, 1985, Volume: 13, Issue:2

    Topics: Analgesics; Anesthesia; Animals; Anticonvulsants; Anura; Blepharoptosis; Blood Pressure; Body Temperature; Chickens; Drug Synergism; Electroshock; Guinea Pigs; Heart Rate; Hexobarbital; In Vitro Techniques; Male; Mice; Motor Activity; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Oxazoles; Pentylenetetrazole; Postural Balance; Rats; Rats, Inbred Strains; Strychnine

1985
Vorticella--a model for chemopharmacodynamic action on smooth muscle.
    Comparative and general pharmacology, 1972, Volume: 3, Issue:11

    Topics: Adenosine; Amides; Anesthetics, Local; Animals; Ciliophora; Culture Media; Cyanides; Ferricyanides; Lanthanum; Lead; Models, Biological; Muscle Contraction; Muscle, Smooth; Nicotine; Oxazoles; Papaverine; Phenazines; Potassium Chloride; Tetrazolium Salts; Time Factors; Vitamin K

1972
Actions of clonidine and 2-(2-methyl-6-ethyl-cyclohexylamino)-2-oxazoline on postganglionic autonomic nerves.
    Archives internationales de pharmacodynamie et de therapie, 1972, Volume: 195, Issue:2

    Topics: Acetylcholine; Animals; Antihypertensive Agents; Autonomic Fibers, Postganglionic; Clonidine; Cyclohexylamines; Depression, Chemical; Electric Stimulation; Guinea Pigs; Heart; Heart Rate; Hexamethonium Compounds; Ileum; Imidazoles; In Vitro Techniques; Muscle Contraction; Neurosecretion; Norepinephrine; Oxazoles; Rabbits; Synaptic Transmission

1972
Action of antibiotics on respiratory tract. II. Dicloxacillin.
    Journal of pharmaceutical sciences, 1970, Volume: 59, Issue:8

    Topics: Acetylcholine; Ampicillin; Animals; Barium; Bronchi; Chlorides; Dicloxacillin; Dogs; Ephedrine; Female; Histamine H1 Antagonists; Isoproterenol; Male; Muscle Contraction; Muscle, Smooth; Oxazoles; Penicillins; Respiration; Respiratory System

1970
Effects of isoxazolium cations on some isolated muscle preparations.
    British journal of pharmacology, 1971, Volume: 43, Issue:3

    Topics: Acetylcholine; Angiotensin II; Animals; Aorta; Cholinesterase Inhibitors; Diaphragm; Diphenhydramine; Electric Stimulation; Guinea Pigs; Histamine H1 Antagonists; Ileum; In Vitro Techniques; Muscle Contraction; Muscle, Smooth; Muscles; Norepinephrine; Oxazoles; Parasympathomimetics; Perchlorates; Pilocarpine; Piperazines; Rabbits; Rats; Serotonin Antagonists

1971
The site of action of ibotenic acid and the identification of two populations of glutamate receptors on insect muscle-fibres.
    Comparative and general pharmacology, 1973, Volume: 4, Issue:16

    Topics: Aminobutyrates; Animals; Basidiomycota; Binding, Competitive; Dose-Response Relationship, Drug; Glutamates; Grasshoppers; In Vitro Techniques; Iontophoresis; Membrane Potentials; Membranes; Muscle Contraction; Muscles; Neural Conduction; Neurons; Oxazoles; Perfusion; Picrotoxin; Quaternary Ammonium Compounds; Receptors, Drug; Serotonin; Time Factors; Tryptamines

1973
General pharmacological properties of 4,5-diphenyl-2-bis-(2-hydroxyethyl)-aminoxazol (ditazol).
    Arzneimittel-Forschung, 1973, Volume: 23, Issue:9

    Topics: Amphetamine; Animals; Anti-Inflammatory Agents; Atropine; Blood Pressure; Cats; Chlorpromazine; Ethanolamines; Female; Gastrointestinal Motility; Guinea Pigs; Heart Rate; In Vitro Techniques; Indomethacin; Lethal Dose 50; Male; Meprobamate; Mice; Motor Activity; Muscle Contraction; Oxazoles; Peptic Ulcer; Phenylbutazone; Rabbits; Rats; Reserpine; Seizures; Sleep

1973
Synthesis and biological activity of some 4-aryl-substituted 4-oxazolin-2-ones.
    Journal of medicinal chemistry, 1972, Volume: 15, Issue:1

    Topics: Animals; Barbiturates; Central Nervous System; Cyclization; Guinea Pigs; Ileum; Injections, Intraperitoneal; Ketones; Lethal Dose 50; Mice; Muscle Contraction; Muscles; Oxazoles; Oxidation-Reduction; Structure-Activity Relationship

1972
Distribution of local anesthetics and the intracellular pH in vascular smooth muscle.
    The Journal of pharmacology and experimental therapeutics, 1972, Volume: 181, Issue:3

    Topics: Anesthetics, Local; Animals; Aorta; Binding Sites; Calcium; Carbon Isotopes; Cocaine; Extracellular Space; Hydrogen-Ion Concentration; In Vitro Techniques; Ketones; Kinetics; Lidocaine; Muscle Contraction; Muscle, Smooth; Norepinephrine; Oxazoles; Potassium; Procaine; Rabbits; Structure-Activity Relationship; Tetracaine

1972
[Study of a new myorelaxant combined with an analgesic: Dorsilon].
    Schweizerische Rundschau fur Medizin Praxis = Revue suisse de medecine Praxis, 1970, Jul-28, Volume: 59, Issue:30

    Topics: Acetaminophen; Adult; Analgesics; Catechols; Drug Synergism; Female; Humans; Male; Middle Aged; Muscle Contraction; Muscle Relaxants, Central; Oxazoles

1970
Actions of procaine on nicotine-induced effects in frog sartorius muscle.
    The Journal of pharmacology and experimental therapeutics, 1968, Volume: 160, Issue:1

    Topics: Animals; Anura; Biological Transport; Calcium; Calcium Isotopes; Carbon Isotopes; Depression, Chemical; Hydrogen-Ion Concentration; In Vitro Techniques; Iodoacetates; Muscle Contraction; Muscles; Nialamide; Nicotine; Oxazoles; Procaine; Stimulation, Chemical; Thigh

1968
[Pharmacological and experimental psychological studies with 2 components of fly agaric (Amanita muscaria)].
    Arzneimittel-Forschung, 1968, Volume: 18, Issue:3

    Topics: Animals; Autonomic Nervous System; Basidiomycota; Behavior, Animal; Blood Pressure; Body Temperature; Conditioning, Classical; Electroencephalography; Guinea Pigs; Humans; Mice; Motor Activity; Muscle Contraction; Oxazoles; Psychological Tests; Psychoses, Substance-Induced; Rabbits; Rats; Reflex, Monosynaptic; Respiration

1968