Page last updated: 2024-10-31

methiothepin and Anochlesia

methiothepin has been researched along with Anochlesia in 2 studies

Methiothepin: A serotonin receptor antagonist in the CENTRAL NERVOUS SYSTEM used as an antipsychotic.
methiothepin : A dibenzothiepine that is 10,11-dihydrodibenzo[b,f]thiepine bearing additional methylthio and 4-methylpiperazin-1-yl substituents at positions 8 and 10 respectively. Potent 5-HT2 antagonist, also active as 5-HT1 antagonist. Differentiates 5-HT1D sub-types. Also displays affinity for rodent 5-HT5B, 5-HT5A, 5-HT7 and 5-HT6 receptors (pK1 values are 6.6, 7.0, 8.4 and 8.7 respectively).

Research

Studies (2)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's1 (50.00)29.6817
2010's1 (50.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Campiani, G1
Butini, S1
Gemma, S1
Nacci, V1
Fattorusso, C1
Catalanotti, B1
Giorgi, G1
Cagnotto, A1
Goegan, M1
Mennini, T1
Minetti, P1
Di Cesare, MA1
Mastroianni, D1
Scafetta, N1
Galletti, B1
Stasi, MA1
Castorina, M1
Pacifici, L1
Ghirardi, O1
Tinti, O1
Carminati, P1
Kołaczkowski, M1
Marcinkowska, M1
Bucki, A1
Pawłowski, M1
Mitka, K1
Jaśkowska, J1
Kowalski, P1
Kazek, G1
Siwek, A1
Wasik, A1
Wesołowska, A1
Mierzejewski, P1
Bienkowski, P1

Other Studies

2 other studies available for methiothepin and Anochlesia

ArticleYear
Pyrrolo[1,3]benzothiazepine-based atypical antipsychotic agents. Synthesis, structure-activity relationship, molecular modeling, and biological studies.
    Journal of medicinal chemistry, 2002, Jan-17, Volume: 45, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Animals; Antipsychotic Agents; Behavior, Animal; Brain; Catalepsy; C

2002
Novel arylsulfonamide derivatives with 5-HT₆/5-HT₇ receptor antagonism targeting behavioral and psychological symptoms of dementia.
    Journal of medicinal chemistry, 2014, Jun-12, Volume: 57, Issue:11

    Topics: Animals; Antidepressive Agents; Antipsychotic Agents; Avoidance Learning; Benzoxazoles; Catalepsy; C

2014