Page last updated: 2024-08-24

loxiglumide and Muscle Contraction

loxiglumide has been researched along with Muscle Contraction in 23 studies

Research

Studies (23)

TimeframeStudies, this research(%)All Research%
pre-19903 (13.04)18.7374
1990's20 (86.96)18.2507
2000's0 (0.00)29.6817
2010's0 (0.00)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
D'Amato, M; Rovati, LC1
Fujii, K; Haruma, K; Kajiyama, G; Kishimoto, S; Kobayashi, H; Machino, H; Miyoshi, A1
Mantovani, P; Milenov, K; Rakovska, A; Sgaragli, G; Valoti, M1
Barbara, G; Barbara, L; Corinaldesi, R; De Giorgio, R; Franzoso, L; Go, VL; Morselli-Labate, AM; Ricci Maccarini, M; Rovati, LC; Stanghellini, V1
Milenov, K; Rakovska, A1
Brotschi, EA; Hilbinger, CL; Kahl, EA; Midis, NA; Vaules, WA1
Endo, T; Nagasaki, M; Taniguchi, H; Yazaki, N1
Adorni Ugolotti, MC; Mantovani, P; Rakowska, A; Valoti, M1
Kondo, T; Liu, F; Naruse, S; Ozaki, T; Sazi, T; Toda, Y1
Hayashi, K; Kannbe, M; Kishimoto, S1
Azpiroz, F; Clavé, P; Cussó, X; D'Amato, M; Farré, A; González, A; Lluís, F; López, R; Moreno, A1
Chijiiwa, Y; Harada, N; Misawa, T; Nawata, H; Yoshinaga, M1
Almegård, B; Bill, A; Stjernschantz, J1
Choudhury, AR; Creutzfeldt, W; Fölsch, UR; Höcker, M; Nitsche, R; Nustede, R; Rovati, LC; Schleser, A; Schmidt, WE; Sostmann, H1
Karaus, M; Niederau, C1
Bennett, A; D'Amato, M; Stamford, IF1
Choudhury, AR; Creutzfeldt, W; Fölsch, UR; Höcker, M; Nitsche, R; Nustede, R; Rovati, LC; Schafmayer, A; Schleser, A; Schmidt, WE1
Biliotti, D; Bontempo, I; Corazziari, E; De Medici, A; Pallotta, N; Ricci, R; Torsoli, A1
Bonato, C; De Fazio, C; Festorazzi, S; Malesci, A; Rovati, L; Setnikar, I; Tacconi, M; Valentini, A1
Baba, H; Fujimura, M; Toda, N1
Fujii, K; Kishimoto, M; Miyoshi, A1
Bogdal, J; Konturek, JW; Konturek, SJ; Kurek, A; Oleksy, J; Rovati, L1
Douglas, BR; Jansen, JB; Jebbink, MC; Lamers, CB; Tjon a Tham, RT1

Trials

2 trial(s) available for loxiglumide and Muscle Contraction

ArticleYear
Cholecystokinin receptor antagonist loxiglumide: influence on bilio-pancreatic secretion and gastrointestinal hormones in man.
    Digestion, 1990, Volume: 46 Suppl 2

    Topics: Adult; Cholecystokinin; Gallbladder; Humans; Male; Muscle Contraction; Muscle, Smooth; Pancreas; Proglumide; Radioimmunoassay; Receptors, Cholecystokinin

1990
Oral administration of loxiglumide (CCK antagonist) inhibits postprandial gallbladder contraction without affecting gastric emptying.
    Digestive diseases and sciences, 1990, Volume: 35, Issue:1

    Topics: Administration, Oral; Adult; Cholecystokinin; Double-Blind Method; Female; Food; Gallbladder; Gastric Emptying; Glutamine; Humans; Male; Muscle Contraction; Proglumide; Random Allocation

1990

Other Studies

21 other study(ies) available for loxiglumide and Muscle Contraction

ArticleYear
CCK-A antagonists: which and how.
    European journal of clinical investigation, 1995, Volume: 25, Issue:3

    Topics: Benzodiazepinones; Devazepide; Gallbladder; Humans; Muscle Contraction; Muscle, Smooth; Proglumide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Stereoisomerism

1995
Inhibitory action of CCK-OP on rat proximal colon.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Acetylcholine; Animals; Atropine; Colon; Fasting; Hexamethonium; Hexamethonium Compounds; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Proglumide; Rats; Receptors, Cholecystokinin; Sincalide

1994
Effect of loxiglumide (CR 1505) on CCK-induced contractions and 3H-acetylcholine release from guinea-pig gallbladder.
    Neuropeptides, 1993, Volume: 25, Issue:5

    Topics: Acetylcholine; Animals; Cholecystokinin; Female; Gallbladder; Guinea Pigs; In Vitro Techniques; Male; Muscle Contraction; Proglumide; Tritium

1993
Effects of dietary fat on postprandial gastrointestinal motility are inhibited by a cholecystokinin type A receptor antagonist.
    Annals of the New York Academy of Sciences, 1994, Mar-23, Volume: 713

    Topics: Adult; Corn Oil; Dietary Fats; Duodenum; Eating; Female; Gastrointestinal Motility; Humans; Infusions, Intravenous; Male; Manometry; Muscle Contraction; Muscle, Smooth; Proglumide; Pyloric Antrum; Random Allocation; Receptors, Cholecystokinin

1994
Neuronal receptors for caerulein in gallbladder.
    Journal of physiology, Paris, 1993, Volume: 87, Issue:6

    Topics: Acetylcholine; Animals; Ceruletide; Gallbladder; Guinea Pigs; Muscle Contraction; Neurons; Proglumide; Receptors, Cholecystokinin

1993
Luminal cholecystokinin and gastrin cause gallbladder contraction.
    The Journal of surgical research, 1996, Volume: 62, Issue:2

    Topics: Animals; Bile; Cholecystokinin; Female; Gallbladder; Gastrins; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Muscle Contraction; Pentagastrin; Proglumide; Receptors, Cholecystokinin; Sincalide

1996
Pharmacological profile of T-0632, a novel potent and selective CCKA receptor antagonist, in vitro.
    European journal of pharmacology, 1996, May-23, Volume: 304, Issue:1-3

    Topics: Amylases; Animals; Benzodiazepinones; Binding, Competitive; Brain; Cell Membrane; Devazepide; Gallbladder; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Indoles; Male; Muscle Contraction; Muscle, Smooth; Pancreas; Proglumide; Protein Binding; Rabbits; Rats; Rats, Sprague-Dawley; Receptors, Cholecystokinin; Sincalide

1996
Ca2+ antagonists reveal a novel inhibitory effect of caerulein on guinea pig ileum.
    Methods and findings in experimental and clinical pharmacology, 1995, Volume: 17, Issue:5

    Topics: Acetylcholine; Animals; Calcium Channel Blockers; Ceruletide; Dibutyryl Cyclic GMP; Electric Stimulation; Female; Gastrointestinal Agents; Guinea Pigs; Hormone Antagonists; Ileum; Male; Muscle Contraction; Muscle, Smooth; Proglumide

1995
Effect of gastrin-releasing peptide (GRP) on guinea pig gallbladder contraction in vitro.
    Journal of gastroenterology, 1995, Volume: 30, Issue:6

    Topics: Acetylcholine; Animals; Atropine; Bombesin; Dose-Response Relationship, Drug; Gallbladder; Gastrin-Releasing Peptide; Guinea Pigs; Hormone Antagonists; In Vitro Techniques; Male; Muscarinic Antagonists; Muscle Contraction; Muscle, Smooth; Peptides; Proglumide; Sincalide

1995
Endogenous CCK inhibits colonic contractions in unrestrained conscious rats.
    Regulatory peptides, 1997, Oct-31, Volume: 72, Issue:2-3

    Topics: Animal Feed; Animals; Colon; Dose-Response Relationship, Drug; Duodenum; Eating; Fasting; Gastrointestinal Motility; Hormone Antagonists; Intubation, Gastrointestinal; Male; Muscle Contraction; Muscle, Smooth; Portal Vein; Proglumide; Radioimmunoassay; Rats; Rats, Wistar; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Reference Values; Sincalide; Telemetry; Transducers

1997
Endogenous cholecystokinin enhances postprandial gastroesophageal reflux in humans through extrasphincteric receptors.
    Gastroenterology, 1998, Volume: 115, Issue:3

    Topics: Adult; Cholecystokinin; Cholestyramine Resin; Eating; Electric Stimulation; Esophagogastric Junction; Esophagus; Gallbladder; Gastroesophageal Reflux; Humans; Hydrogen-Ion Concentration; In Vitro Techniques; Male; Muscle Contraction; Muscle Relaxation; Muscle, Smooth; Proglumide; Receptor, Cholecystokinin A; Receptors, Cholecystokinin; Sincalide

1998
Direct contractile effect of motilin on isolated smooth muscle cells of guinea pig small intestine.
    Life sciences, 1992, Volume: 51, Issue:17

    Topics: Animals; Atropine; Calcium; Cholecystokinin; Guinea Pigs; In Vitro Techniques; Intestine, Small; Male; Motilin; Muscle Contraction; Muscle, Smooth; Proglumide; Substance P

1992
Cholecystokinin contracts isolated human and monkey iris sphincters; a study with CCK receptor antagonists.
    European journal of pharmacology, 1992, Feb-11, Volume: 211, Issue:2

    Topics: Aged; Aged, 80 and over; Animals; Cholecystokinin; Female; Humans; In Vitro Techniques; Iris; Macaca fascicularis; Male; Middle Aged; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide

1992
Role of CCK in regulation of pancreaticobiliary functions and GI motility in humans: effects of loxiglumide.
    The American journal of physiology, 1991, Volume: 260, Issue:2 Pt 1

    Topics: Adult; Bilirubin; Cholecystokinin; Eating; Feces; Gallbladder; Gastrointestinal Motility; Humans; Lipase; Lipid Metabolism; Male; Muscle Contraction; Muscle, Smooth; Pancreas; Pancreatic Juice; Proglumide; Reference Values; Trypsin

1991
Effects of CCK receptor blockade on intestinal motor activity in conscious dogs.
    The American journal of physiology, 1991, Volume: 260, Issue:2 Pt 1

    Topics: Animals; Ceruletide; Cholecystokinin; Digestion; Dogs; Eating; Female; Gastrointestinal Motility; Male; Muscle Contraction; Myoelectric Complex, Migrating; Neostigmine; Proglumide; Receptors, Cholecystokinin

1991
Studies of three non-peptide cholecystokinin antagonists (devazepide, lorglumide and loxiglumide) in human isolated alimentary muscle and guinea-pig ileum.
    British journal of pharmacology, 1991, Volume: 102, Issue:2

    Topics: Animals; Benzodiazepinones; Cholecystokinin; Devazepide; Digestive System; Digestive System Physiological Phenomena; Female; Guinea Pigs; Humans; Ileum; In Vitro Techniques; Male; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide

1991
Effect of loxiglumide on gallbladder contractile response to cerulein and food in humans.
    Gastroenterology, 1990, Volume: 98, Issue:5 Pt 1

    Topics: Adult; Ceruletide; Cholecystokinin; Dose-Response Relationship, Drug; Drug Interactions; Feeding Behavior; Gallbladder; Glutamine; Humans; Male; Muscle Contraction; Proglumide; Reference Values; Time Factors

1990
Mechanism of inhibitory action of peptide YY on cholecystokinin-induced contractions of isolated dog ileum.
    Regulatory peptides, 1990, Feb-04, Volume: 27, Issue:2

    Topics: Animals; Cholecystokinin; Dogs; Female; Gallbladder; Glutamine; Ileum; Isometric Contraction; Male; Muscle Contraction; Peptide YY; Peptides; Proglumide; Sincalide

1990
[Effect of CCK on the large intestine].
    Nihon Heikatsukin Gakkai zasshi, 1989, Volume: 25, Issue:5

    Topics: Animals; Cholecystokinin; Gastrointestinal Motility; Glutamine; Intestine, Large; Male; Muscle Contraction; Muscle, Smooth; Proglumide; Rats; Rats, Inbred Strains

1989
CCK receptor antagonism by loxiglumide and gall bladder contractions in response to cholecystokinin, sham feeding and ordinary feeding in man.
    Gut, 1989, Volume: 30, Issue:8

    Topics: Adolescent; Adult; Cholecystokinin; Food; Gallbladder; Glutamine; Humans; Male; Muscle Contraction; Proglumide; Receptors, Cholecystokinin; Sincalide

1989
The effect of loxiglumide (CR-1505) on basal and bombesin-stimulated gallbladder volume in man.
    European journal of pharmacology, 1989, Jul-18, Volume: 166, Issue:2

    Topics: Adult; Bombesin; Cholecystokinin; Female; Gallbladder; Humans; Male; Muscle Contraction; Muscle, Smooth; Proglumide; Time Factors

1989