lobeline and Amphetamine Abuse

lobeline has been researched along with Amphetamine Abuse in 13 studies

Research

Studies (13)

TimeframeStudies, this research(%)All Research%
pre-19900 (0.00)18.7374
1990's0 (0.00)18.2507
2000's4 (30.77)29.6817
2010's9 (69.23)24.3611
2020's0 (0.00)2.80

Authors

AuthorsStudies
Crooks, PA; Dwoskin, LP; Kangiser, MM; Stairs, DJ; Zheng, G1
Bardo, MT; Crooks, PA; Dwoskin, LP; Lee, NR; Zheng, G1
Crooks, PA; Dwoskin, LP; Nickell, JR; Siripurapu, KB; Vartak, A1
Crooks, PA; Ding, D; Dwoskin, LP; Nickell, JR1
Crooks, PA; Deaciuc, G; Dwoskin, LP; Krishnamurthy, S; Nickell, JR; Norrholm, S; Siripurapu, KB; Zheng, G1
Bardo, MT; Beckmann, JS; Crooks, PA; Denehy, ED; Dwoskin, LP; Horton, DB; Nickell, JR; Siripurapu, KB; Vartak, A1
Crooks, PA; Dwoskin, LP; Horton, DB; Siripurapu, KB; Zheng, G1
Daniels, WM; Dimatelis, JJ; Russell, VA; Stein, DJ1
Alvers, KM; Bardo, MT; Beckmann, JS; Crooks, PA; Dwoskin, LP; Zheng, G1
Bardo, MT; Crooks, PA; Dwoskin, LP; Harrod, SB; Neugebauer, NM; Stairs, DJ1
Eshleman, AJ; Janowsky, A; Johnson, RA; Wilhelm, CJ1
Bardo, MT; Crooks, PA; Dwoskin, LP; Harrod, SB; Klebaur, JE1
Crooks, PA; Dwoskin, LP1

Reviews

2 review(s) available for lobeline and Amphetamine Abuse

ArticleYear
The vesicular monoamine transporter-2: an important pharmacological target for the discovery of novel therapeutics to treat methamphetamine abuse.
    Advances in pharmacology (San Diego, Calif.), 2014, Volume: 69

    Topics: Amphetamine-Related Disorders; Animals; Drug Delivery Systems; Drug Discovery; Humans; Lobeline; Methamphetamine; Protein Binding; Treatment Outcome; Vesicular Monoamine Transport Proteins

2014
A novel mechanism of action and potential use for lobeline as a treatment for psychostimulant abuse.
    Biochemical pharmacology, 2002, Jan-15, Volume: 63, Issue:2

    Topics: Amphetamine-Related Disorders; Central Nervous System; Dopamine; Forecasting; Ganglionic Stimulants; Humans; Lobeline; Methamphetamine

2002

Other Studies

11 other study(ies) available for lobeline and Amphetamine Abuse

ArticleYear
Varenicline and GZ-793A differentially decrease methamphetamine self-administration under a multiple schedule of reinforcement in rats.
    Behavioural pharmacology, 2018, Volume: 29, Issue:1

    Topics: Amphetamine-Related Disorders; Animals; Behavior, Addictive; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Lobeline; Male; Methamphetamine; Rats; Rats, Sprague-Dawley; Reinforcement Schedule; Reinforcement, Psychology; Self Administration; Substance-Related Disorders; Varenicline

2018
New Scaffold for Lead Compounds to Treat Methamphetamine Use Disorders.
    The AAPS journal, 2018, 02-09, Volume: 20, Issue:2

    Topics: Administration, Oral; Amphetamine-Related Disorders; Animals; Cardiotoxicity; Disease Models, Animal; Dopamine; Ether-A-Go-Go Potassium Channels; Humans; Lobeline; Locomotion; Male; Methamphetamine; Molecular Structure; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Treatment Outcome; Vesicular Monoamine Transport Proteins

2018
Quinolyl analogues of norlobelane: novel potent inhibitors of [(3)H]dihydrotetrabenazine binding and [(3)H]dopamine uptake at the vesicular monoamine transporter-2.
    Bioorganic & medicinal chemistry letters, 2015, Jul-01, Volume: 25, Issue:13

    Topics: Amphetamine-Related Disorders; Animals; Binding Sites; Dopamine; Humans; In Vitro Techniques; Kinetics; Lobeline; Methamphetamine; Rats; Structure-Activity Relationship; Synaptic Vesicles; Tetrabenazine; Vesicular Monoamine Transport Proteins

2015
Lobelane inhibits methamphetamine-evoked dopamine release via inhibition of the vesicular monoamine transporter-2.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 332, Issue:2

    Topics: 3,4-Dihydroxyphenylacetic Acid; Amphetamine-Related Disorders; Animals; Corpus Striatum; Dopamine; Dopamine Plasma Membrane Transport Proteins; Drug Evaluation, Preclinical; Lobeline; Male; Methamphetamine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Structure-Activity Relationship; Synaptic Vesicles; Synaptosomes; Vesicular Monoamine Transport Proteins

2010
The novel pyrrolidine nor-lobelane analog UKCP-110 [cis-2,5-di-(2-phenethyl)-pyrrolidine hydrochloride] inhibits VMAT2 function, methamphetamine-evoked dopamine release, and methamphetamine self-administration in rats.
    The Journal of pharmacology and experimental therapeutics, 2010, Volume: 335, Issue:3

    Topics: 3,4-Dihydroxyphenylacetic Acid; Aconitine; Amphetamine-Related Disorders; Animals; Behavior, Animal; Cell Membrane; Conditioning, Operant; Corpus Striatum; Dopamine; Drug Tolerance; Lobeline; Male; Methamphetamine; Nicotine; Protein Binding; Pyrrolidines; Rats; Rats, Sprague-Dawley; Receptors, Nicotinic; Reinforcement, Psychology; Self Administration; Synaptic Vesicles; Tetrabenazine; Vesicular Monoamine Transport Proteins

2010
Novel N-1,2-dihydroxypropyl analogs of lobelane inhibit vesicular monoamine transporter-2 function and methamphetamine-evoked dopamine release.
    The Journal of pharmacology and experimental therapeutics, 2011, Volume: 339, Issue:1

    Topics: Amphetamine-Related Disorders; Animals; Binding, Competitive; Corpus Striatum; Data Interpretation, Statistical; Dopamine; Dopamine Uptake Inhibitors; Kinetics; Lobeline; Male; Methamphetamine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Serotonin; Serotonin Plasma Membrane Transport Proteins; Structure-Activity Relationship; Synaptic Vesicles; Synaptosomes; Vesicular Monoamine Transport Proteins

2011
The effects of lobeline and naltrexone on methamphetamine-induced place preference and striatal dopamine and serotonin levels in adolescent rats with a history of maternal separation.
    Metabolic brain disease, 2012, Volume: 27, Issue:3

    Topics: Age Factors; Amphetamine-Related Disorders; Animals; Animals, Newborn; Corpus Striatum; Female; Lobeline; Male; Maternal Deprivation; Naltrexone; Narcotic Antagonists; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Stress, Psychological; Vesicular Monoamine Transport Proteins

2012
The effect of VMAT2 inhibitor GZ-793A on the reinstatement of methamphetamine-seeking in rats.
    Psychopharmacology, 2012, Volume: 224, Issue:2

    Topics: Amphetamine-Related Disorders; Animals; Drug-Seeking Behavior; Illicit Drugs; Lobeline; Male; Methamphetamine; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Vesicular Monoamine Transport Proteins

2012
Lobelane decreases methamphetamine self-administration in rats.
    European journal of pharmacology, 2007, Sep-24, Volume: 571, Issue:1

    Topics: Amphetamine-Related Disorders; Animals; Central Nervous System Stimulants; Dose-Response Relationship, Drug; Infusions, Intravenous; Lobeline; Male; Methamphetamine; Molecular Structure; Motor Activity; Rats; Rats, Sprague-Dawley; Self Administration; Sucrose

2007
Lobeline effects on tonic and methamphetamine-induced dopamine release.
    Biochemical pharmacology, 2008, Mar-15, Volume: 75, Issue:6

    Topics: Amphetamine-Related Disorders; Cell Line; Cocaine; Dopamine; Dopamine Agents; Dopamine Plasma Membrane Transport Proteins; Dopamine Uptake Inhibitors; Humans; Lobeline; Methamphetamine; Nomifensine; Reserpine; Vesicular Monoamine Transport Proteins

2008
Lobeline attenuates d-methamphetamine self-administration in rats.
    The Journal of pharmacology and experimental therapeutics, 2001, Volume: 298, Issue:1

    Topics: Amphetamine-Related Disorders; Animals; Dopamine; Dopamine Uptake Inhibitors; Dose-Response Relationship, Drug; Lobeline; Male; Methamphetamine; Nicotinic Agonists; Rats; Rats, Sprague-Dawley; Reinforcement, Psychology; Self Administration; Sucrose

2001